CAS: 913827-99-3

CS 2100

CS 2100 is a high-specificity, ethyl-group-containing, blood pressure stabilizer that acts as a serotonin reuptake inhibitor. It has been shown to have efficacy in the treatment of angina and stabilizing cardiac function. CS 2100 has also been used in clinical studies for the treatment of pulmonary embolism, where it was found to reduce the incidence of pulmonary hypertension. CS 2100 binds to serotonin receptors and blocks serotonin reuptake, which enhances its antidepressant effects. CS 2100 also has activity against nt-proBNP (a marker for heart disease) and other markers that are associated with cardiovascular diseases such as sclerosis or coagulation.>>END>>

CS 2100 (1-[[4-Ethyl-5-[5-(4-phenoxyphenyl)-1,2,4-oxadiazol-3-yl]-2-thienyl]methyl]-3-azetidinecarboxylic acid) is an S1P1 agonist.