Histamine Receptor
Histamine receptors are GPCRs that mediate the effects of histamine, a biogenic amine involved in immune responses, gastric acid secretion, and neurotransmission. There are four subtypes of histamine receptors (H1, H2, H3, and H4), each playing distinct roles in allergic reactions, gastric function, and central nervous system activity. Histamine receptor antagonists are widely used in the treatment of allergies, peptic ulcers, and motion sickness. At CymitQuimica, we provide a comprehensive selection of high-quality histamine receptor modulators to support your research in immunology, gastroenterology, and neuropharmacology.
Products of "Histamine Receptor"
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Talastine
CAS:Talastine is an antihistamine compound that can induce an allergic rash.Formula:C19H21N3OPurity:99.30% - 99.37%Color and Shape:SolidMolecular weight:307.39Doxepin hydrochloride
CAS:Doxepin hydrochloride, a dibenzoxepin tricyclic, blocks monoamine reuptake and has anticholinergic and antihistaminic effects. Mechanism partly unknown.Formula:C19H22ClNOPurity:99.57% - 99.91%Color and Shape:White To Off-White PowderMolecular weight:315.837Psoralenoside
CAS:Psoralenoside: a compound from Psoralea fruit; has estrogenic, osteoblastic, antitumor, and antibacterial properties.Formula:C17H18O9Purity:99.03% - 99.49%Color and Shape:SolidMolecular weight:366.32Ref: TM-TN1008
1mg119.00€5mg283.00€10mg418.00€25mg687.00€50mg938.00€100mg1,264.00€1mL*10mM (DMSO)319.00€Buclizine dihydrochloride
CAS:Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic andFormula:C28H33ClN2·2HClPurity:98.05%Color and Shape:Off-White PowderMolecular weight:505.95JNJ-5207852 dihydrochloride
CAS:JNJ-5207852 dihydrochloride is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptorFormula:C20H34Cl2N2OPurity:99.51%Color and Shape:SolidMolecular weight:389.4JNJ-5207852
CAS:JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor.Formula:C20H32N2OPurity:97.19%Color and Shape:SolidMolecular weight:316.48FRG8701
CAS:FRG8701 is a new Histamine H2-receptor antagonist with an IC50 of ranging from 0.25 to 0.43 μM.Formula:C22H30N2O4SPurity:98%Color and Shape:SolidMolecular weight:418.55H3R antagonist 1
CAS:H3R-IN-1 is an effective inverse agonist of the histamine receptor 3 (H3R).Formula:C19H23N3O3Color and Shape:SolidMolecular weight:341.4Clemastine
CAS:Clemastine (Meclastin) is an antagonist of the H1 receptor and exhibits anti-inflammatory effects.Formula:C21H26ClNOPurity:99.83%Color and Shape:SolidMolecular weight:343.89Cetirizine dihydrochloride
CAS:Cetirizine dihydrochloride is a potent non-drowsy antihistamine for allergies and asthma.Formula:C21H27Cl3N2O3Purity:99.4% - 99.97%Color and Shape:SolidMolecular weight:461.81Ranitidine Hydrochloride
CAS:Ranitidine Hydrochloride (AH19065) is a competitive and reversible inhibitor of histamine H2-receptor antagonists with antacid activity.Formula:C13H23ClN4O3SPurity:99.30% - 99.49%Color and Shape:SolidMolecular weight:350.86Ebastine
CAS:Ebastine (Kestine) (trade names Evastin, Kestine, Ebastel, Aleva) is a non-sedating H1 antihistamine.Formula:C32H39NO2Purity:100% - 99.93%Color and Shape:White To Off-White PowderMolecular weight:469.66Azacyclonol
CAS:Azacyclonol (MER 17) is a drug used to diminish hallucinations in psychotic individuals.Formula:C18H21NOPurity:99.46%Color and Shape:Solid PowderMolecular weight:267.37Cyproheptadine hydrochloride sesquihydrate
CAS:Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.Formula:C21H24ClNOPurity:100% - 99.77%Color and Shape:White To Slightly Yellowish Crystalline SolidMolecular weight:341.88Alginic acid
CAS:Alginic acid, a polysaccharide from brown seaweed, has anti-anaphylactic and anti-inflammatory properties and is used in food industry.Formula:C14H22O13Purity:≥98%Color and Shape:SolidMolecular weight:398.317Fexofenadine hydrochloride
CAS:Fexofenadine Hydrochloride is a carboxylated metabolic derivative of terfenadine and long-lasting selective histamine H1 receptor antagonist, withFormula:C32H40ClNO4Purity:100%Color and Shape:White Crystalline PowderMolecular weight:538.12ReN-1869 hydrochloride
CAS:ReN 1869 hydrochloride is a novel, selective antagonist of histamine H1 receptor.Formula:C24H28ClNO2Purity:98%Color and Shape:SolidMolecular weight:397.94Azatadine dimaleate
CAS:Azatadine dimaleate (SCH10649) is an inhibitor for histamine(IC50=6.5 nM) and cholinergic(IC50=10 nM).Formula:C28H30N2O8Purity:100% - 99.70%Color and Shape:PowderMolecular weight:522.55LML134
CAS:LML134 (LML-134) is an inverse agonist of Histamine 3 receptor (H3R)(hH3R cAMP and hH3R bdg with Kis of 0.3 nM and 12 nM).Formula:C19H29N5O3Purity:99.36%Color and Shape:SolidMolecular weight:375.47Ref: TM-T8514
1mg52.00€5mg105.00€10mg170.00€25mg306.00€50mg452.00€100mg672.00€200mg905.00€1mL*10mM (DMSO)117.00€SUN 1334H
CAS:SUN 1334H is a potent, orally active, highly selective antagonist of H1 receptor(Ki of 9.7 nM).Formula:C23H28Cl2F2N2O3Purity:98%Color and Shape:SolidMolecular weight:489.38PF-03654746
CAS:PF-03654746: selective H3 antagonist, boosts cognition in Alzheimer's, may treat allergic rhinitis.Formula:C18H24F2N2OPurity:98.83% - 99.1%Color and Shape:SolidMolecular weight:322.39HTMT dimaleate
CAS:HTMT dimaleate (Histamine Trifluoromethyl Toluidide Dimaleate) is an H1 and H2 receptor agonist.Formula:C27H33F3N4O9Purity:98.51%Color and Shape:SolidMolecular weight:614.57VUF10460
CAS:VUF10460 is a non-imidazole histamine H4 receptor agonist.Formula:C15H19N5Purity:99.44% - 99.57%Color and Shape:SolidMolecular weight:269.34Antazoline hydrochloride
CAS:Antazoline hydrochloride (Phenazoline hydrochloride), a first-generation antihistamine, can bind to the histamine H1 receptor and block the action of endogenousFormula:C17H19N3·HClPurity:98% - 99.53%Color and Shape:White Or Almost White Crystalline PowderMolecular weight:301.82Imetit dihydrobromide
CAS:Imetit dihydrobromide is a high affinity and effective agonist of histamine H3 and H4 receptors (Ki: 0.3 and 2.7 nM). Imetit mimics the histamine effect in triggering a shape change in eosinophils (EC50: 25 nM).Formula:C6H12Br2N4SPurity:98%Color and Shape:SolidMolecular weight:332.06Betahistine dihydrochloride
CAS:Betahistine dihydrochloride (Betahistine 2HCl) is a histamine analog and H1 receptor agonist that serves as a vasodilator.Formula:C8H14Cl2N2Purity:99.34% - 99.88%Color and Shape:White To Light Yellow Crystalline PowderMolecular weight:209.12Diphenhydramine hydrochloride
CAS:DPH: antihistamine for cough, nausea, itching, allergy, Parkinson's, sleep aid, cold remedy.Formula:C17H22ClNOPurity:99.84%Color and Shape:Taste Ph (5% Aqueous Solution) 4-6 (Ntp 1992)Molecular weight:291.82H4 Receptor antagonist 1
CAS:H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM.Formula:C16H17ClN4OPurity:98.81%Color and Shape:SolidMolecular weight:316.79Ref: TM-T5829
2mg46.00€5mg66.00€10mg92.00€25mg177.00€50mg305.00€100mg439.00€500mg938.00€1mL*10mM (DMSO)73.00€Ciproxifan
CAS:Ciproxifan (FUB-359) is a highly effective and specific histamin H3-receptor antagonist (IC50: 9.2 nM).Formula:C16H18N2O2Purity:98.00%Color and Shape:SolidMolecular weight:270.33KSK94
CAS:KSK94 is an H3 receptor antagonist that inhibits sigma-2 receptors , with a Ki value of 75.2 nM, and can be used to study injurious pain.Formula:C25H26N4OPurity:99.56%Color and Shape:SolidMolecular weight:398.5Famotidine
CAS:Famotidine, a histamine H2-blocker, curbs gastric acid production, lowering volume and acidity.Formula:C8H15N7O2S3Purity:98.93% - 99.75%Color and Shape:White To Off-White Crystalline PowderMolecular weight:337.45Enerisant
CAS:Enerisant (TS-091) is a histamine H3 receptor antagonist that promotes pro-cognitive effects and reverses scopolamine-induced cognitive deficits.Formula:C22H30N4O3Purity:99.7%Color and Shape:SoildMolecular weight:398.50Ref: TM-T67828
1mg86.00€5mg180.00€10mg296.00€25mg627.00€50mg810.00€100mg1,140.00€200mg1,510.00€1mL*10mM (DMSO)188.00€Clemizole
CAS:Clemizole is an H1 histamine receptor antagonist, can inhibit NS4B's RNA binding and hepatitis C virus (HCV) replication.Formula:C19H20ClN3Purity:98% - 99.15%Color and Shape:SolidMolecular weight:325.84Ref: TM-T1822
1mg44.00€5mg87.00€10mg106.00€25mg160.00€50mg270.00€100mg487.00€500mg1,026.00€1mL*10mM (DMSO)87.00€Betahistine EP Impurity C
CAS:Betahistine EP Impurity C (NSC19005) is structurally related to Betahistine. Betahistine EP Impurity C is a dimer of Betahistine.Formula:C15H19N3Purity:≥95%Color and Shape:SolidMolecular weight:241.33H3R-IN-1 Hydrochloride
CAS:H3R-IN-1 Hydrochloride is an inverse agonist of histamine receptor 3( H3R ) .Formula:C19H24ClN3O3Purity:98%Color and Shape:SolidMolecular weight:377.86Nedocromil
CAS:Nedocromil (FPL 59002) inhibits the action or formation of multiple mediators. Which including histamine, leukotriene C4 (LTC4), and prostaglandin D2 (PGD2).Formula:C19H17NO7Purity:95.00%Color and Shape:SolidMolecular weight:371.34Meclizine
CAS:Meclizine, also known as Meclozine, is a piperazine class H1 antagonist with antihistamine properties that inhibits the interaction of histamine at H1 receptorsFormula:C25H27ClN2Purity:95.16%Color and Shape:SolidMolecular weight:390.95Brompheniramine maleate
CAS:Brompheniramine maleate (Dimotane) is an antagonist against histamine H1 receptors.Formula:C16H19BrN2·C4H4O4Purity:99.80%Color and Shape:Crystal PowderMolecular weight:435.31Chlorpheniramine maleate
CAS:Chlorpheniramine maleate (NCI-C55265) is a histamine H1 antagonist used in allergic reactions, hay fever, rhinitis, urticaria, and asthma.Formula:C20H23ClN2O4Purity:99.64% - 99.98%Color and Shape:Odorless White Crystalline Solid Or White Powder With A Bitter TasteMolecular weight:390.87Cinnarizine
CAS:Cinnarizine is a piperazine, blocks H1-receptor & Ca-channels, has vasodilating & antiemetic effects, may cause Parkinson-like symptoms.Formula:C26H28N2Purity:99.94%Color and Shape:SolidMolecular weight:368.51Samelisant
CAS:Samelisant (SUVN-G3031), a selective H3 inverse agonist, Ki=8.7/9.8 nM in humans/rats, has anti-narcoleptic properties.Formula:C21H31N3O3Purity:99.09%Color and Shape:SolidMolecular weight:373.49Ref: TM-T9770
1mg111.00€2mg166.00€5mg274.00€10mg439.00€25mg725.00€50mg1,017.00€100mg1,359.00€500mg2,745.00€1mL*10mM (DMSO)283.00€Fexofenadine-d6
CAS:Fexofenadine D6 is an antihistamine pharmaceutical drug.Fexofenadine D6 is deuterium labeled is Fexofenadine.Formula:C32H39NO4Purity:98%Color and Shape:SolidMolecular weight:507.69Dimaprit dihydrochloride
CAS:Dimaprit dihydrochloride: selective H2 agonist, inhibits nNOS (IC50: 49 μM), boosts gastric acid.Formula:C6H15N3S·2HClPurity:99.79%Color and Shape:SolidMolecular weight:234.19Chlorprothixene
CAS:Chlorprothixene (Truxal) is a typical antipsychotic drug of the thioxanthene class, which was the first of the series to be synthesized.Formula:C18H18ClNSPurity:98.77% - 99.69%Color and Shape:Pale Yellow Crystals SolidMolecular weight:315.86Bepotastine
CAS:Bepotastine (Bepotastine free base) free base is a histamine 1 (H1) receptor antagonis.Formula:C21H25ClN2O3Purity:99.96%Color and Shape:SolidMolecular weight:388.89Ref: TM-T7893
2mg39.00€5mg57.00€10mg87.00€25mg156.00€50mg230.00€100mg344.00€200mg512.00€1mL*10mM (DMSO)63.00€Conessine
CAS:Conessine (Conessinum), a steroidal alkaloid isolated from Holarrhena floribunda, interacts with the histamine H3 receptor and has anti-malarial activity.Formula:C24H40N2Purity:99.65%Color and Shape:SolidMolecular weight:356.59Mizolastine
CAS:Mizolastine (SL 850324), an antihistamine with IC50 of 47 nM, treats allergies like hay fever and hives.Formula:C24H25FN6OPurity:98% - 99.75%Color and Shape:SolidMolecular weight:432.49Antazoline
CAS:Antazoline has antihistamine and anticholinergic effects.It used to treat a variety of arrhythmias.Formula:C17H19N3Purity:≥95%Color and Shape:White Crystalline Powder SolidMolecular weight:265.35Mebhydrolin
CAS:Mebhydrolin (Mebhydroline) is a specific histamine H1 receptor antagonist.Formula:C19H20N2Purity:99.73% - ≥98%Color and Shape:SolidMolecular weight:276.38JNJ-39220675
CAS:JNJ-39220675, a selective histamine H3 receptor antagonist, reduces the abuse-related effects of alcohol in rats.Formula:C21H24FN3O2Purity:97.95% - 99.78%Color and Shape:SolidMolecular weight:369.43
