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GNRH Receptor

GNRH Receptor

Gonadotropin-releasing hormone (GnRH) receptors are GPCRs that bind to GnRH, a hormone responsible for regulating the release of luteinizing hormone (LH) and follicle-stimulating hormone (FSH) from the pituitary gland. These receptors are crucial for reproductive function and are targeted in therapies for conditions such as prostate cancer, endometriosis, and infertility. GnRH receptor agonists and antagonists are also used in assisted reproductive technologies. At CymitQuimica, we provide a comprehensive range of high-quality GnRH receptor modulators to support your research in reproductive health, endocrinology, and hormone therapy.

Products of "GNRH Receptor"

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Found 14 products on this category.
  • Relugolix

    CAS:
    Relugolix (RVT-601) is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, with
    Formula:C29H27F2N7O5S
    Purity:98.64% - 99.67%
    Color and Shape:Solid
    Molecular weight:623.63

    Ref: TM-T3630

    1mg
    37.00€
    5mg
    79.00€
    10mg
    116.00€
    25mg
    198.00€
    50mg
    329.00€
    100mg
    512.00€
    500mg
    1,093.00€
    1mL*10mM (DMSO)
    96.00€
  • Goserelin acetate

    CAS:
    Goserelin acetate (Fertilan) is a synthetic long-acting agonist of gonadotropin-releasing hormone, used in treatments of cancer.
    Formula:C61H88N18O16
    Purity:100% - 99.86%
    Color and Shape:White Crystalline Powder
    Molecular weight:1329.46

    Ref: TM-T4102

    2mg
    48.00€
    5mg
    73.00€
    10mg
    96.00€
    25mg
    183.00€
    50mg
    310.00€
    100mg
    467.00€
    1mL*10mM (DMSO)
    155.00€
  • Alarelin Acetate

    CAS:
    Alarelin Acetate is a synthetic GnRH agonist which can directly inhibit proliferation and DNA synthesis of rat GSMC through GnRH receptors.
    Formula:C56H78N16O12
    Purity:100% - 99.81%
    Color and Shape:White Powder
    Molecular weight:1167.34

    Ref: TM-T1494

    5mg
    58.00€
    10mg
    95.00€
    25mg
    115.00€
    50mg
    156.00€
    100mg
    180.00€
    500mg
    452.00€
    1mL*10mM (DMSO)
    120.00€
  • GnRH-R antagonist 1

    CAS:
    Compound 21a: Oral GnRH-R antagonist, IC50=0.57 nM, potent against prostate cancer/prevents LH surges.
    Formula:C31H28F5N7O6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:721.65

    Ref: TM-T72492

    25mg
    2,300.00€
    50mg
    3,022.00€
    100mg
    4,085.00€
  • Abarelix

    CAS:
    Abarelix (PPI 149) is a potent gonadotrophin-releasing hormone (GnRH) antagonist, which is used for prostate cancer treatment.
    Formula:C72H95ClN14O14
    Purity:100%
    Color and Shape:Solid
    Molecular weight:1416.06

    Ref: TM-T10217L

    2mg
    42.00€
    5mg
    62.00€
    10mg
    87.00€
    25mg
    180.00€
    50mg
    283.00€
    100mg
    432.00€
    1mL*10mM (DMSO)
    90.00€
  • GnRH antagonist 2

    CAS:
    GnRH antagonist 2 is a GnRH receptor antagonist, useful for studying endocrine diseases.
    Formula:C28H27F2N9O5
    Purity:98.08%
    Color and Shape:Solid
    Molecular weight:607.57

    Ref: TM-T37003

    1mg
    157.00€
    5mg
    383.00€
    10mg
    604.00€
    25mg
    1,195.00€
    50mg
    1,892.00€
    1mL*10mM (DMSO)
    503.00€
  • Elagolix sodium

    CAS:
    Elagolix sodium (NBI-56418 sodium) is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM, respectively).
    Formula:C32H29F5N3NaO5
    Purity:99.71%
    Color and Shape:Solid
    Molecular weight:653.57

    Ref: TM-T5031

    2mg
    46.00€
    5mg
    66.00€
    10mg
    96.00€
    25mg
    172.00€
    50mg
    273.00€
    100mg
    424.00€
    1mL*10mM (DMSO)
    87.00€
  • Fertirelin

    CAS:
    Fertirelin, or fertirelin acetate, sold under the brand name Ovalyse, is a gonadotropin-releasing hormone agonist (GnRH agonist).
    Formula:C55H76N16O12
    Purity:100%
    Color and Shape:Solid
    Molecular weight:1153.29

    Ref: TM-TP1288

    1mg
    47.00€
    2mg
    63.00€
    5mg
    96.00€
    10mg
    135.00€
    50mg
    177.00€
    100mg
    264.00€
    200mg
    393.00€
    1mL*10mM (DMSO)
    170.00€
  • Linzagolix

    CAS:
    Linzagolix is a small-molecule, non-peptide, orally active gonadotropin-releasing hormone antagonist (GnRH antagonist) which is under development by Kissei
    Formula:C22H15F3N2O7S
    Purity:99.68%
    Color and Shape:Solid
    Molecular weight:508.42

    Ref: TM-T27837

    1mg
    42.00€
    5mg
    92.00€
    10mg
    127.00€
    25mg
    269.00€
    50mg
    439.00€
    1mL*10mM (DMSO)
    93.00€
  • Cetrorelix Acetate

    CAS:
    Cetrorelix Acetate is gonadotropin-releasing hormone (GnRH) receptor antagonist with an IC50 of 1.21 nM.
    Formula:C70H92ClN17O14·xC2H4O2
    Purity:97.96%
    Color and Shape:Solid
    Molecular weight:1491.11

    Ref: TM-T5520

    1mg
    48.00€
    5mg
    85.00€
    10mg
    120.00€
    25mg
    250.00€
    50mg
    401.00€
    100mg
    628.00€
    1mL*10mM (DMSO)
    180.00€
  • Linzagolix choline

    CAS:
    Linzagolix choline is a GnRH antagonist. It can be used to study pain associated with uterine fibroids and endometriosis.
    Formula:C27H28F3N3O8S
    Purity:99.64%
    Color and Shape:Solid
    Molecular weight:611.59

    Ref: TM-T25742

    1mg
    185.00€
    5mg
    459.00€
    10mg
    657.00€
    25mg
    1,026.00€
    50mg
    1,415.00€
    100mg
    1,872.00€
  • (R)-Elagolix

    CAS:
    (R)-Elagolix (NBI-56418) is an orally active, highly selective, short-term potent antagonist of the non-peptide gonadotropin-releasing hormone receptor.
    Formula:C32H30F5N3O5
    Purity:97.63%
    Color and Shape:Solid
    Molecular weight:631.59

    Ref: TM-T11174

    1mg
    38.00€
    2mg
    49.00€
    5mg
    79.00€
    10mg
    111.00€
    25mg
    188.00€
    50mg
    329.00€
    100mg
    487.00€
    200mg
    695.00€
    1mL*10mM (DMSO)
    96.00€
  • Cetrorelix diacetate

    CAS:
    Cetrorelix diacetate (NS-75A) is is a gonadotropin-releasing hormone antagonist.
    Formula:C74H100ClN17O18
    Purity:98.38%
    Color and Shape:Solid
    Molecular weight:1551.17

    Ref: TM-T5520L

    1mg
    52.00€
    5mg
    90.00€
    10mg
    150.00€
    25mg
    291.00€
    50mg
    437.00€
    100mg
    642.00€
    500mg
    1,359.00€
    1mL*10mM (DMSO)
    251.00€
  • Opigolix

    CAS:
    Opigolix is a Gonadotropin-releasing hormone receptor antagonist.
    Formula:C25H19F3N4O5S
    Purity:98.07% - 99.54%
    Color and Shape:Solid
    Molecular weight:544.5

    Ref: TM-T17301

    1mg
    279.00€
    5mg
    685.00€
    10mg
    938.00€
    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,622.00€