CAS 29868-97-1: Pirenzepine hydrochloride
Formula:C19H21N5O2·2ClH
InChI:InChI=1S/C19H21N5O2.2ClH/c1-22-9-11-23(12-10-22)13-17(25)24-16-7-3-2-5-14(16)19(26)21-15-6-4-8-20-18(15)24;;/h2-8H,9-13H2,1H3,(H,21,26);2*1H
InChI key:InChIKey=FFNMBRCFFADNAO-UHFFFAOYSA-N
SMILES:C(CN1CCN(C)CC1)(=O)N2C=3C(NC(=O)C=4C2=CC=CC4)=CC=CN3.Cl
Synonyms:- 11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6H-pyrido[2,3-b][1,4]benzodiazepin-6-one dihydrochloride
- 11-[2-(4-methylpiperazin-1-yl)acetyl]-5H-pyrido[2,3-b][1,4]benzodiazepin-6-one hydrate hydrochloride
- 5,11-Dihydro-11-((4-methylpiperazin-1-yl)acetyl)-6H-pyrido(2,3-b)-(1,4)benzodiazepin-6-one dihydrochloride
- 5,11-Dihydro-11-[(4-methyl-1-piperazinyl)acetyl]-6H-pyrido[2,3-b][1,4]benzodiazepin-6-one dihydrochloride
- 6H-Pyrido[2,3-b][1,4]benzodiazepin-6-one, 5,11-dihydro-11-[(4-methyl-1-piperazinyl)acetyl]-, dihydrochloride
- 6H-Pyrido[2,3-b][1,4]benzodiazepin-6-one, 5,11-dihydro-11-[2-(4-methyl-1-piperazinyl)acetyl]-, hydrochloride (1:2)
- Duogastral
- Durapirenz
- Gasteril
- Gastricur
- Gastrozepin
- See more synonyms
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Found 12 products.
PIRENZEPINE DIHYDROCHLORIDE MONOHYDRATE CRS
CAS:PIRENZEPINE DIHYDROCHLORIDE MONOHYDRATE CRSFormula:C19H23Cl2N5O2Color and Shape:Crystalline Powder. White. Light Yellow. Powder., Crystalline Powder. White. Light Yellow. Powder.Molecular weight:424.3242Pirenzepine dihydrochloride
CAS:Formula:C19H21N5O2·2HClPurity:98.0 - 102.0 % (dried basis)Color and Shape:White to off-white or pale yellow powderMolecular weight:424.32Pirenzepine dihydrochloride
CAS:Pirenzepine is a nonsteroidal anti-inflammatory drug and prokinetic agent used to treat bowel disease. It is also used to treat pancreatic enzyme deficiency, which can result in chronic diarrhea. Pirenzepine has been shown to inhibit protease activity in mouse serum, and it has been reported that this inhibition may be due to its ability to bind with amyloid protein and prevent amyloid aggregation. Pirenzepine also suppresses inflammatory responses by inhibiting the production of inflammatory mediators such as leukotrienes, prostaglandins, and cytokines, thereby providing therapeutic benefits for treating chronic bronchitis and other inflammatory diseases. Pirenzepine is metabolized in the liver by the cytochrome P450 enzyme system into an active form called pirenzepine N-oxide. This active form is then metabolized by hydrolysis or glucuronidation before excretion from the body. The most common sideFormula:C19H23Cl2N5O2Purity:Min. 95%Color and Shape:White PowderMolecular weight:424.32 g/molPirenzepine-d8 Dihydrochloride
CAS:Controlled ProductFormula:C19H15D8Cl2N5O2Color and Shape:NeatMolecular weight:432.37Pirenzepine Dihydrochloride
CAS:Formula:C19H21N5O2·2HClPurity:>98.0%(T)(HPLC)Color and Shape:White to Yellow to Orange powder to crystalMolecular weight:424.33Pirenzepine dihydrochloride
CAS:Formula:C19H23Cl2N5O2Purity:%Color and Shape:SolidMolecular weight:424.3242Pirenzepine-d10 Dihydrochloride
CAS:Controlled ProductApplications Pirenzepine-d10 Dihydrochloride is an analogue of Pirenzepine (P508500), an antiucerative agent that works by inhibiting tricyclic gastric-acid secretion. References Fliri, A . F., et al.: J. Med. Chem., 52, 8038 (2009); Eberlein, W., et al.: Arzneimittel-Forsch., 27, 356 (1977), Hellerr, G., et al.: Verh. Deut. Ges. Inn. Med., 84, 991 (1978), Carmine, A.A., et al.: Drugs, 30,85 (1985), El-Obeid, H.A., et al.: Anal. Profiles Drug Subs., 16, 445 (1987), Homon, C.A., et al.: Ther. Drug Monit., 9, 236 (1987),Formula:C19H12D11Cl2N5O2Color and Shape:BrownMolecular weight:435.39Pirenzepine, Dihydrochloride
CAS:Controlled ProductApplications An antiulcerative. Tricyclic gastric-acid inhibitor. References Eberlein, W., et al.: Arzneimittel-Forsch., 27, 356 (1977), Hellerr, G., et al.: Verh. Deut. Ges. Inn. Med., 84, 991 (1978), Carmine, A.A., et al.: Drugs, 30,85 (1985), El-Obeid, H.A., et al.: Anal. Profiles Drug Subs., 16, 445 (1987), Homon, C.A., et al.: Ther. Drug Monit., 9, 236 (1987),Formula:C19H21N5O2·2ClHColor and Shape:NeatMolecular weight:424.32Pirenzepine dihydrochloride, 99%
CAS:A M1 muscarinic receptor antagonist This Thermo Scientific Chemicals brand product was originally part of the Alfa Aesar product portfolio. Some documentation and label information may refer to the legacy brand. The original Alfa Aesar product / item code or SKU reference has not changed as a part of the brand transition to Thermo Scientific Chemicals.Formula:C19H23Cl2N5O2Purity:99%Color and Shape:Crystals or powder or crystalline powder, White to pale yellowMolecular weight:424.33
