GABA Modulators
GABA modulators are compounds that influence the function of GABA (gamma-aminobutyric acid) receptors, the primary inhibitory neurotransmitter receptors in the central nervous system. These modulators can either enhance or inhibit GABAergic activity, affecting neuronal excitability and synaptic transmission. GABA modulators are crucial in the treatment and study of various neurological and psychiatric disorders, including anxiety, epilepsy, and insomnia. At CymitQuimica, we offer a wide range of GABA modulators to support your research in neuroscience, pharmacology, and neurotherapeutics.
Products of "GABA Modulators"
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EMEDASTINE FUMARATE
CAS:Formula:C25H34N4O9Purity:98%Color and Shape:SolidMolecular weight:534.55885999999993-AMINO-1-METHYL-5-PHENYL-1H-BENZO[E][1,4]DIAZEPIN-2(3H)-ONE
CAS:Purity:95.0%Color and Shape:SolidMolecular weight:265.31600952148447-Fluoro-3,4-dihydro-4-methyl-1H-1,4-benzodiazepine-2,5-dione
CAS:Purity:95.0%Molecular weight:208.192001342773442-[[(2-Amino-5-nitrophenyl)(2-chlorophenyl)methylene]amino]acetic Acid
Formula:C15H12ClN3O4Color and Shape:Neat7-Bromo-3,4-dihydro-1H-benzo[e][1,4]diazepine-2,5-dione
CAS:Purity:97.0%Color and Shape:SolidMolecular weight:255.07099914550786-Amino-5-ethyl-5-(1-methylbutyl)-2,4(3H,5H)-pyrimidinedione
CAS:Controlled ProductApplications 6-Amino-5-ethyl-5-(1-methylbutyl)-2,4(3H,5H)-pyrimidinedione is an impurity of Pentobarbital (P276000), an sedative and hypnotic.Formula:C11H19N3O2Color and Shape:WhiteMolecular weight:225.298-Fluoro-2,3,4,5-tetrahydro-1H-benzo[e][1,4]diazepine
CAS:Purity:97.0%Molecular weight:166.199005126953124-Boc-7,8-Dimethoxy-2,3,4,5-tetrahydro-1H-benzo[e][1,4]diazepine
CAS:Purity:97.0%Molecular weight:308.377990722656253-Amino-4-(2-chlorophenyl)-6-nitroquinolin-2(1H)-one
CAS:Formula:C15H10ClN3O3Purity:98%Color and Shape:SolidMolecular weight:315.7112Mesocarb
CAS:Controlled ProductApplications Mesocarb is a CNS stimulant that acts as a dopamine reuptake inhibitor. Mesocarb is a psychotropic drug. Mesocarb is used to counteract the sedative effects of benzodiazepine drugs. References Gainetdinov, R.R. et al.: Eur. J. Pharmacol., 340, 53 (1997); Kholodov, L.E. et al.: Khim.-Farmat. Zhur., 7, 50 (1973); Valueva, L.N. et al.: Zhur. Nevropatol. Psikh. S. S. Korsak., 82, 1212 (1982);Formula:C18H18N4O2Color and Shape:NeatMolecular weight:322.36Bromazepam-d4
CAS:Controlled ProductApplications Controlled substance (depressant). Anxiolytic. Labelled Bromazepam. References Schwartz, M.A., et al.: J. Pharm. Sci., 62, 1776 (1973), Chalmers, P., et al.: Anesthesia, 39, 370 (1984), Hassan, M.M., et al.: Anal. Profiles Drug Subs., 16, 1 (1987),Formula:C142H4H6BrN3OColor and Shape:NeatMolecular weight:320.18Olanzapine (1mg/ml in Acetonitrile)
CAS:Formula:C17H20N4SColor and Shape:Single SolutionMolecular weight:312.43Flumazenil Carboxylic Acid
CAS:Applications Flumazenil carboxylic acid is a derivative of Flumazenil (F500450), a benzodiazepine antagonist that can prevent or abolish (at the receptor level) the effects of a benzodiazepine. References Brogden, R. & Goa, K.: Drugs, 35, 448 (1988); Klotz, U. & Kanto, J.: Clin. Pharmacokinet., 14, 1 (1988)Formula:C13H10FN3O3Color and Shape:White To Off-WhiteMolecular weight:275.24Clonazepam-d4 (1.0 mg/mL in Methanol)
CAS:Controlled ProductFormula:C152H4H6ClN3O3Color and Shape:Single SolutionMolecular weight:319.74Ketazolam
CAS:Controlled ProductStability Unstable in Solution Applications A psychotropic benzodiazepine derivative with hypnotic and anxiolytic properties. Controlled Substance. References Sethy, V.H. et al.: Naun.-Schmeid. Atch. Pharmacol., 301, 157 (1978); Moore, S. et al.: Curr. Therap. Res., 29, 704 (1981); Gutierrez, S.F. et al.: Cien. Pharmac., 5, 37 (1995);Formula:C20H17ClN2O3Color and Shape:Off White CrystallineMolecular weight:368.81Ketazolam-13C,d3
CAS:Controlled ProductApplications A labelled psychotropic benzodiazepine derivative with hypnotic and anxiolytic properties. Controlled Substance. References Sethy, V.H. et al.: Naun.-Schmeid. Atch. Pharmacol., 301, 157 (1978); Moore, S. et al.: Curr. Therap. Res., 29, 704 (1981); Gutierrez, S.F. et al.: Cien. Pharmac., 5, 37 (1995);Formula:C1913CH14D3ClN2O3Color and Shape:NeatMolecular weight:372.827-Chloro-1-methyl-5-phenyl-[1,2,4]triazolo[4,3-a]quinolin-4-amine
CAS:Applications An impurity of Alprazolam (A575650). The major degradation product in Alprazolam tablets during their stability assay. References Nudelman, N., et al.: J. Pharm. Sci., 91, 1274 (2002), Marin, A., et al.: Anal. Chem., 77, 471 (2005),Formula:C17H13ClN4Color and Shape:White To Off-WhiteMolecular weight:308.76Tilivalline
CAS:Applications Tilivalline, is a metabolite from Klebsiella oxytoca. Tilivalline, is shown to be cytotoxin, and the key event causing Antibiotic-Associated Hemorrhagic Colitis. References Mori, Sh., et al.: Tetrahedron, 47, No.27, 5051 (1991); Nagasaka, T., et al.: Tetrahedron Lett., 14, 1871 (1989);Formula:C20H19N3O2Color and Shape:Light BrownMolecular weight:333.38Pyrrolidin-2-one (2-Pyrrolidone)
CAS:Controlled ProductFormula:C4H7NOColor and Shape:NeatMolecular weight:85.102,3,4,5-Tetrahydro-1H-1,4-benzodiazepine, 95%
CAS:This Thermo Scientific Chemicals brand product was originally part of the Alfa Aesar product portfolio. Some documentation and label information may refer to the legacy brand. The original Alfa Aesar product / item code or SKU reference has not changed as a part of the brand transition to Thermo Scientific Chemicals.Formula:C9H12N2Purity:95%Color and Shape:Yellow with orange to pale brown, Crystals or powder or crystalline powder or lumpy solidMolecular weight:148.217-Amino Clonazepam
CAS:Controlled ProductApplications The major metabolite of Clonazepam (C587080). References Clark, D., et al.: Drugs, 29, 342 (1985), Colmenero, J., et al.: Antimicrob. Agents Chemother., 38, 2798 (1994), Grant, D., et al.: Pharmacology, 61, 204 (2000), Negrusz, A., et al.: Anal. Bioanal. Chem., 376, 1198 (2003),Formula:C15H12ClN3OColor and Shape:YellowMolecular weight:285.73Cloxazolam
CAS:Controlled ProductApplications Cloxazolam is a benzodiazepine derivative with anxiolytic, hypnotic and antihypertensive properties used as an anti-anxiety drug. It is metabolized into the active metabolite Delorezepam (D230675). Controlled Substance. References Oliveira-Silva, D. et al.: Biomed. Chrom., 23, 1266 (2009); Kamioka, T. et al.: Psychopharmacol., 52, 17 (1977); Fischer-Cornelssen, K.A. et al.: Arzneim.-Forsch., 31, 1757 (1981);Formula:C17H14Cl2N2O2Color and Shape:NeatMolecular weight:349.21Nimetazepam-d3
CAS:Controlled ProductApplications Labelled Nimetazepam (N477800). Sedative, hypnotic. Controlled substance. References Inaba, et al.: Chem. Pharm. Bull., 19, 722 (1971), Sakai, S., et al.: Arzneim.-Forsch., 22, 534 (1972),Formula:C16H10D3N3O3Color and Shape:NeatMolecular weight:298.318-Chloro-6-(2-fluorophenyl)-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepine
CAS:Controlled ProductFormula:C17H12ClFN4Color and Shape:NeatMolecular weight:326.765-(2-Bromophenyl)-7-fluoro-1,3-dihydro-2H-1,4-benzodiazepin-2-one (Flubromazepam Isomer)
CAS:Formula:C15H10BrFN2OPirenzepine, Dihydrochloride
CAS:Controlled ProductApplications An antiulcerative. Tricyclic gastric-acid inhibitor. References Eberlein, W., et al.: Arzneimittel-Forsch., 27, 356 (1977), Hellerr, G., et al.: Verh. Deut. Ges. Inn. Med., 84, 991 (1978), Carmine, A.A., et al.: Drugs, 30,85 (1985), El-Obeid, H.A., et al.: Anal. Profiles Drug Subs., 16, 445 (1987), Homon, C.A., et al.: Ther. Drug Monit., 9, 236 (1987),Formula:C19H21N5O2·2ClHColor and Shape:NeatMolecular weight:424.324-Amino-2-methyl-10H-thieno[2,3-b][1,5]-benzodiazapine, Hydrochloride
CAS:Controlled ProductImpurity Olanzapine Impurity 6 HCl Applications Intermediate in the preparation of Olanzapine (O253750). Olanzapine Impurity 6 HCl. References Calligaro, D., et al.: Bioorg. Med. Chem. Lett., 7, 25 (1997),Formula:C12H11N3S·ClHColor and Shape:NeatMolecular weight:265.76Sultiame 100 µg/mL in Acetonitrile
CAS:Formula:C10H14N2O4S2Color and Shape:Single SolutionMolecular weight:290.362-Bromo-2'-(2-chlorobenzoyl)-4'-nitroacetanilide
CAS:Controlled ProductFormula:C15H10BrClN2O4Color and Shape:NeatMolecular weight:397.61Levetiracetam EP Impurity C
CAS:Controlled ProductFormula:C5H5NOColor and Shape:NeatMolecular weight:95.10N-Descarboxymethyl-N-carboxyethyl Lacosamide (Impurity)
CAS:Controlled ProductApplications N-Descarboxymethyl-N-carboxyethyl Lacosamide is an impurity of Lacosamide (L098500), an anticonvulsant drug that enhances sodium channel slow inactivation, and is used to treat patients with epilepsy. References Doty, P., et al.: Neurotherapeutics, 4, 145 (2007); Perucca, E., et al.: Nat. Rev. Drug Discov., 7, 973 (2008); Sake, J., et al.: CNS Drugs, 24, 1055 (2010)Formula:C14H20N2O3Color and Shape:NeatMolecular weight:264.327-Amino Nimetazepam
CAS:Controlled ProductApplications A metabolite of Nimetazepam. Controlled substance. References Nishikawa, M., et al.: Forensic Sci. Int., 66, 149 (1994), Katagi, M., et al.: J. Anal. Toxicol., 24, 354 (2000),Formula:C16H15N3OColor and Shape:NeatMolecular weight:265.31Lixivaptan
CAS:Controlled ProductApplications Drug used in the treatment and prevention of cardiovascular diseases. References Lo, R., et al.: Curr. Clin. Pharmacol., 3, 156 (2008), Ghali, J., et al.: Cardiol., 111, 147 (2008),Formula:C27H21ClFN3O2Color and Shape:NeatMolecular weight:473.93Phenobarbital
CAS:Controlled ProductApplications This is a controlled substance (depressant). Anticonvulsant; sedative; hypnotic. Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package References Goldenthal, E.I., et al.: Toxicol. Appl. Pharmacol., 18, 185 (1971), Chao, M.K.C., et al.: Anal. Profiles Drug Subs., 7, 359 (1978),Formula:C12H12N2O3Color and Shape:White To Off-WhiteMolecular weight:232.247-Amino Clonazepam-d4
CAS:Controlled ProductApplications A labelled major metabolite of Clonazepam (C587080). References Clark, D., et al.: Drugs, 29, 342 (1985), Colmenero, J., et al.: Antimicrob. Agents Chemother., 38, 2798 (1994), Grant, D., et al.: Pharmacology, 61, 204 (2000), Negrusz, A., et al.: Anal. Bioanal. Chem., 376, 1198 (2003),Formula:C152H4H8ClN3OColor and Shape:Yellow To Light Orange ColourMolecular weight:289.754-Hydroxy Midazolam (100 μg/mL in methanol)
CAS:Controlled ProductFormula:C18H13ClFN3OColor and Shape:Single SolutionMolecular weight:341.77Phenazepam
CAS:Controlled ProductApplications A benzodiazepine drug, which is used in the treatment of neurological disorders such as epilepsy, alcohol withdrawal and insomnia. It can be used as a premedication before surgery as it augments the effects of anesthetics and reduces anxiety. References Ogiso, T., et al.: Chem. Pharm. Bull., 37, 446 (1989), Gu, Q., et al.: J. Med. Chem., 36, 1001 (1993), Bekhterev, V.N., et al.: Pharm. Chem. J., 42, 95 (2008),Formula:C15H10BrClN2OColor and Shape:Light YellowMolecular weight:349.61
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