Cannabinoid Receptor
Cannabinoid receptors are GPCRs that mediate the effects of endogenous cannabinoids (endocannabinoids) and phytocannabinoids, such as those found in cannabis. The two main types of cannabinoid receptors, CB1 and CB2, are involved in regulating a wide range of physiological processes, including pain perception, appetite, mood, and immune function. Cannabinoid receptor modulators have therapeutic potential in treating conditions such as chronic pain, epilepsy, and multiple sclerosis. At CymitQuimica, we offer a wide range of high-quality cannabinoid receptor modulators to support your research in neuropharmacology, pain management, and immunology.
Products of "Cannabinoid Receptor"
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Taranabant racemate
CAS:Taranabant racemate is an antagonist and/or inverse agonist of the Cannabinoid-1 (CB1) receptor.Formula:C27H25ClF3N3O2Purity:98%Color and Shape:SolidMolecular weight:515.95AM404
CAS:AM404 is a cannabinoid reuptake inhibitor and a TRPV (1) activator with neuroprotective and anticancer activities that blocks anandamide transport.Formula:C26H37NO2Color and Shape:SolidMolecular weight:395.58Δ8-THC methyl ether
CAS:Δ8-THC methyl ether (compound 3) demonstrates a strong docking score of -10.167 kcal/mol for the CB2 receptor. Additionally, Δ8-THC methyl ether exhibits antinociceptive activity in mice.Formula:C22H32O2Color and Shape:SolidMolecular weight:328.49AEF0117
CAS:AEF0117 is a signaling inhibitor of CB1-SSi that inhibits cannabinoid self-administration and can be used to study cannabis withdrawal.Formula:C29H40O3Purity:99.58%Color and Shape:SolidMolecular weight:436.63AZD1940
CAS:AZD1940 (UNII-0J0035E9FT) is a high affinity CB(1)/CB(2) receptor agonist of the cannabinoid with oral activity. Application in the study of orofacial pain.Formula:C20H29F2N3O2SPurity:99.43%Color and Shape:SolidMolecular weight:413.52Ref: TM-T30252
1mg130.00€5mg311.00€10mg535.00€25mg847.00€50mg1,169.00€100mg1,586.00€1mL*10mM (DMSO)344.00€SR144528
CAS:SR144528 is an antagonist of the CB2 receptor (Ki = 0.6 nM) and inhibits microsomal ACAT activity (IC50 = 3.6 μM).Formula:C29H34ClN3OPurity:99.6%Color and Shape:SolidMolecular weight:476.05CID 16020046
CAS:CID 16020046 (C390-0219) is a selective GPR55 antagonist, inhibiting GPR55 constitutive activity with IC50 of 0.15 μM in yeast.Formula:C25H19N3O4Purity:99.03%Color and Shape:SolidMolecular weight:425.446-Iodopravadoline
CAS:6-Iodopravadoline (AM630) is an antagonist of CB2 (Ki: 31.2 nM). And it shows 165-fold selectivity more than CB1 receptors.Formula:C23H25IN2O3Purity:99.29%Color and Shape:Off-White SolidMolecular weight:504.36Ref: TM-T14204
1mg40.00€2mg50.00€5mg73.00€10mg96.00€25mg210.00€50mg344.00€100mg550.00€1mL*10mM (DMSO)104.00€JD-5037
CAS:JD-5037 is a novel, peripherally restricted CB1R antagonist with an IC50 of 1.5 nM.Formula:C27H27Cl2N5O3SPurity:98.14% - 98.87%Color and Shape:SolidMolecular weight:572.51Ref: TM-T4453
1mg44.00€2mg58.00€5mg95.00€10mg140.00€25mg246.00€50mg369.00€100mg550.00€1mL*10mM (DMSO)106.00€Tedalinab
CAS:Tedalinab is an effective and selective cannabinoid receptor 2 agonist.Formula:C19H21F2N3OPurity:98%Color and Shape:SolidMolecular weight:345.39GP 1a
CAS:GP 1a: potent CB2 receptor agonist (EC50=7.1), 30x CB2 over CB1 preference, boosts P-ERK1/2, aids skin healing, anti-inflammatory.Formula:C23H22Cl2N4OPurity:99.44%Color and Shape:SolidMolecular weight:441.35COR659
CAS:COR659: suppresses alcohol/chocolate intake in rats; enhances GABAB receptor, blocks CB1 receptor.Formula:C16H16ClNO3SPurity:99.56%Color and Shape:SolidMolecular weight:337.82Ref: TM-T36520
1mg52.00€2mg75.00€5mg116.00€10mg178.00€25mg324.00€50mg452.00€100mg620.00€200mg843.00€1mL*10mM (DMSO)128.00€JTE-907
CAS:JTE-907 是一种具有高度选择性和口服活性的 CB2 受体反向激动剂。JTE-907在体内展现出抗炎活性。Formula:C24H26N2O6Purity:100%Color and Shape:SolidMolecular weight:438.47Ref: TM-T19705
1mg56.00€5mg126.00€10mg187.00€25mg329.00€50mg490.00€100mg700.00€1mL*10mM (DMSO)150.00€2-Arachidonoylglycerol
CAS:In the central nervous system, 2-Arachidonoylglycerol is a second endogenous cannabinoid ligandFormula:C23H38O4Purity:95%Color and Shape:LiquidMolecular weight:378.55CB2 PET Radioligand 1
CB2 PET Radioligand 1 (compound [18F]9) is a positron emission tomography (PET) radioligand with high affinity for the human cannabinoid receptor 2 (hCB2, Ki=7.Formula:C20H19F3N4OPurity:98%Color and Shape:SolidMolecular weight:388.39Rimonabant hydrochloride
CAS:Rimonabant hydrochloride (SR 141716A) 是中心大麻素受体 1 的高效选择性反向激动剂, Ki 值为1.8 nM。它也能够抑制分枝杆菌膜蛋白3。Formula:C22H22Cl4N4OPurity:100% - 99.5%Color and Shape:Off-White To White Crystalline PowderMolecular weight:500.25CB1 antagonist 4
CAS:TM38837 is an antagonist of cannabinoid receptor type 1 (CB1), with potential for the treatment of obesity and type 2 diabetes.Formula:C30H25Cl2F3N4OSPurity:100%Color and Shape:SolidMolecular weight:617.51
