Vasopressin Receptor
Vasopressin receptors are a family of G protein-coupled receptors that mediate the effects of vasopressin, a hormone involved in regulating water balance, blood pressure, and kidney function. Vasopressin receptor agonists and antagonists are studied for their roles in treating conditions such as diabetes insipidus, hyponatremia, and heart failure. These receptors are also important targets in research on fluid balance and cardiovascular health. At CymitQuimica, we provide a selection of high-quality vasopressin receptor modulators to support your research in endocrinology, nephrology, and cardiovascular biology.
Products of "Vasopressin Receptor"
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Found 19 products on this category.
V1a/V2 antagonist 1
V1a/V2 antagonist 1 (Compound 18j) is an orally active dual-target antagonist of V1a and V2 receptors, exhibiting high binding affinity toward these receptors [Ki values are hV1a: 0.13 nM, hV2: 0.53 nM, and mV1a: 0.5 nM; IC50 for hV1a is 2.2 nM]. This compound can inhibit oxytocin-induced scratching behavior in mice.Formula:C25H26ClN5O3Color and Shape:SolidMolecular weight:479.96Felypressin acetate
CAS:Felypressin acetate (PLV-2) is an agonist of vasopressin 1 and acts on all arginine vasopressin receptors 1AS.Formula:C48H69N13O13S2Purity:97.06%Color and Shape:SolidMolecular weight:1100.27OPC-51803
CAS:OPC-51803 is an orally available nonapeptidylpressor (AVP) V(2) receptor selective agonist for the treatment of urinary incontinence and nocturia.Formula:C26H32ClN3O2Purity:100% - 100%Color and Shape:SolidMolecular weight:454Ref: TM-T28257
1mg333.00€5mg787.00€10mg1,074.00€25mg1,510.00€50mg1,882.00€100mg2,375.00€500mg4,655.00€Atosiban acetate
CAS:Atosiban acetate (RW22164) is an inhibitor of the hormones oxytocin and vasopressin.Formula:C45H71N11O14S2Purity:99.15% - 99.84%Color and Shape:SolidMolecular weight:1054.24Ref: TM-T5148
5mg73.00€10mg115.00€25mg170.00€50mg207.00€100mg268.00€500mg660.00€1mL*10mM (DMSO)134.00€Argipressin
CAS:Argipressin is a vasoconstrictive and antidiuretic hormone, binding to V1 receptors with Kd ~1.4 nM in rat heart and aortic cells.Formula:C46H65N15O12S2Purity:98%Color and Shape:White PowderMolecular weight:1084.23TASP0390325
CAS:TASP0390325, a potent and orally active V1B receptor antagonist, has antidepressant and anxiolytic activities in rodents.Formula:C25H30Cl2FN5O4Purity:98.62%Color and Shape:SolidMolecular weight:554.44Atosiban
CAS:Atosiban (RW22164), an oxytocin/vasopressin inhibitor, halts premature labor as an intravenous tocolytic, reducing uterine contractions rapidly.Formula:C43H67N11O12S2Purity:98%Color and Shape:SolidMolecular weight:994.19Nelivaptan
CAS:Nelivaptan (SR 149415) is a vasopressin V1b receptor antagonist that can eliminate CHS-induced GE damage.Cost-effective and quality-assured.Formula:C30H32ClN3O8SPurity:98% - 98.39%Color and Shape:SolidMolecular weight:630.11RG7713
CAS:RG7713 (RO 5028442) has been used in trials studying Autistic Disorder.Formula:C25H28ClN3O2Purity:99.74%Color and Shape:SolidMolecular weight:437.96Mozavaptan
CAS:Mozavaptan (OPC-31260) is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively.Formula:C27H29N3O2Purity:98.98% - 99.12%Color and Shape:SolidMolecular weight:427.54E-4177
CAS:E-4177 is an angiotensin II type 1 receptor (AT1R) antagonist and can be used to study cardiovascular diseases.Formula:C24H21N3O2Purity:98.63% - 99.39%Color and Shape:SolidMolecular weight:383.44Tolvaptan
CAS:Tolvaptan (OPC-41061) is an orally bioavailable, selective, arginine vasopressin receptor 2 (V2, AVPR2) antagonist that can be used to treat hyponatremia.Formula:C26H25ClN2O3Purity:97% - 99.91%Color and Shape:SolidMolecular weight:448.94Fedovapagon
CAS:Fedovapagon (VA106483) is a pressin V2 receptor (V2R) agonist for the study of overactive bladder syndrome.Formula:C27H34N4O3Purity:99.33%Color and Shape:SolidMolecular weight:462.58Balovaptan
CAS:Balovaptan (RG7314), a potent brain-penetrant hV1a receptor antagonist, Ki: 1 nM for hV1a, aids autism research.Formula:C22H24ClN5OPurity:99.88%Color and Shape:SolidMolecular weight:409.91Felypressin
CAS:Felypressin, a Lypressin analog with a phenylalanine substitution, acts as a vasoconstrictor with less antidiuretic effect.Formula:C46H65N13O11S2Purity:99.65%Color and Shape:SolidMolecular weight:1040.22LIXIVAPTAN
CAS:Lixivaptan (VPA-985) is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM)Formula:C27H21ClFN3O2Purity:98.36%Color and Shape:SolidMolecular weight:473.93Ref: TM-T7303
1mg43.00€2mg57.00€5mg81.00€10mg127.00€25mg249.00€50mg424.00€100mg625.00€1mL*10mM (DMSO)86.00€Fuscoside
CAS:Fuscoside (OPC-21268) is a non-peptide arginine vasopressin (AVP) receptor VI antagonist with an IC50 value of 0.4 μM.Cost-effective and quality-assured.Formula:C26H31N3O4Purity:97.98% - 99.66%Color and Shape:SolidMolecular weight:449.54Terlipressin Acetate
CAS:Terlipressin Acetate, a highly selective vasopressin V1 receptor agonist, on OGD/R-induced damage in intestinal epithelial cells (IEC-6).Formula:C56H82N16O19S2Purity:98.50% - 99.69%Color and Shape:SolidMolecular weight:1347.5Conivaptan hydrochloride
CAS:Conivaptan hydrochloride (Vaprisol) is an orally active vasopressin V2 and V1A receptor antagonist, used in the therapy of hypervolemic hyponatremia andFormula:C32H26N4O2·HClPurity:98.33% - 99.86%Color and Shape:SolidMolecular weight:535.04
