Adrenergic Receptor
Adrenergic receptors are GPCRs that are activated by catecholamines, such as adrenaline and noradrenaline. These receptors are classified into alpha and beta subtypes, each of which plays a key role in the regulation of heart rate, blood pressure, and the fight-or-flight response. Adrenergic receptor modulators are essential in the treatment of cardiovascular diseases, asthma, and anxiety disorders. At CymitQuimica, we offer a wide range of high-quality adrenergic receptor modulators to support your research in endocrinology, cardiovascular pharmacology, and stress response.
Subcategories of "Adrenergic Receptor"
Products of "Adrenergic Receptor"
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L748337
CAS:L748337 is a β3-adrenoceptor antagonist that inhibits β3-, β2-, and β1-adrenoceptors and inhibits the protective effects of CL316243.Formula:C26H31N3O5SPurity:99.67% - 99.67%Color and Shape:SolidMolecular weight:497.61Tetrahydrozoline
CAS:Tetrahydrozoline (Tetryzoline) is an alpha-adrenergic agonist that causes vasoconstriction and is widely used in the study of nasal and conjunctival congestion.Formula:C13H16N2Purity:97.85% - 99.77%Color and Shape:SolidMolecular weight:200.28Sertindole
CAS:Sertindole, atypical antipsychotic, targets D2, 5-HT1D, 5-HT2A, 5-HT2C receptors (Kds: 2.7, 20, 0.14, 6 nM).Formula:C24H26ClFN4OPurity:99.74%Color and Shape:Off-White To Pale Yellow SolidMolecular weight:440.94ADRA1D receptor antagonist 1 HCl
CAS:ADRA1D receptor antagonist 1 HCl is a selective α1D adrenergic receptor antagonist (Ki: 1.6 nM) with potential antiproliferative activity.Formula:C15H14Cl2N4OPurity:98.13%Color and Shape:SolidMolecular weight:337.2Medetomidine hydrochloride
CAS:Medetomidine hydrochloride (MPV785) is a selective α2-adrenoceptor agonist, with Ki of 1.08 nM, exhibts 1620-fold selectivity over α1-adrenoceptor.Formula:C13H16N2·HClPurity:99.96%Color and Shape:White Or Off White Crystalline PowderMolecular weight:236.74Imiloxan
CAS:Imiloxan (RS-21361) is an α2 adrenergic receptor antagonist used in the treatment of major depressive disorder.Formula:C14H16N2O2Purity:100% - 98.89%Color and Shape:SolidMolecular weight:244.29Tizanidine hydrochloride
CAS:Tizanidine hydrochloride (Tizanidine HCl), an α2-adrenergic receptor agonist, inhibits neurotransmitter release from CNS noradrenergic neurons.Formula:C9H9Cl2N5SPurity:99.96%Color and Shape:Solid WhiteMolecular weight:290.17Ref: TM-T0290
10mg51.00€25mg64.00€50mg95.00€100mg105.00€200mg133.00€500mg212.00€1mL*10mM (DMSO)42.00€SR59230A hydrochloride
CAS:SR59230A hydrochloride (SR59230A HCl) is a beta3-adrenergic receptor antagonist that inhibits ultradian brown adipose tissue thermogenesis.Formula:C21H28ClNO2Purity:99.49%Color and Shape:SolidMolecular weight:361.91Pipoxazole
CAS:Pipoxazole, an adrenergic receptor antagonist, is used potentially for the treatment of depression.Formula:C14H20N4OPurity:97.88% - 99.19%Color and Shape:SolidMolecular weight:260.33Bambuterol hydrochloride
CAS:Bambuterol hydrochloride (KWD-2183 hydrochloride) , a long-acting beta-adrenoceptor agonist, is utilized for the treating of asthma.Formula:C18H30ClN3O5Purity:99.53% - 99.61%Color and Shape:White SolidMolecular weight:403.91Brexpiprazole
CAS:Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.Formula:C25H27N3O2SPurity:99.06% - 99.96%Color and Shape:SolidMolecular weight:433.57Salmeterol
CAS:Salmeterol (GR33343X) is a long-acting agonist of beta2-adrenergic receptor (beta 2AR) used for treatment ofasthma.Formula:C25H37NO4Purity:99.2% - 99.9%Color and Shape:SolidMolecular weight:415.57A 61603
CAS:Cixutumumab (IMC-A12) is a humanized IgG monoclonal antibody targeting the IGF1R with anticancer activity.Formula:C14H20BrN3O3SColor and Shape:SolidMolecular weight:390.3Brefonalol HCl
Brefonalol HCl, ADRA blocker for neurological/cardiovascular issues, treats angina, arrhythmias, hypertension.Formula:C22H29ClN2O2Purity:99.45%Color and Shape:SolidMolecular weight:388.935-Bromoimidazo[1,2-A]Pyrazine
CAS:5-Bromoimidazo[1,2-a]pyrazine inhibits phosphodiesterase and beta-adrenergic receptors.5-Bromoimidazo[1,2-a]pyrazine shows antibronchospastic activity in vitro.Formula:C6H4BrN3Purity:97.04%Color and Shape:SolidMolecular weight:198.02Cyclazosin HCl
CAS:Cyclazosin HCl is an α-adrenergic receptor antagonist that can be used to study non-arteritic ischemic optic neuropathy.Formula:C23H28ClN5O4Purity:99.44%Color and Shape:SolidMolecular weight:473.95Ancarolol
CAS:Ancarolol is a blocking agent of beta-adrenergic.Formula:C18H24N2O4Purity:98%Color and Shape:SolidMolecular weight:332.39Bucumolol
CAS:Bucumolol (Bucumarol) is a β-adrenergic blocking agent and a local anesthetic with antihypertensive activity and can be used to study myocardial infarction.Formula:C17H23NO4Purity:99.70%Color and Shape:SoildMolecular weight:305.371-(2-Pyridyl)piperazine
CAS:1-(2-Pyridyl)piperazine (NSC-13778) is a selective α2-adrenoceptor antagonists.Formula:C9H13N3Purity:98.92%Color and Shape:Clear Colorless To Pale Yellow LiquidMolecular weight:163.22OPC-28326
CAS:OPC-28326: an α2-adrenergic blocker; dilates blood vessels; inhibits α2A/B/C receptors with Ki 2040/285/55 nM.Formula:C26H35N3O2Purity:98.56%Color and Shape:SolidMolecular weight:421.58Ref: TM-T13804
1mg187.00€5mg455.00€10mg620.00€25mg940.00€50mg1,264.00€100mg1,663.00€200mg2,252.00€1mL*10mM (DMSO)567.00€Metoprolol tartrate
CAS:Metoprolol Tartrate is a blocker of the cardioselective β-adrenergic receptor.Formula:C15H25NO3C4H6O6Purity:99.72% - 99.93%Color and Shape:White To Off-White / PowderMolecular weight:684.81Tamsulosin
CAS:Tamsulosin: an alpha1A blocker for easing urination in BPH by relaxing prostate and bladder muscles.Formula:C20H28N2O5SPurity:99.94%Color and Shape:White CrystalsMolecular weight:408.51Ecastolol
CAS:Ecastolol has anti-angina activity and is an adrenergic receptor antagonist.Formula:C26H33N3O6Purity:98.1%Color and Shape:SolidMolecular weight:483.56Ref: TM-T11148
1mg369.00€5mg735.00€10mg938.00€25mg1,473.00€50mg1,882.00€100mg2,670.00€1mL*10mM (DMSO)929.00€Butofilolol
CAS:Butofilolol is a novel beta-blocker with antihypertensive activity and can be used to study hypertension.Formula:C17H26FNO3Purity:100% - 99%Color and Shape:SolidMolecular weight:311.392Brimonidine
CAS:Brimonidine (Bromoxidine) is a drug used as eye drops under the brand names Alphagan and Alphagan-P.Formula:C11H10BrN5Purity:98.60%Color and Shape:Yellow SolidMolecular weight:292.13Ref: TM-T20157
5mg57.00€10mg87.00€25mg173.00€50mg339.00€100mg502.00€500mg1,121.00€1mL*10mM (DMSO)64.00€ICI 118,551 hydrochloride
CAS:ICI 118,551 hydrochloride (ICI 118551 hydrochloride) is a highly selective β2 adrenergic receptor antagonist (Kis: 0.7, 49.5, and 611 nM for β2, β1, and β3Formula:C17H28ClNO2Purity:99.53% - 99.7%Color and Shape:SolidMolecular weight:313.86CGP-20712
CAS:CGP-20712 is a selective β 1-adrenoceptor antagonist with an IC50 of 0.7 nM.Formula:C23H25F3N4O5Purity:100% - 99.40%Color and Shape:SolidMolecular weight:494.46Ref: TM-T30846
1mg333.00€5mg787.00€10mg1,074.00€25mg1,510.00€50mg1,882.00€100mg2,375.00€500mg4,655.00€ORM-10921
CAS:ORM-10921 is an α2C-adrenoceptor antagonist that has shown antipsychotic and antidepressant activity in animal studies.Formula:C18H23NO2Purity:99.46% - 99.75%Color and Shape:SolidMolecular weight:285.38Tamsulosin hydrochloride
CAS:Tamsulosin hydrochloride (Flomax hydrochloride) is the hydrochloride salt of tamsulosin, a sulfonamide derivative with α1 adrenergic antagonist activity.Formula:C20H29ClN2O5SPurity:100% - 99.95%Color and Shape:White To Off-White SolidMolecular weight:444.97Hydrocortisone 17-butyrate
CAS:Hydrocortisone 17-butyrate (Cortisol 17-butyrate) is a glucocorticoid receptor agonist with antiinflammatory, antipruritic and vasoconstrictive effects.Formula:C25H36O6Purity:98% - 99.57%Color and Shape:SolidMolecular weight:432.55Buflomedil hydrochloride
CAS:Buflomedil hydrochloride (Fonzylane), a vasodilator, is used in therapy of claudication or the symptoms of the peripheral arterial disease.Formula:C17H26ClNO4Purity:99.67% - 99.7%Color and Shape:White Or Off-White Crystalline PowderMolecular weight:343.85Naftopidil hydrochloride
CAS:Naftopidil HCl (BM-15275) is a selective alpha1 blocker with Ki: α1a-3.7 nM, α1b-20 nM, α1d-1.2 nM; it also inhibits cell growth.Formula:C24H29ClN2O3Purity:99.50%Color and Shape:SolidMolecular weight:428.95Ref: TM-T9220
1mg44.00€5mg87.00€10mg117.00€25mg202.00€50mg304.00€100mg437.00€200mg612.00€1mL*10mM (DMSO)97.00€Atomoxetine hydrochloride
CAS:Atomoxetine HCl (LY 139603) is a selective non-stimulant ADHD drug that blocks norepinephrine reuptake, enhancing focus and reducing impulsivity.Formula:C17H22ClNOPurity:99.86%Color and Shape:White SolidMolecular weight:291.82Rotigotine Hydrochloride
CAS:Rotigotine HCl, D3-preferential dopamine agonist, is 50x stronger than quinpirole in anti-Parkinson's efficacy.Formula:C19H26ClNOSPurity:99.53% - 99.56%Color and Shape:Almost White To White Crystalline PowderMolecular weight:351.93Ritanserin
CAS:Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.Formula:C27H25F2N3OSPurity:99.45% - 99.89%Color and Shape:SolidMolecular weight:477.57Tiprenolol
CAS:Tiprenolol is a beta adrenergic receptor antagonist.[1]Formula:C13H21NO2SPurity:99.43%Color and Shape:SolidMolecular weight:255.38Ref: TM-T50081
1mg84.00€5mg172.00€10mg249.00€25mg411.00€50mg562.00€100mg787.00€200mg1,035.00€1mL*10mM (DMSO)158.00€Carazolol
CAS:Carazolol (Suacron) is a high-affinity antagonist/partial inverse agonist (also referred to as a beta blocker) of the β-adrenergic receptor.Formula:C18H22N2O2Purity:98.54% - 99.08%Color and Shape:Yellowish SolidMolecular weight:298.38Procaterol hydrochloride
CAS:Short-acting β2-adrenergic receptor agonist used to treat asthma.Formula:C32H48Cl2N4O7Purity:100% - 99.97%Color and Shape:SolidMolecular weight:671.65Doxazosin
CAS:Doxazosin (UK 33274) is a long-lasting inhibitor of α1-adrenoceptors that is widely used to treat benign prostatic hyperplasia and lower urinary tract symptoms.Formula:C23H25N5O5Purity:99.47% - 99.85%Color and Shape:SolidMolecular weight:451.48(±)-Prenalterol
CAS:(±)-Prenalterol (H 80/62) is an agonist of beta-2- and beta-1-adrenergic receptors and is used to study chronic congestive heart failure.Formula:C12H19NO3Purity:99.71%Color and Shape:SolidMolecular weight:225.28(S)-(-)-Propranolol hydrochloride
CAS:(S)-(-)-Propranolol hydrochloride 是一种有效的肾上腺素能受体 (β-adrenergic receptor) 拮抗剂,具有抗高血压活性和潜在的抗癌活性,对β1,β2,和β3受体有抑制作用。(S)-(-)-Propranolol hydrochloride 可改善严重烧伤患者的预后,可用于研究酒精症。Formula:C16H22ClNO2Purity:99.02% - 99.85%Color and Shape:SolidMolecular weight:295.8Dibenamine hydrochloride
CAS:Dibenamine hydrochloride is a competitive and irreversible blocking agent of the β-adrenergic receptor.Formula:C16H19Cl2NPurity:96.43%Color and Shape:Oily Liquid SolidMolecular weight:296.23TAAR1 agonist 3
CAS:TAAR1 agonist 3 is a potent agonist of Trace Amine-Associated Receptor 1 (TAAR1) with a pEC50 value of 7.6. Additionally, it acts as a full agonist at the α2AR with a pEC50 of 6. TAAR1 agonist 3 is utilized in the research of neuropsychiatric disorders.Formula:C10H13NOColor and Shape:SolidMolecular weight:163.22Norepinephrine
CAS:Norepinephrine (Levophed) can stimulate apoptosis in adult rat ventricular myocytes by activation of the β-adrenergic pathway.Formula:C8H11NO3Purity:98.56% - 99.84%Color and Shape:Colorless Micr°Crystals SolidMolecular weight:169.18Trifluoperazine
CAS:Trifluoperazine (trifluoroperazine) is a Dopamine D2 receptor inhibitor(IC50 : 1.2 nM), and Treatment of schizophrenia.Formula:C21H24F3N3SPurity:98.3% - 99.46%Color and Shape:White To Yellowish Crystalline PowderMolecular weight:407.5Indanidine
CAS:Indanidine is a highly selective and potent α-adrenergic agonist with antihypertensive activity.Indanidine is an α-adrenergic antagonist that can be used in theFormula:C11H13N5Purity:100%Color and Shape:SolidMolecular weight:215.25Xamoterol hemifumarate
CAS:Xamoterol hemifumarate is a potent and selective β1-adrenoceptor agonist.Xamoterol hemifumarate is a potential compound for the study of the relationshipFormula:C36H54N6O14Purity:99.79%Color and Shape:White SolidMolecular weight:794.37Yohimbine
CAS:Yohimbine is a nonselective alpha 2-adrenergic receptor (AR) antagonist(IC50 : 0.6 μM)Formula:C21H26N2O3Purity:99.75% - 99.84%Color and Shape:SolidMolecular weight:354.4Tolamolol
CAS:Tolamolol is a selective β-adrenergic blocker that significantly reduces the degree of exercise-induced inhibition of the S-T segment and can be used in theFormula:C19H24N2O4Purity:97.58%Color and Shape:SolidMolecular weight:344.4Pafenolol
CAS:Pafenolol is a P-glycoprotein modulator with a Ki value of 5.5 µM. pafenolol is an orally available and selective beta-adrenergic receptor antagonist.Formula:C18H31N3O3Purity:98.43%Color and Shape:SolidMolecular weight:337.46
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