HIV Protease
HIV Protease inhibitors are a class of antiretroviral drugs that specifically target the protease enzyme of the Human Immunodeficiency Virus (HIV). By inhibiting this enzyme, these compounds prevent the virus from processing its polyproteins into mature, functional proteins, thereby blocking the production of new infectious virions. HIV Protease inhibitors are a cornerstone of highly active antiretroviral therapy (HAART) used to manage HIV/AIDS. At CymitQuimica, we provide a variety of HIV Protease inhibitors to support your research in HIV treatment, drug resistance, and virology.
Products of "HIV Protease"
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Ritonavir
CAS:Ritonavir (ABT 538) inhibits HIV-1/2 proteases; serum proteins limit it but it enhances other HIV drugs by hindering P450 degradation.Formula:C37H48N6O5S2Purity:99.38% - 99.58%Color and Shape:White PowderMolecular weight:720.94Ref: TM-T1525
1g502.00€5mg37.00€10mg49.00€25mg79.00€50mg101.00€100mg145.00€200mg202.00€500mg339.00€1mL*10mM (DMSO)49.00€MK-2048
CAS:MK-2048 is a potent inhibitor of integrase (IN) and INR263K with IC50 of 2.6 nM and 1.5 nM, respectively.Formula:C21H21ClFN5O4Purity:98%Color and Shape:SolidMolecular weight:461.87IMB-301
CAS:IMB-301 is a small molecular inhibitor via virtual screening according to the hA3G model.Formula:C19H17Cl2FN2OPurity:99.72%Color and Shape:SolidMolecular weight:379.26Ref: TM-T9212
1mg48.00€5mg97.00€10mg156.00€25mg259.00€50mg369.00€100mg530.00€200mg720.00€1mL*10mM (DMSO)105.00€Probenecid
CAS:Probenecid (Benemid) is a benzoic acid derivative with antihyperuricemic property.Formula:C13H19NO4SPurity:98.47% - 99.95%Color and Shape:Crystals From Dil Alcohol Pleasant Aftertaste (Ntp 1992)Molecular weight:285.36HIV-1 inhibitor-6
CAS:HIV-1 inhibitor-6 (3-Pyridinecarboxamide, 1,4-dihydro-1-methyl-N-(5-nitro-1,2-benzisothiazol-3-yl)-4-oxo-) is a potent HIV-1 pre-mRNA selective splicingFormula:C14H10N4O4SPurity:98.49%Color and Shape:SolidMolecular weight:330.32TAK-779
CAS:TAK-779 (Takeda 779) is an antagonist of chemokine receptor 5 (CCR5), CCR2b, and CXC chemokine receptor 3 (CXCR3).Formula:C33H39ClN2O2Purity:99.21%Color and Shape:SolidMolecular weight:531.13RN-18
CAS:RN-18 is an inhibitor of HIV-1 viral infectivity factor (IC50: 6 μM in nonpermissive H9 cells).Formula:C20H16N2O4SPurity:97.21% - 98.39%Color and Shape:SolidMolecular weight:380.42Aprepitant
CAS:Aprepitant (Aprepitant') is a Substance P/Neurokinin-1 Receptor Antagonist.Formula:C23H21F7N4O3Purity:98% - 99.68%Color and Shape:Off-White To Light Yellow Cyrstalline SolidMolecular weight:534.43Aplaviroc
CAS:Aplaviroc (AK 602), a SDP derivative, is a CCR5 antagonist. With IC50s of 0.1-0.4 nM for HIV-1Ba-L, HIV-1JRFL and HIV-1MOKW.Formula:C33H43N3O6Purity:98.78% - 99.53%Color and Shape:SolidMolecular weight:577.71HIV-1 inhibitor-81
HIV-1inhibitor-81 (Compound 14g) is an HIV-1 protease inhibitor with a Ki of 1.6 nM. This compound exhibits antiviral activity against HIV-1, with an EC50 value of 250 nM.Formula:C32H44N2O8SColor and Shape:SolidMolecular weight:616.77BMS-488043
CAS:BMS-488043 is a novel and unique oral small molecule HIV fusion inhibitor that inhibits the attachment of Human Immunodeficiency Virus type 1 (HIV-1) to CD4(+)Formula:C22H22N4O5Purity:99.72%Color and Shape:SolidMolecular weight:422.43HIV-1 protease-IN-8
CAS:HIV-1 protease-IN-8 (compound 34b) is a potent inhibitor of the HIV-1 protease enzyme, exhibiting an IC50 of 0.32 nM.Formula:C25H35N3O5SPurity:98%Color and Shape:SolidMolecular weight:489.63Abacavir hydroxyacetate
CAS:Abacavir hydroxyacetate is a nucleoside analog reverse transcriptase inhibitor used in the study of HIV infection.Formula:C16H20N6O3Purity:98.29%Color and Shape:SolidMolecular weight:344.37KM-023
CAS:KM-023 is a new second-generation non-nucleoside reverse transcriptase inhibitor for the study of human immunodeficiency virus (HIV) type 1 infection.Formula:C18H19N3O3Purity:100% - 99.70%Color and Shape:SolidMolecular weight:325.36Ref: TM-T67804
1mg150.00€5mg361.00€10mg542.00€25mg870.00€50mg1,188.00€100mg1,596.00€500mg3,202.00€1mL*10mM (DMSO)359.00€Tenofovir hydrate
CAS:Tenofovir hydrate (GS 1278 hydrate) is a nucleotide reverse transcriptase inhibitor with antiviral activity.Formula:C9H16N5O5PPurity:99.63%Color and Shape:SolidMolecular weight:305.23Bictegravir
CAS:Bictegravir (GS-9883) is a potent inhibitor of HIV-1 integrase (IC50: 7.5 nM).Formula:C21H18F3N3O5Purity:97.6% - 99.51%Color and Shape:SolidMolecular weight:449.38Ref: TM-T4493
1mg50.00€5mg66.00€10mg96.00€25mg185.00€50mg311.00€100mg469.00€500mg1,064.00€1mL*10mM (DMSO)66.00€Zalcitabine
CAS:Zalcitabine (ddC) is a nucleoside analog inhibiting HIV by blocking reverse transcriptase and halting viral DNA synthesis.Formula:C9H13N3O3Purity:99.73% - ≥95%Color and Shape:White To Off-White Crystalline PowderMolecular weight:211.22Fostemsavir Tris
CAS:Fostemsavir Tris (BMS-663068 Tris) is the prodrug of BMS-626529,is a oral, safe and effective inhibitor of HIV-1 attachment.Formula:C29H37N8O11PPurity:99.45%Color and Shape:SolidMolecular weight:704.62Ref: TM-T10570
1mg57.00€5mg120.00€10mg170.00€25mg283.00€50mg432.00€100mg612.00€1mL*10mM (DMSO)180.00€Atazanavir sulfate
CAS:Atazanavir sulfate, an azapeptide HIV-protease inhibitor, treats HIV/AIDS alongside other anti-HIV drugs.Formula:C38H52N6O7·H2SO4Purity:99.31% - 99.40%Color and Shape:SolidMolecular weight:802.93Ref: TM-T0100
5mg47.00€10mg62.00€25mg95.00€50mg120.00€100mg180.00€200mg264.00€500mg449.00€1mL*10mM (DMSO)52.00€Bz-RS-ISer(3-Ph)-Ome
CAS:Bz-RS-ISer(3-Ph)-Ome (Methyl (2R,3S)-3-(benzoylamino)-2-hydroxy-3-phenylpropanoate) is a paclitaxel derivative that inhibits the HSV replication cycle.Formula:C17H17NO4Purity:99.01% - 99.87%Color and Shape:White CrystalMolecular weight:299.32Navuridine
CAS:Navuridine (AZdU) is an oral active inhibitor of HIV reverse transcriptase with a relatively short half-life.Formula:C9H11N5O4Purity:98.9%Color and Shape:SolidMolecular weight:253.22Ref: TM-T21474
5mg74.00€10mg116.00€25mg235.00€50mg373.00€100mg562.00€500mg1,216.00€1mL*10mM (DMSO)82.00€Temsavir
CAS:Temsavir (BMS626529) is a novel attachment inhibitor that targets HIV-1 gp120 and prevents its binding to CD4+ T cells.Formula:C24H23N7O4Purity:98.06%Color and Shape:SolidMolecular weight:473.48Ref: TM-T4665
2mg42.00€5mg64.00€10mg97.00€25mg170.00€50mg293.00€100mg434.00€200mg610.00€1mL*10mM (DMSO)64.00€HIV-1 protease-IN-14
HIV-1protease-IN-14 (compound 5ae) is an effective inhibitor of HIV-1protease, exhibiting Ki values of 0.28 nM and 56.9 nM against WTHIV-1PR and R41THIV-1PR, respectively. This compound also demonstrates low cytotoxicity.Color and Shape:Odour Solid(Iso)-Fosdevirine
CAS:(Iso)-Fosdevirine ( (Iso)-GSK2248761), a reverse transcriptase (NNRTI) inhibitor with anti-HIV activity, is used in the study of neurological diseases.Formula:C20H17ClN3O3PPurity:99.90%Color and Shape:SoildMolecular weight:413.799-Aminoacridine
CAS:9-Aminoacridine is a fluorescent anti-infective dye used clinically as a topical antiseptic and experimentally as a mutagen, due to its interaction with DNA.Formula:C13H10N2Purity:98.74% - 99.93%Color and Shape:Pale Yellow CrystalsMolecular weight:194.23Lersivirine
CAS:Lersivirine (UK-453061)(UK 453061) is a second-generation non-nucleoside reverse transcriptase inhibitor (NNRTI) under development for HIV infection therapy.Formula:C17H18N4O2Purity:98.01%Color and Shape:SolidMolecular weight:310.35Ref: TM-T7700
2mg40.00€5mg60.00€10mg87.00€25mg167.00€50mg255.00€100mg368.00€200mg522.00€1mL*10mM (DMSO)65.00€WAY-639418
CAS:WAY-639418 has potential anti-inflammatory and anti-HIV activity and can be used to study CCR5-mediated inflammatory and immunomodulatory diseases.Formula:C17H16ClN5Purity:100%Color and Shape:SolidMolecular weight:325.8GSK2838232
CAS:GSK2838232 inhibit HIV reverse transcriptase activity across a broad panel of HIV-1 isolates,GSK2838232 is novel human immune virus (HIV) maturation inhibitor.Formula:C48H73ClN2O6Purity:97.97%Color and Shape:SolidMolecular weight:809.56Ref: TM-T15436
1mg70.00€5mg137.00€10mg210.00€25mg464.00€50mg677.00€100mg938.00€1mL*10mM (DMSO)187.00€Bictegravir Sodium
CAS:Bictegravir Sodium is an HIV-1 integrase inhibitor with 7.5 nM IC50, offering strong, selective anti-HIV effects and minimal toxicity.Formula:C21H17F3N3NaO5Purity:98.19%Color and Shape:SolidMolecular weight:471.36Etravirine
CAS:Etravirine (R165335) is a diarylpyrimidine non-nucleoside reverse transcriptase inhibitor.Formula:C20H15BrN6OPurity:97.61% - 99.74%Color and Shape:White To Off-White SolidMolecular weight:435.28Ref: TM-T2551
1g898.00€2mg49.00€5mg74.00€10mg111.00€25mg188.00€50mg279.00€100mg383.00€200mg485.00€1mL*10mM (DMSO)93.00€Dolutegravir
CAS:Dolutegravir (GSK1349572), HIV integrase inhibitor with IC50 of 2.7 nM, partly effective against some raltegravir-resistant HIV strains.Formula:C20H19F2N3O5Purity:98.97% - 99.08%Color and Shape:White To Pale Yellow SolidMolecular weight:419.38Ref: TM-T6198
1g1,111.00€1mg35.00€2mg50.00€5mg74.00€10mg115.00€25mg172.00€50mg274.00€100mg427.00€200mg607.00€500mg850.00€1mL*10mM (DMSO)69.00€INCB-9471
CAS:INCB-9471 is a CCR5 antagonist with anti-HIV activity and inhibits the interaction between HIV-1 gp120.Formula:C30H40F3N5O2Purity:98%Color and Shape:SolidMolecular weight:559.666TAK-220
CAS:TAK-220: Oral CCR5 antagonist. IC50: 3.5 nM (RANTES), 1.4 nM (MIP-1α).Formula:C31H41ClN4O3Purity:98%Color and Shape:SolidMolecular weight:553.14Bis-T-23
CAS:Bis-T-23 is a promoter of actin-dependent dynamin oligomerization, an HIV-I integrase inhibitor, and a Telstar derivative.Formula:C23H20N4O8Purity:96.81% - 98.77%Color and Shape:SolidMolecular weight:480.43Indinavir sulfate
CAS:Indinavir sulfate (L735524 sulfate) is a HIV protease inhibitor.It inhibits the HIV-1 protease with an IC50 value of 0.41 nM and Ki value of 0.24 nM.Formula:C36H49N5O8SPurity:100% - 99.75%Color and Shape:White PowderMolecular weight:711.87Ganoderic acid B
CAS:Ganoderic acid B: quality marker for G. lucidum products, inhibits telomerase & EBV activation, moderates HIV-1 protease.Formula:C30H44O7Purity:99.09% - 99.95%Color and Shape:SolidMolecular weight:516.67Cyclotriazadisulfonamide hydrochloride
CAS:Cyclotriazadisulfonamide HCl blocks HIV entry by hindering CD4 translocation into the ER.Formula:C31H40ClN3O4S2Purity:98%Color and Shape:SolidMolecular weight:618.25Ref: TM-T39264L
1mg185.00€5mg415.00€10mg622.00€25mg1,119.00€50mg1,679.00€100mg2,520.00€200mg3,780.00€Islatravir
CAS:Islatravir (MK-8591) is an effective anti-HIV-1 agent.Formula:C12H12FN5O3Purity:98.77%Color and Shape:SolidMolecular weight:293.25Ref: TM-T16098
1mg80.00€5mg170.00€10mg259.00€25mg454.00€50mg615.00€100mg827.00€200mg1,111.00€1mL*10mM (DMSO)182.00€Vesnarinone
CAS:Vesnarinone (Arkin) (INN) is a mixed phosphodiesterase 3 inhibitor and ion-channel modifier that has modest, dose-dependent, positive inotropic activity, butFormula:C22H25N3O4Purity:96.69% - 98.13%Color and Shape:SolidMolecular weight:395.45PKF050-638
CAS:PKF050-638 disrupts CRM1-NES, inhibits HIV-1 Rev export; selective with IC50=0.04 μM.Formula:C13H13ClN4O2Purity:98%Color and Shape:SolidMolecular weight:292.72LDC4297 hydrochloride
CAS:LDC4297 hydrochloride is a selective and potent CDK7 inhibitor with broad-spectrum antiviral activity, useful for research on viral infections.Formula:C23H29ClN8OColor and Shape:SolidMolecular weight:468.98Ancriviroc
CAS:Ancriviroc (SCH-351125) is an orally bioavailable small molecule chemokine receptor CCR5 antagonist.Cost-effective and quality-assured.Formula:C28H37BrN4O3Purity:97.31% - 99.74%Color and Shape:SolidMolecular weight:557.52Apricitabine
CAS:Apricitabine (SPD754) is a highly selective and orally active HIV-1 reverse transcriptase inhibitor (Ki=0.08 μM), the (-) enantiomer of 2′-deoxy-3′-oxy-4′-Formula:C8H11N3O3SPurity:100%Color and Shape:SolidMolecular weight:229.26Ref: TM-T14313
1mg299.00€5mg535.00€10mg663.00€25mg1,014.00€50mg1,690.00€100mg2,832.00€1mL*10mM (DMSO)625.00€SB 206553 hydrochloride
CAS:SB 206553 hydrochloride is a 5-HT2C inverse agonist and a 5-HT2C/5-HT2B receptor antagonist with anxiolytic activity, useful for studying neurological disordersFormula:C17H17ClN4OPurity:99.56%Color and Shape:SolidMolecular weight:328.84-Chloro-2-(trifluoroacetyl)aniline hydrochloride
CAS:4-Chloro-2-(trifluoroacetyl)aniline hydrochloride is an inhibitor of HIV-1 RT (HIV reverse transcriptase) .Formula:C8H6Cl2F3NOPurity:97.15%Color and Shape:SolidMolecular weight:260.04GSK-364735
CAS:GSK-364735 is an HIV-1 IN inhibitor.Formula:C19H18FN3O4Purity:97.89%Color and Shape:SolidMolecular weight:371.36Tenofovir alafenamide fumarate
CAS:Tenofovir alafenamide fumarate (GS-7340) is an oral anti-HIV drug that prevents infection.Formula:C25H33N6O9PPurity:99.95%Color and Shape:SolidMolecular weight:592.54Amprenavir
CAS:Amprenavir (KVX-478) is a synthetic derivative of hydroxyethylamine sulfonamide that selectively binds to and inhibits human immunodeficiency virus (HIV)Formula:C25H35N3O6SPurity:99.60% - 99.79%Color and Shape:Off-White To Pale YellowMolecular weight:505.63Saquinavir mesylate
CAS:Saquinavir mesylate (Ro 31-8959/003) is an Inhibitor of HIV Proteaseused in antiretroviral therapyFormula:C39H54N6O8SPurity:99.19%Color and Shape:White Or Pale Yellow PowderMolecular weight:766.9NBD-556
CAS:NBD-556 is a small molecule mimetic of CD4. NBD-556 recognizes the HIV-1 envelope protein gp120 and induces restructuring of gp120 analogous to CD4 binding.Formula:C17H24ClN3O2Purity:99.79%Color and Shape:SolidMolecular weight:337.84
