Histamine Receptor
Histamine receptors are GPCRs that mediate the effects of histamine, a biogenic amine involved in immune responses, gastric acid secretion, and neurotransmission. There are four subtypes of histamine receptors (H1, H2, H3, and H4), each playing distinct roles in allergic reactions, gastric function, and central nervous system activity. Histamine receptor antagonists are widely used in the treatment of allergies, peptic ulcers, and motion sickness. At CymitQuimica, we provide a comprehensive selection of high-quality histamine receptor modulators to support your research in immunology, gastroenterology, and neuropharmacology.
Products of "Histamine Receptor"
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Proxyfan
CAS:Proxyfan is a high-affinity protean antagonist/agonist of H3 receptors from full agonist to full inverse agonist, depending on given tissue or brain region.Formula:C13H16N2OPurity:99.68%Color and Shape:SolidMolecular weight:216.28Vapitadine dihydrochloride
CAS:Vapitadine dihydrochloride(R-129160 2HCl) is a novel, potent, selective and non-sedating compound with inhibitory effects on histamine H1.Formula:C17H22Cl2N4OPurity:100% - 99.92%Color and Shape:SolidMolecular weight:369.29Betahistine
CAS:Betahistine treats vertigo and balance issues in Ménière's disease; it's a histamine analog and H1 receptor agonist.Formula:C8H12N2Purity:97.92% - 99.87%Color and Shape:Yellowish Liquid Liquid LiquidMolecular weight:136.19N-Acetylhistamine
CAS:N-Acetylhistamine (N-Omega-acetylhistamine) is a metabolite of histamine.Formula:C7H11N3OPurity:97.72%Color and Shape:SolidMolecular weight:153.18(R)-(-)-α-Methylhistamine dihydrobromide
CAS:(R)-(-)-α-Methylhistamine dihydrobromide is a potent and selective agonist of H3 histamine receptor( Kd of 50.3 nM).Formula:C6H13Br2N3Purity:98%Color and Shape:SolidMolecular weight:287Dimethindene maleate
CAS:Dimethindene maleate (SU 6518) is a histamine H1 antagonist and can be used in studies about the treatment of hypersensitivity reactions, pruritus and rhinitis.Formula:C24H28N2O4Purity:99.87%Color and Shape:SolidMolecular weight:408.49Ref: TM-T21472
1mg35.00€5mg74.00€10mg111.00€25mg250.00€50mg329.00€100mg432.00€200mg615.00€1mL*10mM (DMSO)87.00€H4R antagonist 1
CAS:H4R antagonist 1: selective histamine H4R inhibitor, IC50 27 nM, no affinity for H1R, H2R, H3R.Formula:C11H11BrN8Color and Shape:SolidMolecular weight:335.16H3R antagonist 5
CAS:H3R antagonist 5 (Compound 1b) is a selective inverse agonist of the histamine H3 receptor that can penetrate the blood-brain barrier, with an IC50 of 0.54 nM. It is applicable for research related to the central nervous system.Formula:C23H32N2O4Color and Shape:SolidMolecular weight:400.511Irdabisant
CAS:Irdabisant (CEP-26401) is an H3R antagonist/inverse agonist, BBB permeable, with cognition-enhancing effects for schizophrenia/cognitive research.Formula:C18H23N3O2Purity:99.77%Color and Shape:SolidMolecular weight:313.39Ref: TM-T32191
1mg58.00€5mg134.00€10mg188.00€25mg335.00€50mg470.00€100mg662.00€500mg1,320.00€1mL*10mM (DMSO)93.00€ICI 162,846
CAS:ICI 162,846 is an orally active and potent H2 receptor antagonist that inhibits gastric secretion and may be used in the study of duodenal ulcers.Formula:C11H17F3N6OPurity:99.83%Color and Shape:SolidMolecular weight:306.29H3 receptor-MO-1
CAS:H3 receptor-MO-1 is a potent modulator of the histamine H3 receptor (H3 receptor) and can be used to study neurodegeneration and cognitive disorders.Formula:C20H27N3O2Purity:99.11%Color and Shape:SolidMolecular weight:341.45Pitolisant
CAS:Pitolisant is a potent and selective nonimidazole inverse agonist that acts on the recombinant human histamine H3 receptor with Ki of 0.16 nM.Formula:C17H26ClNOPurity:99.84%Color and Shape:SolidMolecular weight:295.85Ref: TM-T60636
5mg48.00€10mg70.00€25mg120.00€50mg188.00€100mg311.00€500mg747.00€1mL*10mM (DMSO)52.00€Olopatadine hydrochloride
CAS:Olopatadine hydrochloride (ALO4943A) is an antihistamine with mast-cell stabilizing properties used as eye drops in the treatment of ALLERGIC CONJUNCTIVITIS.Formula:C21H23NO3·HClPurity:99.62% - 99.64%Color and Shape:White SolidMolecular weight:373.87Latrepirdine dihydrochloride
CAS:Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets.Formula:C21H25N3·2HClPurity:98.45%Color and Shape:SolidMolecular weight:392.37PF 03654746 FA
PF 03654746 FA is a human histamine receptor H(3) antagonist that can be used to study cognitive impairment and Alzheimer's disease.Formula:C19H26F2N2O3Purity:96.15%Color and Shape:SoildMolecular weight:368.42H1R ligand-1
CAS:H1R ligand-1 (Compound fragment 1) is a high-affinity ligand for the human histamine H1 receptor (H1R). It can serve as a scaffold for synthesizing a series of derivatives to investigate H1R binding kinetics.Formula:C19H23NOColor and Shape:SolidMolecular weight:281.392H4R antagonist 2
CAS:H4R Antagonist 2, a potent Furo[3,2-d]pyrimidine derivative, serves as a histamine H4 receptor antagonist and holds potential for research into rheumatoidFormula:C13H17N5OPurity:98%Color and Shape:SolidMolecular weight:259.31TAAR1 agonist 2
CAS:TAAR1 agonist 2 (compound 30), a full agonist at trace amine-associated receptor 1 (TAAR1) (pEC50=7.5), also displays agonistic properties at H1 receptors and activates various muscarinic acetylcholine receptors, including the M2 receptor (pEC50=5). This compound is utilized in researching neuropsychiatric diseases.Formula:C9H11NOColor and Shape:SolidMolecular weight:149.19Dioxopromethazine
CAS:Dioxopromethazine (Dioxoprothazine) is a drug for the treatment of a cough and expectoration. It also can be used in local anesthesia.Formula:C17H20N2O2SPurity:98%Color and Shape:SolidMolecular weight:316.42JNJ-7777120
CAS:JNJ-7777120 is the first potent and selective non-imidazole histamine H4 receptor antagonist, exhibits >1000-fold selectivity over the other histamin receptors.Formula:C14H16ClN3OPurity:99.83% - 99.96%Color and Shape:SolidMolecular weight:277.75
