Histamine Receptor
Histamine receptors are GPCRs that mediate the effects of histamine, a biogenic amine involved in immune responses, gastric acid secretion, and neurotransmission. There are four subtypes of histamine receptors (H1, H2, H3, and H4), each playing distinct roles in allergic reactions, gastric function, and central nervous system activity. Histamine receptor antagonists are widely used in the treatment of allergies, peptic ulcers, and motion sickness. At CymitQuimica, we provide a comprehensive selection of high-quality histamine receptor modulators to support your research in immunology, gastroenterology, and neuropharmacology.
Products of "Histamine Receptor"
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Samelisant
CAS:Samelisant (SUVN-G3031), a selective H3 inverse agonist, Ki=8.7/9.8 nM in humans/rats, has anti-narcoleptic properties.Formula:C21H31N3O3Purity:99.09%Color and Shape:SolidMolecular weight:373.49Ref: TM-T9770
1mg111.00€2mg166.00€5mg274.00€10mg439.00€25mg725.00€50mg1,017.00€100mg1,359.00€500mg2,745.00€1mL*10mM (DMSO)283.00€Fexofenadine-d6
CAS:Fexofenadine D6 is an antihistamine pharmaceutical drug.Fexofenadine D6 is deuterium labeled is Fexofenadine.Formula:C32H39NO4Purity:98%Color and Shape:SolidMolecular weight:507.69Dimaprit dihydrochloride
CAS:Dimaprit dihydrochloride: selective H2 agonist, inhibits nNOS (IC50: 49 μM), boosts gastric acid.Formula:C6H15N3S·2HClPurity:99.79%Color and Shape:SolidMolecular weight:234.19Chlorprothixene
CAS:Chlorprothixene (Truxal) is a typical antipsychotic drug of the thioxanthene class, which was the first of the series to be synthesized.Formula:C18H18ClNSPurity:98.77% - 99.69%Color and Shape:Pale Yellow Crystals SolidMolecular weight:315.86Bepotastine
CAS:Bepotastine (Bepotastine free base) free base is a histamine 1 (H1) receptor antagonis.Formula:C21H25ClN2O3Purity:99.96%Color and Shape:SolidMolecular weight:388.89Ref: TM-T7893
2mg39.00€5mg57.00€10mg87.00€25mg156.00€50mg230.00€100mg344.00€200mg512.00€1mL*10mM (DMSO)63.00€Conessine
CAS:Conessine (Conessinum), a steroidal alkaloid isolated from Holarrhena floribunda, interacts with the histamine H3 receptor and has anti-malarial activity.Formula:C24H40N2Purity:99.65%Color and Shape:SolidMolecular weight:356.59Mizolastine
CAS:Mizolastine (SL 850324), an antihistamine with IC50 of 47 nM, treats allergies like hay fever and hives.Formula:C24H25FN6OPurity:98% - 99.75%Color and Shape:SolidMolecular weight:432.49Antazoline
CAS:Antazoline has antihistamine and anticholinergic effects.It used to treat a variety of arrhythmias.Formula:C17H19N3Purity:≥95%Color and Shape:White Crystalline Powder SolidMolecular weight:265.35Mebhydrolin
CAS:Mebhydrolin (Mebhydroline) is a specific histamine H1 receptor antagonist.Formula:C19H20N2Purity:99.73% - ≥98%Color and Shape:SolidMolecular weight:276.38JNJ-39220675
CAS:JNJ-39220675, a selective histamine H3 receptor antagonist, reduces the abuse-related effects of alcohol in rats.Formula:C21H24FN3O2Purity:97.95% - 99.78%Color and Shape:SolidMolecular weight:369.43OXOMEMAZINE
CAS:Oxomemazine: a phenothiazine antihistamine H1-blocker with strong antimuscarinic and selective M1 antagonist properties, used in cough research.Formula:C18H22N2O2SPurity:99.49%Color and Shape:SolidMolecular weight:330.44Hydroxyzine dihydrochloride
CAS:Hydroxyzine dihydrochloride treats allergies, pruritus, anxiety; causes drowsiness; also an antiemetic and sedative.Formula:C21H27ClN2O2·2HClPurity:99.46% - 99.79%Color and Shape:Oil PowderMolecular weight:447.83Lodoxamide
CAS:Lodoxamide (Lodoxamidum) is an antiallergic drug acting as a mast-cell stabilizer. It is effective in the treatment of asthma and allergic conjunctivitis.Formula:C11H6ClN3O6Purity:99.13% - 99.81%Color and Shape:SolidMolecular weight:311.63FR-145715
CAS:FR-145715 is a histamine H2 receptor antagonist characterized by its specific anti-Helicobacter pylori activity. This compound is utilized in the study of gastric lesions.Formula:C16H21N5O2SColor and Shape:SolidMolecular weight:347.44Niperotidine
CAS:Niperotidine is an antagonist of histamine H2-receptor.Formula:C20H26N4O5SPurity:98%Color and Shape:SolidMolecular weight:434.51Thonzylamine
CAS:Thonzylamine is an antihistamine/anticholinergic, combined with Clofedanol or Phenylephrine for cold, hay fever, or allergy relief.Formula:C16H22N4OPurity:99.45%Color and Shape:SolidMolecular weight:286.37Levocarnitine propionate hydrochloride
CAS:Levocarnitine propionate hydrochloride (ST-261) is used for the treatment of the deterioration of renal function, congestive heart failure, and other diseases.Formula:C10H20ClNO4Purity:90% - 98%Color and Shape:SolidMolecular weight:253.72Pemirolast potassium
CAS:Pemirolast potassium, a pyrimidinone antiallergic, blocks antigen-induced Ca²⁺ influx in mast cells.Formula:C10H7KN6OPurity:98.91% - 99.63%Color and Shape:Crystals From Dimethylformamide Crystalline SolidMolecular weight:266.31Epinastine hydrochloride
CAS:Epinastine hydrochloride (WAL-801CL HCl) is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.Formula:C16H15N3·HClPurity:99.26% - 99.62%Color and Shape:White SolidMolecular weight:285.77Levocetirizine Dihydrochloride
CAS:Levocetirizine Dihydrochloride is a third-gen antihistamine targeting H1-receptors, treating allergies and urticaria.Formula:C21H27Cl3N2O3Purity:99.75%Color and Shape:White Or Off-White Crystalline PowderMolecular weight:461.81Ref: TM-T22354
1g692.00€10mg50.00€25mg86.00€50mg131.00€100mg188.00€200mg283.00€500mg487.00€1mL*10mM (DMSO)52.00€
