Histamine Receptor
Histamine receptors are GPCRs that mediate the effects of histamine, a biogenic amine involved in immune responses, gastric acid secretion, and neurotransmission. There are four subtypes of histamine receptors (H1, H2, H3, and H4), each playing distinct roles in allergic reactions, gastric function, and central nervous system activity. Histamine receptor antagonists are widely used in the treatment of allergies, peptic ulcers, and motion sickness. At CymitQuimica, we provide a comprehensive selection of high-quality histamine receptor modulators to support your research in immunology, gastroenterology, and neuropharmacology.
Products of "Histamine Receptor"
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ROS 234 dioxalate
CAS:ROS 234 dioxalate is a potent antagonist of H3(pKB of 9.46 for Guinea-pig ileum H3-receptor)Formula:C17H19N5O8Purity:98%Color and Shape:SolidMolecular weight:421.37Bavisant
CAS:Bavisant (JNJ-31001074) is a selective and orally active Human H3 receptor antagonist.Formula:C19H27N3O2Purity:96.06% - 98%Color and Shape:SolidMolecular weight:329.44Ref: TM-TQ0046
1mg43.00€5mg96.00€10mg134.00€25mg221.00€50mg325.00€100mg465.00€500mgTo inquire1mL*10mM (DMSO)94.00€(±)-Tazifylline
CAS:(±)-Tazifylline is a selective and long-acting antagonist of histamine H1 receptor.Formula:C23H32N6O3SPurity:98.97%Color and Shape:SolidMolecular weight:472.6Ref: TM-T10000
1mg148.00€5mg284.00€10mg411.00€25mg645.00€50mg867.00€100mg1,121.00€1mL*10mM (DMSO)369.00€BMY 25368 HCl
CAS:BMY 25368 HCl is a competitive histamine H2 receptor antagonist that antagonizes gastric secretion stimulated by pentagastrin, ethacrynic choline, and food.Formula:C19H26ClN3O3Purity:98.73% - 99.81%Color and Shape:SoildMolecular weight:379.88Lodoxamide tromethamine
CAS:Lodoxamide tromethamine is a mast cell stabilizer with anti-allergic properties and can be used in studies about the treatment of asthma and allergicFormula:C19H28ClN5O12Purity:99.58%Color and Shape:SolidMolecular weight:553.91Mifentidine
CAS:Mifentidine (DA 4577) is an orally available H2 receptor antagonist for the study of gastric emptying and experimental gastric and duodenal ulcers.Formula:C13H16N4Purity:100% - 99.20%Color and Shape:SolidMolecular weight:228.29Clemastine fumarate
CAS:Clemastine fumarate (Meclastine (fumarate)) is a synthetic ethanolamine with anticholinergic, sedative, and histamine H1 antagonistic properties.Formula:C25H30ClNO5Purity:99.52% - 99.8%Color and Shape:Colorless To Faintly Yellow Crystalline Powder Appearance White Or Almost White Crystalline PowderMolecular weight:459.97Fexofenadine
CAS:Fexofenadine, a non-sedating antihistamine, treats allergies like hay fever and urticaria.Formula:C32H39NO4Purity:99.87%Color and Shape:White To Off-White SolidMolecular weight:501.66Ref: TM-T21390
10mg50.00€25mg71.00€50mg97.00€100mg145.00€200mg212.00€500mg373.00€1mL*10mM (DMSO)58.00€NP10679
CAS:NP10679 is a N-methyl-D-aspartate (NMDA) receptor inhibitor of the GluN2B subunit that inhibits histamine H1, hERG channels, and CYPase.Formula:C23H26F3N3O3Purity:99.43%Color and Shape:SolidMolecular weight:449.47Carebastine
CAS:Carebastine, the active metabolite of Ebastine, is an antagonist of the histamine H1 receptor.Formula:C32H37NO4Purity:99.16%Color and Shape:Off-White SolidMolecular weight:499.64Lavoltidine
CAS:Lavoltidine (Loxtidine) is potent and selective H2 receptor antagonist, oral and irreversible,inhibits gastric acid secretion, gastroesophageal reflux disease.Formula:C19H29N5O2Purity:100% - 100%Color and Shape:SolidMolecular weight:359.47Azelastine
CAS:Azelastine (Azelastinum) is a phthalazine derivative, and is an histamine antagonist and mast cell stabilizer.Formula:C22H24ClN3OPurity:99.35%Color and Shape:White Crystal PowderMolecular weight:381.9Benztropine mesylate
CAS:Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSONFormula:C21H25NO·CH4SO3Purity:98.41% - 99.96%Color and Shape:White Crystalline Powder; Odourless Or Almost OdourlessMolecular weight:403.53Levodropropizine
CAS:Levodropropizine ((S)-(-)-Dropropizine) is a histamine receptor inhibitor. It is used as an effective and very well tolerated peripheral antitussive drug.Formula:C13H20N2O2Purity:100% - 99.93%Color and Shape:White Or Off White Crystalline PowderMolecular weight:236.31Diphenhydramine
CAS:Diphenhydramine (Syntedril): first-gen antihistamine for allergies, antiemetic, antitussive, anticholinergic, sedative, treats drug-induced parkinsonism.Formula:C17H21NOPurity:99.49%Color and Shape:SolidMolecular weight:255.35Chlorprothixene hydrochloride
CAS:Chlorprothixene hydrochloride, a typical antipsychotic, blocks 5-HT2, D1-D3, H1, muscarinic, and alpha1 receptors.Formula:C18H18ClNS·HClPurity:99.16%Color and Shape:White PowderMolecular weight:352.322-Pyridylethylamine dihydrochloride
CAS:2-Pyridylethylamine dihydrochloride is a Histamine H1 receptor agonist.Formula:C7H12Cl2N2Purity:99.42%Color and Shape:SolidMolecular weight:195.09Thioperamide maleate
CAS:Thioperamide maleate (MR-12842 maleate) is an effective and selective antagonist of H3 receptor (Ki = 4.3 nM) for inhibition of [3H]histamine synthesis (Ki = 31Formula:C19H28N4O4SPurity:99.88%Color and Shape:SolidMolecular weight:408.52ReN-1869
CAS:ReN-1869 is a novel selective histamine H(1) receptor antagonist with anti-neurogenic pain and anti-inflammatory activity for the study of neurological diseasesFormula:C24H27NO2Purity:99.87% - 99.89%Color and Shape:SolidMolecular weight:361.48Pheniramine maleate
CAS:Pheniramine maleate (Trimetose), an alkylamine derivative with antihistaminic and vasodilatory properties, binds to histamine H1 receptors.Formula:C16H20N2·C4H4O4Purity:99.85%Color and Shape:Physical Description White Powder With A Faint Amine-Like Odor Melting Point 107°CMolecular weight:356.42
