CAS: 1093100-40-3

B-Raf inhibitor 1

Raf inhibitor 1

B-Raf inhibitor 1 is a small molecule that binds to the active conformation of B-Raf, inhibiting its kinase activity. The compound was discovered by screening a library of compounds for conformational specificity and found to be selective for the active conformation of B-Raf. This drug has been shown to inhibit cellular proliferation in vitro and in vivo. Molecular modeling studies have shown that this inhibitor has a high binding affinity for the active conformation of B-Raf. Kinase inhibitors are used as cancer therapy because they inhibit cell growth by blocking the enzyme kinase, which is involved in the transmission of signals from outside to inside cells.

B-Raf inhibitor 1 (B-Raf inhibitor 1) is a potent and selective B-Raf inhibitor.