Cannabinoid Receptor
Cannabinoid receptors are GPCRs that mediate the effects of endogenous cannabinoids (endocannabinoids) and phytocannabinoids, such as those found in cannabis. The two main types of cannabinoid receptors, CB1 and CB2, are involved in regulating a wide range of physiological processes, including pain perception, appetite, mood, and immune function. Cannabinoid receptor modulators have therapeutic potential in treating conditions such as chronic pain, epilepsy, and multiple sclerosis. At CymitQuimica, we offer a wide range of high-quality cannabinoid receptor modulators to support your research in neuropharmacology, pain management, and immunology.
Products of "Cannabinoid Receptor"
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LY2828360
CAS:LY2828360: CB2 agonist, Ki=40.3 nM; biases CB2 over CB1 with EC50s of 20.1 nM and >100 μM.Formula:C22H27ClN6OPurity:98.45% - 99.51%Color and Shape:SolidMolecular weight:426.94FDU-PB-22
CAS:FDU-PB-22, a novel synthetic cannabinoid, undergoes rapid metabolism in human liver microsomes (HLM) with a half-life of 12.4 minutes.Formula:C26H18FNO2Color and Shape:SolidMolecular weight:395.43CB1 antagonist 1
CAS:CB1 antagonist 1 is a CB1 receptor antagonist, used in the research of obesity and metabolic syndrome, neuroinflammatory disorders, cognitive disorders, andFormula:C26H22Cl2N4Purity:98%Color and Shape:SolidMolecular weight:461.39APP-FUBINACA
CAS:APP-FUBINACA is a cannabinoid receptor agonist, classified as a phenylalanine amide-based indazole-3-carboxamide derivative. It exhibits neurostimulatory effects.Formula:C24H21FN4O2Color and Shape:SolidMolecular weight:416.45MJ 15
CAS:MJ 15 is a CB1 receptor antagonist with specificity for the study of obesity-induced diseases.Formula:C23H17Cl3N4OPurity:99.63%Color and Shape:SolidMolecular weight:471.77Afubiata
CAS:ADB-FUBIATA is a synthetic cannabinoid studied for its metabolic profile, along with AFUBIATA, CH-FUBIATA, and CH-PIATA. This in vitro analysis by Watanabe S, et al., examines these compounds, as published in "Arch Toxicol," 2023 Dec;97(12):3085-3094.Formula:C27H29FN2OColor and Shape:SolidMolecular weight:416.53AM281
CAS:AM 281, a cannabinoid antagonist, reduces neurologic dysfunction and mortality rate after cecal ligation and puncture in rats.Formula:C21H19Cl2IN4O2Purity:100% - 99.2%Color and Shape:White To Off-White SolidMolecular weight:557.21Ref: TM-T2264
1mg85.00€5mg172.00€10mg274.00€25mg552.00€50mg792.00€100mg1,093.00€500mg2,175.00€1mL*10mM (DMSO)245.00€PSB-SB-487
CAS:PSB-SB-487 is antagonist of GPR55.Formula:C26H32O4Purity:98.53%Color and Shape:SolidMolecular weight:408.53Ref: TM-T8975
1mg38.00€5mg85.00€10mg126.00€25mg245.00€50mg364.00€100mg507.00€200mg697.00€1mL*10mM (DMSO)93.00€MDA7
CAS:MDA7 is a selective agonist of the cannabinoid receptor 2 (CB2), demonstrating an EC50 of 128 nM in human CB2 receptors and 67.4 nM in rat CB2 receptors. The compound exhibits good affinity for CB2 receptors, with Ki values of 422 nM for humans and 238 nM for rats. In rat models, MDA7 shows analgesic activity.Formula:C22H25NO2Color and Shape:SolidMolecular weight:335.439Drinabant
CAS:Drinabant (AVE-1625) is an orally active CB1 receptor antagonist.Formula:C23H20Cl2F2N2O2SPurity:99.8%Color and Shape:SolidMolecular weight:497.38Ref: TM-T21861
1mg87.00€2mg116.00€5mg170.00€10mg259.00€25mg425.00€50mg598.00€100mg810.00€500mg1,624.00€AM6545
CAS:AM6545 is a CB1 receptor antagonist used in the study of obesity and diabetes.Formula:C26H23Cl2N5O3SPurity:97.03%Color and Shape:SolidMolecular weight:556.46PSNCBAM-1
CAS:PSNCBAM-1 (PSNCBAM 1) is a CB1 receptor negative allosteric modulator (EC50 = 0.1 μM) with hypophagic effects in vivo.Formula:C22H21ClN4OPurity:98.18%Color and Shape:SolidMolecular weight:392.88L-α-lysophosphatidylinositol sodium
CAS:L-α-lysophosphatidylinositol sodium is an endogenous ligand of GPR55 and an endocannabinoid neurotransmitter.Formula:C25H48NaO12PColor and Shape:SolidMolecular weight:594.6Falcarinol
CAS:Falcarinol, also known as Panaxynol, is a naturally occurring compound that acts as an orally active inhibitor of Hsp90.Formula:C17H24OPurity:98%Color and Shape:SolidMolecular weight:244.37AM1241
CAS:AM-1241 is a selective cannabinoid CB2 receptor agonist with Ki of 3.4 nM, exhibits 82-fold selectivity over CB1 receptor.Formula:C22H22IN3O3Purity:98.82% - 99.10%Color and Shape:SolidMolecular weight:503.33Ref: TM-T6755
2mg38.00€5mg51.00€10mg88.00€25mg172.00€50mg290.00€100mg523.00€500mg1,130.00€1mL*10mM (DMSO)93.00€GW 405833
CAS:GW 405833 (L-768242) is an agonist of cannabinoid-2 (CB(2)) receptor-selectiveFormula:C23H24Cl2N2O3Purity:99.82% - 99.93%Color and Shape:SolidMolecular weight:447.35Linoleoyl Ethanolamide
CAS:Linoleoyl Ethanolamide is an endocannabinoid agent.Formula:C20H37NO2Purity:99.97%Color and Shape:SolidMolecular weight:323.51Ref: TM-T8425
1mg35.00€5mg67.00€10mg90.00€25mg164.00€50mg239.00€100mg348.00€200mg522.00€1mL*10mM (DMSO)85.00€Anandamide
CAS:Anandamide ((5Z,8Z,11Z,14Z)-N-(2-Hydroxyethyl)icosa-5,8,11,14-tetraenamide), an immune modulator, acts via not only cannabinoid receptors (CB1 and CB2) but alsoFormula:C22H37NO2Purity:98.76% - 99.22%Color and Shape:Light Yellow OilMolecular weight:347.53Ref: TM-T14046
1mg35.00€2mg49.00€5mg74.00€10mg131.00€25mg246.00€50mg366.00€100mg538.00€200mg752.00€1mL*10mM (DMSO)81.00€exo-Tetrahydrocannabivarin
CAS:exo-Tetrahydrocannabivarin (Compound 12) is an analog of Δ9,11-THC. It weakly binds to cannabinoid receptors (CB) with an IC50 of 1.4 μM. In mice, exo-Tetrahydrocannabivarin exhibits activity related to both motor function and analgesia.Formula:C19H26O2Color and Shape:SolidMolecular weight:286.41Arvanil
CAS:Arvanil (N-Vanillylarachidonamide) is a synthetic capsaicin-amphetamine hybrid that acts as a ligand for VR1 and CB1, offering neuroprotective effects.Formula:C28H41NO3Purity:99.49%Color and Shape:SolidMolecular weight:439.63
