G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
Products of "G-protein Coupled Receptors and 7-TM Receptors"
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ML-335
CAS:ML-335, a μ-δ targeted agonist and MOR/DOR ligand, may lead to isomer-biased drugs with pain-relief properties.Formula:C25H32N2O3Purity:98.52%Color and Shape:SolidMolecular weight:408.53Ref: TM-T23002
2mg40.00€5mg62.00€10mg87.00€25mg170.00€50mg264.00€100mg380.00€200mg540.00€1mL*10mM (DMSO)35.00€Fananserin
CAS:Fananserin: Oral 5-HT2A antagonist (Ki=0.37 nM, rat), blocks human D4 receptor (Ki=2.93 nM).Formula:C23H24FN3O2SPurity:99.78%Color and Shape:SolidMolecular weight:425.52Ref: TM-T15270
2mg42.00€5mg56.00€10mg81.00€25mg116.00€50mg170.00€100mg250.00€200mg369.00€1mL*10mM (DMSO)62.00€(S)-FTY720-phosphonate
CAS:FTY720 (S)-Phosphate, an S1P receptor 1 (S1PR1) agonist, is utilized in studying acute inflammatory diseases, including acute lung injury.Formula:C20H36NO4PPurity:98%Color and Shape:SolidMolecular weight:385.48Pimavanserin tartrate
CAS:Pimavanserin tartrate is a potent 5-HT 2A receptor inverse agonist used to treat Parkinson's disease-related psychosis.Cost-effective and quality-assured.Formula:C50H68F2N6O4·C4H6O6Purity:100% - 99.98%Color and Shape:SolidMolecular weight:1005.2Amosulalol
CAS:Amosulalol is a combined alpha and beta adrenoceptor antagonist.Formula:C18H24N2O5SPurity:98.91%Color and Shape:SolidMolecular weight:380.46Ref: TM-T30027
1mg185.00€2mg279.00€5mg425.00€10mg625.00€25mg938.00€50mg1,311.00€100mg1,795.00€1mL*10mM (DMSO)454.00€Adenosine amine congener
CAS:Adenosine amine congener (ADAC) (ADAC) is an agonist of selective A1 adenosine receptor,.Formula:C28H32N8O6Purity:97.86%Color and Shape:SolidMolecular weight:576.6Efloxate
CAS:Efloxate (Angorlisin), a vasodilator, is utilized in the treatment of chronic coronary insufficiency.Formula:C19H16O5Purity:100%Color and Shape:SolidMolecular weight:324.33Ziprasidone
CAS:Ziprasidone (Geodon) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.Formula:C21H21ClN4OSPurity:100% - 99.53%Color and Shape:Tan SolidMolecular weight:412.94CYM50358
CAS:N-(4-(aminomethyl)-2,6-dimethylphenyl)-5 is a potent, selective antagonist of the sphingosine-1-phosphate receptor 4 (S1P4).Formula:C20H18Cl2N2O2Purity:98.05% - 99.76%Color and Shape:SolidMolecular weight:389.28Gastrin/CCK antagonist 1
CAS:Gastrin/CCK antagonist 1 is a potent gastrin/CCK antagonist for the study of metabolic system-related diseases.Formula:C28H32FN5O4Purity:98.33%Color and Shape:SolidMolecular weight:521.58Pranlukast
CAS:Cysteinyl leukotriene receptor antagonistFormula:C27H23N5O4Purity:Min. 95%Molecular weight:481.5 g/molIodophenpropit dihydrobromide
CAS:Iodophenpropit dihydrobromide: selective histamine H3 antagonist, reversible binding, high affinity (KD: 0.32 nM).Formula:C15H20BrIN4SPurity:98%Color and Shape:SolidMolecular weight:495.22ATI-2341
CAS:ATI-2341, pepducin targeting the CXCR4, is an allosteric agonist activating the Gi to promote inhibition of cAMP production and induce calcium mobilization.Formula:C104H178N26O25S2Color and Shape:SolidMolecular weight:2256.82Maropitant
CAS:Maropitant is a selective neurokinin (NK1) receptor antagonist.Formula:C32H40N2OPurity:97.35% - 99.75%Color and Shape:SolidMolecular weight:468.67BMS-986224
CAS:BMS-986224 is an orally active, potent and selective APJ receptor agonist.BMS-986224 is a candidate compound for the treatment of heart failure.Formula:C24H23ClN4O6Purity:98.61% - 98.82%Color and Shape:SolidMolecular weight:498.92human GALP (3-32)
Human GALP (3-32) (Galanin-like peptide (3-32)) serves as a high-affinity agonist for galanin receptors GalR1 (IC50 = 33 nM) and GalR2 (IC50 = 15 nM), asFormula:C137H213N43O38SPurity:98%Color and Shape:SolidMolecular weight:3102.49(Rac)-Rotigotine hydrochloride
CAS:(Rac)-Rotigotine hydrochloride is a racemate of Rotigotine. Rotigotine is a full agonist of dopamine receptor, a partial the 5-HT1A receptor agonist.Formula:C19H26ClNOSColor and Shape:SolidMolecular weight:351.93GM-60186
GM-60186, a potent inhibitor of the 5-HT receptor 2B (HTR2B) with an IC50 of 257 nM, effectively suppresses the proliferation and migration of colorectal cancer cells.Formula:C30H33FN2O4Color and Shape:SolidMolecular weight:504.59Docosahexaenoic acid ethyl ester
CAS:Docosahexaenoic acid ethyl ester (Ethyl docosahexaenoate) enhances 6-hydroxydopamine-induced neuronal damage by inducing lipid peroxidation in the mouse striatum, and can be used to study oxidative diseases of the retina or neurons.Formula:C24H36O2Color and Shape:SolidMolecular weight:356.54ONO-8130
CAS:ONO-8130 is an orally available antagonist of EP1 receptor.Formula:C25H28N2O5S2Purity:97.82%Color and Shape:SolidMolecular weight:500.63
