Serine/threonin kinase
Serine/threonine kinase inhibitors are compounds that target enzymes responsible for phosphorylating serine and threonine residues on proteins, which play a pivotal role in regulating apoptosis and other cellular processes. These kinases are involved in signaling pathways that control cell growth, division, and programmed cell death. Inhibiting specific serine/threonine kinases can alter the balance between cell survival and apoptosis, making these inhibitors essential tools in cancer research and other areas of cell biology. At CymitQuimica, we provide a comprehensive selection of high-quality serine/threonine kinase inhibitors to support your research in apoptosis, signal transduction, and disease mechanisms.
Products of "Serine/threonin kinase"
Sort by
Found 38 products on this category.
ML-7 hydrochloride
CAS:ML-7 hydrochloride (ML-7 HCl) is a cell-permeable, reversible, effective, ATP-competitive, and specific inhibitor of myosin light chain kinase (Ki: 300 nM);Formula:C15H18ClIN2O2SPurity:99% - 99.26%Color and Shape:White PowderMolecular weight:452.74Ref: TM-T3050
2mg35.00€5mg49.00€10mg74.00€25mg149.00€50mg243.00€100mg353.00€200mg457.00€1mL*10mM (DMSO)50.00€SBC-115076
CAS:SBC-115076 is a potent extracellular proprotein convertase subtilisin kexin type 9 (PCSK9) antagonist.Formula:C31H33N3O5Purity:97.07% - 99.89%Color and Shape:SolidMolecular weight:527.61Ref: TM-T2626
1mg40.00€2mg52.00€5mg85.00€10mg99.00€25mg180.00€50mg325.00€100mg505.00€500mg1,121.00€1mL*10mM (DMSO)92.00€SBC-110736
CAS:SBC-110736 is a proprotein convertase subtilisin kexin type 9 (PCSK9) inhibitorFormula:C26H27N3O2Purity:99.44%Color and Shape:SolidMolecular weight:413.51Ref: TM-T4524
1mg42.00€5mg88.00€10mg127.00€25mg246.00€50mg369.00€100mg620.00€200mg868.00€1mL*10mM (DMSO)87.00€HA-1004
CAS:HA-1004 is a inhibitor of PKG, PKA, PKC and MLC.Formula:C12H15N5O2SPurity:98.91% - 99.03%Color and Shape:SolidMolecular weight:293.34SGC-GAK-1
CAS:SGC-GAK-1 is a selective cyclin G-associated kinase (GAK) inhibitor (Ki: 3.1 nM).Formula:C18H17BrN2O3Purity:99.85%Color and Shape:SolidMolecular weight:389.24FOY 251
CAS:FOY 251 is a proteinase inhibitor, and is an anti-proteolytic active metabolite camostate.Formula:C17H19N3O7SPurity:97.11% - 99.33%Color and Shape:SolidMolecular weight:409.41Ref: TM-T8676
1mg54.00€5mg116.00€10mg187.00€25mg318.00€50mg449.00€100mg638.00€500mg1,264.00€1mL*10mM (DMSO)133.00€CID-797718
CAS:CID-797718 is a protein kinase D1 (PKD1) inhibitor.Formula:C12H11NO3Purity:98.91% - 99.21%Color and Shape:SolidMolecular weight:217.22Ref: TM-T1858
1mg65.00€5mg145.00€10mg212.00€25mg358.00€50mg510.00€100mg702.00€200mg944.00€1mL*10mM (DMSO)160.00€kb-NB77-78
CAS:kb-NB77-78 is an analog of CID797718, which is a by-product of the synthesis of the parental compound, CID755673(PKD1 inhibitor).Formula:C18H25NO3SiPurity:99.54%Color and Shape:SolidMolecular weight:331.48Ref: TM-T1808
1mg34.00€5mg65.00€10mg93.00€25mg180.00€50mg271.00€100mg408.00€200mg567.00€1mL*10mM (DMSO)71.00€CID 2011756
CAS:CID 2011756 is an ATP-competitive and specific PKD1 inhibitor.Formula:C22H21ClN2O3Purity:98.15% - ≥95%Color and Shape:SolidMolecular weight:396.87N-Cyclohexyl-4-[1-(1-piperazinyl)-2,6-naphthyridin-3-yl]-2-pyridinamine
CAS:Novel 2,6-naphthyridine inhibits PKC/PKD, identified by HTS.Formula:C23H28N6Purity:98.35%Color and Shape:SolidMolecular weight:388.51(+)-Isocorydine hydrochloride
CAS:(+)-Isocorydine hydrochloride (Isocorydine HCl) is a eukaryote protein kinases Inhibitor.Formula:C20H24ClNO4Purity:100% - 99.72%Color and Shape:SolidMolecular weight:377.87Ref: TM-T4291
1mg113.00€2mg170.00€5mg284.00€10mg411.00€25mg758.00€50mg1,223.00€100mg1,689.00€500mgTo inquire1mL*10mM (DMSO)304.00€PKD-IN-1 dihydrochloride (956121-30-5 free base)
CAS:CRT0066101 dihydrochloride is an inhibitor of PKD.Formula:C18H21Cl3N4OPurity:99.50%Color and Shape:SolidMolecular weight:415.75SBC-115337
CAS:SBC-115337 is a PCSK9 inhibitor.Formula:C29H19N3O4Purity:99.41%Color and Shape:SolidMolecular weight:473.48TAO Kinase inhibitor 2
CAS:TAO Kinase inhibitor 2 is a TAO kinase inhibitor with an IC50 of 50-500 nM. TAO Kinase inhibitor 2 inhibits KIAA1361 and JIK with IC50s of 50-500 nM.Formula:C25H24N2O3Purity:98.73%Color and Shape:SoildMolecular weight:400.47IPR-803
CAS:IPR-803 is an effective inhibitor of the uPAR·uPA protein-protein interaction (PPI) with anti-tumor activity.Formula:C27H23N3O4Purity:95%Color and Shape:SolidMolecular weight:453.49BMT-124110 Formate
BMT-124110 Formate is a selective AAK1 inhibitor (IC50: 0.9 nM) with anti-injury sensory activity.BMT-124110 Formate inhibits the BMP-2-inducible protein kinaseFormula:C22H20N2O2Purity:99.17%Color and Shape:SoildMolecular weight:344.41Ref: TM-T10572L
1mg185.00€5mg409.00€10mg605.00€25mg938.00€50mg1,293.00€100mg1,738.00€500mg3,496.00€1mL*10mM (DMSO)426.00€SRPKIN-1
CAS:SRPKIN-1 is a covalent and irreversible inhibitor of SRPK1/2 (IC50s: 35.6 and 98 nM, respectively).Formula:C27H21FN2O3SPurity:98%Color and Shape:SolidMolecular weight:472.53PKR-IN-C51
CAS:PKR-IN-C51 is ATP-competitive protein kinase R (PKR) inhibitor that inhibits intracellular PKR activation and autophosphorylation. Ser/Thr kinase.Formula:C23H21N5Purity:98.94%Color and Shape:SolidMolecular weight:367.45Ref: TM-T24647
2mg97.00€5mg156.00€10mg225.00€25mg376.00€50mg558.00€100mg797.00€200mg1,103.00€1mL*10mM (DMSO)165.00€Cetraxate hydrochloride
CAS:Cetraxate hydrochloride (DV10062) is an oral gastrointestinal medication. It has a cytoprotective effect.Formula:C17H24ClNO4Purity:99.75%Color and Shape:SolidMolecular weight:341.83PCSK9-IN-10
CAS:PCSK9-IN-10: potent oral PCSK9 inhibitor (IC50 = 6.4 µM), upregulates LDLR, curbs atherosclerosis, for hyperlipidemia research.Formula:C18H23N5O4Purity:98.85%Color and Shape:SoildMolecular weight:373.41Ref: TM-T72025
2mg42.00€5mg64.00€10mg92.00€25mg178.00€50mg281.00€100mg414.00€200mg585.00€1mL*10mM (DMSO)65.00€6-(Dimethylamino)purine
CAS:6-(Dimethylamino)purine (N,N-Dimethyladenine) is a serine threonine protein kinase and CDK inhibitorFormula:C7H9N5Purity:99.01% - 99.77%Color and Shape:SolidMolecular weight:163.18GAK inhibitor 49
CAS:GAK inhibitor 49 is a highly selective and ATP-competitive cyclin G associated kinase (GAK) inhibitor (IC50: 56 nM; Ki: 0.54 nM ).Formula:C20H22N2O5Purity:98.71%Color and Shape:SolidMolecular weight:370.4Ref: TM-T8535
1mg57.00€5mg117.00€10mg187.00€25mg315.00€50mg454.00€100mg620.00€200mg835.00€1mL*10mM (DMSO)135.00€SPHINX31
CAS:SPHINX31 is a potent inhibitor of serine/arginine-rich protein kinase 1 (SRPK1; IC50: 5.9 nM).Formula:C27H24F3N5O2Purity:100% - 99.3%Color and Shape:SolidMolecular weight:507.51Ref: TM-T5194
1mg40.00€5mg84.00€10mg97.00€25mg180.00€50mg269.00€100mg430.00€500mg998.00€1mL*10mM (DMSO)87.00€PKD-IN-1
CAS:CRT0066101 is an inhibitor of PKD.Formula:C18H19ClN4OPurity:98%Color and Shape:SolidMolecular weight:342.82Camostat mesylate
CAS:Camostat mesylate (FOY-S980) is a trypsin-like protease inhibitor and inhibits airway epithelial sodium channel (ENaC) function.Formula:C21H26N4O8SPurity:100% - 99.85%Color and Shape:Crystalline SolidMolecular weight:494.52Ref: TM-T2391
10mg50.00€25mg72.00€50mg87.00€100mg123.00€200mg175.00€500mg298.00€1mL*10mM (DMSO)52.00€R-IMPP
CAS:R-IMPP is an inhibitor of PCSK9 translation.Formula:C24H27N3O2Purity:99.47%Color and Shape:SolidMolecular weight:389.49Ref: TM-T4058
1mg48.00€2mg59.00€5mg93.00€10mg147.00€25mg296.00€50mg527.00€100mg758.00€1mL*10mM (DMSO)80.00€kb NB 142-70
CAS:kb NB 142-70 is a selective protein kinase D (PKD) inhibitor (IC50 values are 28.3, 58.7 and 53.2 nM for PKD1, 2 and 3 respectively).Formula:C11H9NO2S2Purity:99.57% - ≥95%Color and Shape:SolidMolecular weight:251.32Ref: TM-T2062
1mg48.00€2mg64.00€5mg95.00€10mg154.00€25mg331.00€50mg522.00€100mg748.00€1mL*10mM (DMSO)96.00€BioE-1115
CAS:BioE-1115 is a selective and potent inhibitor of serine-threonine protein kinase (PASK, IC50 = 4 nM). BioE-1115 is a potent inhibitor of CK2α (IC50 = 10 μM).Formula:C19H18FN3O2Purity:97.38%Color and Shape:SolidMolecular weight:339.36WNK463
CAS:WNK463 is a pan-WNK-kinase inhibitor. It effectively inhibits the in vitro kinase activity of all four WNK family members (WNK1/2/3/4).Formula:C21H24F3N7O2Purity:100% - ≥95%Color and Shape:SolidMolecular weight:463.46HTH-01-091
CAS:HTH-01-091 is a potent and selective maternal embryonic leucine zipper kinase (MELK) inhibitor (IC50: 10.5 nM).HTH-01-091 inhibits PIM1/2/3, RIPK2, DYRK3,Formula:C26H28Cl2N4O2Purity:98.40%Color and Shape:SolidMolecular weight:499.43Ref: TM-T24152
1mg281.00€5mg692.00€10mg938.00€25mg1,454.00€50mg1,882.00€100mg2,375.00€1mL*10mM (DMSO)775.00€Benzamidine hydrochloride
CAS:Benzamidine hydrochloride (Benzamidine HCl) is a reversible inhibitor of serine proteases, including trypsin, plasmin, and thrombin.Formula:C7H9ClN2Purity:99.25% - 99.97%Color and Shape:White To Off-White PowderMolecular weight:156.61WNK-IN-11
CAS:WNK-IN-11 (Allosteric WNK Kinase Inhibitor) is an allosteric With-No-Lysine (WNK) kinase inhibitor,WNK1(IC50 : 4 nM)Formula:C21H21Cl2N5OSPurity:98.32%Color and Shape:SolidMolecular weight:462.4Ref: TM-T5456
1mg92.00€5mg180.00€10mg296.00€25mg500.00€50mg722.00€100mg1,017.00€500mg2,023.00€1mL*10mM (DMSO)198.00€1-NM-PP1
CAS:1-NM-PP1 (PP1 Analog II) is a cell-permeable PP1 analog that acts as a potent and selective inhibitor of mutant kinases over their wild-type progenitors.Formula:C20H21N5Purity:98% - 98.93%Color and Shape:White Cyrstalline SolidMolecular weight:331.41Ref: TM-T2153
1mg50.00€2mg66.00€5mg88.00€10mg139.00€25mg286.00€50mg532.00€100mg705.00€1mL*10mM (DMSO)95.00€CID755673
CAS:CID755673 inhibits PKD (IC50: 182 nM), with selectivity over PLK1, AKT, CAMKIIα, CAK, PKC.Formula:C12H11NO3Purity:97.68% - 99.84%Color and Shape:SolidMolecular weight:217.22SM1-71
CAS:SM1-71 is a TAK1 inhibitor that inhibits MKNK2 and RSK2.SM1-71 acts as a kinase probe with anticancer activity.Formula:C24H26ClN7OPurity:96%Color and Shape:SolidMolecular weight:463.96MS-444
CAS:MS-444 (BE-34776) is an MLCK and HuR inhibitor with antitumor activity that can be used to study triple-negative breast cancer and colorectal cancer.Formula:C13H10O4Purity:99.45% - 99.45%Color and Shape:SolidMolecular weight:230.22LP-935509
CAS:LP-935509 is a selective, brain-permeable, small molecule competitive inhibitor of articulin-2-associated kinase 1 (AAK1).Cost-effective and quality-assured.Formula:C20H24N6O3Purity:98.82% - 99.64%Color and Shape:SolidMolecular weight:396.44Ref: TM-T15781
1mg39.00€2mg51.00€5mg84.00€10mg131.00€25mg251.00€50mg469.00€100mg683.00€1mL*10mM (DMSO)92.00€CRT0066101 dihydrochloride
CAS:CRT0066101 dihydrochloride is an effective and selective PKD inhibitor (IC50s: 1, 2.5 and 2 nM for PKD1, 2, and 3).Formula:C18H22N6O·2HClPurity:99.85%Color and Shape:SolidMolecular weight:411.33
![N-Cyclohexyl-4-[1-(1-piperazinyl)-2,6-naphthyridin-3-yl]-2-pyridinamine](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT9256.webp&w=3840&q=75)
