Histamine Receptor
Histamine receptors are GPCRs that mediate the effects of histamine, a biogenic amine involved in immune responses, gastric acid secretion, and neurotransmission. There are four subtypes of histamine receptors (H1, H2, H3, and H4), each playing distinct roles in allergic reactions, gastric function, and central nervous system activity. Histamine receptor antagonists are widely used in the treatment of allergies, peptic ulcers, and motion sickness. At CymitQuimica, we provide a comprehensive selection of high-quality histamine receptor modulators to support your research in immunology, gastroenterology, and neuropharmacology.
Products of "Histamine Receptor"
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Adriforant
CAS:Adriforant (PF-3893787,ZPL-3893797) is a competitive histamine receptor 4 h4 antagonist that antagonizes histamine-induced phosphorylation of ERK, inflammation.Formula:C13H22N6Purity:99.84%Color and Shape:SolidMolecular weight:262.35KP136
CAS:KP136 is an orally effective antiallergic compound (IC50: 76.1 μg/mL for histamine release and 63 ug/mL for degranulation).Formula:C16H18N4O3Purity:98.16% - 99.86%Color and Shape:SolidMolecular weight:314.34Oxmetidine
CAS:Oxmetidine (SKF 92994) is an H2R antagonist that inhibits transmembrane calcium flux in the cardiovascular system and is used in the study of duodenal ulcers.Formula:C19H21N5O3SPurity:99.67%Color and Shape:SolidMolecular weight:399.47Ref: TM-T68122
1mg378.00€5mg895.00€10mg1,216.00€25mg1,786.00€50mg2,442.00€100mg3,287.00€500mg6,603.00€Histamine
CAS:Histamine (Ergamine) is an amine derived by enzymatic decarboxylation of HISTIDINE.Formula:C5H9N3Purity:100% - 96.63%Color and Shape:Needles From Chloroform SolidMolecular weight:111.15Terfenadine
CAS:Terfenadine, metabolized to fexofenadine by CYP3A4, is a non-sedative antihistamine targeting H1 receptors.Formula:C32H41NO2Purity:98.76% - 99.75%Color and Shape:SolidMolecular weight:471.67WZ4141
CAS:WZ4141 is an intermediate in compound synthesis.Formula:C16H13N3O2Purity:98%Color and Shape:SolidMolecular weight:279.29MK-0249 FA
MK-0249 FA is an H3 inverse agonist that can be used to study attention-deficit, hyperactivity disorder and cognitive disorders in adults.Formula:C24H26F3N3O4Purity:100%Color and Shape:SolidMolecular weight:477.48Vapitadine
CAS:Vapitadine is a non-sedative antihistamine compound that relieves itching caused by atopic dermatitis.Formula:C17H20N4OPurity:100% - 100%Color and Shape:SoildMolecular weight:296.37Hydroxyzine
CAS:Hydroxyzine (Hydroxyzine free base) is an antagonist of histamine H1-receptor.Formula:C21H27ClN2O2Purity:99.54% - ≥95%Color and Shape:Oil SolidMolecular weight:374.9JNJ 10191584 maleate
CAS:JNJ 10191584 maleate (VUF6002 maleate) is an orally active and selective antagonist of H4 receptor (Ki = 26 nM).Formula:C17H19ClN4O5Purity:99.82%Color and Shape:SolidMolecular weight:394.81Nα-Methylhistamine FA
Nα-Methylhistamine FA is a histamine H3 receptor agonistFormula:C7H13N3O2Purity:100%Color and Shape:SolidMolecular weight:171.2Amitriptyline hydrochloride
CAS:Amitriptyline hydrochloride (Annoyltin) is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptiveFormula:C20H24ClNPurity:97% - 99.94%Color and Shape:Crystals White To Off-White PowderMolecular weight:313.86Donetidine
CAS:Donetidine is a histamine H2 receptor antagonist used to treat digestive disorders.Formula:C20H25N5O3SPurity:99.12%Color and Shape:SolidMolecular weight:415.51Mepyramine maleate
CAS:Mepyramine maleate is a mild hypnotic, local anesthetic, and H1 histamine antagonist for allergies and colds.Formula:C21H27N3O5Purity:99.51% - 99.7%Color and Shape:White Crystalline PowderMolecular weight:401.47Abt-288
CAS:ABT-288 is a selective and potent H3 antagonist for the treatment of mild to moderate Alzheimer's dementia.Formula:C23H24N4OPurity:98% - 98.84%Color and Shape:SolidMolecular weight:372.46Levocetirizine
CAS:Levocetirizine is a Histamine-1 Receptor Antagonist. The mechanism of action of levocetirizine is as a Histamine H1 Receptor Antagonist.Formula:C21H25ClN2O3Purity:98% - 99.9%Color and Shape:White PowderMolecular weight:388.89Cetirizine Impurity B dihydrochloride
CAS:Cetirizine Impurity B dihydrochloride is a Cetirizine antihistamine byproduct with anti-allergic properties.Formula:C19H23Cl3N2O2Purity:99.24%Color and Shape:SolidMolecular weight:417.76BMY-25271
CAS:BMY-25271 is an antagonist of histamine H2 receptor.Formula:C12H19N5O2S2Purity:98%Color and Shape:SolidMolecular weight:329.44Iodophenpropit dihydrobromide
CAS:Iodophenpropit dihydrobromide: selective histamine H3 antagonist, reversible binding, high affinity (KD: 0.32 nM).Formula:C15H20BrIN4SPurity:98%Color and Shape:SolidMolecular weight:495.22Pitolisant hydrochloride
CAS:Pitolisant hydrochloride (Ciproxidine) is a potent and selective inverse agonist of the histamine H3 receptor(Ki : 0.16 nM).Formula:C17H27Cl2NOPurity:99.26% - 99.72%Color and Shape:SolidMolecular weight:332.31Ref: TM-T7176
5mg50.00€10mg74.00€25mg124.00€50mg197.00€100mg311.00€200mg467.00€500mg747.00€1mL*10mM (DMSO)52.00€
