CGRP Receptor
CGRP receptors are involved in the transmission of pain and the regulation of blood flow. CGRP is a neuropeptide that plays a critical role in migraine pathophysiology by dilating blood vessels and modulating pain signaling pathways. Targeting CGRP receptors has become a promising approach in the development of migraine therapies. At CymitQuimica, we offer a range of CGRP receptor modulators to support your research in pain management, neurobiology, and vascular health.
Products of "CGRP Receptor"
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Found 16 products on this category.
CGRP antagonist 6
CGRP Antagonist 6 (Compound 23) is a potent CGRP receptor antagonist (Ki: 0.84 nM). It is utilized in the study of migraines.Color and Shape:Odour SolidVazegepant hydrochloride
CAS:Vazegepant hydrochloride (Vazegepant HCl) is the first intranasal gepant for the acute treatment of migraine and has announced a positive phase II/III study.Formula:C36H47ClN8O3Purity:98.93%Color and Shape:SolidMolecular weight:675.3Ref: TM-T8682
1mg107.00€5mg227.00€10mg334.00€25mg565.00€50mg805.00€100mg1,111.00€1mL*10mM (DMSO)329.00€β-CGRP, human acetate
β-CGRP, human acetate is one of calcitonin peptides and acts via the complex of receptor-activity-modifying protein (RAMP) and calcitonin-receptor-like receptorFormula:C164H271N51O50S3Purity:99.35%Color and Shape:SolidMolecular weight:3853.46Vazegepant
CAS:Vazegepant is an intranasal CGRP receptor antagonist utilized for conducting acute migraine research.Formula:C36H46N8O3Purity:98.61%Color and Shape:SolidMolecular weight:638.80Calcitonin-13C6,15N4 TFA
Calcitonin-13CIC6,15NIC4(salmon) (Salmon calcitonin-13CIC6,15NIC4) TFA is a version of calcitonin(salmon) labeled with carbon-13 and nitrogen-15. This hormone regulates calcium and acts dualistically as an agonist to both amylin and calcitonin receptors, promoting bone formation while inhibiting bone resorption.Formula:C1401C5H240N4315NO48S2·5C2HF3O2Color and Shape:SolidMolecular weight:4007.93Telcagepant
CAS:Telcagepant (MK-0974) is an oral calcitonin gene-related peptide receptor (CGRP) antagonist that blocks CGRP receptors, migraines and for pain relief.Formula:C26H27F5N6O3Purity:98.98%Color and Shape:SolidMolecular weight:566.52Atogepant
CAS:Atogepant (MK-8031) is an orally available, selective and potent calcitonin gene-related peptide receptor (CGRP) antagonist for the study of migraine.Formula:C29H23F6N5O3Purity:99.66%Color and Shape:SolidMolecular weight:603.52Ref: TM-T26682
1mg156.00€5mg264.00€10mg329.00€25mg655.00€50mg1,169.00€100mg1,700.00€200mg2,300.00€1mL*10mM (DMSO)354.00€MK-3207 Hydrochloride
CAS:MK-3207 Hydrochloride (MK-3207 HCl) is a potent CGRP receptor antagonist with IC50 and Kiof 0.12 nM and 0.022 nM, highly selective versus human AM1, AM2, CTR, and AMY3. Phase 2.Formula:C31H30ClF2N5O3Purity:98%Color and Shape:SolidMolecular weight:594.05Olcegepant
CAS:Olcegepant (BIBN-4096) is an effective and selective non-peptide calcitonin gene-related peptide 1 (CGRP1) receptor antagonist (IC50 of 0.03 nM and Ki of 14.4Formula:C38H47Br2N9O5Purity:96.08%Color and Shape:SolidMolecular weight:869.65ML230
CAS:ML230 is a selective ATP-binding cassette (ABC) transporter ABCG2 inhibitor.Formula:C25H21N5O3Purity:98%Color and Shape:SolidMolecular weight:439.47Rimegepant
CAS:View and buy Rimegepant from TargetMol.BMS-927711 is a highly potent, oral calcitonin gene-related peptide (CGRP) receptor antagonist with a Ki value of 0.027 nM.Cited in 1 publications.Formula:C28H28F2N6O3Purity:99.1% - 99.8%Color and Shape:SolidMolecular weight:534.56Calcitonin (salmon)
CAS:Calcitonin (salmon), a calcium regulating hormone, is used to treat osteoporosis in women who are at least 5 years past menopause.Formula:C145H240N44O48S2Purity:99.41% - 99.80%Color and Shape:PowderMolecular weight:3431.85Ubrogepant
CAS:Ubrogepant (MK-1602) is an antagonist of calcitonin gene-related peptide receptor that can be used in the acute treatment of migraine studies.Formula:C29H26F3N5O3Purity:99.79%Color and Shape:SolidMolecular weight:549.54Ref: TM-T17194
1mg153.00€5mg378.00€10mg597.00€25mg929.00€50mg1,225.00€100mg1,681.00€1mL*10mM (DMSO)487.00€Erenumab
CAS:Erenumab: human antibody blocking CGRP receptors to prevent migraines.Purity:99.43% (SEC-HPLC) - > 95%Color and Shape:LiquidMolecular weight:146.2 kDaSUN B8155
CAS:SUN B8155 is a CT receptor agonist that induces cAMP formation in cells expressing recombinant human CT receptor.Formula:C14H15N3O3Purity:99.38% - 99.38%Color and Shape:SolidMolecular weight:273.29Galcanezumab
CAS:Galcanezumab: humanized IgG4 antibody that targets CGRP for migraine and cluster headache prevention/treatment.Purity:> 95%Color and Shape:LiquidMolecular weight:144.08 kDa
