Histamine Receptor
Histamine receptors are GPCRs that mediate the effects of histamine, a biogenic amine involved in immune responses, gastric acid secretion, and neurotransmission. There are four subtypes of histamine receptors (H1, H2, H3, and H4), each playing distinct roles in allergic reactions, gastric function, and central nervous system activity. Histamine receptor antagonists are widely used in the treatment of allergies, peptic ulcers, and motion sickness. At CymitQuimica, we provide a comprehensive selection of high-quality histamine receptor modulators to support your research in immunology, gastroenterology, and neuropharmacology.
Products of "Histamine Receptor"
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Noberastine
CAS:Noberastine (R 64947) is a novel histamine H1 antagonist with potent and specific peripheral antihistamine activity.Formula:C17H21N5OPurity:100% - 99.67%Color and Shape:SolidMolecular weight:311.38Dalcotidine
CAS:Dalcotidine (KU 1257), a histamine H2/H9 blocker, inhibits acid secretion; Ki=0.040, KB=0.041, aids ulcer healing, may lower relapse.Formula:C18H29N3O2Purity:98.34%Color and Shape:SolidMolecular weight:319.44Ref: TM-T31195
1mg94.00€5mg205.00€10mg303.00€25mg490.00€50mg710.00€100mg998.00€200mg1,349.00€1mL*10mM (DMSO)205.00€Acrivastine
CAS:Acrivastine (Acrivastin) is a short-acting histamine 1 receptor antagonist.Formula:C22H24N2O2Purity:100% - 99.73%Color and Shape:SolidMolecular weight:348.44Ref: TM-T4551
1g792.00€5mg37.00€10mg51.00€25mg99.00€50mg160.00€100mg221.00€500mg553.00€1mL*10mM (DMSO)40.00€Chlorphenoxamine
CAS:Chlorphenoxamine (Contristamine) is an antihistamine and anticholinergic used as an antipruritic and antiparkinsonian agent.Formula:C18H22ClNOPurity:99.44%Color and Shape:SolidMolecular weight:303.83Fexofenadine hydrochloride
CAS:Fexofenadine hydrochloride (Terfenidine carboxylate hydrochloride) is a second generation antihistamine that is used for the treatment of allergic rhinitis,Formula:C32H39NO4·HClPurity:99.39% - ≥95%Color and Shape:SolidMolecular weight:538.13Azelastine hydrochloride
CAS:Azelastine hydrochloride (Astelin) is a phthalazinone derivative with antihistaminergic activity.Formula:C22H24ClN3O·HClPurity:100% - 99.97%Color and Shape:White Crystalline PowderMolecular weight:418.36Chloropyramine hydrochloride
CAS:Chloropyramine hydrochloride (Alergosan) is a histamine receptor H1 antagonist.Formula:C16H20ClN3·HClPurity:99.45% - 99.8%Color and Shape:SolidMolecular weight:326.26Dexchlorpheniramine Maleate
CAS:Dexchlorpheniramine Maleate, an antihistamine with anticholinergic effects, treats allergies like hay fever. It's the active isomer of chlorpheniramine.Formula:C20H23ClN2O4Purity:99.58%Color and Shape:White Or Almost White Crystalline PowderMolecular weight:390.86Mirtazapine
CAS:Mirtazapine is a unique tetracyclic antidepressant, may cause temporary liver enzyme elevation, and is linked to rare liver injury.Formula:C17H19N3Purity:99.98%Color and Shape:SolidMolecular weight:265.35Tripelennamine hydrochloride
CAS:Tripelennamine hydrochloride (Pyribenzamine hydrochloride) is a histamine H1 antagonist with low sedative action but frequent gastrointestinal irritation.Formula:C16H21N3·HClPurity:100% - 99.54%Color and Shape:White SolidMolecular weight:291.82KSK94 FA
KSK94 FA is a potent histamine H3 receptor antagonist that inhibits H3 receptors and is used in the study of neuropathic pain and obesity.Formula:C26H28N4O3Purity:98.13%Color and Shape:SoildMolecular weight:444.53H3 receptor antagonist 1
CAS:H3 receptor antagonist 1 is used in the study of neurological diseases, histamine H3 receptor antagonist.Formula:C20H28F2N2OPurity:98%Color and Shape:SolidMolecular weight:350.45PF-03654746 Tosylate
CAS:PF-03654746 Tosylate is selective antagonist of histamine H3 receptor with high brain penetration.Formula:C25H32F2N2O4SPurity:98%Color and Shape:SolidMolecular weight:494.6Clobenpropit dihydrobromide
CAS:Clobenpropit dihydrobromide is a potent antagonist and inverse agonist of histamine H3R (histamine H3LR,pEC50 of 8.07)Formula:C14H19Br2ClN4SPurity:99.86%Color and Shape:SolidMolecular weight:470.7Metiamide
CAS:Metiamide (SK&F 92058) is a histamine H2-receptor antagonist .Formula:C9H16N4S2Purity:97.41%Color and Shape:SolidMolecular weight:244.38Bromodiphenhydramine hydrochloride
CAS:Bromodiphenhydramine hydrochloride is a new antihistaminic in the control of cutaneous.Formula:C17H21BrClNOPurity:97.31%Color and Shape:SolidMolecular weight:370.71UR-AK49
CAS:UR-AK49 (compound 11) is an agonist for the human histamine H1 and H2 receptors. It exhibits an EC50 of 23 nM in the GTPase assay involving hH2R-Gsalpha fusion protein expressed in Sf9 insect cells. UR-AK49 is applicable in neurologically related research.Formula:C16H27N5OColor and Shape:SolidMolecular weight:305.42Doxylamine succinate
CAS:Doxylamine Succinate is a pyridine derivate histamine H1 antagonist with pronounced sedative properties.Formula:C21H28N2O5Purity:99.61%Color and Shape:5 1 (Ntp 1992)Molecular weight:388.46MK-0249
CAS:MK-0249 is a potent antagonist of histamine H3 receptor (human H3, Ki : 1.7 nM).Formula:C23H24F3N3O2Purity:99.79%Color and Shape:SolidMolecular weight:431.45Mianserin
CAS:Mianserin, an H1 receptor reverse agonist, is a psychoactive compound in the tetracyclic antidepressant (TeCA) treatment family.Formula:C18H20N2Purity:99.39%Color and Shape:SolidMolecular weight:264.36
