Ephrin Receptor
Ephrin receptor inhibitors target Eph receptors, a family of receptor tyrosine kinases that interact with membrane-bound ephrin ligands. Ephrin signaling is crucial for cell positioning, tissue patterning, and angiogenesis. Dysregulation of this pathway is implicated in cancer, neurodegenerative diseases, and developmental disorders. At CymitQuimica, we provide Ephrin receptor inhibitors to support your research in developmental biology, oncology, and neurobiology.
Products of "Ephrin Receptor"
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Found 15 products on this category.
UniPR1449
UniPR1449 is an EphA2 receptor antagonist with a KD of 3.8±2.4 μM, which is significant in cancer pathophysiology [1].Purity:98%Color and Shape:Odour SolidTesevatinib
CAS:Tesevatinib (XL-647) is an oral, multi-targeted tyrosine kinase inhibitor.Cost-effective and quality-assured.Formula:C24H25Cl2FN4O2Purity:97.89% - 97.89%Color and Shape:SolidMolecular weight:491.39Ref: TM-TQ0166
1mg107.00€2mg156.00€5mg236.00€10mg457.00€25mg750.00€50mg1,026.00€1mL*10mM (DMSO)255.00€JI-101
CAS:JI-101 (CGI-1842) is an oral multi-kinase inhibitor that targets VEGFR-2, PDGFR-β, and EphB4.Formula:C22H20BrN5O2Purity:99.35% - 99.41%Color and Shape:SolidMolecular weight:466.33UniPR1447
CAS:UniPR1447 is a dual antagonist for both EphA2 and EphB2 receptors, exhibiting an IC50 value of 6.6 μM against EphA2-ephrin-A1 binding [1].Formula:C36H50N2O4Purity:98%Color and Shape:SolidMolecular weight:574.79AWL-II-38.3
CAS:AWL-II-38.3 is a highly potent EphA3 inhibitor with potent kinase inhibitory activity against EphA3.Cost-effective and quality-assured.Formula:C23H18F3N5O3Purity:99.87% - 99.87%Color and Shape:SolidMolecular weight:469.42Ref: TM-T38511
1mg81.00€5mg170.00€10mg264.00€25mg543.00€50mg780.00€100mg1,074.00€500mg2,167.00€1mL*10mM (DMSO)177.00€ALW-II-41-27
CAS:ALW-II-41-27 (Eph receptor tyrosine kinase inhibitor), an Eph receptor tyrosine kinase inhibitor, is used for cancer therapy.Formula:C32H32F3N5O2SPurity:97.01% - 99.52%Color and Shape:SolidMolecular weight:607.69Ref: TM-T4344
1mg69.00€2mg97.00€5mg170.00€10mg264.00€25mg437.00€50mg640.00€100mg910.00€1mL*10mM (DMSO)240.00€123C4
CAS:123C4 is a potent, selective and competitive agonist of the receptor tyrosine kinase EPHA4 (Ki=0.65 μM)[1].Formula:C43H47ClN8O6Purity:98.94%Color and Shape:SolidMolecular weight:807.34Ref: TM-TP1561
1mg144.00€5mg311.00€10mg512.00€25mg815.00€50mg1,093.00€100mg1,473.00€1mL*10mM (DMSO)507.00€Ehp-inhibitor-2
CAS:Ehp-inhibitor-2 is an Eph family tyrosine kinase inhibitor targeting Eph receptors.Formula:C17H13N5OPurity:98.02%Color and Shape:SolidMolecular weight:303.32Ref: TM-T5452
1mg47.00€2mg58.00€5mg87.00€10mg153.00€25mg249.00€50mg369.00€100mg545.00€1mL*10mM (DMSO)97.00€ALW-II-49-7
CAS:ALW-II-49-7 is a selective and potent inhibitor of EphB2 kinase with an EC50 value of 40 nM in cell.Formula:C21H17F3N4O2Purity:99.84%Color and Shape:SoildMolecular weight:414.38Ref: TM-T67736
1mg71.00€5mg166.00€10mg243.00€25mg439.00€50mg647.00€100mg920.00€500mg1,853.00€1mL*10mM (DMSO)177.00€UniPR505
CAS:UniPR505 is a potent EphA2 antagonist (IC50: 0.95 µM), a novel 3α-carbamoyloxy derivative with antiangiogenic properties.Formula:C39H57N3O5Purity:99.23%Color and Shape:SolidMolecular weight:647.89LDN-211904 oxalate
CAS:LDN-211904 oxalate (LDN211904 oxalate) is a selective and efficient EphB3 inhibitor with antitumor activity, useful in neurodegenerative disease research.Formula:C21H21ClN4O5Purity:99.87%Color and Shape:SolidMolecular weight:444.87Eph inhibitor 2
CAS:Eph inhibitor 2 is an Eph family tyrosine kinase inhibitor targeting Eph receptors.Formula:C18H15N5OPurity:99.01%Color and Shape:SolidMolecular weight:317.34Ref: TM-T5451
1mg95.00€2mg125.00€5mg188.00€10mg284.00€25mg515.00€50mg742.00€100mg1,035.00€500mg2,080.00€1mL*10mM (DMSO)187.00€NVP-BHG712
CAS:NVP-BHG712 is a specific EphB4 inhibitor with ED50 of 25 nM that discriminates between VEGFR and EphB4 inhibition; also shows activity against c-Raf, c-Src andFormula:C26H20F3N7OPurity:97.32%Color and Shape:SolidMolecular weight:503.48Ref: TM-T6348
1mg35.00€5mg79.00€10mg111.00€25mg212.00€50mg393.00€100mg587.00€200mg833.00€1mL*10mM (DMSO)88.00€UniPR500
CAS:UniPR500, a derivative of UniPR129, is a competitive antagonist for the EphA2 receptor, with a Ki of 0.78 μM. It reduces the binding of biotinylated Ephrin-A1 to EphA2 in a dose-dependent manner, exhibiting an IC50 value of 1.1 μM.Formula:C36H51N3O4Color and Shape:SolidMolecular weight:589.808NVP-BHG712 isomer
CAS:NVP-BHG712 isomer shows conserved non-bonded binding to EPHA2 and EPHB4.Formula:C26H20F3N7OPurity:99.14%Color and Shape:SolidMolecular weight:503.48Ref: TM-T19487
1mg43.00€2mg56.00€5mg88.00€10mg150.00€25mg259.00€50mg376.00€100mg560.00€1mL*10mM (DMSO)87.00€
