Receptor de andrógenos
El receptor de andrógenos (AR) es un receptor hormonal nuclear que se activa al unirse a andrógenos, como la testosterona y la dihidrotestosterona. Este receptor juega un papel crucial en el desarrollo y mantenimiento de las características masculinas, así como en la regulación de varios procesos fisiológicos, incluyendo el crecimiento muscular, la libido y la densidad ósea. Los inhibidores del receptor de andrógenos son ampliamente estudiados en el contexto del cáncer de próstata, donde la señalización del AR a menudo está sobreexpresada. En CymitQuimica, ofrecemos una gama de moduladores del receptor de andrógenos de alta calidad para apoyar su investigación en endocrinología, biología del cáncer y regulación hormonal.
Productos de "Receptor de andrógenos"
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BMS-641988
CAS:BMS-641988 is a novel nonsteroidal androgen receptor antagonist for the treatment of prostate cancer.Fórmula:C20H20F3N3O5SPureza:100% - 100%Forma y color:SoildPeso molecular:471.45N-desmethyl Enzalutamide
CAS:N-desmethyl Enzalutamide (N-desmethyl MDV 3100) is the active Enzalutamide metabolite.It is the active metabolite of Enzalutamide.Fórmula:C20H14F4N4O2SPureza:99.74%Forma y color:SolidPeso molecular:450.41Ref: TM-T19450
2mg34,00€5mg52,00€10mg74,00€25mg138,00€50mg255,00€100mg375,00€200mg532,00€1mL*10mM (DMSO)58,00€Enzalutamide
CAS:Enzalutamide (MDV3100) is an androgen receptor (AR) antagonist (IC50=36 nM in LNCaP).Fórmula:C21H16F4N4O2SPureza:100% - 99.7%Forma y color:SolidPeso molecular:464.44Ref: TM-T6002
5mg48,00€10mg56,00€25mg74,00€50mg96,00€100mg154,00€200mg187,00€500mg274,00€1mL*10mM (DMSO)52,00€Triptophenolide
CAS:Triptophenolide (Hypolide) is a compound isolated from Tripterygium wilfordii Hook with anti-inflammatory activity.Fórmula:C20H24O3Pureza:98.07% - ≥95%Forma y color:White PowderPeso molecular:312.4Anti-Androgen receptor Antibody (7Q574)
Anti-Androgen receptor Antibody (7Q574) is an antibody targeting Androgen receptor. Anti-Androgen receptor Antibody (7Q574) can be used in ELISA, WB, IHC.Forma y color:Odour LiquidGLPG0492
CAS:GLPG0492 is a novel selective androgen receptor modulator.Fórmula:C19H14F3N3O3Pureza:98.27%Forma y color:SolidPeso molecular:389.33Ref: TM-T11410L
1mg74,00€5mg164,00€10mg235,00€25mg378,00€50mg543,00€100mg730,00€200mg938,00€1mL*10mM (DMSO)170,00€Androgen receptor degrader-5
CAS:Androgen receptor degrader-5 (compound 14k) demonstrates superior capabilities, specifically in androgen receptor degradation and antiproliferative activity, showcasing its promising properties.Fórmula:C29H25F4N5O2Forma y color:SolidPeso molecular:551.53GDC-2992
CAS:GDC-2992 is a selective and oral AR (androgen receptor) degrader that, degrades AR and inhibits proliferation in VCaP cells, prostate cancer (CRPC).Fórmula:C45H51ClN8O5Forma y color:SoildPeso molecular:819.39Androgen receptor degrader-2
CAS:Androgen Receptor Degrader-2 (Compound 9) is a potent degrader of androgen receptors, with potential application in cancer research [1].Fórmula:C16H16ClN3O4Pureza:98%Forma y color:SolidPeso molecular:349.77UT-34
CAS:UT-34 is a selective and orally active antagonist of second-generation pan-androgen receptor (AR) and degrader(IC50s of 211.7 nM, 262.4 nM and 215.7 nM for wildFórmula:C15H12F4N4O2Pureza:98.12%Forma y color:SolidPeso molecular:356.27Ref: TM-T13273
1mg52,00€5mg119,00€10mg187,00€25mg354,00€50mg533,00€100mg825,00€1mL*10mM (DMSO)131,00€Ailanthone
CAS:Ailanthone (Δ13-Dehydrochaparrinone) is an effective inhibitor of both full-length androgen receptor (AR) (IC50: 69 nM) and constitutively active truncated ARFórmula:C20H24O7Pureza:99.71% - 99.96%Forma y color:SolidPeso molecular:376.4ARD-266
CAS:ARD-266 is a PROTAC degrader based on the von Hippel-Lindau E3 ligase that induces the degradation of AR proteins and is useful in prostate cancer research.Fórmula:C52H59ClN6O7Pureza:99.89%Forma y color:SolidPeso molecular:915.51Andarine
CAS:Andarine (GTx-007) (S-4) is an active partial agonist and an investigational selective androgen receptor modulator (SARM).Fórmula:C19H18F3N3O6Pureza:99.84%Forma y color:Pale Yellow SolidPeso molecular:441.36DSRM-3716
CAS:Isoquinoline, 5-iodo- (9CI) is a potent and selective inhibitor of SARM1(IC50 = 75 nM) by preventing axonal degeneration and by allowing functional recovery ofFórmula:C9H6INPureza:99.74%Forma y color:SolidPeso molecular:255.063,3'-Diindolylmethane
CAS:3,3'-Diindolylmethane (DIM), a small molecule compound, is a proposed Y preventive agent.Fórmula:C17H14N2Pureza:100%Forma y color:SolidPeso molecular:246.31Ligandrol
CAS:Ligandrol is a novel nonsteroidal, oral SARM that binds to the androgen receptor with high affinity (Ki: 1 nM) and selectivity.Fórmula:C14H12F6N2OPureza:100%Forma y color:SolidPeso molecular:338.25Masofaniten
CAS:Masofaniten (EPI-7386) is an orally active androgen receptor (AR) inhibitor with antitumor activity for the study of prostate and breast cancer.Fórmula:C24H24Cl2N4O4SPureza:98.42% - 98.66%Forma y color:SolidPeso molecular:535.44Nilutamide
CAS:Nilutamide, a nonsteroidal anti-androgen, treats prostate cancer by blocking androgen receptors, not affecting other hormone receptors.Fórmula:C12H10F3N3O4Pureza:98.45% - 98.67%Forma y color:Crystalline SolidPeso molecular:317.22Enzalutamide carboxylic acid
CAS:Enzalutamide carboxylic acid is an antagonist of androgen receptor (AR) .Fórmula:C20H13F4N3O3SPureza:97.88%Forma y color:SolidPeso molecular:451.39Ref: TM-T8217
1mg66,00€2mg93,00€5mg126,00€10mg187,00€25mg315,00€50mg439,00€100mg648,00€1mL*10mM (DMSO)140,00€Androgen receptor-IN-5
CAS:Androgen receptor-IN-5 is a potent inhibitor of the androgen receptor with anticancer properties.Fórmula:C22H10Cl2F4N4OSPureza:98%Forma y color:SolidPeso molecular:525.31
