GPR
G protein-coupled receptors (GPRs) are a large family of cell surface receptors that play a crucial role in transmitting signals from hormones, neurotransmitters, and other extracellular ligands into the cell. GPRs are involved in a wide range of physiological processes, including hormone regulation, immune response, and sensory perception. Modulating GPR activity is a key strategy in the development of therapeutics for various diseases, including endocrine disorders, cardiovascular diseases, and neurological conditions. At CymitQuimica, we offer a selection of high-quality GPR modulators to support your research in cell signaling, endocrinology, and drug discovery.
Products of "GPR"
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GPR41 agonist-1
CAS:GPR41 agonist-1 is a GPR41 agonist, used for studying metabolic diseases such as diabetes and obesity.Formula:C24H23N3O4Purity:98.40%Color and Shape:SolidMolecular weight:417.46AMG-009
CAS:AMG-009 is a prostaglandin D2 antagonist. For CRTH2 and DP receptors, the IC50s are 3 nM and 12 nM, respectively.Formula:C26H26Cl2N2O7SPurity:97.88%Color and Shape:SolidMolecular weight:581.47WAY-298630
CAS:Fluorophenoxy benzimidazole, a CRTH2 blocker, IC50 < 10 μM for rhinitis, COPD, arthritis, eczema, conjunctivitis.Formula:C17H15FN2O3SPurity:97.13%Color and Shape:SolidMolecular weight:346.38Bimatoprost acid
CAS:Bimatoprost acid (17-phenyl trinor PGF2α) is a metabolically stable analog of PGF2α and has a potential antagonistic activity for the FP receptor.Formula:C23H32O5Purity:99.29%Color and Shape:SolidMolecular weight:388.5Ref: TM-T20939
1mg133.00€5mg304.00€10mg452.00€25mg740.00€50mg1,026.00€100mg1,388.00€1mL*10mM (DMSO)325.00€CRTh2 antagonist 1
CAS:CRTh2 antagonist 1 is a CRTh2 antagonist (IC50: 89 nM).Formula:C23H25N3O5SPurity:97.39%Color and Shape:SolidMolecular weight:455.53Ref: TM-T10084
1mg115.00€5mg255.00€10mg374.00€25mg562.00€50mg787.00€100mg1,074.00€500mg2,147.00€1mL*10mM (DMSO)283.00€Questiomycin A
CAS:Questiomycin A: crème fraiche antibiotic with antibacterial, anticancer effects; inhibits GRP78.Formula:C12H8N2O2Purity:98% - 99.07%Color and Shape:SolidMolecular weight:212.2Ginsenoside Rb2
CAS:Ginsenoside Rb2 (Ginsenoside C) found in species of Panax, upregulating GPR120 gene expression.Formula:C53H90O22Purity:99.01% - 99.66%Color and Shape:White PowderMolecular weight:1079.27CAY10595
CAS:CAY10595 is an antagonist of the CRTh2 (DP2) receptor with a Ki of 10 nM.Formula:C20H13Cl2FN2O5Purity:100% - 99.71%Color and Shape:SolidMolecular weight:451.23Latanoprost
CAS:Latanoprost (Xalatan) is a prostaglandin F2alpha analogue and a prostanoid selective FP receptor agonist with an ocular hypertensive effect.Formula:C26H40O5Purity:99.69% - 99.78%Color and Shape:Pale Yellow OilMolecular weight:432.59Ref: TM-T2528
1mg47.00€2mg59.00€5mg88.00€10mg142.00€25mg274.00€50mg408.00€100mg603.00€500mg1,293.00€1mL*10mM (DMSO)87.00€AM-4668
CAS:AM-4668, a GPR40 (FFA1) agonist with oral availability, was optimized to reduce central nervous system (CNS) permeability, and reduced blood glucose level.Formula:C24H19F3N2O4SPurity:100% - 99.92%Color and Shape:SolidMolecular weight:488.48AF64394
CAS:AF64394 is a selective inverse agonist of GPR3(pIC50 : 7.3)Formula:C21H20ClN5OPurity:97.22%Color and Shape:SolidMolecular weight:393.87GPCR agonist-2
CAS:GPCR agonist-2 (4-(Cyclopropylamino)-3-nitrobenzoic acid) is an agonist of the orphan human GPCR GPR109B.Formula:C10H10N2O4Purity:99.94%Color and Shape:SolidMolecular weight:222.2NE 52-QQ57
CAS:NE 52-QQ57 is a selective, and orally available antagonist of GPR4(IC50 : 70 nM),with anti-inflammatory activity.Formula:C24H28N6OPurity:98.63%Color and Shape:SolidMolecular weight:416.52Ref: TM-T11461
1mg73.00€5mg160.00€10mg235.00€25mg394.00€50mg587.00€100mg835.00€1mL*10mM (DMSO)170.00€6-OAU
CAS:6-OAU is a GPR84 agonist, activates it in HEK293 cells with a 105 nM EC50.Formula:C12H21N3O2Purity:99.01% - 99.68%Color and Shape:SolidMolecular weight:239.31Ref: TM-T2036
1mg160.00€2mg215.00€5mg329.00€10mg472.00€25mg753.00€50mg1,074.00€100mg1,444.00€1mL*10mM (DMSO)301.00€TAK-041
CAS:TAK-041 (NBI-1065846) is a potent and selective GPR139 agonist.Formula:C18H15F3N4O3Purity:99.95%Color and Shape:SolidMolecular weight:392.33Ref: TM-T9317
1mg37.00€5mg144.00€10mg225.00€25mg452.00€50mg723.00€100mg1,130.00€200mg1,501.00€1mL*10mM (DMSO)159.00€Grp94 Inhibitor-1
CAS:Grp94 Inhibitor-1 is a potent, selective Grp94 inhibitor (IC50 : 2 nM).Formula:C22H28N2O2Purity:97.02%Color and Shape:SolidMolecular weight:352.47BTB09089
CAS:BTB09089 (GPR65 agonist ) is a T cell death-associated gene 8 (TDAG8/GPR65)-specific agonist.BTB09089 induces TDAG8 expression and regulates cytokine productionFormula:C14H12Cl2N4OS2Purity:100%Color and Shape:SoildMolecular weight:387.31Acifran
CAS:Acifran (AY 25712) is an HM74A/GPR109A and GPR109B agonist and displays antihyperlipidemic activity.Formula:C12H10O4Purity:98.65%Color and Shape:SolidMolecular weight:218.21APD597
CAS:APD597 (JNJ-38431055) is a GPR119 agonist, used in the treatment of type 2 diabetes.Formula:C21H29N5O6SPurity:99.63% - 99.78%Color and Shape:SolidMolecular weight:479.55GPR81 agonist 1
CAS:GPR81 agonist 1 is a GPR81 agonist that improves glycaemic control in insulin-resistant mouse models for the study of diabetes and obesity.Formula:C22H30N4O2S2Purity:99.68%Color and Shape:SolidMolecular weight:446.63
