CAS: 186543-64-6

LY 344864 racemate

Ly 344864 is a peptide agonist of the β-adrenergic receptor, which is expressed in cells of the heart and blood vessels. It activates these receptors by binding to them and stimulating intracellular signaling pathways. Ly 344864 has been shown to be a high-affinity ligand for the β-adrenergic receptor, with a Kd value of 0.3 nM in competition binding assays. This means that Ly 344864 binds to the receptor with high affinity and selectivity, without activating other receptors or ion channels. Ly 344864 has also been shown to inhibit voltage-gated potassium channels in vitro, suggesting that it may have potential as an antihypertensive agent.

LY 344864 racemate is a 5-HT1F receptor agonist.