
GNRH Receptor
Gonadotropin-releasing hormone (GnRH) receptors are GPCRs that bind to GnRH, a hormone responsible for regulating the release of luteinizing hormone (LH) and follicle-stimulating hormone (FSH) from the pituitary gland. These receptors are crucial for reproductive function and are targeted in therapies for conditions such as prostate cancer, endometriosis, and infertility. GnRH receptor agonists and antagonists are also used in assisted reproductive technologies. At CymitQuimica, we provide a comprehensive range of high-quality GnRH receptor modulators to support your research in reproductive health, endocrinology, and hormone therapy.
Products of "GNRH Receptor"
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Found 14 products on this category.
Relugolix
CAS:Relugolix (RVT-601) is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, withFormula:C29H27F2N7O5SPurity:98.64% - 99.67%Color and Shape:SolidMolecular weight:623.63Ref: TM-T3630
1mg37.00€5mg79.00€10mg116.00€25mg198.00€50mg329.00€100mg512.00€500mg1,093.00€1mL*10mM (DMSO)96.00€Goserelin acetate
CAS:Goserelin acetate (Fertilan) is a synthetic long-acting agonist of gonadotropin-releasing hormone, used in treatments of cancer.Formula:C61H88N18O16Purity:100% - 99.86%Color and Shape:White Crystalline PowderMolecular weight:1329.46Alarelin Acetate
CAS:Alarelin Acetate is a synthetic GnRH agonist which can directly inhibit proliferation and DNA synthesis of rat GSMC through GnRH receptors.Formula:C56H78N16O12Purity:100% - 99.81%Color and Shape:White PowderMolecular weight:1167.34Ref: TM-T1494
5mg58.00€10mg95.00€25mg115.00€50mg156.00€100mg180.00€500mg452.00€1mL*10mM (DMSO)120.00€GnRH-R antagonist 1
CAS:Compound 21a: Oral GnRH-R antagonist, IC50=0.57 nM, potent against prostate cancer/prevents LH surges.Formula:C31H28F5N7O6SPurity:98%Color and Shape:SolidMolecular weight:721.65Abarelix
CAS:Abarelix (PPI 149) is a potent gonadotrophin-releasing hormone (GnRH) antagonist, which is used for prostate cancer treatment.Formula:C72H95ClN14O14Purity:100%Color and Shape:SolidMolecular weight:1416.06GnRH antagonist 2
CAS:GnRH antagonist 2 is a GnRH receptor antagonist, useful for studying endocrine diseases.Formula:C28H27F2N9O5Purity:98.08%Color and Shape:SolidMolecular weight:607.57Elagolix sodium
CAS:Elagolix sodium (NBI-56418 sodium) is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM, respectively).Formula:C32H29F5N3NaO5Purity:99.71%Color and Shape:SolidMolecular weight:653.57Fertirelin
CAS:Fertirelin, or fertirelin acetate, sold under the brand name Ovalyse, is a gonadotropin-releasing hormone agonist (GnRH agonist).Formula:C55H76N16O12Purity:100%Color and Shape:SolidMolecular weight:1153.29Ref: TM-TP1288
1mg47.00€2mg63.00€5mg96.00€10mg135.00€50mg177.00€100mg264.00€200mg393.00€1mL*10mM (DMSO)170.00€Linzagolix
CAS:Linzagolix is a small-molecule, non-peptide, orally active gonadotropin-releasing hormone antagonist (GnRH antagonist) which is under development by KisseiFormula:C22H15F3N2O7SPurity:99.68%Color and Shape:SolidMolecular weight:508.42Cetrorelix Acetate
CAS:Cetrorelix Acetate is gonadotropin-releasing hormone (GnRH) receptor antagonist with an IC50 of 1.21 nM.Formula:C70H92ClN17O14·xC2H4O2Purity:97.96%Color and Shape:SolidMolecular weight:1491.11Linzagolix choline
CAS:Linzagolix choline is a GnRH antagonist. It can be used to study pain associated with uterine fibroids and endometriosis.Formula:C27H28F3N3O8SPurity:99.64%Color and Shape:SolidMolecular weight:611.59(R)-Elagolix
CAS:(R)-Elagolix (NBI-56418) is an orally active, highly selective, short-term potent antagonist of the non-peptide gonadotropin-releasing hormone receptor.Formula:C32H30F5N3O5Purity:97.63%Color and Shape:SolidMolecular weight:631.59Ref: TM-T11174
1mg38.00€2mg49.00€5mg79.00€10mg111.00€25mg188.00€50mg329.00€100mg487.00€200mg695.00€1mL*10mM (DMSO)96.00€Cetrorelix diacetate
CAS:Cetrorelix diacetate (NS-75A) is is a gonadotropin-releasing hormone antagonist.Formula:C74H100ClN17O18Purity:98.38%Color and Shape:SolidMolecular weight:1551.17Ref: TM-T5520L
1mg52.00€5mg90.00€10mg150.00€25mg291.00€50mg437.00€100mg642.00€500mg1,359.00€1mL*10mM (DMSO)251.00€Opigolix
CAS:Opigolix is a Gonadotropin-releasing hormone receptor antagonist.Formula:C25H19F3N4O5SPurity:98.07% - 99.54%Color and Shape:SolidMolecular weight:544.5