Adenosine Receptor
Adenosine receptors are a class of GPCRs that respond to the endogenous nucleoside adenosine. These receptors are involved in regulating various physiological processes, including cardiovascular function, sleep-wake cycles, and immune responses. Adenosine receptor modulators have therapeutic potential in treating conditions such as cardiac arrhythmias, inflammation, and neurodegenerative diseases. At CymitQuimica, we provide a selection of high-quality adenosine receptor modulators to support your research in cardiovascular biology, neuroscience, and immunology.
Products of "Adenosine Receptor"
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Nitrobenzylthioinosine
CAS:Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.Formula:C17H17N5O6SPurity:98.83% - 99.69%Color and Shape:Off-White SolidMolecular weight:419.41hA3AR agonist 2
hA3AR agonist 2 is a potent activator of A3AR, with a Ki value of 3.5 nM.Formula:C11H14ClN5O2SColor and Shape:SolidMolecular weight:315.78A2AR-agonist-1
CAS:A2AR-agonist-1 targets A2A Receptor/ENT1 for neuroprotection; potent with Ki of 4.39 (A2AR), 3.47 (ENT1).Formula:C20H22N6O4Purity:99.82%Color and Shape:SolidMolecular weight:410.43Ref: TM-T10212
1mg96.00€2mg134.00€5mg188.00€10mg284.00€25mg452.00€50mg645.00€100mg867.00€500mg1,691.00€1mL*10mM (DMSO)217.00€CHEMBL241987
CAS:CHEMBL241987 targets the Adenosine receptor A3 (human)Formula:C16H11N3OPurity:99.81%Color and Shape:SolidMolecular weight:261.28Ref: TM-T8598
2mg35.00€5mg50.00€10mg66.00€25mg108.00€50mg162.00€100mg235.00€200mg349.00€1mL*10mM (DMSO)50.00€ZM241385
CAS:ZM-241385 is a high-affinity antagonist ligand selective for the adenosine A2A receptor.Formula:C16H15N7O2Purity:95.28% - 99.69%Color and Shape:SolidMolecular weight:337.34Ref: TM-T7021
5mg57.00€10mg82.00€25mg133.00€50mg233.00€100mg432.00€200mg652.00€500mg1,026.00€1mL*10mM (DMSO)57.00€Tonapofylline
CAS:Tonapofylline, orally active, selectively blocks A1 adenosine receptor (Ki: 7.4 nM), used in heart failure research.Formula:C22H32N4O4Purity:99.52%Color and Shape:SolidMolecular weight:416.51Namodenoson
CAS:Namodenoson (2-Cl-IB-MECA) is an adenosine A3 receptor agonist.Formula:C18H18ClIN6O4Purity:98.97%Color and Shape:SolidMolecular weight:544.73ATL444
CAS:ATL444 is an adenosine receptor antagonist with affinity (Ki values) for rA1AR, rA2AAR, rA2BAR, and rA3AR of 7.0, 2.5, 61.8, and >1000 nM, respectively.Formula:C17H19N5OColor and Shape:SolidMolecular weight:309.37SCH442416
CAS:SCH442416: selective A2A adenosine receptor antagonist; Ki: 0.048 nM (human), 0.5 nM (rat).Formula:C20H19N7O2Purity:99.58%Color and Shape:SolidMolecular weight:389.41Ref: TM-T23336
1mg48.00€2mg63.00€5mg93.00€10mg139.00€25mg281.00€50mg449.00€100mg658.00€1mL*10mM (DMSO)97.00€FSCPX
CAS:FSCPX is a potent and selective irreversible antagonist of the A1 adenosine receptor (A1AR), exhibiting low nanomolar binding potency.Formula:C23H27FN4O6SPurity:98.00%Color and Shape:SolidMolecular weight:506.55Ref: TM-T39039
1mg111.00€5mg273.00€10mg409.00€25mg695.00€50mg929.00€100mg1,244.00€200mg1,681.00€1mL*10mM (DMSO)116.00€AZD4635
CAS:AZD4635 (HTL1071) is a new-type adenosine 2A receptor (A2AR) inhibitor(Ki=1.7 nM).Formula:C15H11ClFN5Purity:99.15% - 99.90%Color and Shape:SolidMolecular weight:315.73Ref: TM-T4265
1mg37.00€2mg52.00€5mg79.00€10mg116.00€25mg188.00€50mg296.00€100mg457.00€500mg1,008.00€1mL*10mM (DMSO)87.00€BAY-545
CAS:BAY-545 is an antagonist of A2B adenosine receptor(IC50 : 59 nM).Formula:C18H22F3N3O4SPurity:98.05%Color and Shape:SolidMolecular weight:433.45Ref: TM-T8512
1mg88.00€5mg170.00€10mg248.00€25mg444.00€50mg638.00€100mg889.00€200mg1,198.00€1mL*10mM (DMSO)182.00€Kira8 Hydrochloride
CAS:Kira8 Hydrochloride is a mono-selective IRE1α inhibitor that allosterically attenuates IRE1α RNase activity with an IC50 of 5.9 nM.Formula:C31H30Cl2N6O3SPurity:98%Color and Shape:SolidMolecular weight:637.58A2A receptor antagonist 1
CAS:A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.Formula:C16H12FN5OPurity:99.29% - 99.76%Color and Shape:SolidMolecular weight:309.3Ref: TM-T37792
1mg37.00€5mg64.00€10mg92.00€25mg185.00€50mg284.00€100mg419.00€500mg883.00€1mL*10mM (DMSO)47.00€Norisoboldine
CAS:Norisoboldine, potential rheumatoid arthritis therapy, protects joints and modulates immunity by inhibiting MAPKs, not NF-κB.Formula:C18H19NO4Purity:98.12%Color and Shape:SolidMolecular weight:313.35Adenosine amine congener
CAS:Adenosine amine congener (ADAC) (ADAC) is an agonist of selective A1 adenosine receptor,.Formula:C28H32N8O6Purity:97.86%Color and Shape:SolidMolecular weight:576.6Theophylline monohydrate
CAS:Theophylline monohydrate (Quibron) appears to inhibit phosphodiesterase and prostaglandin production, regulate calcium flux and intracellular calciumFormula:C7H8N4O2·H2OPurity:99.78%Color and Shape:SolidMolecular weight:198.18Nelonicline
CAS:Nelonicline is a selective agonist of neuronal nicotinic receptors.Formula:C17H19N3OSPurity:98%Color and Shape:SolidMolecular weight:313.42Alloxazine
CAS:Alloxazine (Isoalloxazine) is an A2 receptor antagonist, which is approximately 10-fold more selective for the A2B receptor than for the A2A receptor.Formula:C10H6N4O2Purity:99.75%Color and Shape:SolidMolecular weight:214.18N6-Cyclohexyladenosine
CAS:N6-Cyclohexyladenosine (CHA) is a selective agonist of A1 receptor with EC50 of 8.2 Nm.Formula:C16H23N5O4Purity:99.84% - 99.98%Color and Shape:SolidMolecular weight:349.38Xanthine amine congener trihydrochloride
CAS:Xanthine amine congener trihydrochloride: potent adenosine antagonist, reverses effects of N6-cyclohexyladenosine on urine, sodium excretion, heart rate.Formula:C21H29ClN6O4Purity:97.85%Color and Shape:SolidMolecular weight:464.95CCPA
CAS:CCPA (2-chloro-N(6)cyclopentyladenosine) is a potent and selective agonist of adenosine A1 receptorFormula:C15H20ClN5O4Purity:99.10%Color and Shape:Off-White To Light Yellow SolidMolecular weight:369.8PF-02575799
CAS:PF-02575799 is an inhibitor of microsomal triglyceride transfer protein (MTP) (IC50: 0.77±0.29 nM).Formula:C42H37FN4O4Purity:98%Color and Shape:SolidMolecular weight:680.77Piclidenoson
CAS:Piclidenoson (CF-101), a selective agonist of adenosine A3 receptor(EC50 values of 0.11 μM), induces robust anti-inflammatory effect in psoriasis patients.Formula:C18H19IN6O4Purity:100% - ≥95%Color and Shape:SolidMolecular weight:510.29Ref: TM-T7188
2mg42.00€5mg62.00€10mg89.00€25mg183.00€50mg298.00€100mg464.00€200mg663.00€1mL*10mM (DMSO)70.00€ANR 94
CAS:ANR94 is a potent hAA2AR antagonist (Ki 46 nM) with potential for Parkinson's research.Formula:C9H13N5OPurity:98.21%Color and Shape:SolidMolecular weight:207.23Ref: TM-T22031
2mg42.00€5mg64.00€10mg97.00€25mg188.00€50mg329.00€100mg465.00€200mg655.00€1mL*10mM (DMSO)63.00€CGS 15943
CAS:CGS 15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor.Formula:C13H8ClN5OPurity:99.63%Color and Shape:SolidMolecular weight:285.695-Iodotubercidin
CAS:5-Iodotubercidin (NSC-113939) is a potent adenosine kinase inhibitor with IC50 of 26 nM.Formula:C11H13IN4O4Purity:99.98%Color and Shape:Tan SolidMolecular weight:392.15Ref: TM-T6745
1mg46.00€2mg57.00€5mg92.00€10mg155.00€25mg343.00€50mg509.00€100mg735.00€1mL*10mM (DMSO)97.00€Regadenoson
CAS:Regadenoson (CVT-3146) is a selective A2A receptor agonist that increases coronary blood flow with a longer half-life than adenosine.Formula:C15H18N8O5Purity:99.57% - 99.81%Color and Shape:Off-White SolidMolecular weight:390.35Ref: TM-T2671
2mg47.00€5mg65.00€10mg92.00€25mg173.00€50mg273.00€100mg416.00€500mg935.00€1mL*10mM (DMSO)72.00€MIPS521
CAS:MIPS521 ({2-Amino-4-[3,5-bis(trifluoromethyl)phenyl]thiophen-3-yl}(4-chlorophenyl)methanone) is a positive allosteric modulator of the A1R.Formula:C19H10ClF6NOSPurity:99.76%Color and Shape:SolidMolecular weight:449.8Ref: TM-T9330
1mg38.00€2mg49.00€5mg79.00€10mg111.00€25mg188.00€50mg329.00€100mg512.00€1mL*10mM (DMSO)87.00€PSB 1115
CAS:PSB 1115 is an A2B receptor antagonist and can counteract the inhibitory effect of NECA.Formula:C14H14N4O5SPurity:100% - 99.24%Color and Shape:SolidMolecular weight:350.351-Ethyl-6-aminouracil
CAS:1-Ethyl-6-aminouracil (6-AMINO-1-ETHYL-1H-PYRIMIDINE-2,4-DIONE) is an intermediate in the synthesis of a series of new substituted Xanthines which have highFormula:C6H9N3O2Purity:99.29%Color and Shape:SolidMolecular weight:155.15A2B receptor antagonist 1
CAS:A2B receptor antagonist 1 (EXAMPLE 9B) is a potent A2B adenosine receptor antagonist.Formula:C21H24N6O2Purity:98.83%Color and Shape:SolidMolecular weight:392.45Ref: TM-T10058
1mg369.00€5mg735.00€10mg938.00€25mg1,473.00€50mg1,882.00€100mg2,670.00€1mL*10mM (DMSO)843.00€ISAM-140
CAS:ISAM-140 is a potent and highly selective antagonist of A2B adenosine receptor.Formula:C19H19N3O3Purity:97.41%Color and Shape:SolidMolecular weight:337.37N-[(4-Aminophenyl)methyl]adenosine
CAS:N-[(4-Aminophenyl)methyl]adenosine is an adenosine receptor inhibitor (Ki: 29 nM for Rat ecto-5′-Nucleotidase).Formula:C17H20N6O4Purity:98.75%Color and Shape:SolidMolecular weight:372.38Ref: TM-T16166
1mg92.00€5mg188.00€10mg283.00€25mg558.00€50mg885.00€100mg1,415.00€1mL*10mM (DMSO)240.00€FK-453
CAS:FK-453 is a potent antagonist of non-xanthine adenosine A1 receptor with diuretic and renal vasodilatory activity.Formula:C23H25N3O2Purity:99.69%Color and Shape:SolidMolecular weight:375.46Enprofylline
CAS:Enprofylline (Enprofilina), a bronchodilator, acts primarily as a competitive nonselective phosphodiesterase inhibitor.Formula:C8H10N4O2Purity:98.37%Color and Shape:SolidMolecular weight:194.19Ref: TM-T21389
2mg44.00€5mg65.00€10mg93.00€25mg149.00€50mg226.00€100mg335.00€200mg465.00€1mL*10mM (DMSO)63.00€5'-N-Ethylcarboxamidoadenosine
CAS:NECA, an adenosine receptor agonist, boosts brain extravasation of fluorescein and dextran without affecting the blood-brain barrier.Formula:C12H16N6O4Purity:≥95%Color and Shape:PowderMolecular weight:308.29Proxyphylline
CAS:Proxyphylline (7-(2-Hydroxypropyl)theophylline) is a dual of adenosine A1/A2a receptor inhibitor and phosphodiesterase (PDE) inhibitor.Formula:C10H14N4O3Purity:99.48%Color and Shape:SolidMolecular weight:238.24GS-9667
CAS:GS-9667, a selective and partial agonist of the A(1) adenosine receptor (AR), represents an effective therapy for Type 2 diabetes (T2DM) and dyslipidemia viaFormula:C21H24FN5O4SPurity:99.76% - 99.76%Color and Shape:SolidMolecular weight:461.51Adenosine A1 receptor activator T62
CAS:Adenosine A1 receptor activator T62 is an allosteric enhancer of adenosine A1 receptor, and it produces antinociception in animal models of acute pain and alsoFormula:C15H14ClNOSPurity:97.83%Color and Shape:SolidMolecular weight:291.8Ref: TM-T14127
1mg87.00€5mg183.00€10mg273.00€25mg439.00€50mg598.00€100mg810.00€200mg1,074.00€1mL*10mM (DMSO)280.00€Adenosine 5'-monophosphate monohydrate
CAS:Adenosine 5'-monophosphate monohydrate (5'-AMP) , also known as 5'-adenylic acid, is a nucleotide that is used as a monomer in RNA.Formula:C10H14N5O7P·H2OPurity:97.68% - 98.49%Color and Shape:White PowderMolecular weight:365.248-Chloro caffeine
CAS:8-Chloro caffeine binds to adenosine receptors with a Ki of 30 µM. It enhances UV-induced chromosomal aberrations in the Cl-I type Chinese hamster embryo lung cells. 8-Chloro caffeine is a derivative of the methylxanthine alkaloid caffeine.Formula:C8H9ClN4O2Color and Shape:SolidMolecular weight:228.64ST-1535
CAS:ST 1535: potent, oral A2A adenosine receptor antagonist with antiparkinsonian and antitremor effects, promising for Parkinson's research.Formula:C12H16N8Purity:99.64% - 99.71%Color and Shape:SolidMolecular weight:272.31SDZ WAG 994
CAS:SDZ WAG 994 is an A1 adenosine receptor agonist.Formula:C17H25N5O4Purity:99.82%Color and Shape:SolidMolecular weight:363.41Ref: TM-T23347
1mg66.00€5mg120.00€10mg175.00€25mg316.00€50mg455.00€100mg620.00€200mg835.00€1mL*10mM (DMSO)127.00€2-Chloroadenosine
CAS:2-Chloroadenosine (CADO) is a metabolically stable analog of adenosine that binds to adenosine A1, A2A, and A3 receptors( Ki:300, 80, and 1,900 nM, respectivelyFormula:C10H12ClN5O4Purity:99.23%Color and Shape:White PowderMolecular weight:301.69Adenosine receptor antagonist 4
CAS:Adenosine receptor antagonist 4 is an adenosine receptor antagonist.Formula:C10H13N3Purity:98.59% - 99.58%Color and Shape:Off-White PowderMolecular weight:175.23Adenosine receptor agonist 1
Compound 6m, an A3 adenosine receptor (AR) partial agonist, exhibits a K i value of 6.7 nM as an adenosine receptor agonist.Formula:C12H14ClN5O2SeColor and Shape:SolidMolecular weight:374.68AB928
CAS:AB928 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. It has immunomodulatory activity[1].Formula:C23H22N8OPurity:100% - 98.55%Color and Shape:SolidMolecular weight:426.47Ref: TM-T14078
1mg50.00€5mg124.00€10mg197.00€25mg389.00€50mg462.00€100mg663.00€1mL*10mM (DMSO)134.00€DPCPX
CAS:DPCPX (PD 116948) is an A1 adenosine receptor antagonistFormula:C16H24N4O2Purity:99.23% - 99.93%Color and Shape:White SolidMolecular weight:304.39MRS-1706
CAS:MRS-1706: Ki of 1.39nM for A2B; selective inverse agonist; also affects A2A, A1, A3.Formula:C27H29N5O5Purity:97.95%Color and Shape:SolidMolecular weight:503.55Ref: TM-T16136
1mg37.00€2mg52.00€5mg79.00€10mg119.00€25mg240.00€50mg472.00€100mg687.00€1mL*10mM (DMSO)88.00€
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