CAS: 1793080-72-4

VX-150 is a highly selective NaV1.8 inhibitor relative to the other sodium channel subtypes (>400-fold).

VX-150 is a medicinal compound that acts as a potent inhibitor of kinases, which are enzymes that play a critical role in the regulation of cellular processes such as apoptosis and protein synthesis. This inhibitor has been shown to be effective against various types of cancer cells, including those found in human and Chinese patients. VX-150 works by binding to the kinase domain of the target protein, thereby blocking its activity and inhibiting tumor growth. This analog has been found to be particularly effective against urinary tract tumors and is being investigated as a potential anticancer agent.

VX-150