GPR
G protein-coupled receptors (GPRs) are a large family of cell surface receptors that play a crucial role in transmitting signals from hormones, neurotransmitters, and other extracellular ligands into the cell. GPRs are involved in a wide range of physiological processes, including hormone regulation, immune response, and sensory perception. Modulating GPR activity is a key strategy in the development of therapeutics for various diseases, including endocrine disorders, cardiovascular diseases, and neurological conditions. At CymitQuimica, we offer a selection of high-quality GPR modulators to support your research in cell signaling, endocrinology, and drug discovery.
Products of "GPR"
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Fezagepras sodium
CAS:Fezagepras sodium (Setogepram sodium salt) is an orally active GPR40 agonist and is an antagonist or inverse agonist for GPR84, with anti-fibrotic, anti-Formula:C13H17NaO2Purity:99.59%Color and Shape:SolidMolecular weight:228.26Ref: TM-T12375
1mg43.00€5mg96.00€10mg140.00€25mg255.00€50mg374.00€100mg542.00€500mg1,093.00€1mL*10mM (DMSO)96.00€Palosuran hydrochloride 540769-28-6(free base)
Palosuran hydrochloride 540769-28-6(free base)(ACT-058362 hydrochloride) is a new potent and specific antagonist of the human UT receptor with an IC50 of 3.6±0.Formula:C25H31ClN4O2Purity:99.75%Color and Shape:SolidMolecular weight:454.99Ramatroban
CAS:Ramatroban (BAY u3405) (BAY u3405) is a thromboxane A(2) (TxA(2)) antagonist marketed for allergic rhinitis.Formula:C21H21FN2O4SPurity:98.12% - 99.96%Color and Shape:Crystalline SolidMolecular weight:416.47Ref: TM-T2396
5mg38.00€10mg57.00€25mg95.00€50mg170.00€100mg274.00€200mg354.00€500mg597.00€1mL*10mM (DMSO)63.00€Ogremorphin
CAS:Ogremorphin (GPR68-IN-1) is a potent inhibitor of GPR68, exhibiting an EC50 of 170 nM.it is utilized in the study of autoimmune chronic inflammatory diseases [1Formula:C21H17N3OSPurity:99.65% - 99.65%Color and Shape:SolidMolecular weight:359.44DJ-V-159
CAS:DJ-V-159 is a GPRC6A agonist, targeting the G protein-coupled receptor family C group 6 member A (GPRC6A).Formula:C24H12F6N4O2Purity:99.85% - 99.96%Color and Shape:SolidMolecular weight:502.37LY2881835
CAS:LY2881835 is a potent and selective GPR40 agonist.Formula:C33H33NO3Purity:97.65% - 97.65%Color and Shape:SolidMolecular weight:491.62APD668
CAS:APD668 is a potent GPR119 agonist with EC50 of 2.7 nM and 33 nM for hGPR119 and ratGPR119, respectively.Formula:C21H24FN5O5SPurity:99.45% - 99.97%Color and Shape:SolidMolecular weight:477.51GPR40/FFAR1 modulator 1
CAS:GPR40/FFAR1 modulator 1 is a Gq-coupled free fatty acid receptor 1 (GPR40/FFAR1) agonist and allosteric modulator.Formula:C21H19N5O3Purity:99.72%Color and Shape:SolidMolecular weight:389.41NOX-6-18
CAS:NOX-6-18 (GPR132-B-160) is a GPR132 antagonist with insulin-promoting activity and reduced weight gain.Formula:C18H17NO5SPurity:99.29%Color and Shape:SoildMolecular weight:359.4hGPR91 antagonist 3
CAS:hGPR91 antagonist 3 is an hGPR91 antagonist. hGPR91 antagonist 3 can be used to study diseases in hypertension and retinal angiogenesis.Formula:C23H18F4N4O2Purity:98.82% - 98.82%Color and Shape:SolidMolecular weight:458.41Latanoprost acid
CAS:Latanoprost acid is a prostanoid receptor agonist that blocks RANKL and can be used to reduce intraocular pressure.Formula:C23H34O5Purity:96.97%Color and Shape:Pale Yellow OilMolecular weight:390.51Ref: TM-T15718
1mg57.00€5mg145.00€10mg226.00€25mg454.00€50mg672.00€100mg924.00€200mg1,225.00€1mL*10mM (DMSO)160.00€GSK1292263
CAS:GSK1292263 is a GPR119 agonist and has been investigated for the treatment of DIABETES MELLITUS, TYPE 2.Formula:C23H28N4O4SPurity:98.34% - 99.46%Color and Shape:SolidMolecular weight:456.56NCRW0005-F05
CAS:NCRW0005-F05 is a potent agonist of orphan G-protein coupled receptor GPR139 with an IC 50 value of 0.21 μM.Formula:C16H13F2NO2Purity:99.48%Color and Shape:SolidMolecular weight:289.28P2Y2R/GPR17 antagonist 1
CAS:P2Y2R/GPR17 antagonist 1 (Compound 14m) is a dual P2Y2R (IC50: 3.17 μM) and GPR17 (IC50: 1.67 μM) antagonist.Formula:C19H13ClN2O6SPurity:98.21%Color and Shape:SolidMolecular weight:432.83YL-365
YL-365 is a highly potent and selective GPR34 antagonist that exhibits excellent activity in neuropathic pain models for the study of neurologic diseases.Purity:98.51%Color and Shape:Odour Solid7-FluorotryptaMine HCl
CAS:7-FluorotryptaMine HCl is a potent aromatic monoamine GPRC5A agonist that induces GPRC5A-mediated β-arrestin recruitment.7-FluorotryptaMine HCl can be used toFormula:C10H12ClFN2Purity:98.06%Color and Shape:SolidMolecular weight:214.67GW9508
CAS:GW9508(GW 9508) is a potent and selective agonist for FFA1 (GPR40), stimulates insulin secretion in a glucose-sensitive manner.Formula:C22H21NO3Purity:97.89% - 99.19%Color and Shape:SolidMolecular weight:347.41GPR40 Agonist 2
CAS:GPR40 Agonist 2 is a GPR40 agonist. It can be used in the research of diabetes.Formula:C24H30O3Purity:98%Color and Shape:SolidMolecular weight:366.49Myristyl nicotinate
CAS:Myristyl nicotinate (Tetradecyl nicotinate) is an ester prodrug being developed for delivery of nicotinic acid (NIC) into the skin for prevention of actinicFormula:C20H33NO2Purity:99.50%Color and Shape:SolidMolecular weight:319.48LY2922470
CAS:LY2922470: Selective GPR40 agonist; EC50=7nM (human), 1nM (mouse), 3nM (rat); lowers glucose, boosts insulin/GLP-1.Formula:C28H29NO4SPurity:93.34% - 96%Color and Shape:SolidMolecular weight:475.6Ref: TM-T15810
1mg115.00€5mg236.00€10mg355.00€25mg617.00€50mg879.00€100mg1,198.00€1mL*10mM (DMSO)248.00€
