Adrenergic Receptor
Adrenergic receptors are GPCRs that are activated by catecholamines, such as adrenaline and noradrenaline. These receptors are classified into alpha and beta subtypes, each of which plays a key role in the regulation of heart rate, blood pressure, and the fight-or-flight response. Adrenergic receptor modulators are essential in the treatment of cardiovascular diseases, asthma, and anxiety disorders. At CymitQuimica, we offer a wide range of high-quality adrenergic receptor modulators to support your research in endocrinology, cardiovascular pharmacology, and stress response.
Subcategories of "Adrenergic Receptor"
Products of "Adrenergic Receptor"
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Apraclonidine hydrochloride
CAS:Apraclonidine hydrochloride (ALO 2145) is an α2-adrenergic agonist and a weak α-1 adrenergic receptor agonist.Formula:C9H11Cl3N4Purity:98.01%Color and Shape:SolidMolecular weight:281.57N-Nitroso Atenolol
CAS:N-Nitroso Atenolol is a derivative of Atenolol. At concentrations ranging from 0.1 to 1 mM, it induces DNA fragmentation in rat hepatocytes.Formula:C14H21N3O4Color and Shape:SolidMolecular weight:295.33Clonidine hydrochloride
CAS:Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.Formula:C9H10Cl3N3Purity:99.16% - 99.99%Color and Shape:SolidMolecular weight:266.55Dronedarone
CAS:Dronedarone (SR 33589) is an amiodarone analogue which has an effective and promising treatment for Atrial fibrillation.Formula:C31H44N2O5SPurity:98.85% - 99.58%Color and Shape:SolidMolecular weight:556.76ZK-90055 hydrochloride
CAS:ZK-90055 hydrochloride is a β2 adrenergic receptor agonist used to study asthma.Formula:C16H23ClN2O4Purity:99.67%Color and Shape:SolidMolecular weight:342.82Esmolol acid hydrochloride
CAS:Esmolol acid (ASL-8123) hydrochloride is a mild antagonist of β-adrenergic receptors. It inhibits the heart rate and diastolic pressure responses induced by Isoproterenol in a dose-dependent manner and is applicable for renal failure research.Formula:C15H24ClNO4Color and Shape:SolidMolecular weight:317.81Metipranolol
CAS:Metipranolol (Betamann) is a type of β- Adrenergic receptors( β- A potent antagonist of adrenergic receptor on guinea pig atria β 1- Adrenergic receptors and rat uterus β The 2-adrenergic receptor exhibited the beta blocking potentials (pA2) of 8.3 and 8.4, respectively. It is also a potent substituent in the 3H DHA binding assay, with a ligand concentration of 0.7 nM and a Ki of 39 ± 24 nM.Formula:C17H27NO4Purity:98.37%Color and Shape:SolidMolecular weight:309.4Talipexole dihydrochloride
CAS:Talipexole dihydrochloride (Domnin) is a dopamine D2 receptor agonist, α2-adrenoceptor agonist, and 5-HT3 receptor antagonist in both rat cortical andFormula:C10H17Cl2N3SPurity:98.64%Color and Shape:Light Yellow SolidMolecular weight:282.23Ref: TM-T14490
2mg38.00€5mg56.00€10mg89.00€25mg154.00€50mg264.00€100mg424.00€200mg613.00€500mg949.00€1mL*10mM (DMSO)63.00€Tizanidine
CAS:Tizanidine, an α2-adrenergic receptor agonist, suppresses the release of neurotransmitters from central nervous system (CNS) noradrenergic neurons.Formula:C9H8ClN5SPurity:99.75%Color and Shape:White SolidMolecular weight:253.71Phentolamine Analogue 1
CAS:Phentolamine Analogue 1 is an analogue of phentolamine. Phentolamine is a nonselective antagonist of α-adrenergic.Formula:C17H19N3OPurity:98.54%Color and Shape:SolidMolecular weight:281.35Ref: TM-T12444
1mg86.00€5mg172.00€10mg259.00€25mg425.00€50mg598.00€100mg810.00€200mg1,074.00€1mL*10mM (DMSO)172.00€Rilmenidine Phosphate
CAS:Rilmenidine Phosphate is a selective I(1) imidazoline receptor agonist, used to treat hypertension.Formula:C10H19N2O5PPurity:99.87% - ≥95%Color and Shape:SolidMolecular weight:278.24Ref: TM-T6641
1mg40.00€5mg88.00€10mg137.00€25mg264.00€50mg418.00€100mg627.00€500mg1,301.00€1mL*10mM (DMSO)87.00€Carteolol hydrochloride
CAS:Carteolol hydrochloride is a nonselective beta-blocker used to treat hypertension, arrhythmias, angina, and glaucoma.Formula:C16H24N2O3·HClPurity:99.84% - 99.91%Color and Shape:SolidMolecular weight:328.83Ref: TM-T1282
10mg37.00€25mg52.00€50mg79.00€100mg111.00€200mg165.00€500mg268.00€1mL*10mM (DMSO)55.00€BRL 44408 Maleate Salt
CAS:BRL 44408 Maleate is an α2A-adrenoceptor antagonist with antidepressant and analgesic activity.Formula:C17H21N3O4Purity:98.71%Color and Shape:SolidMolecular weight:331.37Milveterol HCl
CAS:Milveterol HCl is a long-acting β(2) -adrenergic receptor agonist for the potential treatment of chronic obstructive pulmonary disease (COPD).Formula:C25H30ClN3O4Purity:98.2%Color and Shape:SolidMolecular weight:471.982-(1-Piperazinyl)pyrimidine
CAS:2-(1-Piperazinyl)pyrimidine is used as an anti-anxiety drug.Formula:C8H12N4Purity:98.46%Color and Shape:Liquid - Crystal - LumpMolecular weight:164.21Tulobuterol hydrochloride
CAS:Tulobuterol hydrochloride (Hokunalin) is a long-acting beta2-adrenergic receptor agonist.Formula:C12H19Cl2NOPurity:99.24% - 99.96%Color and Shape:Appearance White Crystalline PowderMolecular weight:264.19Batefenterol
CAS:Batefenterol (GSK961081) is a muscarinic antagonist and β2-agonist with high affinity (Ki: 1.4/1.3/3.7 nM).Formula:C40H42ClN5O7Purity:97.94% - 98.4%Color and Shape:SolidMolecular weight:740.24Vatinoxan hydrochloride
CAS:Vatinoxan hydrochloride is an antagonist of the peripheral α2 adrenergic receptors.Formula:C20H27ClN4O4SPurity:98%Color and Shape:SolidMolecular weight:454.97Nemazoline Free Base
CAS:Nemazoline Free Base: a long-lasting nasal decongestant, better than oxymetazoline, with no systemic effects or toxicity in dogs and rats.Formula:C10H11Cl2N3Purity:99.03% - 99.18%Color and Shape:SolidMolecular weight:244.12Tamsolusin Hydrochloride
CAS:Tamsolusin Hydrochloride (YM 12617) is a highly selective alpha-1A adrenergic receptor antagonist used in the treatment of benign prostatic hypertrophy.Formula:C20H29ClN2O5SPurity:99.92%Color and Shape:SoildMolecular weight:444.97MG 1
CAS:MG 1 is a potent alpha-1 adrenergic receptor antagonist.Formula:C17H25N3O2Purity:100% - 99.73%Color and Shape:SolidMolecular weight:303.4Amosulalol
CAS:Amosulalol is a combined alpha and beta adrenoceptor antagonist.Formula:C18H24N2O5SPurity:98.91%Color and Shape:SolidMolecular weight:380.46Ref: TM-T30027
1mg185.00€2mg279.00€5mg425.00€10mg625.00€25mg938.00€50mg1,311.00€100mg1,795.00€1mL*10mM (DMSO)454.00€Moprolol
CAS:Moprolol ((±)-Moprolol) is a beta-adrenergic receptor antagonist utilized in research pertaining to essential hypertension [1] [2] [3].Formula:C13H21NO3Purity:98%Color and Shape:SolidMolecular weight:239.31Nylidrin hydrochloride
CAS:Nylidrin HCl inhibits IgG1-induced histamine release in guinea pigs and IgE-induced release in rat mast cells & human basophils.Formula:C19H26ClNO2Purity:99.35%Color and Shape:SolidMolecular weight:335.87(R)-Terazosin
CAS:R-Terazosin is the active R-enantiomer and potent α1-adrenoceptor antagonist (Ki: α1a 6.51 nM, α1b 1.01 nM, α1d 1.97 nM).Formula:C19H25N5O4Purity:98.87% - 98.96%Color and Shape:SolidMolecular weight:387.43Ref: TM-T12643
1mg47.00€2mg64.00€5mg96.00€10mg145.00€25mg240.00€50mg353.00€100mg495.00€500mgTo inquire1mL*10mM (DMSO)105.00€Lofexidine
CAS:Lofexidine is a selective α2-receptor agonist, Lofexidine reduces narcotic withdrawal symptoms.Formula:C11H12Cl2N2OPurity:98.78%Color and Shape:SolidMolecular weight:259.132-Methoxyidazoxan monohydrochloride
CAS:L-Albizziin (2-Methoxyidazoxan monohydrochloride) is a highly potent selective antagonist of the alpha 2r adrenergic receptor.Formula:C12H14N2O3·HClPurity:98.99%Color and Shape:SolidMolecular weight:270.72Meranzin
CAS:Meranzin, a bioactive from TCM CSS, targets alpha 2-adrenoceptor, affects AMPA-ERK1/2-BDNF pathway, and may prevent atherosclerosis and depression.Formula:C15H16O4Purity:95.08% - 99.3%Color and Shape:SolidMolecular weight:260.29LUN42518 HCl 47142-51-8(free base)
LUN42518 HCl is an analogue of phentolamine. Phentolamine is a nonselective alpha-adrenergic antagonist.Formula:C17H20ClN3OPurity:99.96%Color and Shape:SolidMolecular weight:317.81Ref: TM-T8738
1mg88.00€5mg172.00€10mg259.00€25mg425.00€50mg598.00€100mg810.00€200mg1,074.00€1mL*10mM (DMSO)170.00€Esprolol
CAS:Esprolol (ACC-9369 free base) is a novel beta-adrenergic antagonist used to study exertional angina.Formula:C17H27NO4Purity:100% - 99.16%Color and Shape:SoildMolecular weight:309.4KUL-7211 racemate
CAS:KUL 7211, a selective β-adrenoceptor agonist, exists as a racemate, referred to as KUL 7211 racemate, which is the mixture of its enantiomers.Formula:C19H23NO5Purity:98%Color and Shape:SolidMolecular weight:345.39Nicergoline
CAS:Nicergoline (Nicergolinum) is an ergot derivative used to treat senile dementia and other disorders with vascular origins.Formula:C24H26BrN3O3Purity:100% - 99.53%Color and Shape:SolidMolecular weight:484.39Ref: TM-T1132
5mg35.00€10mg51.00€25mg67.00€50mg85.00€100mg104.00€200mg145.00€500mg234.00€1mL*10mM (DMSO)57.00€Betaxolol hydrochloride
CAS:Betaxolol HCl (SL 75212) is a cardioselective beta-blocker for hypertension without reported liver injury.Formula:C18H30ClNO3Purity:99.48% - 99.56%Color and Shape:SolidMolecular weight:343.89Phenoxybenzamine hydrochloride
CAS:Phenoxybenzamine hydrochloride: non-selective, irreversible alpha-blocker; antihypertensive, vasodilator, may cause tachycardia, potential carcinogen.Formula:C18H23Cl2NOPurity:100% - 98.04%Color and Shape:Antihypertensive DrugMolecular weight:340.3Atenolol
CAS:Atenolol (Tenormin) is a selective β1 receptor antagonist.Formula:C14H22N2O3Purity:99.07% - 99.95%Color and Shape:White Crystalline Powder SolidMolecular weight:266.3361Levobunolol hydrochloride
CAS:Levobunolol hydrochloride 是一种非选择性的 β-肾上腺素受体阻滞剂,可用于治疗青光眼和上斜肌肌障碍的研究。Formula:C17H26ClNO3Purity:100% - 98.49%Color and Shape:SolidMolecular weight:327.85Blonanserin
CAS:Blonanserin (AD-5423), approved in Japan (2008), is an atypical antipsychotic with fewer side effects like EPS, sedation, or hypotension.Formula:C23H30FN3Purity:99.85%Color and Shape:SolidMolecular weight:367.5Falintolol
CAS:Falintolol is a novel beta-adrenergic antagonist with antihypertensive effects and can be used to study glaucoma.Formula:C12H24N2O2Purity:100% - 100%Color and Shape:SolidMolecular weight:228.33D2343
CAS:D2343 is an agonist of β2-adrenoceptor. It also is an inhibitor of α1- adrenoceptor.Formula:C20H27NO3Purity:98%Color and Shape:SolidMolecular weight:329.43Guanadrel
CAS:Guanadrel is an antihypertensive agent.Formula:C10H19N3O2Purity:98%Color and Shape:SolidMolecular weight:213.28Dabelotine
CAS:Dabelotine (UNII-6RY56RB98P) is an adrenergic agonist used in the study of dementia.Formula:C15H22N2O2Purity:98.55%Color and Shape:SolidMolecular weight:262.35BMY 7378 dihydrochloride
CAS:BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.Formula:C22H33Cl2N3O3Purity:97.32% - 99.08%Color and Shape:SolidMolecular weight:458.42RS 100329 hydrochloride
CAS:RS 100329 hydrochloride is an antagonist of α1A-adrenergic receptor.Formula:C20H26ClF3N4O3Purity:100%Color and Shape:SolidMolecular weight:462.89Ajmalicine
CAS:Ajmalicine (Raubasine): Blocks α1-adrenoceptor, non-competitive nicotine receptor inhibitor (IC50=72.3 μM), anti-hypertensive, sedative.Formula:C21H24N2O3Purity:96.9%Color and Shape:SolidMolecular weight:352.43Azepexole hydrochloride
CAS:Azepexole hydrochloride (4H-Oxazolo[4,5-d]azepin-2-amine, 6-ethyl-5,6,7,8-tetrahydro-, hydrochloride (1:1)) is a potent α2-Adrenoceptor agonist with anaestheticFormula:C9H16ClN3OPurity:98.03% - 99.72%Color and Shape:SoildMolecular weight:217.7Methylhexanamine hydrochloride
CAS:Methylhexanamine hydrochloride is a fatty amine and vasoconstrictor that functions as a nasal decongestant when inhaled through the nasal mucosa.Formula:C7H18ClNColor and Shape:SolidMolecular weight:151.68Talinolol
CAS:(±)-Talinolol is a selective β1 adrenoceptor antagonist well known for its cardioprotective and antihypertensive activity.Formula:C20H33N3O3Purity:98.80%Color and Shape:SolidMolecular weight:363.49Ref: TM-T21640
2mg35.00€5mg50.00€10mg96.00€25mg188.00€50mg329.00€100mg565.00€200mg818.00€1mL*10mM (DMSO)55.00€Tetrahydrozoline hydrochloride
CAS:Tetrahydrozoline hydrochloride (Murine Plus) is an imidazoline derivative with alpha receptor agonist activity.Formula:C13H16N2·HClPurity:99.90%Color and Shape:Off-White SolidMolecular weight:236.74Indacaterol maleate
CAS:Indacaterol maleate (QAB149) is an ultra-long-acting β-adrenoceptor agonist.Formula:C28H32N2O7Purity:99.03% - 99.67%Color and Shape:SolidMolecular weight:508.56Bedoradrine sulfate
CAS:Bedoradrine sulfate (MN-221 sulfate) is a novel, highly selective β2-adrenoceptor agonist.Cost-effective and quality-assured.Formula:C24H32N2O5H2O4SPurity:99.31%Color and Shape:SolidMolecular weight:477.56
