HIV Protease
HIV Protease inhibitors are a class of antiretroviral drugs that specifically target the protease enzyme of the Human Immunodeficiency Virus (HIV). By inhibiting this enzyme, these compounds prevent the virus from processing its polyproteins into mature, functional proteins, thereby blocking the production of new infectious virions. HIV Protease inhibitors are a cornerstone of highly active antiretroviral therapy (HAART) used to manage HIV/AIDS. At CymitQuimica, we provide a variety of HIV Protease inhibitors to support your research in HIV treatment, drug resistance, and virology.
Products of "HIV Protease"
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(S)-BI-1001
CAS:(S)-BI-1001 is an active S-enantiomer of BI-1001. (S)-BI-1001 has antiviral potency against HIV-1 integrase (IC50: 28 nM, and EC50: 450 nM and a Kd: 4.7 μM).Formula:C19H15BrClNO3Purity:98%Color and Shape:SolidMolecular weight:420.68Censavudine
CAS:Censavudine (OBP-601) is an HIV-1/2 treatment and prevention drug, a reverse transcriptase inhibitor with EC50 of 30-890 nM.Formula:C12H12N2O4Purity:98%Color and Shape:SolidMolecular weight:248.23Salmeterol Xinafoate
CAS:Salmeterol Xinafoate (GR 33343X xinafoate) is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma.Formula:C36H45NO7Purity:98% - 98.24%Color and Shape:White SolidMolecular weight:603.75Doravirine
CAS:Doravirine (MK-1439) is a non-nucleoside reverse transcriptase inhibitor, used in the treatment of HIV/AIDS.Formula:C17H11ClF3N5O3Purity:99.65% - 99.79%Color and Shape:SolidMolecular weight:425.75Ref: TM-T3632
1mg49.00€2mg69.00€5mg97.00€10mg170.00€25mg335.00€50mg520.00€100mg750.00€500mg1,549.00€1mL*10mM (DMSO)131.00€Atevirdine
CAS:Atevirdine is an HIV-1 reverse transcriptase inhibitor with antiviral activity for the study of the AIDS dementia complex (ADC).Formula:C21H25N5O2Purity:98.75%Color and Shape:SolidMolecular weight:379.46Opaviraline
CAS:Opaviraline (GW-420867X) is a potent reverse transcriptase inhibitor that inhibits Human immunodeficiency virus 1 and has the potential to treat HIV infection.Formula:C14H17FN2O3Purity:100%Color and Shape:SolidMolecular weight:280.29Ref: TM-T28255
1mg378.00€5mg922.00€10mg1,225.00€25mg1,853.00€50mg2,490.00€100mg3,353.00€1mL*10mM (DMSO)823.00€Lamivudine
CAS:Lamivudine (BCH-189) is a reverse transcriptase inhibitor and ZALCITABINE analog in which a sulfur atom replaces the 3' carbon of the pentose ring.Formula:C8H11N3O3SPurity:100% - 99.56%Color and Shape:White Crystalline PowderMolecular weight:229.26Pentosan Polysulfate Sodium (W/W 43%)
CAS:Pentosan Polysulfate Sodium: anti-HIV, anti-inflammatory, aids cartilage, treats interstitial cystitis.Purity:98%Color and Shape:SolidMolecular weight:N/ALenacapavir
CAS:Lenacapavir (GS-6207) is the first HIV-1 capsid inhibitor approved by the U.S. Food and Drug Administration, the European Medicines Agency, and Health Canada for the treatment of MDR HIV-1 infection.Cost-effective and quality-assured.Formula:C39H32ClF10N7O5S2Purity:100.00% - 99.61%Color and Shape:SolidMolecular weight:968.28Gamibetal
CAS:Gamibetal (4-Amino-3-hydroxybutyric Acid) is used as a chiral reagent in the synthesis of antiepileptic and hypotensive drug GABOB and analogues.Formula:C4H9NO3Purity:99.96%Color and Shape:White Crystalline PowderMolecular weight:119.12Bryostatin 1
CAS:Bryostatin 1, a marine macrolide, permeates CNS and modulates PKC, with strong affinity for Munc13-1 (Ki: 8.07 nM and 0.45 nM).Formula:C47H68O17Purity:98%Color and Shape:SolidMolecular weight:905.03Amylmetacresol
CAS:Amylmetacresol treats sore throat, pharyngitis, tonsillitis, laryngitis, influenza A, and SARS-CoV.Formula:C12H18OPurity:99.66%Color and Shape:SolidMolecular weight:178.27AzddMeC
CAS:AzddMeC (Az-Dcme) is an HIV-1 reverse transcriptase and HIV-1 replication inhibitor with antiretroviral activity.AzddMeC is used in the study of HIV-1 infectionFormula:C10H14N6O3Purity:97.65% - 99.62%Color and Shape:SolidMolecular weight:266.26Emtricitabine
CAS:Emtricitabine is a nucleoside reverse transcriptase inhibitor with anti-human immunodeficiency virus (HIV) and hepatitis B virus activity.Cost-effective and quality-assured.Formula:C8H10FN3O3SPurity:100% - 99.78%Color and Shape:White PowderMolecular weight:247.25Clathrin-IN-1
CAS:Pitstop 2 inhibits clathrin-mediated endocytosis, targeting clathrin's terminal domain, with potential in cancer research.Formula:C20H13BrN2O3S2Purity:99.91%Color and Shape:SolidMolecular weight:473.36Ref: TM-T9063
1mg52.00€2mg77.00€5mg96.00€10mg149.00€25mg259.00€50mg378.00€100mg560.00€500mg1,216.00€1mL*10mM (DMSO)111.00€Des(benzylpyridyl) Atazanavi
CAS:The N-dealkylated metabolite (M1) of Atazanavir, a HIV protease inhibitor.Formula:C26H43N5O7Purity:98% - 99.75%Color and Shape:SolidMolecular weight:537.65Elvitegravir
CAS:Elvitegravir (JTK-303) is an HIV integrase inhibitor and CYP2C9 inducer.Formula:C23H23ClFNO5Purity:98.35% - 99.73%Color and Shape:SolidMolecular weight:447.88Saquinavir
CAS:Saquinavir (Ro 31-8959) is a potent HIV protease inhibitor, is an antiretroviral drug used together with other medications to treat or prevent HIV/AIDS.Formula:C38H50N6O5Purity:100% - 99.50%Color and Shape:SolidMolecular weight:670.84Cytochalasin A
CAS:Cytochalasin A, a cell-penetrating fungal toxin, blocks HIV-1 protease (IC50 = 3 μM) and hinders actin and microtubule assembly. It's an antibiotic.Formula:C29H35NO5Purity:98%Color and Shape:White Crystalline PowderMolecular weight:477.59Cosalane
CAS:Cosalane (NSC 658586) is an HIV replication inhibitor and an inhibitor of chemokine receptor 7 (CCR7) signalling in humans and mice.Formula:C45H60Cl2O6Purity:100% - 98.82%Color and Shape:SolidMolecular weight:767.86Fosamprenavir Calcium Salt
CAS:Fosamprenavir Calcium Salt (GW433908G) (GW433908G) is a phosphate ester prodrug of the antiretroviral protease inhibitor Amprenavir, with improved solubility.Formula:C25H34CaN3O9PSPurity:99.59%Color and Shape:White Microcrystalline NeedlesMolecular weight:623.67Isoescin IA
CAS:Isoescin IA is a triterpenoid saponin isolated from the seeds of Aesculus chinensis. It has anti-HIV-1 protease activity.Formula:C55H86O24Purity:98.18%Color and Shape:SolidMolecular weight:1131.26(Rac)-Telinavir
CAS:N1 compound with anti-HIV activity; contains dimethyl, phenyl, quinoline groups.Formula:C33H44N6O5Purity:99.30%Color and Shape:SolidMolecular weight:604.74gp120-α4β7 binding inhibitor 11
CAS:gp120-α4β7 binding inhibitor 11 is an anti-HIV agent.Formula:C26H27N3O2Purity:97.61%Color and Shape:SolidMolecular weight:413.51Ref: TM-T67737
1mg115.00€5mg255.00€10mg375.00€25mg562.00€50mg792.00€100mg1,064.00€200mg1,444.00€1mL*10mM (DMSO)278.00€Tenofovir alafenamide
CAS:Tenofovir alafenamide (GS-7340) is a nucleotide reverse transcriptase inhibitor (NRTI) and a novel ester prodrug of the antiretroviral tenofovir.Formula:C21H29N6O5PPurity:99% - 99.81%Color and Shape:SolidMolecular weight:476.47Terameprocol
CAS:Terameprocol (EM-1421), a synthetic NDGA derivative, shows potent anti-HIV, antiangiogenic, and anticancer properties.Formula:C22H30O4Purity:99.38%Color and Shape:SolidMolecular weight:358.473-Deazaadenosine
CAS:3-Deazaadenosine, an inhibitor of S-adenosylhomocysteine hydrolase with a Ki of 3.9 μM, exhibits anti-inflammatory, anti-proliferative, and anti-HIV activity.Formula:C11H14N4O4Purity:98%Color and Shape:SolidMolecular weight:266.25CA inhibitor 1
CAS:CA inhibitor 1 (GS-6207 analog) is a potent inhibitor of the HIV capsid.Formula:C41H36ClF8N7O5S2Purity:98%Color and Shape:SolidMolecular weight:958.34PF-3450074
CAS:PF-3450074 (PF-74) is a specific HIV-1 inhibitor, blocking viral replication and uncoating at submicromolar EC50=8-640 nM.Formula:C27H27N3O2Purity:99.92%Color and Shape:SolidMolecular weight:425.52Nelfinavir Mesylate
CAS:Nelfinavir Mesylate (Viracept) is an effective HIV protease inhibitor (Ki: 2 nM).Formula:C33H49N3O7S2Purity:95.81% - 98.27%Color and Shape:A White Or Almost White PowderMolecular weight:663.89HIV-1 protease-IN-11
CAS:HIV-1 protease-IN-11 (compound 34a), an HIV-1 protease inhibitor, demonstrates potent inhibition with an IC50 of 0.41 nM and maintains substantial efficacyFormula:C26H37N3O5SPurity:98%Color and Shape:SolidMolecular weight:503.65CCR5 antagonist 1
CAS:CCR5 antagonist 1 is a CCR5 antagonist extracted from WO 2004054974 A2. It can inhibit HIV replication.Formula:C39H46ClF2N5O3SPurity:98%Color and Shape:SolidMolecular weight:738.33CDK9-IN-1
CAS:CDK9-IN-1 is a selective and potent CDK9 inhibitor with antiviral activity used in the study of PRRSV infections.Formula:C26H21N5O4SPurity:98.52%Color and Shape:SolidMolecular weight:499.54HIV-1 integrase inhibitor 8
CAS:HIV-1 integrase inhibitor 8 is an inhibitor of HIV-1 integrase. Integration is a required step in HIV replication [1].Formula:C21H24O2Purity:98.01%Color and Shape:SolidMolecular weight:308.41Tenofovir diphosphate TEA
CAS:Tenofovir diphosphate TEA (TFV-DP TEA) is an ATP-competitive DNA polymerase inhibitor that inhibits HIV-1 reverse transcriptase that\has anti-HIV/HBV potential.Formula:C9H16N5O10P3·C6H15NPurity:93.45% - 98.51%Color and Shape:SolidMolecular weight:548.36PMEDAP
CAS:PMEDAP is a potent inhibitor of Moloney murine sarcoma virus (MSV)-induced tumor formation and associated mortality and an inhibitor of human immunodeficiencyFormula:C8H13N6O4PPurity:98.12%Color and Shape:SolidMolecular weight:288.2Reverse transcriptase-IN-1
CAS:Reverse transcriptase-IN-1 is a diarylbenzopyrimidine (DABP) analogue and a potent inhibitor of HIV-1 nonnucleoside reverse transcriptase with an IC50of 13.7Formula:C25H17N7O2Purity:99.14%Color and Shape:SolidMolecular weight:447.45Ref: TM-T12715
1mg64.00€5mg131.00€10mg183.00€25mg311.00€50mg449.00€100mg615.00€200mg833.00€1mL*10mM (DMSO)143.00€PNU-103017
CAS:PNU-103017 is an inhibitor of HIV protease.Formula:C28H28N2O5SPurity:98%Color and Shape:SolidMolecular weight:504.6Delavirdine mesylate
CAS:Delavirdine mesylate (BHAP-U 90152 (mesylate)) is a non-nucleoside reverse transcriptase inhibitor (NNRTI).Formula:C23H32N6O6S2Purity:99.99%Color and Shape:Light Brown SolidMolecular weight:552.67Rilpivirine
CAS:Rilpivirine (R278474) is a diarylpyrimidine derivative and reverse transcriptase inhibitor with antiviral activity against HIV-1 that is used in the treatmentFormula:C22H18N6Purity:97.22% - 98.83%Color and Shape:SolidMolecular weight:366.42Ref: TM-T2330
2mg38.00€5mg55.00€10mg88.00€25mg145.00€50mg243.00€100mg359.00€500mg842.00€1mL*10mM (DMSO)80.00€Darunavir Ethanolate
CAS:Darunavir Ethanolate (UIC 94017) is an HIV PROTEASE INHIBITOR that is used in the treatment of AIDS and HIV INFECTIONS.Formula:C29H43N3O8SPurity:99.84%Color and Shape:SolidMolecular weight:593.74Ref: TM-T3335
5mg37.00€10mg52.00€25mg80.00€50mg111.00€100mg165.00€200mg236.00€500mg399.00€1mL*10mM (DMSO)48.00€Stercobilin hydrochloride (mixture of isomers)
CAS:Stercobilin hydrochloride (mixture of isomers) is a bile pigment metabolized by intestinal bacteria and also acts as an inhibitor of HIV protease (HIVProtease) with a Ki of 4 μM. This compound can induce pro-inflammatory activity in mouse macrophage RAW264 cells, including the production of TNF-α and IL-1β. Stercobilin hydrochloride (mixture of isomers) is utilized in research on inflammation and viral infections.Formula:C33H47ClN4O6Color and Shape:SolidMolecular weight:631.20HIV-IN-6
CAS:HIV-IN-6, an anti-HIV agent, blocks replication by targeting SFKs like Hck involved with Nef protein.Formula:C20H16N4O3SPurity:97.12%Color and Shape:SolidMolecular weight:392.43Oxindole
CAS:Oxindole (Indolin-2-one) is an aromatic heterocyclic building block. 2-indolinone derivatives have become lead compounds in the research of kinase inhibitors.Oxindole structure has been used in receptor tyrosine kinases (RTKs) inhibitors such as SU4984 and intedanib, the RTK family represents an important therapeutic target for anti-cancer drug development.Formula:C8H7NOPurity:99.34%Color and Shape:Off-White Crystalline PowderMolecular weight:133.15Rolipram
CAS:Rolipram (SB 95952) is a phosphodiesterase 4 inhibitor with antidepressant properties.Formula:C16H21NO3Purity:99.22% - 99.26%Color and Shape:SolidMolecular weight:275.34Rosamultin
CAS:Rosamultin has antioxidant, antiinflammatory/antinociceptive properties,and has anti-human immunodeficiency virus (HIV) activity.Formula:C36H58O10Purity:98% - 99.83%Color and Shape:SolidMolecular weight:650.84Cabotegravir
CAS:Cabotegravir (S/GSK1265744) (GSK744, GSK1265744) is a long-acting HIV integrase inhibitor and inhibits the HIV-1 integrase catalyzed strand transfer reaction (Formula:C19H17F2N3O5Purity:98.55% - 99.92%Color and Shape:SolidMolecular weight:405.35Arg-Val-(Nle-p-nitro)-Phe-Glu-Ala-Nle-NH2
CAS:Arg-Val-(Nle-p-nitro)-Phe-Glu-Ala-Nle-NH2 is a fluorogenic substrate for the HIV-1 protease, facilitating the assessment of enzyme activity [1].Formula:C40H66N12O11Purity:98%Color and Shape:SolidMolecular weight:891.03L 756423
CAS:L756423 is a potent, selective HIV protease inhibitor (Ki=0.049 nM), effective against HIV spread in MT25 lymphocytes at 0.1-0.5 nM, useful for AIDS research.Formula:C39H48N4O5Purity:100% - 100%Color and Shape:SolidMolecular weight:652.82Mavorixafor trihydrochloride
CAS:Mavorixafor trihydrochloride blocks CXCR4 (IC50: 13 nM) and suppresses T-tropic HIV-1 replication (IC50: 1-9 nM). It's orally active.Formula:C21H30Cl3N5Purity:98.00%Color and Shape:SolidMolecular weight:458.86NBD-557
CAS:NBD-557 is a potentially HIV-1 inhibitor.Formula:C17H24BrN3O2Purity:99.52%Color and Shape:SolidMolecular weight:382.3Ref: TM-T7382
1mg48.00€5mg97.00€10mg156.00€25mg301.00€50mg437.00€100mg620.00€200mg843.00€1mL*10mM (DMSO)105.00€Bellidifolin
CAS:Bellidoferin: anti-oxidant, protects liver, fights inflammation/tumors, aids nerve injury, blocks MAO A, may improve type-2 diabetes, antifungal.Formula:C14H10O6Purity:99.79% - 99.81%Color and Shape:SolidMolecular weight:274.23Ref: TM-T3822
1mg96.00€5mg225.00€10mg323.00€25mg537.00€50mg752.00€100mg1,035.00€1mL*10mM (DMSO)202.00€Talviraline
CAS:Talviraline (Bay 10-8979) is an RNA-induced DNA polymerase inhibitor.Talviraline is a potent inhibitor of HIV-1-induced cell killing and HIV-1 replication in aFormula:C15H20N2O3S2Purity:99.82%Color and Shape:SolidMolecular weight:340.46Lopinavir
CAS:Lopinavir (ABT-378) is a peptidomimetic HIV protease inhibitor that retains activity against HIV protease with the Val 82 mutation.Formula:C37H48N4O5Purity:98% - 99.62%Color and Shape:White Crystalline SolidMolecular weight:628.83-Deazaadenosine hydrochloride
CAS:3-Deazaadenosine HCl blocks SAH hydrolase (Ki: 3.9 μM), with anti-inflammatory, anti-proliferative, and anti-HIV effects.Formula:C11H15ClN4O4Purity:98.48%Color and Shape:SolidMolecular weight:302.71Ref: TM-T10111
1mg126.00€5mg216.00€10mg374.00€25mg620.00€50mg868.00€100mg1,169.00€1mL*10mM (DMSO)149.00€Maraviroc
CAS:Maraviroc: a CCR5 antagonist blocking HIV-1 entry; IC50s-MIP-1α: 3.3nM, MIP-1β: 7.2nM, RANTES: 5.2nM.Formula:C29H41F2N5OPurity:100% - 99.55%Color and Shape:Brown SolidMolecular weight:513.67Ref: TM-T6016
5mg51.00€10mg95.00€25mg160.00€50mg273.00€100mg492.00€200mg633.00€500mg998.00€1mL*10mM (DMSO)59.00€HIV-1 inhibitor-53
CAS:HIV-1 Inhibitor-53 targets HIV-1 protease (IC50: 1.93 nM) and reverse transcriptase (IC50: 2.35 μM), aiding AIDS research.Formula:C30H34N2O8SPurity:98%Color and Shape:SolidMolecular weight:582.66Raltegravir potassium
CAS:Raltegravir potassium (MK 0518 potassium salt) salt(MK0518 potassium salt) is a potent integrase (IN) inhibitor, used to treat HIV infection.Formula:C20H20FN6O5·KPurity:98% - 99.55%Color and Shape:Off-White SolidMolecular weight:482.51Nevirapine
CAS:Nevirapine (NVP) is a benzodiazepine non-nucleoside reverse transcriptase inhibitor.Formula:C15H14N4OPurity:99.58% - 99.59%Color and Shape:White Or Off-White Crystalline PowderMolecular weight:266.3Ro24-7429
CAS:Ro24-7429: oral HIV-1 Tat antagonist, RUNX1 inhibitor with anti-HIV, antifibrotic, and anti-inflammatory properties.Formula:C14H13ClN4Purity:99.29% - 99.85%Color and Shape:SolidMolecular weight:272.73Ref: TM-T28578
1mg92.00€5mg187.00€10mg298.00€25mg507.00€50mg730.00€100mg1,026.00€500mg2,877.00€1mL*10mM (DMSO)215.00€HIV-1 protease-IN-7
CAS:HIV-1 protease-IN-7 (compound 16) is an orally active inhibitor of HIV-1 protease, exhibiting an IC50 of 3.52 nM and an EC50 of 37 nM [1].Formula:C68H104N10O12SPurity:98%Color and Shape:SolidMolecular weight:1285.68Dolutegravir intermediate-1
CAS:Dolutegravir intermediate-1 is a synthetic precursor for HIV-1 treatment from patent WO 2016125192 A2.Formula:C13H17NO8Purity:99.52%Color and Shape:SolidMolecular weight:315.28AMD 3465
CAS:AMD 3465 (GENZ-644494) blocks CXCR4, hinders X4 HIV replication (IC50: 1-10 nM), ineffective against R5 viruses, IC50: 0.75 nM (12G5 mAb), 18 nM (CXCL12AF647).Formula:C24H38N6Purity:98%Color and Shape:SolidMolecular weight:410.60Didanosine
CAS:Didanosine (ddI) is a nucleoside reverse transcriptase inhibitor analog of adenosine (IC50: 0.49 μM).Formula:C10H12N4O3Purity:99.64%Color and Shape:White Crystalline PowderMolecular weight:236.23Obefazimod
CAS:Obefazimod (ABX-464) is a potent anti-HIV agent. ABX464 inhibits HIV-1 replication in stimulated peripheral blood mononuclear cells (PBMCs).Formula:C16H10ClF3N2OPurity:99.86%Color and Shape:SolidMolecular weight:338.71Ref: TM-T8311
2mg39.00€5mg62.00€10mg87.00€25mg187.00€50mg301.00€100mg437.00€200mg617.00€1mL*10mM (DMSO)65.00€Trovirdine
CAS:Trovirdine (LY300046) is a thiourea non-nucleoside reverse transcriptase inhibitor.Formula:C13H13BrN4SPurity:98.12% - 98.50%Color and Shape:SolidMolecular weight:337.24HIV-1 inhibitor-54
CAS:HIV-1 inhibitor-54: potent anti-HIV (EC50: 32 nM), targets WT HIV-1 IIIB in MT-4 cells for infection research.Formula:C27H30N6O4SPurity:97.61% - 98.61%Color and Shape:SoildMolecular weight:534.63Pepstatin
CAS:Pepstatin (Pepsin Inhibitor S 735A) is a specific and orally aspartate protease inhibitor that also inhibits HIV protease activity. Cost effective and quality assured.Formula:C34H63N5O9Purity:96.74% - 99.94%Color and Shape:SolidMolecular weight:685.89
