LPA Receptor
Lysophosphatidic acid (LPA) receptors are a group of GPCRs that respond to LPA, a bioactive lipid involved in cell proliferation, migration, and survival. LPA signaling plays a crucial role in various physiological processes, including wound healing, vascular development, and cancer metastasis. Modulation of LPA receptor activity is being explored for therapeutic applications in cancer, fibrosis, and inflammatory diseases. At CymitQuimica, we offer a range of high-quality LPA receptor modulators to support your research in cell signaling, oncology, and inflammatory disorders.
Products of "LPA Receptor"
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H2L5186303
CAS:H2L5186303 is an LPA2 antagonist and can be used in studies about asthma treatment.Formula:C26H20N2O8Purity:97.23%Color and Shape:SolidMolecular weight:488.45Ref: TM-T22835
1mg35.00€5mg64.00€10mg104.00€25mg226.00€50mg335.00€100mg470.00€500mg938.00€1mL*10mM (DMSO)75.00€ONO-7300243
CAS:ONO-7300243 is an antagonist of lysophosphatidic acid receptor 1 (LPA1; IC50 : 0.16 μM).Formula:C28H31NO5Purity:99.66%Color and Shape:SolidMolecular weight:461.55H2L 5765834
CAS:H2L 5765834 is a lysophosphatidic acid receptors antagonistFormula:C21H12N2O7Purity:99.47% - ≥98%Color and Shape:SolidMolecular weight:404.33Ref: TM-T22834
1mg62.00€5mg119.00€10mg187.00€25mg354.00€50mg525.00€100mg747.00€1mL*10mM (DMSO)131.00€Tetradecyl Phosphonate
CAS:Tetradecyl Phosphonate 是溶血磷脂酸 1 (LPA1)、LPA2 和 LPA3 受体的泛拮抗剂。Formula:C14H31O3PPurity:99.95%Color and Shape:White To Off-White PowderMolecular weight:278.37Radioprotectin-1
CAS:Radioprotectin-1 is a selective agonist of LPA2 with EC50 of 25 nM for murine LPA2 GPCR and exerts radioprotective and radiomitigative action.Formula:C23H19ClN2O6SPurity:98.75% - 99.43%Color and Shape:SolidMolecular weight:486.92Ref: TM-T12684
1mg81.00€5mg170.00€10mg259.00€25mg425.00€50mg562.00€100mg775.00€1mL*10mM (DMSO)187.00€Ki16425
CAS:Ki16425 (Debio 0719) is a competitive, potent and reversible antagonist to LPA1, LPA2 and LPA3 with Ki of 0.34 μM, 6.5 μM and 0.93 μM, respectively.Formula:C23H23ClN2O5SPurity:97.60% - 97.78%Color and Shape:SolidMolecular weight:474.96TAK-615
CAS:TAK-615 is commonly used to study pulmonary fibrosis and is a negative allosteric modulator of LPA1 receptors.Formula:C25H22FNO4Purity:99.36%Color and Shape:SolidMolecular weight:419.44Ref: TM-T9699
1mg75.00€5mg169.00€10mg259.00€25mg429.00€50mg605.00€100mg815.00€500mg1,624.00€1mL*10mM (DMSO)180.00€LPA1 receptor antagonist 1
CAS:LPA1 receptor antagonist 1(LPA1 R antagonist 1) is a lysophosphatidic acid receptor antagonist for the study of idiopathic pulmonary fibrosis.Formula:C28H26N4O4Purity:99.46% - 99.58%Color and Shape:SolidMolecular weight:482.53ASP6432
CAS:ASP6432 is an antagonist of type 1 lysophosphatidic acid receptor (LPA1). For human LPA1 and rat LPA1, the IC50s are 11 nM and 30 nM , respectively.Formula:C26H32KN4O6S2Color and Shape:SolidMolecular weight:599.78Edg-2 receptor inhibitor 1
CAS:Edg-2 receptor inhibitor 1 (SAR-100842) is an Edg-2 receptor inhibitor extracted (IC50: <0.1 μM).Formula:C27H27NO5Purity:99.47%Color and Shape:SolidMolecular weight:445.51Ref: TM-T4521
1mg97.00€2mg170.00€5mg274.00€10mg426.00€25mg663.00€50mg947.00€100mg1,264.00€1mL*10mM (DMSO)288.00€TC LPA5 4
CAS:TC LPA5 4 is a LPA5 receptor antagonist.Formula:C23H23ClN2O3Purity:99.05%Color and Shape:SolidMolecular weight:410.89GRI977143
CAS:GRI977143: selective LPA2 agonist (EC50=3.3μM), blocks caspases 3/7/8/9, limits DNA fragmentation.Formula:C22H17NO4SPurity:98.07%Color and Shape:SolidMolecular weight:391.44AM095 free acid
CAS:AM095 (free acid) is a potent LPA1 receptor antagonist (IC50s: 0.98 and 0.73 μM for recombinant human or mouse LPA1).Formula:C27H24N2O5Purity:99.88%Color and Shape:SolidMolecular weight:456.49Ref: TM-T10293
1mg39.00€2mg51.00€5mg84.00€10mg119.00€25mg210.00€50mg354.00€100mg550.00€200mg792.00€1mL*10mM (DMSO)92.00€DBIBB
CAS:DBIBB: non-lipid LPA2 receptor agonist, treats acute radiation syndrome, aids in organic synthesis/drug research.Formula:C23H20N2O6SPurity:97.18% - 97.26%Color and Shape:SolidMolecular weight:452.48Ref: TM-T22070
1mg42.00€5mg93.00€10mg134.00€25mg264.00€50mg378.00€100mg553.00€500mg1,111.00€1mL*10mM (DMSO)93.00€BMS-986278
CAS:BMS-986278 is an orally active and potent hemophosphatidic acid receptor 1 (LPA1) antagonist with Kb values of 6.9 nM and 4.0 nM for human and mouse LPA1,Formula:C22H31N5O5Purity:99.86%Color and Shape:SolidMolecular weight:445.51Ki16198
CAS:Ki16198, a methyl ester derivative of Ki16425, blocks LPA1/3, weak on LPA2; inactive on LPA4/5/6. Ki values: 0.34 μM (LPA1), 0.93 μM (LPA3).Formula:C24H25ClN2O5SPurity:97.6%Color and Shape:SolidMolecular weight:488.98LPA2 antagonist 1
CAS:LPA2 antagonist 1 is a potent LPA2 antagonist.Formula:C20H23Cl2N5O2S2Purity:99.85%Color and Shape:SolidMolecular weight:500.47UCM-05194
CAS:UCM-05194: potent LPA1 agonist, best for neuropathic pain relief (Emax 118%, EC50 0.24 μM, KD 19.6 nM, inactive at LPA2-6/autotaxin).Formula:C19H30BrO6PPurity:90% - 91.22%Color and Shape:SolidMolecular weight:465.32AM095
CAS:AM095 is a potent LPA1 receptor antagonist with IC50 values of 0.98 and 0.73 μM for recombinant human or mouse LPA1 respectively.Formula:C27H23N2NaO5Purity:99.62%Color and Shape:SolidMolecular weight:478.47BMS-986020
CAS:BMS-986020 (AM152) is a selective antagonist of LPA1.Formula:C29H26N2O5Purity:100% - 98.82%Color and Shape:SolidMolecular weight:482.53
