Adrenergic Receptor
Adrenergic receptors are GPCRs that are activated by catecholamines, such as adrenaline and noradrenaline. These receptors are classified into alpha and beta subtypes, each of which plays a key role in the regulation of heart rate, blood pressure, and the fight-or-flight response. Adrenergic receptor modulators are essential in the treatment of cardiovascular diseases, asthma, and anxiety disorders. At CymitQuimica, we offer a wide range of high-quality adrenergic receptor modulators to support your research in endocrinology, cardiovascular pharmacology, and stress response.
Subcategories of "Adrenergic Receptor"
Products of "Adrenergic Receptor"
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Detomidine hydrochloride
CAS:Detomidine hydrochloride (MPV-253 AII) produce dose-dependent sedative and analgesic effects, mediatated by activation of α2 catecholamine receptors.Formula:C12H14N2·HClPurity:99.97%Color and Shape:SolidMolecular weight:222.71Terazosin hydrochloride dihydrate
CAS:Terazosin hydrochloride dihydrate (Heitrin dihydrate) is a selective α1-adrenoceptor antagonist, used for treatment of symptoms of an enlarged prostate (BPH).Formula:C19H25N5O4·HCl·2H2OPurity:99.81%Color and Shape:White Or Off-White Crystalline PowderMolecular weight:459.92Arbutamine
CAS:Arbutamine (GP 21213) is a β-adrenoceptor agonist with alpha-1-sympathomimetic activity that can be used to study cardiac stress.Formula:C18H23NO4Purity:95.06%Color and Shape:SolidMolecular weight:317.38Nardeterol HCl
Nardeterol HCl is a β-adrenergic receptor partial agonist used in the study of the central nervous system.CAS 번호13460-73-83-4Formula:C20H25ClFN3O2Purity:97.36% - 98%Color and Shape:SoildMolecular weight:393.88Droxidopa
CAS:Droxidopa (L-DOPS), an oral prodrug, treats symptomatic orthostatic hypotension from neurogenic autonomic failure.Formula:C9H11NO5Purity:98% - 98.12%Color and Shape:SolidMolecular weight:213.19Guanabenz hydrochloride
CAS:Guanabenz hydrochloride (NE56490) is an orally active α2-adrenoceptor agonist with hypotensive effects.Formula:C8H9Cl3N4Purity:99.45%Color and Shape:SolidMolecular weight:267.54Clonidine
CAS:Clonidine (Kapvay): central alpha-adrenergic agonist, antihypertensive, often combined, not tied to liver issues.Formula:C9H9Cl2N3Purity:99.44% - 99.88%Color and Shape:Crystals SolidMolecular weight:230.09Salbutamol hemisulfate
CAS:Salbutamol hemisulfate (Albuterol Sulfate) is a short-acting β2-adrenergic receptor agonist with an IC50 of 8.93 μM.Formula:C13H21NO3H2O4SPurity:99.35%Color and Shape:White Or Almost White Odourless PowderMolecular weight:576.7Todralazine hydrochloride
CAS:Todralazine hydrochloride, a β2AR blocker with antioxidant properties, is used in hypertension studies.Formula:C11H13ClN4O2Purity:98.32%Color and Shape:SolidMolecular weight:268.7Mirtazapine
CAS:Mirtazapine is a unique tetracyclic antidepressant, may cause temporary liver enzyme elevation, and is linked to rare liver injury.Formula:C17H19N3Purity:99.98%Color and Shape:SolidMolecular weight:265.35Dobutamine hydrochloride
CAS:Dobutamine hydrochloride (Dobutamine (hydrochloride)) is a catecholamine that acts as a β-adrenergic receptor agonist with potent positive inotropic effects.Formula:C18H24ClNO3Purity:97.15% - 99.94%Color and Shape:SolidMolecular weight:337.84N-Methyldopamine hydrochloride
CAS:N-Methyldopamine hydrochloride (Ephinine hydrochloride) is an α and β agonist, with indirect sympathomimetic effects similar to dopamine.Formula:C9H14ClNO2Color and Shape:SolidMolecular weight:203.67Neldazosin
CAS:Neldazosin is used as a potent α1-adrenoceptor antagonist.Formula:C18H25N5O4Purity:100% - 99.87%Color and Shape:SolidMolecular weight:375.42Ref: TM-T61535
1mg200.00€5mg504.00€10mg727.00€25mg1,121.00€50mg1,510.00€100mg2,043.00€500mg4,075.00€1mL*10mM (DMSO)525.00€Detomidine carboxylic acid
CAS:Detomidine carboxylic acid, a urine metabolite of detomidine, is a synthetic α2-agonist, animal analgesic, with cardiac, respiratory, and diuretic effects.Formula:C12H12N2O2Purity:98%Color and Shape:SolidMolecular weight:216.24Harmane
CAS:Harmane (Loturine) is a bio-active β-Carboline and monoamine oxidase inhibitor found in coffee and tobacco smoke.Formula:C12H10N2Purity:100% - 97.89%Color and Shape:Off-White SolidMolecular weight:182.22nifenalol.HCl
CAS:Nifenalol.HCl(INPEA) is a antagonist of β-adrenergic receptor.Formula:C11H17ClN2O3Purity:99.96%Color and Shape:SolidMolecular weight:260.72Bedoradrine
CAS:Bedoradrine (MN-221) free base is a novel, highly selective β2-adrenoceptor agonist.Cost-effective and quality-assured.Formula:C24H32N2O5Purity:100%Color and Shape:SolidMolecular weight:428.52Brimonidine Tartrate
CAS:Brimonidine Tartrate (AGN190342 tartrate) is a quinoxaline derivative and adrenergic α-2 receptor agonist (EC50: 0.45 nM).Formula:C15H16BrN5O6Purity:99.95%Color and Shape:Off-White Crystalline SolidMolecular weight:442.22(±)-N-Methylcoclaurine
CAS:N-Methylcoclaurine (±) acts as a selective antagonist at the α2-adrenoceptor [1].Formula:C18H21NO3Purity:98%Color and Shape:SolidMolecular weight:299.36(S)-Bucindolol
CAS:(S)-Bucindolol is an enantiomer of bucindolol, specifically a β1-adrenergic receptor antagonist. It is primarily utilized in research related to heart failure.Formula:C22H25N3O2Color and Shape:SolidMolecular weight:363.45Pimozide
CAS:Pimozide: antipsychotic that blocks type 2 dopamine, alpha-adrenergic, and 5-HT2 receptors, reducing tics and delusions.Formula:C28H29F2N3OPurity:100% - 99.85%Color and Shape:SolidMolecular weight:461.55Aclidinium
CAS:Aclidinium, a dual-action compound, serves as a long-acting muscarinic antagonist and a β2-adrenoceptor (β2-AR) agonist, exhibiting bronchodilator properties. It effectively reduces lung hyperinflation, enhances lung function, and prolongs exercise endurance time. This compound is commonly utilized in studies focusing on chronic obstructive pulmonary disease (COPD).Formula:C26H30NO4S2Color and Shape:SolidMolecular weight:484.65Pardoprunox hydrochloride
CAS:Pardoprunox hydrochloride (SLV-308 hydrochloride) is a novel partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist, D2 (pKi = 8.1)Formula:C12H16ClN3O2Purity:98.73% - 99.13%Color and Shape:SolidMolecular weight:269.73Labetalone hydrochloride
CAS:Labetalone hydrochloride, a Labetalol impurity, is an orally active alpha and beta-adrenoceptor blocker.Formula:C19H23ClN2O3Purity:99.06%Color and Shape:SolidMolecular weight:362.85Tolazoline
CAS:Tolazoline (Benzalolin), a vasodilator, treats vessel spasms and reverses 5-HT2A drug overdose effects.Formula:C10H12N2Purity:97.51%Color and Shape:SolidMolecular weight:160.22Nebivolol hydrochloride
CAS:Nebivolol hydrochloride is a beta-1 blocker and vasodilator treating hypertension and heart failure in the elderly.Formula:C22H25F2NO4·HClPurity:100% - 99.77%Color and Shape:White To Off-White PowderMolecular weight:441.9Ref: TM-T0154
10mg50.00€25mg69.00€50mg96.00€100mg163.00€200mg268.00€500mg464.00€1mL*10mM (DMSO)46.00€RS 17053 hydrochloride
CAS:RS 17053 hydrochloride: selective α1A adrenoceptor antagonist, pKi 9.1, pA2 9.8.Formula:C24H30Cl2N2O2Purity:99.27%Color and Shape:SolidMolecular weight:449.41Phenylephrine
CAS:Phenylephrine ((R)-(-)-Phenylephrine) is a selective α1-adrenoceptor agonist ( pKi: 5.86, 4.87 and 4.70 for α1D, α1B, and α1A receptors respectively).Formula:C9H13NO2Purity:99.87% - 99.89%Color and Shape:SolidMolecular weight:167.21Bucindolol Formate
Bucindolol is a β1-adrenergic blocker with sympathomimetic activity, used in heart failure research.Formula:C23H27N3O4Purity:99.11% - 99.61%Color and Shape:SolidMolecular weight:409.48Ref: TM-T10631L
1mg185.00€5mg415.00€10mg613.00€25mg938.00€50mg1,311.00€100mg1,768.00€500mg3,535.00€1mL*10mM (DMSO)465.00€Higenamine hydrochloride
CAS:Higenamine HCl is a β2 adrenoreceptor agonist active in fat and muscle tissue.Formula:C16H18ClNO3Purity:98.75% - 99.80%Color and Shape:White PowderMolecular weight:307.772Indacaterol
CAS:Indacaterol (Onbrez; Arcapta) is a β2-Adrenergic Agonist. The mechanism of action of indacaterol is as an Adrenergic beta2-Agonist.Formula:C24H28N2O3Purity:100.00% - 99.63%Color and Shape:SolidMolecular weight:392.49Dexmedetomidine
CAS:Dexmedetomidine: a central alpha-2 adrenergic agonist for general anesthesia.Formula:C13H16N2Purity:100% - 99.74%Color and Shape:SolidMolecular weight:200.28Fluparoxan hydrochloride
CAS:Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmentalFormula:C10H11ClFNO2Purity:99.44%Color and Shape:SoildMolecular weight:231.65Synephrine
CAS:Synephrine (Oxedrine) is sympathetic alpha-adrenergic agonist used as a vasoconstrictor in circulatory failure, asthma, nasal congestion, and glaucoma.Formula:C9H13NO2Purity:100% - 99.63%Color and Shape:SolidMolecular weight:167.21AR-08
CAS:AR-08 is a potent α2-adrenergic receptor agonist for the study of ADHD and attention deficit.Formula:C12H12N6Purity:99.7%Color and Shape:SolidMolecular weight:240.26Rauwolscine hydrochloride
CAS:Rauwolscine HCl, a natural α2-adrenergic antagonist (Ki: 12 nM) & weak 5-HT1A agonist, also blocks 5-HT2B (Ki: 14.3 nM), affects mood/behavior.Formula:C21H27ClN2O3Purity:100% - 99.95%Color and Shape:White SolidMolecular weight:390.9Upidosin
CAS:Upidosin (SB-216469), a uroselective α1 blocker: Ki α1a=0.34 nM, α1b=3.9 nM, α1d=1.5 nM, α2=33.3 nM.Formula:C31H33N3O4Purity:99.26%Color and Shape:SolidMolecular weight:511.61Picumeterol
CAS:Picumeterol(GR 114297A) is a potent and selective β2 adrenergic receptor agonist. In vitro and in vivo trials, Picumeterol produced long-lasting airway smooth muscle relaxation. Picumeterol is a pure R enantiomer that can be used to improve lung function and reduce airway hyperreactivity in patients with asthma.Formula:C21H29Cl2N3O2Purity:98%Color and Shape:SolidMolecular weight:426.38Prazosin
CAS:Prazosin (Prazosine), an α1-blocker, acts as an inverse agonist at alpha-1 adrenergic receptors and is used to treat hypertension.Formula:C19H21N5O4Purity:99.86%Color and Shape:White To Tan Powder SolidMolecular weight:383.4Taprizosin
CAS:Taprizosin(UK-338003) is a selective and orally active α1-adrenoceptor antagonist for vasodilatation in the treatment of benign prostatic hyperplasia.Formula:C25H26N6O4SPurity:97.01% - 99.11%Color and Shape:SolidMolecular weight:506.58Mapenterol hydrochloride
CAS:Mapenterol hydrochloride is an agonist of β2-adrenergic receptor.Formula:C14H21Cl2F3N2OPurity:99.31% - 99.96%Color and Shape:SolidMolecular weight:361.23Ref: TM-T40622
1mg52.00€5mg107.00€10mg158.00€25mg263.00€50mg378.00€100mg548.00€500mg1,093.00€1mL*10mM (DMSO)113.00€Midaglizole hydrochloride
CAS:Midaglizole hydrochloride (DG5128) is an α2-adrenoceptor antagonist with 7.4x more affinity than α1-adrenoceptors (pKi=6.28).Formula:C16H19Cl2N3Purity:100% - 98.73%Color and Shape:SolidMolecular weight:324.25Ref: TM-T11015
1mg57.00€5mg126.00€10mg198.00€25mg324.00€50mg439.00€100mg562.00€200mg743.00€1mL*10mM (DMSO)160.00€Olodaterol
CAS:Olodaterol is a novel, long-acting beta2-adrenergic agonist (LABA) that exerts its pharmacological effect by binding and activating beta2-adrenergic receptorsFormula:C21H26N2O5Purity:98.9%Color and Shape:SolidMolecular weight:386.45GUANABENZ
CAS:GUANABENZ is a Central alpha-2 Adrenergic Agonist. The mechanism of action of guanabenz is as an Adrenergic alpha2-Agonist.Formula:C8H8Cl2N4Purity:98.31%Color and Shape:White Solid From Acetonitrile SolidMolecular weight:231.08Ref: TM-T5471
2mg35.00€5mg48.00€10mg65.00€25mg104.00€50mg148.00€100mg215.00€200mg319.00€1mL*10mM (DMSO)50.00€Pardoprunox
CAS:Pardoprunox (SLV-308) is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties.Formula:C12H15N3O2Purity:98%Color and Shape:SolidMolecular weight:233.27L755507
CAS:L755507 is an effective, selective agonist of β3-AR(IC50=35 nM).Formula:C30H40N4O6SPurity:99% - 99.88%Color and Shape:SolidMolecular weight:584.73Nefazodone hydrochloride
CAS:Nefazodone hydrochloride (Serzone) is a serotoninergic modulating antidepressant that is used in therapy of depression, aggressive behavior and panic disorder.Formula:C25H33Cl2N5O2Purity:99% - 99.86%Color and Shape:White SolidMolecular weight:506.47Ref: TM-T3275
5mg47.00€10mg70.00€25mg120.00€50mg216.00€100mg325.00€200mg472.00€500mg775.00€1mL*10mM (DMSO)77.00€Piperoxan hydrochloride
CAS:Piperoxan hydrochloride (Benodaine hydrochloride) is an α2 adrenoceptor antagonist.Formula:C14H20ClNO2Purity:99.61%Color and Shape:SolidMolecular weight:269.77Ref: TM-T4526
2mg42.00€5mg65.00€10mg96.00€25mg135.00€50mg170.00€100mg212.00€200mg315.00€1mL*10mM (DMSO)58.00€Pamatolol
CAS:Pamatolol is a selective and potent beta-adrenoceptor antagonist that has not shown sympathomimetic activity in ex vivo experiments.Formula:C16H26N2O4Purity:100%Color and Shape:SolidMolecular weight:310.39Naphazoline
CAS:Naphazoline (Naphcon-a) is a sympathomimetic compound with marked alpha adrenergic activity.Formula:C14H14N2Purity:99.25%Color and Shape:White Crystalline Powder SolidMolecular weight:210.27
