Cannabinoid Receptor
Cannabinoid receptors are GPCRs that mediate the effects of endogenous cannabinoids (endocannabinoids) and phytocannabinoids, such as those found in cannabis. The two main types of cannabinoid receptors, CB1 and CB2, are involved in regulating a wide range of physiological processes, including pain perception, appetite, mood, and immune function. Cannabinoid receptor modulators have therapeutic potential in treating conditions such as chronic pain, epilepsy, and multiple sclerosis. At CymitQuimica, we offer a wide range of high-quality cannabinoid receptor modulators to support your research in neuropharmacology, pain management, and immunology.
Products of "Cannabinoid Receptor"
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OMDM-5
CAS:OMDM-5 is a potent vanilloid receptor type 1 (TRPV1, EC50 = 75 nM) agonist, showing weak ligand activity at cannabinoid type 1 receptor (CB1, Ki=4.9 μM).Formula:C26H44N2O3Purity:99.72%Color and Shape:SolidMolecular weight:432.64Ref: TM-T12306
1mg87.00€5mg187.00€10mg284.00€25mg452.00€50mg645.00€100mg867.00€200mg1,130.00€1mL*10mM (DMSO)221.00€A-836339
CAS:A-836339: Potent cannabinoid, CB2-focused (Ki=0.64nM), lesser CB1 affinity (Ki=270nM); analgesic, anti-inflammatory in mice.Formula:C16H26N2O2SPurity:99.94%Color and Shape:SolidMolecular weight:310.45Ref: TM-T7375
2mg48.00€5mg92.00€10mg164.00€25mg266.00€50mg393.00€100mg557.00€200mg753.00€1mL*10mM (DMSO)94.00€CB2R agonist 3
CB2R agonist 3, a potent activator of cannabinoid receptor 2 (CB2R), exhibits an EC50 value of 0.37μM, indicative of its significant role in the immune system [Purity:98%Color and Shape:Odour SolidN-Arachidonyldopamine
CAS:N-Arachidonyldopamine (NADA) is a selective and potent endogenous CB1 receptor agonist (Ki: 250 nM).N-Arachidonyldopamine is also a potent and selective TRPV1Formula:C28H41NO3Purity:97.65%Color and Shape:SolidMolecular weight:439.63BML-190
CAS:BML-190 (Indomethacin morpholinylamide) 是一种 CB2 受体的配体,其对 CB2 受体 (Ki:435 nM) 和 CB1受体 (Ki> 2 μM)。Formula:C23H23ClN2O4Purity:97.70%Color and Shape:SolidMolecular weight:426.89CB1 antagonist 2
CAS:CB1 antagonist 2 (AM4113) is caimabinoid 1 (CB1) antagonist which inhibits CB1 in vivo with an IC50 of 25.5 nM.Formula:C17H12Cl3N3OPurity:99.75%Color and Shape:SolidMolecular weight:380.66Δ8-THC-C8
CAS:Δ8-THC-C8 is a semi-synthetic cannabinoid. It acts as an agonist for the cannabinoid receptor 1 (CB1) with an EC50 value of 13.8 nM.Formula:C24H36O2Color and Shape:SolidMolecular weight:356.54AM841
CAS:AM841, a high-affinity electrophilic ligand, covalently interacts with a cysteine residue in helix six, thus activating the CB1 cannabinoid receptor.Formula:C26H39NO3SPurity:98%Color and Shape:SolidMolecular weight:445.66CB2 receptor agonist 9
CAS:CB2 receptor agonist 9 (Compound 33) is an orally active agonist of cannabinoid receptor 2 (CB2 receptor) with an EC50 of 16.2 nM. It inhibits the expression of TNF-α, IL-1β, and IL-6, demonstrating anti-inflammatory activity in a DSS-induced acute colitis model in mice.Formula:C16H23N3O2SColor and Shape:SolidMolecular weight:321.44CB2R/FAAH modulator-1
CAS:CB2R/FAAH modulator-1: agonizes CB2R, inhibits FAAH (IC50=4 μM), alters cytokine production; used in inflammation research. Ki: CB2R=14.8 nM, CB1R=241.3 nM.Formula:C24H27NO2Purity:100%Color and Shape:SoildMolecular weight:361.48Ref: TM-T67896
1mg77.00€5mg158.00€10mg225.00€25mg338.00€50mg472.00€100mg645.00€200mg868.00€1mL*10mM (DMSO)163.00€CB2 modulator 1
CAS:CB2 modulator 1 is a potent CB2 modulator. It can be used for the research for immune disorders, osteoporosis, inflammation, renal ischemia.Formula:C18H19F3N4O2Purity:99.02%Color and Shape:SolidMolecular weight:380.36Ref: TM-T10696
1mg35.00€5mg56.00€10mg79.00€25mg114.00€50mg167.00€100mgTo inquire1mL*10mM (DMSO)64.00€Evofolin B
CAS:Evofolin B is a natural compound isolated from the stem bark of Zanthoxylum ailanthoides.Formula:C17H18O6Purity:98%Color and Shape:SolidMolecular weight:318.32JHU 75528
CAS:JHU 75528 (JHU-75528) is a novel PET tracer with inhibitory effects on CB that can be used to study the cannabinoid system in schizophrenic patients.Formula:C23H21Cl2N5O2Purity:99.97%Color and Shape:SolidMolecular weight:470.35CB2R/FAAH modulator-3
CAS:CB2R/FAAH modulator-3 (compound 27) is a modulator targeting at CB2R and FAAH.Formula:C22H31NO2Purity:99.02%Color and Shape:SoildMolecular weight:341.49Ref: TM-T67747
2mg38.00€5mg58.00€10mg90.00€25mg164.00€50mg259.00€100mg383.00€200mg545.00€1mL*10mM (DMSO)64.00€AM251
CAS:AM251: potent CB1 blocker (IC50: 8 nM), 306x CB2 selective; GPR55 activator (EC50: 39 nM).Formula:C22H21Cl2IN4OPurity:97.38% - 97.88%Color and Shape:A Crystalline SolidMolecular weight:555.24Pregnenolone acetate
CAS:Pregnenolone acetate inhibits CB1 receptors, blocking THC effects and shielding the brain from cannabis intoxication.Formula:C23H34O3Purity:99.66%Color and Shape:White To Light Yellow Crystalline PowderMolecular weight:358.51Rimonabant
CAS:Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.Formula:C22H21Cl3N4OPurity:98% - 99.91%Color and Shape:White Or Almost White Crystalline PowderMolecular weight:463.79GW 833972A
CAS:GW 833972A: selective CB2 agonist; reduces neural depolarization and citric acid cough in animals.Formula:C18H14Cl2F3N5OPurity:99.93%Color and Shape:SoildMolecular weight:444.24ML-193
CAS:ML-193: GPR55 antagonist, IC50 221nM, 27x selective over GPR35/CB1/CB2, may aid Parkinson's symptoms.Formula:C28H25N5O4SPurity:97.74%Color and Shape:SolidMolecular weight:527.59AM-2232
CAS:AM-2232 (UNII-40KCH8YIKP) is a potent and unselective agonist of the cannabinoid receptors.Formula:C24H20N2OPurity:99.37%Color and Shape:SolidMolecular weight:352.43
