Adenosine Receptor
Adenosine receptors are a class of GPCRs that respond to the endogenous nucleoside adenosine. These receptors are involved in regulating various physiological processes, including cardiovascular function, sleep-wake cycles, and immune responses. Adenosine receptor modulators have therapeutic potential in treating conditions such as cardiac arrhythmias, inflammation, and neurodegenerative diseases. At CymitQuimica, we provide a selection of high-quality adenosine receptor modulators to support your research in cardiovascular biology, neuroscience, and immunology.
Products of "Adenosine Receptor"
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MRS-3777 hemioxalate
CAS:MRS-3777 hemioxalate, a selective adenosine A3 receptor antagonist, reverses the anti-injury perception effects of its corresponding agonist and serves as a valuable tool for studying inflammatory pain.Formula:C17H19N5OC2H2O4Purity:97.10%Color and Shape:SolidMolecular weight:354.39Quercetin-3'-o-phosphate TEA
Quercetin-3'-o-phosphate TEA (Quercetin 3'-phosphate TEA) is an adenosine A receptor antagonist that can be used to prevent and treat metabolic disorders.Formula:C21H26NO10PPurity:95.50%Color and Shape:SoildMolecular weight:483.41GS-6201
CAS:GS-6201 (CVT-6883) is a selective antagonist of adenosine A2B receptor.Formula:C21H21F3N6O2Purity:98.32% - 99.74%Color and Shape:SolidMolecular weight:446.43Ref: TM-T15418
1mg38.00€5mg79.00€10mg127.00€25mg261.00€50mg423.00€100mg635.00€200mg887.00€1mL*10mM (DMSO)87.00€A2B receptor antagonist 2
CAS:A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).Formula:C12H15N5Purity:100%Color and Shape:SolidMolecular weight:229.28Inosine
CAS:Inosine (NSC-20262) is a purine nucleoside that has hypoxanthine linked by the N9 nitrogen to the C1 carbon of ribose.Formula:C10H12N4O5Purity:99.51% - 99.78%Color and Shape:SolidMolecular weight:268.23A3AR agonist 2
Compound 19, a selective A3 Adenosine Receptor (A3AR) agonist (K i : 22.1 nM), effectively stimulates β-arrestin2 recruitment with an EC 50 value of 4.36 nM.Formula:C34H34N6O6Purity:98%Color and Shape:SolidMolecular weight:622.67PSB-603
CAS:PSB-603 is a selective antagonist of Adenosine A2B receptor(Ki = 0.553 nM) with anti-inflammatory effects.Formula:C24H25ClN6O4SPurity:97.13%Color and Shape:SolidMolecular weight:529.01Ref: TM-T23203
1mg37.00€5mg97.00€10mg160.00€25mg344.00€50mg562.00€100mg938.00€200mg1,264.00€1mL*10mM (DMSO)111.00€LUF6096
CAS:LUF6096 (CF-602) is a potent allosteric enhancer of the adenosine A3 receptor, exhibiting the capability to enhance agonist binding allosterically whileFormula:C22H21Cl2N3OPurity:100%Color and Shape:SolidMolecular weight:414.33LAS38096
CAS:LAS38096 is an A2B adenosine receptor antagonist (Ki : 17 nM) that is potent, selective and efficient .Formula:C17H12N6OPurity:98.71% - 99.16%Color and Shape:SolidMolecular weight:316.32A3AR antagonist 5
CAS:A3AR antagonist 5 (Compound 16) acts as a selective antagonist for the human adenosine A3 receptor (human adenosine A3 receptor), with an affinity expressed as a pC value of 4.542 μM.Formula:C18H16N2O2SColor and Shape:SolidMolecular weight:324.40Selodenoson
CAS:Selodenoson (RG-14202) is a selective adenosine A1 receptor agonist used to slow the heart rate in patients with atrial fibrillation and to treat arrhythmias.Formula:C17H24N6O4Purity:99.33%Color and Shape:SolidMolecular weight:376.41Adenosine antagonist-1
CAS:Adenosine antagonist-1 acts as an adenosine A3 receptor (AA3R) antagonist.Formula:C18H13N7SPurity:100% - 97%Color and Shape:SolidMolecular weight:359.41A1/A3 AR antagonist 3
CAS:A1/A3 AR Antagonist 3 is a dual A1R/A3R antagonist that demonstrates high affinity within the low-micromolar to nanomolar range, and is potentially useful inFormula:C22H19N5O3Purity:98%Color and Shape:SolidMolecular weight:401.42Theobromine
CAS:Theobromine (3,7-Dimethylxanthine), a xanthine alkaloid, is used as a bronchodilator and as a vasodilator.Formula:C7H8N4O2Purity:99.63% - 99.89%Color and Shape:White To Yellow Crystalline PowderMolecular weight:180.16Theophylline
CAS:Theophylline (1,3-Dimethylxanthine) is a methyl xanthine derivative from tea with diuretic, smooth muscle relaxant, bronchial dilation, cardiac and centralFormula:C7H8N4O2Purity:99.47% - 99.97%Color and Shape:White Solid PowderMolecular weight:180.16N 0861
CAS:N 0861 is a selective adenosine A1 receptor antagonist that attenuates renal insufficiency during adenosine-controlled hypotension in rats.Formula:C13H17N5Purity:99.81%Color and Shape:SolidMolecular weight:243.31KFM19
CAS:KFM19 is a potent and selective adenosine receptor (A1-receptor) antagonist (IC50 : 50 nM) for the study of neurological disorders.Formula:C16H22N4O3Purity:99.18%Color and Shape:SolidMolecular weight:318.37Zaladenant
CAS:Zaladenant is an adenosine receptor antagonist with antitumor properties.Formula:C19H15F3N6OColor and Shape:SolidMolecular weight:400.357GR79236
CAS:GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions.Formula:C15H21N5O5Color and Shape:SolidMolecular weight:351.36CPI-444
CAS:CPI-444 (V81444) is an antagonist of the adenosine A2A receptor.It reduces tumor area in mouse model of murine Her2/neu-expressing breast cancer.Formula:C20H21N7O3Purity:98.78%Color and Shape:SolidMolecular weight:407.43ST3932
CAS:ST3932 is a ST1535 metabolite, is a adenosine A2A receptor antagonist(Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively).Formula:C12H16N8OPurity:98%Color and Shape:SolidMolecular weight:288.31A2AR-antagonist-1
CAS:Oral A2AR-antagonist-1, IC50 29 nM; anti-tumor, stable in mice (t1/2 86.1 min), boosts T cells, impedes LAG-3/TIM-3.Formula:C27H25N5O2Purity:98%Color and Shape:SolidMolecular weight:451.52Binodenoson
CAS:Binodenoson (WRC 0470), a selective A2A adenosine receptor agonist, aids in coronary imaging.Formula:C17H25N7O4Purity:99.84%Color and Shape:SolidMolecular weight:391.42Ref: TM-T9516
1mg103.00€5mg246.00€10mg369.00€25mg620.00€50mg825.00€100mg1,130.00€200mg1,549.00€1mL*10mM (DMSO)271.00€VUF 5574
CAS:VUF 5574 is a selective antagonist of adenosine A3 receptor with a Ki of 4.03 nM for the recombinant human receptor.Formula:C21H17N5O2Purity:97.63%Color and Shape:SolidMolecular weight:371.39DPTN dihydrochloride
CAS:DPTN dihydrochloride is a potent and selective A3AR antagonist with Ki values of 1.65, 9.61 and 8.53 nM in human, mouse and rat, respectively.Formula:C22H20Cl2N4OSPurity:100%Color and Shape:SoildMolecular weight:459.39PD 117519
CAS:PD 117519 (CI947) is an agonist of adenosine receptorFormula:C19H21N5O4Purity:99.98%Color and Shape:SolidMolecular weight:383.4GW-493838
CAS:GW-493838 is a potent adenosine A1A receptor agonist for the treatment of dyslipidemia and neuropathic pain, with analgesic effects on post-herpetic neuralgiaFormula:C21H21ClFN7O4Purity:99.70% - 99.76%Color and Shape:SolidMolecular weight:489.89Ref: TM-T27509
1mg152.00€5mg365.00€10mg520.00€25mg780.00€50mg1,054.00€100mg1,425.00€500mg2,793.00€1mL*10mM (DMSO)420.00€Ticlopidine hydrochloride
CAS:Ticlopidine hydrochloride (Ticlodix) is an effective inhibitor of platelet aggregation commonly used in the placement of STENTS in CORONARY ARTERIES.Formula:C14H15Cl2NSPurity:99.82% - 99.98%Color and Shape:White PowderMolecular weight:300.25ABT-702 dihydrochloride
CAS:ABT-702 dihydrochloride is a potent adenosine kinase (AK) inhibitor.Formula:C22H21BrCl2N6OPurity:98.89% - 99%Color and Shape:SolidMolecular weight:536.25Ref: TM-T4668
1mg62.00€2mg87.00€5mg119.00€10mg187.00€25mg350.00€50mg530.00€100mg748.00€500mg1,578.00€1mL*10mM (DMSO)140.00€YT 146
CAS:YT 146 is a biochemical.Formula:C18H25N5O4Purity:98.81% - 99.72%Color and Shape:SolidMolecular weight:375.42PSB 0777 ammonium hydrate
PSB 0777 ammonium hydrate is a potent and selective adenosine A2A receptor full agonist, exhibiting K i values of 44.4 nM for rat A2A receptors and 360 nM forFormula:C18H20N5O7S2·NH4·75H2OPurity:98%Color and Shape:SolidMolecular weight:532.09Aminophylline
CAS:Aminophylline (Phyllocontin) is a competitive nonselective phosphodiesterase inhibitor giving a bronchodilatory effect.Formula:C7H8O2·C2H8N2Purity:99.31%Color and Shape:White Or Slightly Yellowish Granules Or Powder SolidMolecular weight:420.43Istradefylline
CAS:Istradefylline (KW-6002)(Ki of 2.2 nM) is a selective adenosine A2A receptor (A2AR) antagonist, which is under development in Phase 3 trails.Formula:C20H24N4O4Purity:98.18% - 99.95%Color and Shape:SolidMolecular weight:384.43N6-(2-Phenylethyl)adenosine
CAS:N6-(2-Phenylethyl)adenosine (N6-Phenethyladenosine) is an adenosine derivative and an agonist of adenosine receptors with Ki values of 11.8 nM and 30.1 nM forFormula:C18H21N5O4Purity:99.94%Color and Shape:SolidMolecular weight:371.398-Cyclopentyl-1,3-dimethylxanthine
CAS:8-Cyclopentyl-1,3-dimethylxanthine (CPT) is a potent antagonist of adenosine A1 receptor.Formula:C12H16N4O2Purity:100% - 98.58%Color and Shape:SolidMolecular weight:248.28Apadenoson TFA
Apadenoson TFA is a potent adenosine A2A receptor (A2AR) agonist that can be used to improve survival in patients infected with SARS.Formula:C25H31F3N6O8Purity:98.40%Color and Shape:SoildMolecular weight:600.55Evodenoson
CAS:Evodenoson (ATL313), a potent A2aR agonist, treats eye diseases, tumors, and immune disorders; potential for glaucoma and blood cancer studies.Formula:C23H29N7O6Purity:100% - 99.74%Color and Shape:SolidMolecular weight:499.52Xanthine amine congener
CAS:Xanthine amine congener is an Adenosine receptor antagonist.Formula:C21H28N6O4Purity:99.7%Color and Shape:SolidMolecular weight:428.48CGS 21680 Hydrochloride
CAS:CGS 21680 Hydrochloride (CGS 21680 HCl)(IC50=22 nM), an adenosine receptor agonist, exhibits 140-fold potency in A2 receptor over A1 receptor.Formula:C23H29N7O6·HClPurity:96.74% - 98.81%Color and Shape:SolidMolecular weight:535.98Ref: TM-T6441
1mg40.00€2mg52.00€5mg86.00€10mg115.00€25mg226.00€50mg410.00€100mg607.00€1mL*10mM (DMSO)90.00€Trabodenoson
CAS:Trabodenoson (INO-8875) is a selective and potent adenosine A1 receptor agonist, an adenosine analog, for the study of primary open-angle glaucoma.Formula:C15H20N6O6Purity:99.94%Color and Shape:SolidMolecular weight:380.36Ref: TM-T34914
1mg131.00€2mg187.00€5mg311.00€10mg467.00€25mg747.00€50mg1,017.00€100mg1,359.00€1mL*10mM (DMSO)344.00€Tecadenoson
CAS:Tecadenoson (CVT-510) is a selective agonist of A1 adenosine receptor.Formula:C14H19N5O5Purity:98.83%Color and Shape:SolidMolecular weight:337.33Ref: TM-T17023
1mg50.00€5mg116.00€10mg178.00€25mg306.00€50mg434.00€100mg562.00€200mg743.00€1mL*10mM (DMSO)128.00€N6-Cyclopentyladenosine
CAS:N6-Cyclopentyladenosine (CPA) is a selective agonist of the adenosine A1 receptor and can be used to mimic the action of the adenosine A1 receptor, with Ki's ofFormula:C15H21N5O4Purity:99.84%Color and Shape:SolidMolecular weight:335.36Vipadenant
CAS:Vipadenant (CEB-4520)(BIIB-014) is an adenosine A2a antagonist with Ki of 1.3 nM; less potent for A1(Ki=69 nM).Formula:C16H15N7OPurity:97.25% - 97.36%Color and Shape:SolidMolecular weight:321.34Ref: TM-T2373
1mg40.00€2mg52.00€5mg87.00€10mg119.00€25mg210.00€50mg350.00€100mg522.00€500mg1,130.00€1mL*10mM (DMSO)359.00€Tozadenant
CAS:Tozadenant (SYN115) is an adenosine A2A receptor antagonist(Ki of 11.5 nM and 6 nM on human and rhesus,respectively)Formula:C19H26N4O4SPurity:98%Color and Shape:SolidMolecular weight:406.5Ref: TM-T7320
2mg38.00€5mg58.00€10mg96.00€25mg162.00€50mg273.00€100mg393.00€200mg563.00€1mL*10mM (DMSO)64.00€Doxofylline
CAS:Doxofylline (Doxophylline) is a methylxanthine derivative with the presence of a dioxolane group in position 7.Formula:C11H14N4O4Purity:99.09% - 99.98%Color and Shape:SolidMolecular weight:266.25Preladenant
CAS:Preladenant (SCH-420814) is an orally bioavailable antagonist of the adenosine A2A receptor (Ki: 1.1 nM) and has >1000-fold selectivity over all other adenosineFormula:C25H29N9O3Purity:97.32% - 98.18%Color and Shape:SolidMolecular weight:503.56APNEA
CAS:APNEA ((2R,3R,4S,5R)-2-[6-[2-(4-aminophenyl)ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol) is a non-selective agonist of adenosine A3 receptor.Formula:C18H22N6O4Purity:99.58%Color and Shape:SolidMolecular weight:386.41Amp579 TFA
Amp579 TFA is a novel adenosine A1/A2a receptor agonist that induces acute and delayed preconditioning against myocardial shock in vivo.Formula:C24H29ClF3N5O5SPurity:96.67%Color and Shape:SoildMolecular weight:592.03Derenofylline
CAS:Derenofylline is a selective and potent adenosine A(1) antagonist in vitro (Ki=1 nM)Formula:C18H20N4OPurity:98.09%Color and Shape:SolidMolecular weight:308.38Capadenoson
CAS:Capadenoson (BAY 68-4986) is a selective adenosine-A1 receptor agonist.Formula:C25H18ClN5O2S2Purity:98.85% - 99.62%Color and Shape:SolidMolecular weight:520.03
