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CAS 121204-87-3: (ala,1,3,11,15)-endothelin-1

Formula:C109H163N25O32S
InChI:InChI=1/C109H163N25O32S/c1-16-56(9)86(113)104(159)134-88(57(10)17-2)106(161)129-78(43-64-47-115-69-28-22-21-27-67(64)69)108(163)166-109(164)79(46-84(141)142)128-97(152)72(39-53(3)4)124-99(154)75(44-65-48-114-52-116-65)122-90(145)59(12)118-96(151)73(41-62-25-19-18-20-26-62)125-98(153)74(42-63-30-32-66(138)33-31-63)126-105(160)87(55(7)8)133-92(147)61(14)117-94(149)71(121-95(150)70(29-23-24-37-110)120-100(155)76(45-83(139)140)123-93(148)68(112)36-38-167-15)34-35-85(143)165-107(162)77(40-54(5)6)127-102(157)82(51-137)132-103(158)81(50-136)131-91(146)60(13)119-101(156)80(49-135)130-89(144)58(11)111/h18-22,25-28,30-33,47-48,52-61,65,68,70-82,86-88,115,135-138H,16-17,23-24,29,34-46,49-51,110-113H2,1-15H3,(H,117,149)(H,118,151)(H,119,156)(H,120,155)(H,121,150)(H,122,145)(H,123,148)(H,124,154)(H,125,153)(H,126,160)(H,127,157)(H,128,152)(H,129,161)(H,130,144)(H,131,146)(H,132,158)(H,133,147)(H,134,159)(H,139,140)(H,141,142)/t56-,57-,58-,59-,60-,61-,65?,68-,70-,71-,72-,73-,74-,75-,76-,77-,78-,79-,80-,81-,82-,86-,87-,88-/m0/s1
SMILES:CC[C@H](C)[C@@H](C(=N[C@@H]([C@@H](C)CC)C(=N[C@@H](Cc1c[nH]c2ccccc12)C(=O)OC(=O)[C@H](CC(=O)O)N=C([C@H](CC(C)C)N=C([C@H](CC1C=NC=N1)N=C([C@H](C)N=C([C@H](Cc1ccccc1)N=C([C@H](Cc1ccc(cc1)O)N=C([C@H](C(C)C)N=C([C@H](C)N=C([C@H](CCC(=O)OC(=O)[C@H](CC(C)C)N=C([C@H](CO)N=C([C@H](CO)N=C([C@H](C)N=C([C@H](CO)N=C([C@H](C)N)O)O)O)O)O)N=C([C@H](CCCCN)N=C([C@H](CC(=O)O)N=C([C@H](CCSC)N)O)O)O)O)O)O)O)O)O)O)O)O)O)N
Synonyms:
  • (Ala131115)-Endothelin-1
  • H-Ala-Ser-Ala-Ser-Ser-Leu-Met-Asp-Lys-Glu-Ala-Val-Tyr-Phe-Ala-His-Leu-Asp-Ile-Ile-Trp-OH
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Found 4 products.
  • [Ala1,3,11,15]-Endothelin 1
    Glentham
    + Info

    [Ala1,3,11,15]-Endothelin 1

    CAS:
    Formula:C109H163N25O32S
    Purity:≥ 95.0%
    Color and Shape:White solid
    Molecular weight:2367.67

    Ref: 7W-GK1126

    ne
    To inquire
  • (Ala1·3·11·15)-Endothelin-1 trifluoroacetate salt
    Biosynth
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    (Ala1·3·11·15)-Endothelin-1 trifluoroacetate salt

    CAS:
    (Ala1·3·11·15)-Endothelin-1 trifluoroacetate salt H-Ala-Ser-Ala-Ser-Ser-Leu-Met-Asp-Lys-Glu-Ala-Val-Tyr-Phe-Ala-His-Leu) is a phorbol ester, which is an analog of endothelin. It has been shown to inhibit the production of proinflammatory cytokines and chemokines in vitro and in vivo. This compound also inhibits the migration and proliferation of vascular endothelial cells, which may be due to its ability to suppress Ca2+ concentration. (Ala1·3·11·15)-Endothelin -1 trifluoroacetate salt H-) can also be used as a fluorescent marker for immunohistochemical studies on tissues such as vessels and gastrointestinal tissues. The localization of this drug can be observed by microscopy techniques such as
    Formula:C109H163N25O32S
    Purity:Min. 95%
    Molecular weight:2,367.68 g/mol

    Ref: 3D-FA108867

    1mg
    349.00€
    2mg
    550.00€
    5mg
    1,019.00€
    10mg
    1,707.00€
    500µg
    315.00€
  • (Ala¹·³·¹¹·¹⁵)-Endothelin-1
    Bachem
    + Info

    (Ala¹·³·¹¹·¹⁵)-Endothelin-1

    CAS:
    4 Ala ET-1, linear analog of ET-1 is a selective agonist for ET-B receptors.
    Formula:C109H163N25O32S
    Purity:95.5%
    Color and Shape:White Powder
    Molecular weight:2367.71

    Ref: 01-4030582

    1mg
    203.00€
    0.5mg
    116.00€
  • [Ala1,3,11,15]-Endothelin
    Targetmol
    + Info

    [Ala1,3,11,15]-Endothelin

    CAS:
    Selective ETB endothelin receptor agonist (IC50 values are 0.33 and 2200 nM for displacing [125I]-ET-1 from ETB and ETA receptors respectively).
    Formula:C109H163N25O32S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:2368

    Ref: TM-TP2099

    5mg
    477.00€