
Proteases/Proteasome
Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.
Subcategories of "Proteases/Proteasome"
- Acetyl-CoA Carboxylase
- Cysteine Protease
- DPP-4
- Glutaminase
- HCV Protease
- HIV Protease
- p97
- PAI-1
- Protease-activated Receptor
- Protease Inhibitors
- Proteasome
- Serine Protease
Show 4 more subcategories
Products of "Proteases/Proteasome"
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Arg-Val-(Nle-p-nitro)-Phe-Glu-Ala-Nle-NH2
CAS:Arg-Val-(Nle-p-nitro)-Phe-Glu-Ala-Nle-NH2 is a fluorogenic substrate for the HIV-1 protease, facilitating the assessment of enzyme activity [1].Formula:C40H66N12O11Purity:98%Color and Shape:SolidMolecular weight:891.03Hinokiflavone
CAS:Hinokiflavone, a novel modulator of pre-mRNA splicing activity both in vitro and in cellulo, inhibits the assembly of the spliceosome, particularly blocking theFormula:C30H18O10Purity:97.6% - 98.67%Color and Shape:SolidMolecular weight:538.46TTP-8307
CAS:TTP-8307 is an antiviral compound that inhibits the replication of rhinoviruses and enteroviruses and is used in the study of viral infections.Formula:C27H21FN4OPurity:99.14%Color and Shape:SolidMolecular weight:436.48Ref: TM-T13221
1mg105.00€5mg250.00€10mg401.00€25mg780.00€50mg1,169.00€100mg1,890.00€200mg2,547.00€1mL*10mM (DMSO)303.00€YH-306
CAS:YH-306 (TRV055 acetate ) is a modulator of the FAK signaling pathway that acts by suppressing colorectal tumor growth and metastasis.Formula:C19H18N2O2Purity:97.87%Color and Shape:SolidMolecular weight:306.36Platycodin D3
CAS:Platycodin D3 is a NF-κB inhibitor, it could as expectorants in diverse inflammatory pulmonary diseases, it can regulate the production and secretion of airwayFormula:C63H102O33Purity:98.91% - 99.69%Color and Shape:SolidMolecular weight:1387.46Dabigatran etexilate
CAS:Dabigatran etexilate (BIBR 1048) is a thrombin inhibitor, which acts by binding and blocking thrombogenic activity and the prevention of thrombus formation.Formula:C34H41N7O5Purity:98.19% - 99.12%Color and Shape:White PowderMolecular weight:627.73PMSF
CAS:Phenylmethanesulfonyl fluoride (PMSF (Phenylmethylsulfonyl fluoride)) is an enzyme inhibitor that inactivates IRC-50 arvin, subtilisin, and the fatty acidFormula:C7H7FO2SPurity:97.75% - 99.9%Color and Shape:White To Cream SolidMolecular weight:174.194-Butylresorcinol
CAS:4-Butylresorcinol (Butylresorcinol) is a potent inhibitor of tyrosinase(IC50 : 11.27 μM), and is used in cosmetics as a depigmenting agent.Formula:C10H14O2Purity:98.64% - ≥95%Color and Shape:Light Beige Solid PowderMolecular weight:166.22Petesicatib
CAS:Petesicatib is an inhibitor of cathepsin S. Petesicatib used in the research of immune diseases.Formula:C25H23F6N5O4SPurity:≥98%Color and Shape:SolidMolecular weight:603.54Ref: TM-T16474
1mg127.00€5mg305.00€10mg492.00€25mg938.00€50mg1,454.00€100mg1,882.00€1mL*10mM (DMSO)406.00€Mavorixafor trihydrochloride
CAS:Mavorixafor trihydrochloride blocks CXCR4 (IC50: 13 nM) and suppresses T-tropic HIV-1 replication (IC50: 1-9 nM). It's orally active.Formula:C21H30Cl3N5Purity:98.00%Color and Shape:SolidMolecular weight:458.86UK-370106
CAS:UK-370106 is a potent and highly selective inhibitor of MMP-3 with IC50 of 23 nM and MMP-12 with IC50 of 42 nM, and potently inhibits cleavage of [3H]-Formula:C35H44N2O5Purity:98%Color and Shape:SolidMolecular weight:572.73Bellidifolin
CAS:Bellidoferin: anti-oxidant, protects liver, fights inflammation/tumors, aids nerve injury, blocks MAO A, may improve type-2 diabetes, antifungal.Formula:C14H10O6Purity:99.79% - 99.81%Color and Shape:SolidMolecular weight:274.23Ref: TM-T3822
1mg96.00€5mg225.00€10mg323.00€25mg537.00€50mg752.00€100mg1,035.00€1mL*10mM (DMSO)202.00€DS-1040 Tosylate
CAS:DS-1040 Tosylate is a thrombin-activated fibrinolysis inhibitor (TAFI) inhibitor and a fibrinolysis enhancer, used for researching thromboembolic diseases.Formula:C23H35N3O5SColor and Shape:SolidMolecular weight:465.61Talviraline
CAS:Talviraline (Bay 10-8979) is an RNA-induced DNA polymerase inhibitor.Talviraline is a potent inhibitor of HIV-1-induced cell killing and HIV-1 replication in aFormula:C15H20N2O3S2Purity:99.82%Color and Shape:SolidMolecular weight:340.462-Cyanopyrimidine
CAS:2-Cyanopyrimidine (m-Hydroxyphenylpropionic acid) is inhibitor of cathepsin K(IC50 : 170 nM)Formula:C5H3N3Purity:99.27%Color and Shape:Crystalline SolidMolecular weight:105.1CA inhibitor 1
CAS:CA inhibitor 1 (GS-6207 analog) is a potent inhibitor of the HIV capsid.Formula:C41H36ClF8N7O5S2Purity:98%Color and Shape:SolidMolecular weight:958.34PF-3450074
CAS:PF-3450074 (PF-74) is a specific HIV-1 inhibitor, blocking viral replication and uncoating at submicromolar EC50=8-640 nM.Formula:C27H27N3O2Purity:99.92%Color and Shape:SolidMolecular weight:425.52Aderbasib
CAS:Aderbasib (INCB007839) is an ADAM10 and ADAM17 inhibitor with antitumor activity, used in cancer and cardiovascular disease research.Formula:C21H28N4O5Color and Shape:SolidMolecular weight:416.47Cystamine
CAS:Cystamine (2,2'-Disulfanediyldiethanamine) is an inhibitor of transglutaminase and inhibits caspase-3 with an IC50 value of 23.6 μM.Formula:C4H12N2S2Purity:99.41%Color and Shape:SolidMolecular weight:152.28Ceritinib
CAS:Ceritinib (LDK378) is an ALK inhibitor with selective, ATP-competitive, and oral activity. Ceritinib has antitumor activity. Cost-effective and quality-assured.Formula:C28H36ClN5O3SPurity:100% - 99.77%Color and Shape:SolidMolecular weight:558.14Bacoside A
CAS:Bacoside A shows potential anti-cancer effects, cytoprotection, EAE inhibition, and vasorelaxation abilities.Formula:C41H68O13Purity:98%Color and Shape:SolidMolecular weight:768.98E-64d [for Biochemical Research]
CAS:Formula:C17H30N2O5Purity:>95.0%(HPLC)Color and Shape:White to Almost white powder to crystalMolecular weight:342.44GS-9256
CAS:GS-9256 is a selective inhibitor of the HCV NS3 protease, exhibiting favorable pharmacokinetic properties and antiviral activity [1].Formula:C46H56ClF2N6O8PSPurity:98%Color and Shape:SolidMolecular weight:957.46Levovirin
CAS:Levovirin (L-Ribavirin) is a guanosine nucleoside analog that has immunomodulatory activity and is used in the study of hepatitis C virus infection.Formula:C8H12N4O5Purity:100% - 99.96%Color and Shape:SolidMolecular weight:244.203-Deazaadenosine hydrochloride
CAS:3-Deazaadenosine HCl blocks SAH hydrolase (Ki: 3.9 μM), with anti-inflammatory, anti-proliferative, and anti-HIV effects.Formula:C11H15ClN4O4Purity:98.48%Color and Shape:SolidMolecular weight:302.71Ref: TM-T10111
1mg126.00€5mg216.00€10mg374.00€25mg620.00€50mg868.00€100mg1,169.00€1mL*10mM (DMSO)149.00€Maraviroc
CAS:Maraviroc: a CCR5 antagonist blocking HIV-1 entry; IC50s-MIP-1α: 3.3nM, MIP-1β: 7.2nM, RANTES: 5.2nM.Formula:C29H41F2N5OPurity:100% - 99.55%Color and Shape:Brown SolidMolecular weight:513.67Ref: TM-T6016
5mg51.00€10mg95.00€25mg160.00€50mg273.00€100mg492.00€200mg633.00€500mg998.00€1mL*10mM (DMSO)59.00€Epitheaflagallin 3-O-gallate
CAS:Epitheaflagallin 3-O-gallate: potential antiobesity, antiperiodontal agent; inhibits tumor growth by blocking angiogenesis.Formula:C27H20O13Purity:98%Color and Shape:SolidMolecular weight:552.44Aloesin
CAS:Aloesin, a C-glycosylated chromone from aloe, blocks tyrosinase (IC50=0.9mM) in melanin production.Formula:C19H22O9Purity:98% - 99.58%Color and Shape:SolidMolecular weight:394.37Collagenase Type V
Collagenase Type V, an endopeptidic matrix metalloproteinase MMP from the bacterium Clostridium histolyticum, can be used for islet tissue isolation.Color and Shape:Odour SolidTrichosanatine
CAS:Trichosanatine and squamosamide, as potential candidates as lead compounds for further study in drug development process with the PP2A- α protein.Formula:C27H28N2O4Purity:98%Color and Shape:SolidMolecular weight:444.52Saikosaponin B2
CAS:Saikosaponin B2 inhibits HCV, blocks viral binding to hepatoma cells, and induces melanoma differentiation, enhancing tyrosinase and melanogenesis.Formula:C42H68O13Purity:99.59% - 99.88%Color and Shape:SolidMolecular weight:780.98Z-Gly-Pro-Arg-4MβNA
CAS:Z-Gly-Pro-Arg-4MβNA is a thrombin substrate that, upon cleavage by thrombin, releases 4-methoxy-2-naphthylamine (4MβNA).Formula:C32H39N7O6Purity:98%Color and Shape:SolidMolecular weight:617.7Artemisinin
CAS:Artemisinin (Qinghaosu) is a natural sesquiterpene lactone. Artemisinin has anti-malarial, neuroprotective and anti-tumor effects. Cost-effective and quality-assured.Formula:C15H22O5Purity:100% - 99.87%Color and Shape:Crystalline SolidMolecular weight:282.33HIV-1 inhibitor-53
CAS:HIV-1 Inhibitor-53 targets HIV-1 protease (IC50: 1.93 nM) and reverse transcriptase (IC50: 2.35 μM), aiding AIDS research.Formula:C30H34N2O8SPurity:98%Color and Shape:SolidMolecular weight:582.66Nevirapine
CAS:Nevirapine (NVP) is a benzodiazepine non-nucleoside reverse transcriptase inhibitor.Formula:C15H14N4OPurity:99.58% - 99.59%Color and Shape:White Or Off-White Crystalline PowderMolecular weight:266.3Bestatin Hydrochloride
CAS:Formula:C16H25ClN2O4Purity:98%Color and Shape:SolidMolecular weight:344.8337CCR5 antagonist 1
CAS:CCR5 antagonist 1 is a CCR5 antagonist extracted from WO 2004054974 A2. It can inhibit HIV replication.Formula:C39H46ClF2N5O3SPurity:98%Color and Shape:SolidMolecular weight:738.33Z-Pro-Pro-CHO
CAS:Z-Pro-Pro-CHO acts as a prolyl oligopeptidase inhibitor with half-maximal inhibitory concentrations (IC50) of 0.16 μM for human prolyl oligopeptidase and 0.01Formula:C18H22N2O4Purity:98%Color and Shape:SolidMolecular weight:330.38Efegatran sulfate
CAS:Efegatran sulfate (LY294468 sulfate) is a potent thrombin inhibitor used in the treatment of thrombotic disorders.Formula:C21H34N6O7SPurity:≥98% - ≥98%Color and Shape:SolidMolecular weight:514.6CM-352
CAS:CM-352 is a metalloproteinase inhibitor that reduces brain damage and improves functional recovery in rat models of cerebral hemorrhage.Formula:C24H29N3O6SPurity:99.36%Color and Shape:SolidMolecular weight:487.57Dabigatran Etexilate Mesylate
CAS:Dabigatran Etexilate Mesylate (BIBR 1048MS) is the orally active prodrug of dabigatran. Dabigatran is a reversible and selective, direct thrombin inhibitor.Formula:C34H41N7O5·CH4O3SPurity:99.91%Color and Shape:SolidMolecular weight:723.84Ref: TM-T5133
5mg42.00€10mg57.00€25mg74.00€50mg95.00€100mg111.00€200mg169.00€500mg240.00€1mL*10mM (DMSO)64.00€NM107
CAS:NM107, a ribonucleoside, inhibits HCV NS5B polymerase. It has broad antiviral properties with EC50 of 1.85 μM in wild-type cells.Formula:C10H15N3O5Purity:98%Color and Shape:White To Off-White PowderMolecular weight:257.24MRS1177
CAS:MRS1177 is an effective and selective antagonist of the human Adenosine A3 receptor (hA3AR) (Ki: 0.3 nM).Formula:C20H12ClN5O2Purity:98%Color and Shape:SolidMolecular weight:389.79Methyl rosmarinate
CAS:Methyl rosmarinate, from Rabdosia serra, inhibits tyrosinase (IC50: 0.28 mM), α-glucosidase, MMP-1, and has antioxidant, antifungal properties.Formula:C19H18O8Purity:97.52% - 99.62%Color and Shape:SolidMolecular weight:374.34Ref: TM-TN1928
1mg74.00€5mg165.00€10mg259.00€25mg435.00€50mg630.00€100mg880.00€1mL*10mM (DMSO)173.00€GLS1 Inhibitor-4
CAS:GLS1 Inhibitor-4 (41e) has 11.86 nM IC50, strong binding, disrupts glutamine metabolism, induces apoptosis, and shows antitumor effects.Formula:C29H27F3N10O2S2Purity:98%Color and Shape:SolidMolecular weight:668.72Collagenase Type IV
Collagenase Type IV is an MMP-18 primarily degrades collagen type IV and VII and basement membranes (e.g., neural tissue, renal tissue) mild activity.Color and Shape:Odour SolidMirificin
CAS:Mirificin (BCP10902) is an active ingredient in Tongmai formula (TMF) which is a well-known Chinese medicinal preparation. Anti-oxidant.Formula:C26H28O13Purity:99.33% - 99.8%Color and Shape:SolidMolecular weight:548.49Ubenimex
CAS:Formula:C16H24N2O4Purity:>98.0%(HPLC)Color and Shape:White to Almost white powder to crystalMolecular weight:308.38Eltrombopag
CAS:Eltrombopag (SB-497115-GR), an orally active thrombopoietin receptor agonist with megakaryopoiesis stimulating activity, binds to and stimulates the plateletFormula:C25H22N4O4Purity:99.27%Color and Shape:Orange To Red SolidMolecular weight:442.471,10-Phenanthroline Monohydrate [for Biochemical Research]
CAS:Formula:C12H8N2·H2OPurity:>99.0%(T)Color and Shape:White powder to crystalMolecular weight:198.23HIV-1 integrase inhibitor 8
CAS:HIV-1 integrase inhibitor 8 is an inhibitor of HIV-1 integrase. Integration is a required step in HIV replication [1].Formula:C21H24O2Purity:98.01%Color and Shape:SolidMolecular weight:308.41Monobenzone
CAS:Monobenzone (Benoquin) is a Depigmenting Agent.Formula:C13H12O2Purity:99.87%Color and Shape:Lustrous Leaflets From Water SolidMolecular weight:200.23Aclacinomycin A hydrochloride
CAS:Aclacinomycin A (Aclarubicin) hydrochloride is a fluorescent molecule and the first described non-peptidic inhibitor showing discrete specificity for the CTRL (Formula:C42H54ClNO15Purity:98%Color and Shape:SolidMolecular weight:848.33Ref: TM-T10238
5mgTo inquire10mgTo inquire25mgTo inquire50mgTo inquire100mgTo inquire200mgTo inquire1mL*10mM (DMSO)To inquireVCH-916 free acid(1200133-34-1 free base)
CAS:VCH-916 is a novel nonnucleoside HCV NS5B polymerase inhibitor.Formula:C26H37NO4SPurity:98.45%Color and Shape:SolidMolecular weight:459.64Ref: TM-TQ0122L
1mg74.00€2mg97.00€5mg140.00€10mg188.00€25mg339.00€50mg552.00€100mg792.00€1mL*10mM (DMSO)150.00€BI-1230
CAS:BI-1230 is a potent inhibitor of HCV NS3 protease, exhibiting efficacy in the low nanomolar range, and notably suppresses viral replication.Formula:C42H52N6O9SPurity:98%Color and Shape:SolidMolecular weight:816.96TGase2-IN-1
CAS:TGase2-IN-1 (Compound 22) is an orally effective TGase2 inhibitor with an IC50 of 1.12 µM. It inhibits TGase2 in human retinal microvascular endothelial cells with a strikingly lower IC50 of 0.07 µM. The oral bioavailability of TGase2-IN-1 is 74.6%. Additionally, it can suppress retinal vascular leakage in a mouse model of diabetes induced by Streptozotocin.Formula:C23H25N3O3Color and Shape:SolidMolecular weight:391.46Cathepsin Inhibitor 2
CAS:Cathepsin Inhibitor 2 is a potent Cathepsin S inhibitor (Ki: <20 nM).Formula:C19H21F6N3OPurity:98%Color and Shape:SolidMolecular weight:421.38Temocapil
CAS:Temocapril is an inhibitor of tyrosine kinase.Formula:C23H28N2O5S2Purity:97.8%Color and Shape:White PowderMolecular weight:476.61IK-862
CAS:IK-862 is a selective TACE inhibitor with potential anti-inflammatory and anticancer activity for the study of neuritis.Formula:C25H27N3O4Purity:98.72% - 99.39%Color and Shape:SolidMolecular weight:433.5MK-0608
CAS:MK-0608 is an orally bioavailable HCV replication inhibitor in vitro(EC50 = 0.3 μM and EC90=1.3 μM in the subgenomic-replicon assay).Formula:C12H16N4O4Purity:98.48%Color and Shape:SolidMolecular weight:280.28Ref: TM-T16088
1mg81.00€2mg96.00€5mg170.00€10mg274.00€25mg525.00€50mg753.00€100mg1,035.00€1mL*10mM (DMSO)183.00€Excisanin A
CAS:ExcisaninA may be a potent inhibitor of AKT signaling pathway in tumor cells, it can inhibit invasion by suppressing MMP-2 and MMP-9 expression, it may be aFormula:C20H30O5Purity:98%Color and Shape:SolidMolecular weight:350.45S 3304
CAS:S 3304 is a novel matrix metalloproteinases inhibitor which is specific for MMP-2 and MMP-9.Formula:C24H20N2O4S2Purity:98.09%Color and Shape:SolidMolecular weight:464.56Ref: TM-T16966
1mg58.00€5mg160.00€10mg259.00€25mg429.00€50mg605.00€100mg815.00€200mg1,093.00€1mL*10mM (DMSO)163.00€Reverse transcriptase-IN-1
CAS:Reverse transcriptase-IN-1 is a diarylbenzopyrimidine (DABP) analogue and a potent inhibitor of HIV-1 nonnucleoside reverse transcriptase with an IC50of 13.7Formula:C25H17N7O2Purity:99.14%Color and Shape:SolidMolecular weight:447.45Ref: TM-T12715
1mg64.00€5mg131.00€10mg183.00€25mg311.00€50mg449.00€100mg615.00€200mg833.00€1mL*10mM (DMSO)143.00€MMP-9-IN-1
CAS:MMP-9-IN-1 is an inhibitor of specific matrix metalloproteinase-9 (MMP-9).Formula:C16H17F2N3O3SPurity:99.21%Color and Shape:SolidMolecular weight:369.39Ref: TM-T8310
1mg96.00€2mg139.00€5mg227.00€10mg359.00€25mg607.00€50mg847.00€100mg1,169.00€1mL*10mM (DMSO)221.00€ZM223 hydrochloride (2031177-48-5 free base)
ZM223 hydrochloride is an orally active, potent non-covalent inhibitor of NEDD8 activating enzyme (NAE), and with excellent anticancer activity.Formula:C23H18ClF3N4O2S2Purity:98%Color and Shape:SolidMolecular weight:538.99Teneligliptin
CAS:Teneligliptin (MP-513), potent DPP-4 inhibitor, IC50 ~1 nM, blocks DPP-4 in human/rat plasma and recombinant forms.Formula:C22H30N6OSPurity:99.73%Color and Shape:SolidMolecular weight:426.58Ref: TM-T37522
1mgTo inquire5mg35.00€10mg52.00€25mg74.00€50mg97.00€100mg173.00€200mgTo inquire1mL*10mM (DMSO)50.00€Incyclinide
CAS:Incyclinide (COL-3) is a matrix metalloproteinase (MMP) inhibitor.Formula:C19H17NO7Purity:97.99%Color and Shape:SolidMolecular weight:371.34Tyrosinase-IN-36
Tyrosinase-IN-36 is a moderately potent inhibitor of tyrosine, exhibiting an inhibition percentage of 42.75% compared to kojic acid at a concentration of 100 μM and possesses antioxidant activity.Color and Shape:Odour SolidDabigatran ethyl ester
CAS:Dabigatran ethyl ester (Dabigatran (ethyl ester)) is an emerging oral anticoagulant and it also is a direct inhibitor of thrombin activity.Formula:C27H29N7O3Purity:97.63%Color and Shape:SolidMolecular weight:499.56Diprotin A
CAS:Diprotin A (Ile-Pro-Ile) (Ile-Pro-Ile) is a dipeptidyl peptidase IV (DPP-IV) inhibitor.Formula:C17H31N3O4Purity:99.29%Color and Shape:White PowderMolecular weight:341.45Ginkgolide C
CAS:Ginkgolide C (BN-52022), a natural product, can enhance the cardiac function of rats in the body.Formula:C20H24O11Purity:99.71% - 99.98%Color and Shape:White PowderMolecular weight:440.4Phepropeptin B
CAS:Phepropeptin B is a secondary metabolite derived from microorganisms, functioning as a proteasome (proteasome) inhibitor with an IC50 value of 11 μg/mL.Formula:C40H56N6O6Color and Shape:SolidMolecular weight:716.91Eltrombopag Olamine
CAS:Eltrombopag Olamine (Eltrombopag diethanolamine salt) is the orally active ethanolamine salt of eltrombopag, a small-molecule, nonpeptide thrombopoietinFormula:C29H36N6O6Purity:99.59% - 99.89%Color and Shape:SolidMolecular weight:564.63Ref: TM-T6825
2mg43.00€5mg64.00€10mg90.00€25mg140.00€50mg177.00€100mg230.00€200mg340.00€500mg563.00€1mL*10mM (DMSO)90.00€MUN57694
CAS:MUN57694 is an inhibitor of 26S proteasome.Formula:C23H25N3O4Purity:99%Color and Shape:SolidMolecular weight:407.46Ref: TM-T9090
1mg40.00€5mg80.00€10mg116.00€25mg212.00€50mg316.00€100mg447.00€200mg627.00€1mL*10mM (DMSO)96.00€Obefazimod
CAS:Obefazimod (ABX-464) is a potent anti-HIV agent. ABX464 inhibits HIV-1 replication in stimulated peripheral blood mononuclear cells (PBMCs).Formula:C16H10ClF3N2OPurity:99.86%Color and Shape:SolidMolecular weight:338.71Ref: TM-T8311
2mg39.00€5mg62.00€10mg87.00€25mg187.00€50mg301.00€100mg437.00€200mg617.00€1mL*10mM (DMSO)65.00€Trovirdine
CAS:Trovirdine (LY300046) is a thiourea non-nucleoside reverse transcriptase inhibitor.Formula:C13H13BrN4SPurity:98.12% - 98.50%Color and Shape:SolidMolecular weight:337.24HZ-1157
CAS:HZ-1157 (DHFR-inhibitor) is a hepatitis C virus (HCV) inhibitor with inhibitory activities toward HCV NS3/4A protease.Formula:C12H16N4OPurity:98.23%Color and Shape:SolidMolecular weight:232.28UPGL00004
CAS:UPGL00004: potent GAC inhibitor, IC50=29 nM, Kd=27 nM, suppresses triple-negative breast cancer cell growth.Formula:C25H26N8O2S2Purity:97.44%Color and Shape:SolidMolecular weight:534.66Ginsenoside F4
CAS:Ginsenoside F4 induces apoptosis in JK cells by causing mitochondrial dysfunction and altering Bax and Bcl-2 levels.Formula:C42H70O12Purity:98%Color and Shape:SolidMolecular weight:767.01Feniralstat
CAS:Feniralstat (KVD-824) is a selective and potent kallikrein (kallikrein) inhibitor, useful in immune system diseases and cardiovascular disease research.Formula:C26H25F2N5O4Purity:99.52%Color and Shape:SolidMolecular weight:509.51JG26
CAS:JG26 is a potent inhibitor of ADAM17, which can inhibit ADAM8, ADAM17, ADAM10 and MMP-12, with IC50 values of 12 nM, 1.9 nM, 150 nM and 9.4 nM, respectively,Formula:C19H22Br2N4O6SPurity:100.00% - 98.92%Color and Shape:SolidMolecular weight:594.27MMP2-IN-3
CAS:MMP2-IN-3 is a potent inhibitor of matrix metalloproteinases (MMP-2) (IC50: 31 μM).Formula:C23H21N3OPurity:99.13%Color and Shape:SolidMolecular weight:355.43Ref: TM-T61271
1mg87.00€5mg192.00€10mg293.00€25mg477.00€50mg662.00€100mg889.00€200mg1,198.00€1mL*10mM (DMSO)205.00€Immunoproteasome activator 1
CAS:Immunoproteasome Activator 1 (compound A) is a selective immunoproteasome activator that enhances the presentation of individual MHC-I binding peptides by over 100 times. It binds to the proteasomal structural subunit PSMA1 and facilitates the association of the proteasome activators PA28α/β (PSME1/PSME2) with the immunoproteasome.Formula:C24H23N3O3Color and Shape:SolidMolecular weight:401.46Ledipasvir
CAS:Ledipasvir (GS-5885) is a Hepatitis C Virus NS5A Inhibitor.Formula:C49H54F2N8O6Purity:99.46%Color and Shape:SolidMolecular weight:889Ref: TM-T6200
1mg38.00€2mg49.00€5mg79.00€10mg88.00€25mg159.00€50mg256.00€100mg444.00€500mg1,017.00€1mL*10mM (DMSO)88.00€FK706
CAS:FK706, a human neutrophil elastase inhibitor (IC50: 83 nM, Ki: 4.2 nM), also blocks mouse and porcine elastases. Anti-inflammatory.Formula:C26H33F3N4NaO7Color and Shape:SolidMolecular weight:593.556CPA inhibitor
CAS:CPA inhibitor (Carboxypeptidase inhibitor) is a potent carboxypeptidase A (CPA) inhibitor with a Ki of 0.32 μM.Formula:C18H19NO4Purity:100%Color and Shape:SolidMolecular weight:313.35Ref: TM-T10876
1mg57.00€5mg125.00€10mg163.00€25mg278.00€50mg405.00€100mgTo inquire1mL*10mM (DMSO)138.00€Y-29794 Tosylate
CAS:Y-29794 Tosylate (Y-29794) is an orally active, effective, and specific non-peptide-prolyl endopeptidase (PPCE) inhibitor.Formula:C30H42N2O4S3Purity:99.10%Color and Shape:SolidMolecular weight:590.86Ref: TM-T35233
1mg52.00€2mg74.00€5mg96.00€10mg137.00€25mg217.00€50mg391.00€100mg582.00€500mg1,254.00€1mL*10mM (DMSO)159.00€Benzoic acid, 4-[[6-[(aminoiminomethyl)amino]-1-oxohexyl]oxy]-, ethylester, monomethanesulfonate
CAS:Formula:C17H27N3O7SPurity:98%Color and Shape:SolidMolecular weight:417.4772Gly-Pro-pNA hydrochloride
CAS:Gly-Pro-pNA hydrochloride (Gly-Pro p-nitroanilide hydrochloride) is a dipeptidyl peptidase inhibitor that inhibits dipeptidyl peptidase II, dipeptidyl peptidaseFormula:C13H17ClN4O4Purity:99.41%Color and Shape:SolidMolecular weight:328.75BRD-6929
CAS:BRD-6929, a brain-targeted HDAC1/2 inhibitor (IC50 1/8 nM), enhances gnidimacrin's anti-HIV effect, useful in mood behavior studies.Formula:C19H17N3O2SPurity:99.05%Color and Shape:SolidMolecular weight:351.42Ref: TM-T10603
5mg50.00€10mg90.00€25mg170.00€50mg305.00€100mg442.00€200mg620.00€1mL*10mM (DMSO)51.00€Abietic Acid
CAS:Abietic Acid (Sylvic acid) is a diterpene extracted from Pimenta racemosavar. Cost-effective and quality-assured.Formula:C20H30O2Purity:90.59% - 92.6%Color and Shape:Physical Description Yellowish Resinous Powder (Ntp 1992)Molecular weight:302.45JNJ-10311795
CAS:JNJ-10311795 (RWJ-355871) is an inhibitor of neutrophil elastase G and mast cell chymase, demonstrating significant anti-inflammatory effects.Formula:C40H35N2O6PPurity:99.19%Color and Shape:SolidMolecular weight:670.69ML281
CAS:ML281 is a potent and selective STK33 inhibitor with IC50 of 14 nM.Formula:C22H19N3O2SPurity:99.12% - 99.77%Color and Shape:SolidMolecular weight:389.47Ref: TM-T3423
1mg35.00€5mg80.00€10mg97.00€25mg188.00€50mg311.00€100mg500.00€500mg1,093.00€1mL*10mM (DMSO)88.00€Methyl 2-amino-5-bromobenzoate
CAS:Methyl 2-amino-5-bromobenzoate (Methyl 5-Bromoanthranilate) is an HCV NS5b RNA polymerase inhibitor with antimicrobial activity.Formula:C8H8BrNO2Purity:98.05%Color and Shape:SolidMolecular weight:230.06L-Homocysteine
CAS:L-Homocysteine is a biological thiol associated with various diseases and conditions. It serves as a marker for atherosclerosis.Formula:C4H9NO2SPurity:99.91%Color and Shape:SolidMolecular weight:135.19Micrococcin P1
CAS:Micrococcin P1 is a macrocyclic peptide antibiotic and is a potent hepatitis C virus (HCV) inhibitor(EC50 range of 0.1-0.5 μM)Formula:C48H49N13O9S6Purity:98%Color and Shape:SolidMolecular weight:1144.36Triolein
CAS:Glyceryl Trioleate has been investigated for the treatment of Adrenoleukodystrophy.Formula:C57H104O6Purity:98.28% - 99.99%Color and Shape:Clear Yellowish LiquidMolecular weight:885.43Paritaprevir free base
CAS:Paritaprevir (ABT-450) is an oral HCV NS3/NS4A protease inhibitor with potential against genotype 1, disrupting viral replication.Formula:C40H43N7O7SPurity:95% - 99.26%Color and Shape:SolidMolecular weight:765.89CGS 27023A
CAS:CGS 27023A is a non-peptidic, potent, and orally active stromelysin inhibitor.Formula:C18H24ClN3O5SPurity:99.08%Color and Shape:SolidMolecular weight:429.92ZD-0892
CAS:ZD-0892: potent, selective neutrophil elastase inhibitor; Ki 6.7 nM (human), 200 nM (porcine).Formula:C24H32F3N3O5Purity:95% - 99.53%Color and Shape:SolidMolecular weight:499.52PR 39 (porcine) acetate
PR 39 (porcine) acetate is a noncompetitive, reversible and allosteric proteasome inhibitor.Purity:98%Color and Shape:LiquidMolecular weight:N/ADolutegravir sodium
CAS:Dolutegravir sodium (GSK-1349572A) salt(DTG; GSK1349572) is an HIV integrase inhibitor(IC50: 2.7 nM), modest activity against raltegravir-resistant signatureFormula:C20H18F2N3NaO5Purity:98% - 99.74%Color and Shape:SolidMolecular weight:441.36EDTA, Disodium Salt, Dihydrate
CAS:EDTA disodium dihydrate chelates metals, inhibits proteases, and aids in protein purification; doesn't affect cellulase.Formula:C10H18N2Na2O10Purity:99.97%Color and Shape:SolidMolecular weight:372.24Beclabuvir
CAS:Beclabuvir blocks HCV NS5B polymerase at thumb site 1, effective on genotypes 1, 3, 4, 5 with IC50 <28 nM.Formula:C36H45N5O5SPurity:99.87% - 99.93%Color and Shape:SolidMolecular weight:659.84Sulochrin
CAS:Sulochrin shows antifungal and antibacterial activities, it can inhibit hepatitis C virus (HCV) infection in a dose-dependent manner without any apparentFormula:C17H16O7Purity:98%Color and Shape:SolidMolecular weight:332.3ISOGINKGETIN
CAS:ISOGINKGETIN (4',4'''-Dimethylamentoflavone), a compound derived from the leaves of Ginkgo biloba, to up-regulate adiponectin secretion.Formula:C32H22O10Purity:98% - 99.72%Color and Shape:SolidMolecular weight:566.51Davelizomib
CAS:Davelizomib is a proteasome inhibitor that exhibits antineoplastic activity [1].Formula:C21H26BF2N3O7Purity:98%Color and Shape:SolidMolecular weight:481.25Notoginsenoside T5
CAS:TPNS from San-Chi root (Araliaceae) treats atherosclerosis by lowering lipids and modifying vascular CD40/MMP-9, suggesting clinical use.Formula:C41H68O12Purity:98%Color and Shape:SolidMolecular weight:752.983Viscumneoside III
CAS:Viscumneoside III, a dihydroflavone O-glycoside, is a potent Tyrosinase inhibitor with an IC50 of 0.5 mM. Viscumneoside III has anti-angina pectoris.Formula:C27H32O15Purity:98%Color and Shape:SolidMolecular weight:596.53Aloin
CAS:Aloin (Aloin-A)(mixture of A&B), a natural anthracycline from Aloe vera, is a tyrosinase inhibitor.Formula:C21H22O9Purity:98.28%Color and Shape:Yellow PowderMolecular weight:418.39Mizoribine
CAS:Mizoribine (NSC-289637) belongs to the family of 1-Ribosyl-imidazolecarboxamides. Mizoribine has been investigated for the treatment of Rheumatoid Arthritis.Formula:C9H13N3O6Purity:98.38% - 99.95%Color and Shape:White To Off-White Crystalline PowderMolecular weight:259.22Isatoribine
CAS:Isatoribine(ANA245) free base is a potent TLR7 receptor agonist with anti-hepatitis C virus infection activity for the study of HCV infection.Formula:C10H12N4O6SPurity:100% - 99.73%Color and Shape:SolidMolecular weight:316.29CIL62
CAS:CIL62 is a caspase-3/7-independent inducer of cell death. The mechanism of action of CIL62 is Necrostatin-1 dependent cell death [1].Formula:C23H26O5Purity:97.07%Color and Shape:SolidMolecular weight:382.45Ref: TM-T8468
1mg52.00€5mg116.00€10mg170.00€25mg335.00€50mg562.00€100mg758.00€200mg1,017.00€1mL*10mM (DMSO)128.00€HIV-1 Inhibitor 18A
CAS:HIV-1 Inhibitor 18A (HIV-1 Inhibitor-18A) specifically inhibits the entry of multiple HIV-1 isolates.Formula:C14H11N5O2SPurity:91.64%Color and Shape:SolidMolecular weight:313.33Ref: TM-T24141
1mg115.00€5mg227.00€10mg313.00€25mg535.00€50mg752.00€100mg1,064.00€1mL*10mM (DMSO)217.00€Sirpiglenastat
CAS:Sirpiglenastat (DRP-104) is a glutamine antagonist, a prodrug of DON, with antitumor activity that acts by suppressing the adaptive immune system.Formula:C22H27N5O5Purity:98.01% - 98.37%Color and Shape:SolidMolecular weight:441.48Atazanavir Sulfate
CAS:Formula:C38H52N6O7·H2SO4Purity:>98.0%(HPLC)Color and Shape:White to Almost white powder to crystalMolecular weight:802.94Melagatran
CAS:Melagatran is an orally available, direct synthetic thrombin inhibitor that does not require endogenous cofactors other than thrombin.Cost-effective and quality-assured.Formula:C22H31N5O4Purity:100% - 98.37%Color and Shape:SolidMolecular weight:429.51Ref: TM-T11994
1mg513.00€5mg1,198.00€10mg1,549.00€25mg2,337.00€50mg3,125.00€100mg4,246.00€1mL*10mM (DMSO)1,130.00€BMS-561392 Formic acid
BMS-561392 Formic acid is a selective inhibitor of TACE and reduces TNFalpha levels.Formula:C28H34N4O6Purity:97.25%Color and Shape:SoildMolecular weight:522.59Ref: TM-T30531L
1mg185.00€5mg424.00€10mg627.00€25mg938.00€50mg1,311.00€100mg1,795.00€500mg3,600.00€1mL*10mM (DMSO)520.00€Pseudane IX
CAS:Pseudane IX (2-nonyl-1H-quinolin-4-one) reduces infection of Huh 7.5 cells by hepatitis C virus (HCV) with an IC50 of 1.4 μg/ml.Formula:C18H25NOPurity:99.71%Color and Shape:SolidMolecular weight:271.4TG2-IN-3h
CAS:TG2-IN-3h is a highly selective, potent, cell-permeable fluorescent irreversible tissue transglutaminase (tg2) inhibitorFormula:C21H26N4O4SPurity:99.34% - 99.76%Color and Shape:SolidMolecular weight:430.52MEGA-9
CAS:MEGA-9 (Nonanoyl-N-Methylglucamide) solubilizes membrane protein and can be used as a nonionic detergent.Formula:C16H33NO6Purity:99.59%Color and Shape:SolidMolecular weight:335.44Emtricitabine S-oxide
CAS:Emtricitabine treats HIV; its degradation byproduct is Emtricitabine S-oxide.Formula:C8H10FN3O4SPurity:98%Color and Shape:SolidMolecular weight:263.25PSI
CAS:PSI is a proteasome inhibitor.Formula:C32H50N4O8Purity:97% - 98.33%Color and Shape:SolidMolecular weight:618.76Methylchloroisothiazolinone/Methylisothiazolinone Mixture
CAS:Methylchloroisothiazolinone/Methylisothiazolinone Mixture (Kathon 886MW),a preservative, activates MMPs in human bronchial epithelial cells.Formula:C8H9ClN2O2S2Color and Shape:SolidMolecular weight:264.75Sovaprevir
CAS:Sovaprevir is a non-structural 3 (NS3) protease inhibitor with antiviral activity for the treatment of HCV infection.Formula:C43H53N5O8SPurity:99.10%Color and Shape:SolidMolecular weight:799.97Ref: TM-T28830
1mg266.00€5mg655.00€10mg934.00€25mg1,388.00€50mg1,872.00€100mg2,517.00€1mL*10mM (DMSO)1,035.00€TS-021
CAS:TS-021 is a selective dipeptidyl peptidase 4 (DPP-4) inhibitor with antidiabetic activity for the study of type 2 diabetes.Formula:C17H24FN3O5SPurity:100% - 100%Color and Shape:SolidMolecular weight:401.45RJF02215
CAS:RJF02215, an MMP-9 inhibitor, exhibits growth inhibitory activity against the ovarian cancer cell line SKOV3. It is utilized in tumor research.Formula:C17H12ClN3OS3Color and Shape:SolidMolecular weight:405.95Salicylanilide
CAS:Salicylanilide (2-Hydroxybenzanilide)s are a group of compounds with antiviral potency, antibacterial and antifungal activities.Formula:C13H11NO2Purity:99.55%Color and Shape:White To Off-White Crystalline PowderMolecular weight:213.23hTYR/AbTYR-IN-1
CAS:hTYR/AbTYR-IN-1 is a dual hTYR/AbTYR inhibitor with inhibitory effects on hTYR and AbTYR, with IC50s of 5.4 μM and 3.52 μM, respectively.Formula:C18H20N2O3Purity:99.59%Color and Shape:SoildMolecular weight:312.36Heparin
CAS:Heparin (Adomiparin) is a mucopolysaccharide sulfate that has shown partial anti-inflammatory activity in in vivo studies.Formula:C26H42N2O37S5Purity:98%Color and Shape:White Or Pale-Colored Amorphous Powder SolidMolecular weight:1134.9Oxindole
CAS:Oxindole (Indolin-2-one) is an aromatic heterocyclic building block. 2-indolinone derivatives have become lead compounds in the research of kinase inhibitors.Oxindole structure has been used in receptor tyrosine kinases (RTKs) inhibitors such as SU4984 and intedanib, the RTK family represents an important therapeutic target for anti-cancer drug development.Formula:C8H7NOPurity:99.34%Color and Shape:Off-White Crystalline PowderMolecular weight:133.15TCH-165
CAS:TCH-165 boosts 20S proteasome levels, enhancing IDP breakdown.Formula:C39H37N3O3Purity:98.2% - 98.75%Color and Shape:SolidMolecular weight:595.73Ref: TM-T17011
1mg74.00€5mg160.00€10mg250.00€25mg455.00€50mg682.00€100mg938.00€1mL*10mM (DMSO)265.00€KW-2450 Formate
KW-2450 Formate is an IGF-1R/IR tyrosine kinase inhibitor with antitumor effects that acts through inhibition of Aurora A and B kinases.KW-2450 Formate inhibits the growth of TNBC xenografts and induces tetraploid accumulation.Formula:C29H31N5O5SPurity:99.34%Color and Shape:SolidMolecular weight:561.65Thiamine disulfide
CAS:Thiamine disulfide (Algoneurina) , also known as thiamin or vitamin B1, is a vitamin found in food and manufactured as a dietary supplement and medication.Formula:C24H34N8O4S2Purity:99.18%Color and Shape:CoaMolecular weight:562.71Chlorcyclizine
CAS:CHLORCYCLIZINE is a histamine H1 antagonist and a potent hepatitis C virus (HCV) entry inhibitor.Formula:C18H21ClN2Purity:98% - 98.75%Color and Shape:SolidMolecular weight:300.83UK 356618
CAS:UK 356618 is a potent and selective inhibitor of matrix metalloprotease-3 (IC50: 5.9 nM).Formula:C34H43N3O4Purity:98%Color and Shape:SolidMolecular weight:557.72Cabotegravir
CAS:Cabotegravir (S/GSK1265744) (GSK744, GSK1265744) is a long-acting HIV integrase inhibitor and inhibits the HIV-1 integrase catalyzed strand transfer reaction (Formula:C19H17F2N3O5Purity:98.55% - 99.92%Color and Shape:SolidMolecular weight:405.35Tyrosinase-IN-35
CAS:Tyrosinase-IN-35 (compound 6g), exhibiting a IC 50 value of 2.09 μM, serves as a more effective inhibitor of human tyrosinase compared to Kojic Acid (IC 50: 16.38 μM). At concentrations of 4 μM and 8 μM, this compound effectively lowers melanin levels in melanoma B16F10 cells in vitro.Formula:C17H15N5OSColor and Shape:SolidMolecular weight:337.40DRB
CAS:DRB is a nucleoside analog that inhibits several carboxyl-terminal domain (CTD) kinases including casein kinase II (IC50 range of 4-10 μM)Formula:C12H12Cl2N2O4Purity:99.46%Color and Shape:White To Off-White Crystalline SolidMolecular weight:319.14Collagenase Type II
Collagenase Type II, an endopeptidic MMP-8, preferentially degrades type I collagen tissues requiring high digestive efficiency pancreas and liver.Color and Shape:Odour SolidU18666A
CAS:U18666A is a cell-permeable drug and is a cholesterol synthesis and transport inhibitor.Formula:C25H42ClNO2Purity:98.99%Color and Shape:SolidMolecular weight:424.06Ref: TM-T17190
1mg35.00€2mg47.00€5mg70.00€10mg97.00€25mg185.00€50mg301.00€100mg454.00€200mg650.00€1mL*10mM (DMSO)77.00€CASP3 Activator 1541
CAS:CASP3 Activator 1541 is an activator of the proenzyme forms of caspase-3, and induces cell death.Formula:C24H17N3O4Purity:98.84%Color and Shape:SolidMolecular weight:411.41L 756423
CAS:L756423 is a potent, selective HIV protease inhibitor (Ki=0.049 nM), effective against HIV spread in MT25 lymphocytes at 0.1-0.5 nM, useful for AIDS research.Formula:C39H48N4O5Purity:100% - 100%Color and Shape:SolidMolecular weight:652.82TAPI1
CAS:TAPI1 (TAPI) , an ADAM17/TACE inhibitor, inhibits shedding of cytokine receptors.Formula:C26H37N5O5Purity:≥95%Color and Shape:SolidMolecular weight:499.6Setrobuvir
CAS:Setrobuvir (ANA-598) is an orally active non-nucleoside HCV NS5B polymerase inhibitor with inhibitory effects on de novo RNA synthesis and primer extension withFormula:C25H25FN4O6S2Purity:100% - 99%Color and Shape:SolidMolecular weight:560.62Ref: TM-T28762
1mg229.00€5mg570.00€10mg812.00€25mg1,216.00€50mg1,663.00€100mg2,242.00€500mg4,494.00€1mL*10mM (DMSO)737.00€Efavirenz
CAS:Efavirenz (DMP 266) is an HIV-1 inhibitor, affecting reverse transcriptase and various cytochrome P450 enzymes.Formula:C14H9ClF3NO2Purity:99.2% - 99.83%Color and Shape:White To Slightly Pink Crystalline PowderMolecular weight:315.67Ref: TM-T2393
1g404.00€5mg42.00€10mg52.00€25mg71.00€50mg89.00€100mg116.00€500mg273.00€1mL*10mM (DMSO)49.00€Doxycycline hydrochloride
CAS:Doxycycline hydrochloride (Hyclate) is a synthetic tetracycline derivative with similar antimicrobial activity.Formula:C22H24N2O8·HClPurity:98.77%Color and Shape:Yellow Hygroscopic Crystalline PowderMolecular weight:480.9Atazanavir
CAS:Formula:C38H52N6O7Purity:>95.0%(HPLC)Color and Shape:White to Light yellow powder to crystalMolecular weight:704.87Mk-6186 HCl
MK-6186 HCl, a novel non-nucleoside reverse transcriptase inhibitor with antiviral activity, can be used to study HIV.Formula:C21H13Cl3N6OPurity:98.19%Color and Shape:SoildMolecular weight:471.73Trelagliptin
CAS:Trelagliptin (SYR-472) is a highly specific and long-acting DPP-4 inhibitor.Formula:C18H20FN5O2Purity:98.88%Color and Shape:SolidMolecular weight:357.38ACH-806
CAS:ACH-806 is an NS4A antagonist. It can inhibit Hepatitis C Virus (HCV) replication with an EC50 of 14 nM.Formula:C19H20F3N3O2SPurity:98%Color and Shape:SolidMolecular weight:411.44Sofosbuvir impurity K
CAS:Sofosbuvir impurity K is an diastereoisomer of Sofosbuvir.Sofosbuvir is an HCV RNA replication inhibitor, with potent anti-hepatitis C virus activity.Formula:C22H29ClN3O9PPurity:98%Color and Shape:SolidMolecular weight:545.91NBD-557
CAS:NBD-557 is a potentially HIV-1 inhibitor.Formula:C17H24BrN3O2Purity:99.52%Color and Shape:SolidMolecular weight:382.3Ref: TM-T7382
1mg48.00€5mg97.00€10mg156.00€25mg301.00€50mg437.00€100mg620.00€200mg843.00€1mL*10mM (DMSO)105.00€Ilomastat
CAS:Formula:C20H28N4O4Purity:>95.0%(HPLC)(qNMR)Color and Shape:White to Light yellow powder to crystalMolecular weight:388.472-Amino-6-bromopyridine
CAS:2-Amino-6-bromopyridine has inhibitory effect on HIV-68 protease.Formula:C5H5BrN2Purity:99.87%Color and Shape:SolidMolecular weight:173.013,3′-Bisdemethylpinoresinol
CAS:3,3′-Bisdemethylpinoresinol, a natural lignin derivative, exhibits MMP-1 inhibitory activity in UVA-irradiated human dermal fibroblasts and can be isolated fromFormula:C18H18O6Purity:98%Color and Shape:SolidMolecular weight:330.33LY 3000328
CAS:LY 3000328 (Cathepsin S inhibitor) is a selective inhibitor of cathepsin S.Cost-effective and quality-assured.Formula:C25H29FN4O5Purity:97.83% - 99.54%Color and Shape:SolidMolecular weight:484.52Ref: TM-TQ0116
1mg96.00€2mg137.00€5mg210.00€10mg278.00€25mg487.00€50mg708.00€100mg998.00€1mL*10mM (DMSO)220.00€NNRTIs-IN-3
NNRTIs-IN-3 (compound 8) is an HIV-1 non-nucleoside reverse transcriptase inhibitor, displaying potent efficacy with an EC50 value of 0.01 µM [1].Formula:C17H20ClN5OPurity:98%Color and Shape:SolidMolecular weight:345.83NP-313
CAS:NP-313 (NSC-4264) is a potent antithrombotic that blocks platelet aggregation via thromboxane A2 synthesis inhibition and targets SOCC-mediated Ca2+ efflux.Formula:C12H8ClNO3Purity:98.97%Color and Shape:SolidMolecular weight:249.65Ac-VRPR-AMC
CAS:Ac-VRPR-AMC is a fluorogenic substrate for metacaspase activity assays, facilitating the detection and measurement of metacaspase activity [1].Formula:C34H51N11O7Purity:98%Color and Shape:SolidMolecular weight:725.842-PMPA
CAS:2-PMPA (2-(Phosphonomethyl)pentanedioic acid) is a potent and selective inhibitor of glutamate carboxypeptidase II (GCPII) (IC50=300 pM).Formula:C6H11O7PPurity:98% - 99.50%Color and Shape:SolidMolecular weight:226.12Tyrosinase-IN-32
Tyrosinase-IN-32 (compound 11), a hydroxamate-based alkaloid extracted from black pepper (Piper nigrum L.), functions as an inhibitor of mushroom tyrosinase. In addition to its inhibitory properties, it exhibits antioxidant activity.Formula:C15H19NO3Color and Shape:SolidMolecular weight:261.32ABT530
CAS:ABT530 (Pibrentasvir) is an HCV NS5A inhibitor with EC50s ranging from 1.4-5.0 pM against HCV replicons containing NS5A from genotypes 1-6.Formula:C57H65F5N10O8Purity:99.15% - 99.93%Color and Shape:SolidMolecular weight:1113.18MMP-3 Inhibitor
CAS:MMP-3 Inhibitor is a peptide matrix metalloproteinase-3 (MMP-3) inhibitor with a Ki value of 95 nM.MMP-3 inhibitor has anticancer and antitumor activity.Formula:C27H46N10O9SPurity:98.87%Color and Shape:SolidMolecular weight:686.78Ref: TM-T37048
1mg81.00€5mg208.00€10mg309.00€25mg525.00€50mg757.00€100mg1,035.00€500mg2,110.00€1mL*10mM (DMSO)221.00€Isoangustone A
CAS:Isoangustone A has antitumor activity, it can induce G1 cycle arrest in DU145 human prostate and 4T1 murine mammary cancer cells, it inhibits cell proliferationFormula:C25H26O6Purity:98%Color and Shape:SolidMolecular weight:422.47MMP13-IN-3
CAS:MMP13-IN-3 is an oral, selective MMP-13 inhibitor with IC50 of 1 nM, >1000x selective, for osteoarthritis treatment.Formula:C24H22N4O5Purity:99.05%Color and Shape:SolidMolecular weight:446.46Ref: TM-T16124
1mg87.00€5mg216.00€10mg354.00€25mg620.00€50mg847.00€100mg1,169.00€1mL*10mM (DMSO)240.00€N-α-Tosyl-L-lysine chloromethyl ketone hydrochloride
CAS:N-alpha-Tosyl-L-lysine chloromethyl ketone hydrochloride inhibits trypsin-like proteases and IFN-γ activities.Formula:C14H22Cl2N2O3SPurity:97.44%Color and Shape:PowderMolecular weight:369.31TNF Protease Inhibitor 2
CAS:TAPI-2 is a broad-spectrum inhibitor of MMP (IC50: 20 μM), tumour necrosis factorα-converting enzyme (TACE) and a disintegrin and metalloproteinase (ADAM).Formula:C19H37N5O5Purity:98%Color and Shape:SolidMolecular weight:415.53MG-132
CAS:Formula:C26H41N3O5Purity:>95.0%(qNMR)Color and Shape:White to Light yellow powder to crystalMolecular weight:475.63Z-Leu-Leu-Tyr-COCHO
CAS:Z-Leu-Leu-Tyr-COCHO is a potent inhibitor of chymotrypsin-like activity, exhibiting a Ki value of 3.0 nM [1].Formula:C30H39N3O7Purity:98%Color and Shape:SolidMolecular weight:553.65Emivirine
CAS:Emivirine (MKC-442) is a potent and selective nonnucleoside reverse transcriptase inhibitor of human immunodeficiency virus type 1.Formula:C17H22N2O3Purity:99.68%Color and Shape:SolidMolecular weight:302.37Benzylsulfonyl Fluoride [for Biochemical Research]
CAS:Formula:C7H7FO2SPurity:>98.0%(GC)Color and Shape:White to Almost white powder to crystalMolecular weight:174.19BI 224436
CAS:BI 224436 is an inhibitor of HIV-1 noncatalytic site integrase. With EC50 values of less than 15 nM against different HIV-1 laboratory strains.Formula:C27H26N2O4Color and Shape:SolidMolecular weight:442.51HIV-1 protease-IN-9
CAS:HIV-1 protease-IN-9 (compound 5b), a potent HIV-1 protease inhibitor, exhibits strong antiviral efficacy with a dissociation constant (K_i) of 0.028 nM and aFormula:C37H41N7O4SPurity:98%Color and Shape:SolidMolecular weight:679.83CDK9-IN-30
CAS:CDK9-IN-30 is one of the Tat peptide derivatives and inhibits HIV-1 long terminal repeat-activated transcription.Formula:C16H20FNO3Purity:99.76%Color and Shape:SolidMolecular weight:293.33Ref: TM-T9632
1mg56.00€5mg119.00€10mg187.00€25mg316.00€50mg472.00€100mg658.00€500mg1,378.00€1mL*10mM (DMSO)114.00€GLPG2451
CAS:GLPG2451 potentiates F508del CFTR at low temp (EC50: 11.1 nM), aiding cystic fibrosis treatment.Formula:C16H16F3N3O5SColor and Shape:SolidMolecular weight:419.38Trisodium Hydrogen Ethylenediaminetetraacetate Hydrate [for Biochemical Research]
CAS:Formula:C10H13N2Na3O8·xH2OPurity:>98.0%(T)Color and Shape:White to Almost white powder to crystalMolecular weight:358.19 (as Anhydrous)Benzoic acid, 4-[(aminoiminomethyl)amino]-, 6-(aminoiminomethyl)-2-naphthalenyl ester, dimethanesulfonate
CAS:Formula:C21H25N5O8S2Purity:98%Color and Shape:SolidMolecular weight:539.5819MMP-2 Inhibitor-4
MMP-2Inhibitor-4 (Compound 5g) is an MMP-2 inhibitor with an IC50 of 152.62 nM. It effectively reduces MMP-2 levels in K562 cell lines by stably binding to the active site of MMP-2 and exhibits strong anti-angiogenic effects in ACHN cell lines. MMP-2Inhibitor-4 shows potential for research in chronic myelogenous leukemia (CML).Formula:C19H23N3O5SMolecular weight:405.468Sofosbuvir impurity H
Sofosbuvir impurity H, an diastereoisomer of Sofosbuvir, is the impurity of Sofosbuvir.Formula:C29H33FN3O10PPurity:98%Color and Shape:SolidMolecular weight:633.56Licraside
CAS:Licraside is a tyrosinase inhibitor with an IC50 of 0.072 mM for monophenolase and can be used in studies about antibrowning and depigmenting agents.Formula:C26H30O13Purity:99.85%Color and Shape:SolidMolecular weight:550.51Raltegravir potassium
CAS:Raltegravir potassium (MK 0518 potassium salt) salt(MK0518 potassium salt) is a potent integrase (IN) inhibitor, used to treat HIV infection.Formula:C20H20FN6O5·KPurity:98% - 99.55%Color and Shape:Off-White SolidMolecular weight:482.51Cilastatin
CAS:Cilastatin (MK0791): protects imipenem from renal breakdown; inhibits leukotriene D4 metabolism.Formula:C16H26N2O5SPurity:97.76% - 99.71%Color and Shape:SolidMolecular weight:358.45Ref: TM-T2583
5mg35.00€10mg44.00€25mg63.00€50mg88.00€100mg124.00€200mg188.00€500mg325.00€1mL*10mM (DMSO)55.00€Flovagatran
CAS:Flovagatran (TGN 255) is a potent, and selective inhibitor of thrombin and parenteral direct factor II.Flovagatran is used to study venous thromboembolism.Formula:C27H36BN3O7Purity:99.56%Color and Shape:SolidMolecular weight:525.4Ro24-7429
CAS:Ro24-7429: oral HIV-1 Tat antagonist, RUNX1 inhibitor with anti-HIV, antifibrotic, and anti-inflammatory properties.Formula:C14H13ClN4Purity:99.29% - 99.85%Color and Shape:SolidMolecular weight:272.73Ref: TM-T28578
1mg92.00€5mg187.00€10mg298.00€25mg507.00€50mg730.00€100mg1,026.00€500mg2,877.00€1mL*10mM (DMSO)215.00€Caspase-3 activator 3
Caspase-3 activator 3 (compound 2h) effectively induces apoptosis in HL-60 and K562 cells by substantially activating caspase-3, demonstrating antileukemicPurity:98%Color and Shape:Odour Solid3-Aminobenzene-1,2-diol
CAS:3-Aminobenzene-1,2-diol (compound C8) is an inhibitor of matrix metalloproteinases (MMP), with IC50 values of 20, 26, 16, and 16.3 μM against MMP-2, MMP-8, MMP-9, and MMP-14, respectively.Formula:C6H7NO2Color and Shape:SolidMolecular weight:125.132-Benzylsuccinic acid
CAS:2-Benzylsuccinic acid (DL-Benzylsuccinic acid) is a bacterial xenobiotic metabolite.Formula:C11H12O4Purity:≥95%Color and Shape:SolidMolecular weight:208.21HIV-1 protease-IN-7
CAS:HIV-1 protease-IN-7 (compound 16) is an orally active inhibitor of HIV-1 protease, exhibiting an IC50 of 3.52 nM and an EC50 of 37 nM [1].Formula:C68H104N10O12SPurity:98%Color and Shape:SolidMolecular weight:1285.68Aderamastat
CAS:Aderamastat (FP-025) is an orally active matrix metalloproteinase 12 (MMP-12) inhibitor indicated for the study of allergic asthma, COPD and pulmonary fibrosis.Formula:C21H18N2O4SPurity:99.35%Color and Shape:SolidMolecular weight:394.44PF 00356231
CAS:PF 00356231 is a selectivity inhibitor MMP-12 and can be used in studies about the treatment of emphysema and chronic obstructive pulmonary disease (COPD).Formula:C25H20N2O3SPurity:99.35%Color and Shape:SolidMolecular weight:428.5R-1479
CAS:R-1479 (4'-Azidocytidine) is an RdRp inhibitor with an IC50 value of 1.28 μM for HCV RNA replication in the HCV subgenomic replicon system.Formula:C9H12N6O5Purity:99.68% - 99.95%Color and Shape:SolidMolecular weight:284.23Ref: TM-TQ0162
1mg135.00€2mg187.00€5mg329.00€10mg472.00€25mg753.00€50mg1,074.00€100mg1,444.00€1mL*10mM (DMSO)363.00€Trypsin Inhibitor, soybean
CAS:Trypsin Inhibitor, soybean is a trypsin inhibitor extracted from leguminous plants.Color and Shape:SolidPhepropeptin C
CAS:Phepropeptin C is a microbial secondary metabolite that acts as a proteasome (proteasome) inhibitor, with an IC50 of 12.5 μg/mL.Formula:C38H60N6O6Color and Shape:SolidMolecular weight:696.92Dolutegravir intermediate-1
CAS:Dolutegravir intermediate-1 is a synthetic precursor for HIV-1 treatment from patent WO 2016125192 A2.Formula:C13H17NO8Purity:99.52%Color and Shape:SolidMolecular weight:315.28Isoderrone
CAS:Isoderrone inhibits α-glucosidase and PTP1B; IC50 = 22.7 uM, potential type 2 diabetes drug.Formula:C20H16O5Purity:98%Color and Shape:SolidMolecular weight:336.34Tenofovir alafenamide hemifumarate
CAS:Tenofovir alafenamide hemifumarate (GS-7340 hemifumarate) is an oral phosphonoamidate prodrug of the HIV reverse transcriptase nucleotide inhibitor tenofovir.Formula:C21H29N6O5PC4H4O4Purity:99.33% - 99.96%Color and Shape:SolidMolecular weight:534.51Glucosamine
CAS:Glucosamine (Chitosamine) is an amino sugar and a prominent precursor in the biochemical synthesis of glycosylated proteins and lipids.Formula:C6H13NO5Purity:99.80% - 99.80%Color and Shape:CoaMolecular weight:179.17S-Methylglutathione
CAS:S-Methylglutathione (S-Methyl glutathione) is a 1-chloro-2,4-dinitrobenzene coupling inhibitor, an XOCl scavenger, and inhibitor of glyoxalase 1.Formula:C11H19N3O6SPurity:98%Color and Shape:SolidMolecular weight:321.35