Bombesin Receptor
Bombesin receptors are a group of GPCRs that are activated by bombesin-like peptides, which are involved in regulating gastrointestinal function, energy balance, and cell proliferation. These receptors are of particular interest in cancer research, as they are often overexpressed in certain types of tumors. Bombesin receptor antagonists are studied for their potential as cancer therapeutics. At CymitQuimica, we provide a selection of high-quality bombesin receptor modulators to support your research in oncology, gastrointestinal physiology, and receptor signaling.
Products of "Bombesin Receptor"
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Found 8 products on this category.
MK-5046
CAS:MK-5046 is a novel BRS-3 agonist, binding to BRS-3 with high affinity (mouse Ki = 1.6 nM, human Ki = 25 nM).Formula:C20H18F6N4OPurity:98.56%Color and Shape:SolidMolecular weight:444.37ML-18
CAS:ML-18 is a non-peptide bombesin receptor subtype-3 (BRS-3) antagonist with an IC50 of 4.8 μM.Formula:C32H35N5O5Purity:100% - 98.62%Color and Shape:SolidMolecular weight:569.65Ref: TM-T4540
1mg35.00€5mg64.00€10mg92.00€25mg178.00€50mg279.00€100mg449.00€200mg620.00€1mL*10mM (DMSO)80.00€CD80-IN-3
CAS:CD80-IN-3 is a potent CD80 inhibitor and inhibits CD80/CD28 interaction (Kd: 125 nM; EC50: 630 nM).Formula:C17H10FN3O3Purity:98.08%Color and Shape:SolidMolecular weight:323.28Ref: TM-T10722
1mg80.00€5mg187.00€10mg305.00€25mg494.00€50mg682.00€100mg847.00€1mL*10mM (DMSO)207.00€kuwanon G
CAS:Kuwanon G (Moracenin B) may be used to treat the type II diabetes mellitus as a dual inhibitor of PTP1B and α-glucosidase and as an insulin sensitiser.Formula:C40H36O11Purity:98% - 98.47%Color and Shape:SolidMolecular weight:692.71Ref: TM-T3S1612
1mg66.00€5mg145.00€10mg210.00€25mg339.00€50mg492.00€100mg662.00€200mg892.00€1mL*10mM (DMSO)188.00€Kuwanon H
CAS:Kuwanon H is a potent non-peptide GRP receptor antagonist with a Ki of 290 nM, useful in GRP-related studies.Formula:C45H44O11Purity:97.99%Color and Shape:SolidMolecular weight:760.82RC-3095 TFA
CAS:RC-3095 TFA (RC-3095 (TFA)) is a bombesin/gastrin-releasing peptide (BN/GRP) antagonist with potential anticancer activity.Formula:C58H80F3N15O11Purity:98%Color and Shape:SolidMolecular weight:1220.34PD176252
CAS:PD176252 is a BB1 and BB2 antagonist, GRPR inhibitor, and FPR1/FPR2 agonist that inhibits the growth and proliferation of a wide range of cancer cells.Formula:C32H36N6O5Purity:99.18%Color and Shape:SolidMolecular weight:584.67PD 168368
CAS:PD 168368 is a mixed neuromodulin B receptor (NMB-R) antagonist and potent FPR1/FPR2/FPR3 agonist that inhibits the gastrin-releasing peptide receptor.Formula:C31H34N6O4Purity:98.44%Color and Shape:SolidMolecular weight:554.64
