Receptor de vasopresina
Los receptores de vasopresina son una familia de receptores acoplados a proteínas G que median los efectos de la vasopresina, una hormona involucrada en la regulación del equilibrio hídrico, la presión arterial y la función renal. Los agonistas y antagonistas de los receptores de vasopresina se estudian por su papel en el tratamiento de afecciones como la diabetes insípida, la hiponatremia y la insuficiencia cardíaca. Estos receptores también son objetivos importantes en la investigación sobre el equilibrio de líquidos y la salud cardiovascular. En CymitQuimica, ofrecemos una selección de moduladores de receptores de vasopresina de alta calidad para apoyar su investigación en endocrinología, nefrología y biología cardiovascular.
Productos de "Receptor de vasopresina"
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Hay 19 productos en esta categoría.
V1a/V2 antagonist 1
V1a/V2 antagonist 1 (Compound 18j) is an orally active dual-target antagonist of V1a and V2 receptors, exhibiting high binding affinity toward these receptors [Ki values are hV1a: 0.13 nM, hV2: 0.53 nM, and mV1a: 0.5 nM; IC50 for hV1a is 2.2 nM]. This compound can inhibit oxytocin-induced scratching behavior in mice.Fórmula:C25H26ClN5O3Forma y color:SolidPeso molecular:479.96Felypressin acetate
CAS:Felypressin acetate (PLV-2) is an agonist of vasopressin 1 and acts on all arginine vasopressin receptors 1AS.Fórmula:C48H69N13O13S2Pureza:97.06%Forma y color:SolidPeso molecular:1100.27OPC-51803
CAS:OPC-51803 is an orally available nonapeptidylpressor (AVP) V(2) receptor selective agonist for the treatment of urinary incontinence and nocturia.Fórmula:C26H32ClN3O2Pureza:100% - 100%Forma y color:SolidPeso molecular:454Ref: TM-T28257
1mg333,00€5mg787,00€10mg1.074,00€25mg1.510,00€50mg1.882,00€100mg2.375,00€500mg4.655,00€Atosiban acetate
CAS:Atosiban acetate (RW22164) is an inhibitor of the hormones oxytocin and vasopressin.Fórmula:C45H71N11O14S2Pureza:99.15% - 99.84%Forma y color:SolidPeso molecular:1054.24Ref: TM-T5148
5mg73,00€10mg115,00€25mg170,00€50mg207,00€100mg268,00€500mg660,00€1mL*10mM (DMSO)134,00€Argipressin
CAS:Argipressin is a vasoconstrictive and antidiuretic hormone, binding to V1 receptors with Kd ~1.4 nM in rat heart and aortic cells.Fórmula:C46H65N15O12S2Pureza:98%Forma y color:White PowderPeso molecular:1084.23TASP0390325
CAS:TASP0390325, a potent and orally active V1B receptor antagonist, has antidepressant and anxiolytic activities in rodents.Fórmula:C25H30Cl2FN5O4Pureza:98.62%Forma y color:SolidPeso molecular:554.44Atosiban
CAS:Atosiban (RW22164), an oxytocin/vasopressin inhibitor, halts premature labor as an intravenous tocolytic, reducing uterine contractions rapidly.Fórmula:C43H67N11O12S2Pureza:98%Forma y color:SolidPeso molecular:994.19Nelivaptan
CAS:Nelivaptan (SR 149415) is a vasopressin V1b receptor antagonist that can eliminate CHS-induced GE damage.Cost-effective and quality-assured.Fórmula:C30H32ClN3O8SPureza:98% - 98.39%Forma y color:SolidPeso molecular:630.11RG7713
CAS:RG7713 (RO 5028442) has been used in trials studying Autistic Disorder.Fórmula:C25H28ClN3O2Pureza:99.74%Forma y color:SolidPeso molecular:437.96Mozavaptan
CAS:Mozavaptan (OPC-31260) is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively.Fórmula:C27H29N3O2Pureza:98.98% - 99.12%Forma y color:SolidPeso molecular:427.54E-4177
CAS:E-4177 is an angiotensin II type 1 receptor (AT1R) antagonist and can be used to study cardiovascular diseases.Fórmula:C24H21N3O2Pureza:98.63% - 99.39%Forma y color:SolidPeso molecular:383.44Tolvaptan
CAS:Tolvaptan (OPC-41061) is an orally bioavailable, selective, arginine vasopressin receptor 2 (V2, AVPR2) antagonist that can be used to treat hyponatremia.Fórmula:C26H25ClN2O3Pureza:97% - 99.91%Forma y color:SolidPeso molecular:448.94Fedovapagon
CAS:Fedovapagon (VA106483) is a pressin V2 receptor (V2R) agonist for the study of overactive bladder syndrome.Fórmula:C27H34N4O3Pureza:99.33%Forma y color:SolidPeso molecular:462.58Balovaptan
CAS:Balovaptan (RG7314), a potent brain-penetrant hV1a receptor antagonist, Ki: 1 nM for hV1a, aids autism research.Fórmula:C22H24ClN5OPureza:99.88%Forma y color:SolidPeso molecular:409.91Felypressin
CAS:Felypressin, a Lypressin analog with a phenylalanine substitution, acts as a vasoconstrictor with less antidiuretic effect.Fórmula:C46H65N13O11S2Pureza:99.65%Forma y color:SolidPeso molecular:1040.22LIXIVAPTAN
CAS:Lixivaptan (VPA-985) is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM)Fórmula:C27H21ClFN3O2Pureza:98.36%Forma y color:SolidPeso molecular:473.93Ref: TM-T7303
1mg43,00€2mg57,00€5mg81,00€10mg127,00€25mg249,00€50mg424,00€100mg625,00€1mL*10mM (DMSO)86,00€Fuscoside
CAS:Fuscoside (OPC-21268) is a non-peptide arginine vasopressin (AVP) receptor VI antagonist with an IC50 value of 0.4 μM.Cost-effective and quality-assured.Fórmula:C26H31N3O4Pureza:97.98% - 99.66%Forma y color:SolidPeso molecular:449.54Terlipressin Acetate
CAS:Terlipressin Acetate, a highly selective vasopressin V1 receptor agonist, on OGD/R-induced damage in intestinal epithelial cells (IEC-6).Fórmula:C56H82N16O19S2Pureza:98.50% - 99.69%Forma y color:SolidPeso molecular:1347.5Conivaptan hydrochloride
CAS:Conivaptan hydrochloride (Vaprisol) is an orally active vasopressin V2 and V1A receptor antagonist, used in the therapy of hypervolemic hyponatremia andFórmula:C32H26N4O2·HClPureza:98.33% - 99.86%Forma y color:SolidPeso molecular:535.04
