Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC
- Adiponectin receptor
- ATPase
- Calcium Channel
- CFTR
- CGRP Receptor
- Chloride channel
- GABA Receptor
- Monoamine Transporter
- Monocarboxylate transporter
- Na-K-Cl cotransporter
- NKCC
- NPC1L1
- OAT
- OCT
- P-gp
- Potassium Channel
- Proton pump
- SGLT
- Sodium Channel
- TRP/TRPV Channel
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Products of "Membrane Transporter/Ion Channel"
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TRPA1-IN-2
CAS:TRPA1-IN-2 is a potent and orally active TRPA1 inhibitor with an IC50 value of 0.04 µM.TRPA1-IN-2 has anti-inflammatory activity.Formula:C24H25F3N4OPurity:98.05%Color and Shape:SoildMolecular weight:442.48Ref: TM-T77511
1mg85.00€5mg187.00€10mg284.00€25mg482.00€50mg672.00€100mg905.00€200mg1,216.00€1mL*10mM (DMSO)207.00€Digitoxin
CAS:Digitoxin (Digitoxinum) is an effective Na+/K+-ATPase inhibitor (EC50 value: 0.78 μM).Formula:C41H64O13Purity:98.23% - 98.54%Color and Shape:Very Small Elongated Rectangular Plates From Dilute Alcohol 1998)Molecular weight:764.94Propafenone
CAS:Propafenone: a drug for ventricular arrhythmias with mild beta-blocker activity, prolongs refractory period, and reduces heart automaticity.Formula:C21H27NO3Purity:99.02%Color and Shape:SolidMolecular weight:341.44Fenamic acid
CAS:Fenamic acid (N-Phenylanthranilic acid) is a chloride channel blocker that causes renal papillary necrosis in rats.Formula:C13H11NO2Purity:99.60%Color and Shape:White To Off-White Crystalline PowderMolecular weight:213.2319(2S)-6-Prenylnaringenin
CAS:(2S)-6-Prenylnaringenin (6-Prenylnaringenin) is an isomer of the potent phytoestrogen, 8-prenylnaringenin.Formula:C20H20O5Purity:99.47%Color and Shape:SolidMolecular weight:340.37ASP2905
CAS:ASP-2905 is a potent and selective inhibitor of potassium channel Kv12.2 encoded by the Kcnh3/BEC1 gene.Formula:C20H17FN8Purity:97.29%Color and Shape:SolidMolecular weight:388.4Ref: TM-T9070
1mg35.00€2mg48.00€5mg70.00€10mg96.00€25mg188.00€50mg311.00€100mg512.00€1mL*10mM (DMSO)77.00€DL-Menthol
CAS:DL-Menthol ((±)-Menthol) is a racemic mixture of the monoterpene alcohols (-)-menthol and (+)-menthod, which have been found in Cannabis.Formula:C10H20OPurity:99.74%Color and Shape:White Crystals /89-78-1/ Physical Description White Crystalline Solid With A Peppermint Odor And Taste (Ntp 1992)Molecular weight:156.27FEMA-4809
CAS:FEMA-4809 activates TRPM8, the ion channel for cold sensation, and is used as a cooling agent.Formula:C17H17N3O2SPurity:99.19%Color and Shape:SolidMolecular weight:327.4Ref: TM-T27308
1mg35.00€5mg78.00€10mg116.00€25mg190.00€50mg269.00€100mg383.00€200mg525.00€1mL*10mM (DMSO)88.00€GX 201
CAS:GX 201 is a selective NaV1.7 inhibitor, IC50 of < 3.2 nM for hNaV1.7.Formula:C25H27ClF4N2O4SPurity:99.46%Color and Shape:SolidMolecular weight:563CFTR corrector 12
CAS:CFTR corrector 12 is a CFTR corrector that rescues all mutant proteins except M760R ABCA3 and can be used to study cystic fibrosis.Formula:C19H21ClN4O2S2Purity:99.78%Color and Shape:SolidMolecular weight:436.98Verdinexor
CAS:Verdinexor (KPT-335) (KPT-335), a specific XPO1/CRM1 inhibitor, are orally bioavailable.Formula:C18H12F6N6OPurity:98% - 99.68%Color and Shape:SolidMolecular weight:442.32Ref: TM-T6123
1mg35.00€5mg111.00€10mg187.00€25mg341.00€50mg567.00€100mg905.00€200mg1,216.00€1mL*10mM (DMSO)123.00€Methionine
CAS:Methionine (D-Methionine) (MRX-1024; D-Methionine) is an effective chemoprotective agent which can also inhibit the neuronal activity through GABAA receptorFormula:C5H11NO2SPurity:99.13% - 99.62%Color and Shape:SolidMolecular weight:149.21Elexacaftor
CAS:Elexacaftor (VX-445) is a cystic fibrosis transmembrane conductance regulator (CFTR) corrector.Cost-effective and quality-assured.Formula:C26H34F3N7O4SPurity:98.87% - 99.87%Color and Shape:SolidMolecular weight:597.65Ref: TM-T14935
1mg87.00€2mg137.00€5mg243.00€10mg393.00€25mg772.00€50mg1,074.00€100mg1,444.00€1mL*10mM (DMSO)320.00€CGP37157
CAS:CGP37157 (7-Chloro-5-(2-chlorophenyl)-1,5-dihydro-4,1-benzothiazepine-2(3H)-one) is a Na+/Ca2+ exchanger inhibitor, inhibits Na+-induced Ca2+ release fromFormula:C15H11Cl2NOSPurity:99.04%Color and Shape:SolidMolecular weight:324.22Lingdolinurad
CAS:Lingdolinurad is a uric acid transporter protein inhibitor targeting hURAT1 for the study of hyperuricemia or gout.Formula:C17H12BrN3O2Purity:98.70%Color and Shape:SolidMolecular weight:370.2Ref: TM-T79854
1mg185.00€5mg459.00€10mg657.00€25mg1,026.00€50mg1,415.00€100mg1,872.00€1mL*10mM (DMSO)469.00€TC-I 2014
CAS:TC-I 2014 shows antiallodynic properties in pain models.Formula:C23H19F6N3OPurity:98.75%Color and Shape:SolidMolecular weight:467.41Ref: TM-T17006
1mg60.00€5mg127.00€10mg202.00€25mg406.00€50mg655.00€100mg1,074.00€200mg1,454.00€1mL*10mM (DMSO)133.00€Amentoflavone
CAS:Amentoflavone (3',8''-Biapigenin), as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications.Formula:C30H18O10Purity:98.21% - 99.22%Color and Shape:Odourless Whitish SolidMolecular weight:538.46SCS
CAS:SCS is a GABAA receptor antagonist.Formula:C14H12N2O3Purity:98.89%Color and Shape:SolidMolecular weight:256.26FFN 206 dihydrochloride
CAS:FFN 206 dihydrochloride: fluorescent VMAT2 marker, detects subcellular sites, non-inhibitory to DAT.Formula:C12H15ClN2O2Purity:100% - 98.57%Color and Shape:SolidMolecular weight:254.71Fengabine
CAS:Fengabine (SL-79229) is a GABA receptor agonist with antidepressant activity and is used to treat depression.Formula:C17H17Cl2NOPurity:98.54%Color and Shape:SolidMolecular weight:322.23Desmethylflunitrazepam
CAS:Desmethylflunitrazepam (Norflunitrazepam) is a benzodiazepine derivative and an active metabolite of Flunitrazepam.Formula:C15H10FN3O3Color and Shape:SolidMolecular weight:299.26Flufenamic acid
CAS:Flufenamic acid (Arlef) is an anthranilic acid derivative with analgesic, anti-inflammatory, and antipyretic properties.Formula:C14H10F3NO2Purity:98.68%Color and Shape:White To Light Yellow Crystalline PowderMolecular weight:281.23Eniporide
CAS:Eniporide is a Na(+)/H(+) exchange inhibitor.Formula:C14H16N4O3SPurity:95.09% - 96.78%Color and Shape:SolidMolecular weight:320.37Ref: TM-T2089
1mg35.00€5mg77.00€10mg119.00€25mg197.00€50mg295.00€100mg426.00€200mg602.00€1mL*10mM (DMSO)88.00€AMG9810
CAS:AMG 9810 blocks capsaicin's action on TRPV1; human IC50=24.5 nM, rat IC50=85.6 nM.Formula:C21H23NO3Purity:99.79% - 99.83%Color and Shape:SolidMolecular weight:337.41μ-Conotoxin Sx IIIA
CAS:μ-Conotoxin Sx IIIA is a biologically active peptide that functions as a blocker of NaV1.4 channels.Formula:C86H152N34O26S6Purity:98%Color and Shape:SolidMolecular weight:2270.73Vigabatrin Hydrochloride
CAS:Vigabatrin Hydrochloride (γ-Vinyl-GABA hydrochloride) is a structural analog of the GABA, irreversibly inhibiting the catabolism of GABA by GABA transaminase.Formula:C6H11NO2·HClPurity:98%Color and Shape:SolidMolecular weight:165.62JYL 1421
CAS:JYL 1421 (SC 0030) is an antagonist of TRPV1 receptor (IC50 = 8 nM).Formula:C20H26FN3O2S2Purity:98.83%Color and Shape:SolidMolecular weight:423.57Ref: TM-T15634
1mg70.00€5mg187.00€10mg305.00€25mg612.00€50mg938.00€100mg1,491.00€200mg1,985.00€1mL*10mM (DMSO)173.00€RN-1747
CAS:RN-1747: TRPV4 agonist (EC50: human 0.77 μM, mouse 4.0 μM, rat 4.1 μM), TRPM8 antagonist (IC50: 4 μM).Formula:C17H18ClN3O4SPurity:99.29%Color and Shape:SolidMolecular weight:395.86Ref: TM-T16763
5mg44.00€10mg74.00€25mg126.00€50mg188.00€100mg316.00€200mg452.00€1mL*10mM (DMSO)47.00€Flecainide acetate
CAS:Flecainide acetate (R-818) is a class Ic antiarrhythmic agent used to prevent and treat tachyarrhythmias (abnormal fast rhythms of the heart).Formula:C19H24F6N2O5Purity:99.42%Color and Shape:SolidMolecular weight:474.39Pentetrazol
CAS:Pentylenetetrazol is a GABA(A) receptor antagonist, that displays activity as a central nervous system and respiratory stimulant.Formula:C6H10N4Purity:100% - 99.95%Color and Shape:Bitter Taste Aqueous Solutions Neutral To Litmus (Ntp 1992)Molecular weight:138.17Istaroxime hydrochloride
CAS:Istaroxime hydrochloride (PST2744 hydrochloride) is a Na+/K+-ATPase inhibitor and SERCA 2 activator, and is a novel positive inotropic compound.Formula:C21H33ClN2O3Color and Shape:SolidMolecular weight:396.95Apamin acetate
Apamin acetate: Selective Ca2+-activated K+ channel blocker, 18-amino acid bee venom peptide, promotes synapse repair, anti-inflammatory.Purity:96.97%Color and Shape:SolidSulcardine 2HCl
CAS:Sulcardine 2HCl is a multi-ion channel blocker that blocks the properties of hERG and hNav1.5 channels and can be used to study atrial fibrillation.Formula:C24H35Cl2N3O4SPurity:98.45% - 99.51%Color and Shape:SoildMolecular weight:532.523(+)-Tetrabenazine
CAS:(+)-Tetrabenazine ((3R,11bR)-Tetrabenazine) is a reversible vesicular monoamine transporter 2 (VMAT-2) inhibitor, inhibits transport by VMAT2 with 10-foldFormula:C19H27NO3Purity:98.31%Color and Shape:SolidMolecular weight:317.42Vm24-toxin
CAS:Vm24-toxin, a peptide toxin isolated from the Mexican scorpion Vaejovis mexicanus smithi, serves as an inhibitor of the Kv1.3 potassium channel [1].Formula:C157H253N51O45S9Purity:98%Color and Shape:SolidMolecular weight:3863.59HC067047 Hydrochloride(883031-03-6 free base)
CAS:HC-067047 hydrochloride, a TRPV4 antagonist, selectively inhibits human, rat, and mouse currents with IC50s: 486 nM, 133 nM, and 17 nM.Formula:C26H29ClF3N3O2Purity:99.95%Color and Shape:SolidMolecular weight:507.98Ref: TM-T4680L
1mg88.00€5mg172.00€10mg259.00€25mg425.00€50mg598.00€100mg810.00€200mg1,074.00€1mL*10mM (DMSO)217.00€Orphenadrine hydrochloride
CAS:Orphenadrine hydrochloride (Mephenamin) is a muscarinic antagonist used to treat drug-induced parkinsonism and to relieve pain from muscle spasm.Formula:C18H23NO·HClPurity:99.88%Color and Shape:Liquid About 5 5 Bitter Numbing Taste (Ntp 1992)Molecular weight:305.85Mtb ATP synthase-IN-1
CAS:Mtb ATP synthase-IN-1 is a potent, low-toxicity M. tuberculosis inhibitor with good oral bioavailability and metabolic stability.Formula:C17H13N3O4Purity:98.28%Color and Shape:SolidMolecular weight:323.30Bacoside A3
CAS:Bacoside A3 is one of the components of Bacopa monnieri (L.) Wettst.Formula:C47H76O18Purity:99.67%Color and Shape:SolidMolecular weight:929.19-Hydroxycanthin-6-one
CAS:9-Hydroxycanthin-6-one might be the active component that contributed to the aphrodisiac effect of E.Formula:C14H8N2O2Purity:98%Color and Shape:SolidMolecular weight:236.23Mambalgin-3
Mambalgin-3, an acid-sensitive ion channel 1 (ASIC1) inhibitor, has potential applications in analgesia research [1].Formula:C274H433N85O83S10Purity:98%Color and Shape:SolidMolecular weight:6566.54Aneratrigine
CAS:Aneratrigine is a blocker of the sodium channel protein type 9 subunit alpha, utilized in research on neuropathic pain diseases [1].Formula:C19H20ClF2N5O2S2Purity:98%Color and Shape:SolidMolecular weight:487.97α-Cyano-4-hydroxycinnamic acid
CAS:α-Cyano-4-hydroxycinnamic acid (α-Cyano-4-hydroxycinnamic acid(α-CHCA)) (α-CHCA) is an inhibitor of monocarboxylate transporter 1 (MCT1) that blocks pyruvateFormula:C10H7NO3Purity:99.8% - 99.86%Color and Shape:PowderMolecular weight:189.17TRAM-34
CAS:TRAM-34 (Triarylmethane-34), an effective and specific inhibitor of the intermediate-conductance Ca2+-activated K+ channel, does not block cytochrome P450.Formula:C22H17ClN2Purity:99.01% - 99.76%Color and Shape:SolidMolecular weight:344.84Spinoxin
CAS:Spinoxin, a 34-residue peptide neurotoxin extracted from the venom of Heterometrus spinifer, is characterized by four disulfide bridges.Formula:C147H236N48O46S9Purity:98%Color and Shape:SolidMolecular weight:3700.33ATX-II TFA
ATX-II TFA, a specific Na+ channel modulator toxin, is derived from the venom of the sea anemone (Anemonia sulcata).Purity:98%Color and Shape:Odour SolidXE991
CAS:XE991 is a Kv7 (KCNQ) channel blocker.XE 991 dihydrochloride inhibits Kv7.1 (KCNQ1) and M-current and can be used in the study of neurological disorders.Formula:C26H20N2OPurity:99.51%Color and Shape:SolidMolecular weight:376.45Ref: TM-T78570
1mg48.00€5mg96.00€10mg153.00€25mg283.00€50mg522.00€100mg838.00€500mg1,681.00€1mL*10mM (DMSO)105.00€GS 39783
CAS:GS 39783 is a positive allosteric modulator (PAM) of GABABR, which reduces the motivational properties of alcohol and the conditioned reinforcement andFormula:C15H23N5O2SPurity:99.94%Color and Shape:SolidMolecular weight:337.44RN9893
CAS:RN9893 is a selective and potent TRPV4 receptor antagonist with IC50 values of 320, 420 and 660 nM for TRPV4 receptors in mouse, human and rat, respectively.Formula:C21H23F3N4O5SPurity:99.89%Color and Shape:SolidMolecular weight:500.49Tiludronate disodium
CAS:Tiludronate disodium: osteoclast inhibitor for metabolic bone disorder research.Formula:C7H7ClNa2O6P2SPurity:100% - 100%Color and Shape:Fine White To Off-White Crystalline PowderMolecular weight:362.57
