CaMK
Calcium/Calmodulin-Dependent Protein Kinase (CaMK) inhibitors are compounds that block the activity of CaMK, a kinase involved in regulating various cellular processes, including synaptic plasticity, memory formation, and gene expression in the nervous system. CaMK plays a critical role in translating calcium signals into cellular responses, and its dysregulation is associated with neurological disorders. Inhibitors of CaMK are valuable tools for studying synaptic signaling, learning, and memory. At CymitQuimica, we offer CaMK inhibitors to support your research in synaptic plasticity, cognitive function, and neuropharmacology.
Products of "CaMK"
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Perphenazine
CAS:Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.Formula:C21H26ClN3OSPurity:99.3% - 99.72%Color and Shape:SolidMolecular weight:403.97Rottlerin
CAS:Rottlerin (NSC-56346), a Mallotus Philippinensis extract, inhibits PKC (3-100 μM IC50); triggers apoptosis by activating caspase 3.Formula:C30H28O8Purity:97.41% - 99.44%Color and Shape:Orange To Brown PowderMolecular weight:516.54Praeruptorin A
CAS:Praeruptorin A ((+)-Praeruptorin A) has the potential to inhibit migration/fusion of preosteoclasts in vitro and bone erosion in vivo by targeting calmodulinFormula:C21H22O7Purity:99.63% - 99.65%Color and Shape:SolidMolecular weight:386.4KN-93
CAS:KN-93 is a selective inhibitor of Ca2+/calmodulin-dependent kinase II (CaMKII), competitively blocking CaM binding to the kinase.Formula:C26H29ClN2O4SPurity:99.78% - 99.86%Color and Shape:White SolidMolecular weight:501.04Ref: TM-T2697
1mg57.00€2mg79.00€5mg113.00€10mg155.00€25mg305.00€50mg378.00€100mg552.00€1mL*10mM (DMSO)127.00€CaMKIIα-PHOTAC
CaMKIIα-PHOTAC is a photochemically targeted chimera (PHOTAC) that specifically targets Ca2+/calmodulin-dependent protein kinase II α (CaMKIIα).Formula:C54H58Cl2N10O11Purity:98%Color and Shape:SolidMolecular weight:1094Autocamtide-2-related inhibitory peptide, myristoylated acetate(201422-04-0 free base)
Myristoylated autocamtide-2-related inhibitory peptide acetate is a cell-permeable CaM kinase II inhibitor.Formula:C80H146N22O22Purity:97.03%Color and Shape:SolidMolecular weight:1768.15CALP1 acetate
CALP1 acetate is a calmodulin (CaM) agonist (Kd of 88 µM) that binds to the CaM EF-hand/Ca2+-binding site.Formula:C42H79N9O12Purity:99.63%Color and Shape:SolidMolecular weight:902.13Rimacalib
CAS:Rimacalib is an inhibitor of Ca2+/calmodulin-dependent protein kinase II (IC50s: ~1 μM for CaMKIIα and ~30 μM for CaMKIIγ).Formula:C22H23FN4O2Purity:98%Color and Shape:SolidMolecular weight:394.44Psoralenoside
CAS:Psoralenoside: a compound from Psoralea fruit; has estrogenic, osteoblastic, antitumor, and antibacterial properties.Formula:C17H18O9Purity:99.03% - 99.49%Color and Shape:SolidMolecular weight:366.32Ref: TM-TN1008
1mg119.00€5mg283.00€10mg418.00€25mg687.00€50mg938.00€100mg1,264.00€1mL*10mM (DMSO)319.00€Tanshinone IIA sulfonate sodium
CAS:Tanshinone IIA sulfonate sodium, a water-soluble derivative from Salvia miltiorrhiza, modulates P2X7 receptors and inhibits hypoxia effects on rat arteries.Formula:C19H17O6S·NaPurity:97.95% - 99.04%Color and Shape:SolidMolecular weight:396.39Trifluoperazine
CAS:Trifluoperazine (trifluoroperazine) is a Dopamine D2 receptor inhibitor(IC50 : 1.2 nM), and Treatment of schizophrenia.Formula:C21H24F3N3SPurity:98.3% - 99.46%Color and Shape:White To Yellowish Crystalline PowderMolecular weight:407.5CAMKIV Protein, Human, Recombinant (GST)
CAMKIV Protein, Human, Recombinant (GST) is expressed in Baculovirus insect cells with GST tag.Color and Shape:Lyophilized PowderMolecular weight:79 kDa (predicted); 100 kDa (reducing conditions)Elziverine
CAS:Elziverine: oral calmodulin antagonist, inhibits Ca-induced acanthocyte formation, potential for neurological and cognitive disorder treatment.Formula:C32H37N3O5Purity:98.43%Color and Shape:SolidMolecular weight:543.65W-7 hydrochloride
CAS:W-7 hydrochloride (W-7 HCl), a calmodulin antagonist, inhibits Ca2+-calmodulin-dependent myosin light chain kinase and phosphodiesterase, W-7 hydrochlorideFormula:C16H22Cl2N2O2SPurity:99.63%Color and Shape:White Crystalline SolidMolecular weight:377.32STO-609
CAS:STO-609 inhibits CaM-KKα/KKβ (Ki: 80/15 ng/mL), is specific, cell-permeable, and targets Ca2+/calmodulin-dependent protein kinase kinase.Formula:C19H10N2O3Purity:97.14% - 98.95%Color and Shape:SolidMolecular weight:314.29Ref: TM-T3546
1mg42.00€5mg88.00€10mg127.00€25mg264.00€50mg423.00€100mg655.00€500mg1,359.00€1mL*10mM (DMSO)113.00€KN-92 hydrochloride
CAS:KN-92 hydrochloride is an inactive derivative of KN-93.Formula:C24H26Cl2N2O3SPurity:99.68%Color and Shape:SolidMolecular weight:493.45A-7 hydrochloride
CAS:A-7 hydrochloride is a calmodulin antagonist and causes alterations in the subpopulation of CD44+CD24- in MDA-MB-231 cells.Formula:C20H30Cl2N2O2SPurity:99.54%Color and Shape:SolidMolecular weight:433.44W-9 hydrochloride
CAS:W-9 hydrochloride is a calmodulin antagonist.Formula:C16H22Cl2N2O2SPurity:98.9%Color and Shape:SolidMolecular weight:377.33Ref: TM-T23525
1mg35.00€2mg44.00€5mg64.00€10mg96.00€25mg183.00€50mg284.00€100mg411.00€500mgTo inquire1mL*10mM (DMSO)70.00€Syntide 2 acetate(108334-68-5 free base)
Syntide-2 acetate is a synthetic peptide recognized as a substrate by Ca2+/calmodulin-dependent protein kinase II (CaMKII; Km = 12 μM).Formula:C70H126N20O20Purity:99.74%Color and Shape:SolidMolecular weight:1567.85FO-4-15
CAS:FO-4-15 is an activator of mGluR1/CaMKIIα. It exhibits protective effects against H2O2 in human neuroblastoma (SH-SY5Y) cells. In mice with Alzheimer's disease, FO-4-15 enhances cognitive function by activating the mGluR1/CaMKIIα pathway, reducing Aβ accumulation, Tau hyperphosphorylation, and synaptic damage.Formula:C18H20N4O4SColor and Shape:SolidMolecular weight:388.44
