Transferasa
Las transferasas son una gran clase de enzimas que catalizan la transferencia de grupos funcionales, como grupos metilo, glicosilo y fosfato, de una molécula a otra. Los inhibidores de transferasas se utilizan para estudiar una amplia gama de procesos biológicos, incluyendo la transducción de señales, el metabolismo y la expresión génica. Estos inhibidores son herramientas esenciales en áreas de investigación como el cáncer, las enfermedades metabólicas y la epigenética, donde está implicada la disfunción de la actividad de las transferasas. En CymitQuimica, ofrecemos una selección integral de inhibidores de transferasas para apoyar su investigación en enzimología, señalización celular y mecanismos de enfermedad.
Productos de "Transferasa"
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Hay 46 productos en esta categoría.
3-O-Methyltolcapone
CAS:3-O-Methyltolcapone (Ro 40-7591) is a metabolite of Tolcapone which is a potent COMT inhibitor.Fórmula:C15H13NO5Pureza:98%Forma y color:SolidPeso molecular:287.27Opicapone
CAS:Opicapone (BIA 9-1067), a potent COMT inhibitor for Parkinson's studies, lowers cell ATP (IC50: 98 μM).Fórmula:C15H10Cl2N4O6Pureza:97.39% - 99.36%Forma y color:SolidPeso molecular:413.17Alendronate sodium trihydrate
CAS:Alendronate sodium hydrate (MK 217), a nitrogen bisphosphonate, inhibits bone loss, treats and prevents osteoporosis.Fórmula:C4H12NO7P2·3H2O·NaPureza:99.66% - 99.90%Forma y color:White Crystalline SolidPeso molecular:325.12AMP-Deoxynojirimycin
CAS:AMP-Deoxynojirimycin (AMP-DNM) is a ceramide glucosyltransferase and GCase 2 inhibitor for the study of Parkinson's and diabetes.Fórmula:C22H39NO5Pureza:100%Forma y color:SolidPeso molecular:397.55PD 128042
CAS:PD 128042 (CI 976) is a potent orally active and selective ACAT inhibitor(IC50: 73 nM) and a potent lysophospholipid acyltransferase(LPAT) inhibitor.Fórmula:C23H39NO4Pureza:99.44%Forma y color:SolidPeso molecular:393.56Ref: TM-T22665
1mg35,00€5mg67,00€10mg114,00€25mg245,00€50mg406,00€100mg677,00€200mg935,00€1mL*10mM (DMSO)97,00€Prenyl-IN-1
CAS:Prenyl-IN-1 inhibits prenylation selectively, counters oxidative stress in Parkinson's.Fórmula:C28H24ClN5O2Pureza:100%Forma y color:SolidPeso molecular:497.98Cycloleucine
CAS:Cycloleucine is an antagonist of NMDA receptor associated glycine receptor with a Ki of 600 μM.Fórmula:C6H11NO2Pureza:98.13%Forma y color:SolidPeso molecular:129.16Pradigastat
CAS:Pradigastat (LCQ-908) is a diacylglycerol acyltransferase 1 (DGAT1) inhibitor for the treatment of constipation and can be used in the study of obesityFórmula:C25H24F3N3O2Pureza:95.21% - 95.21%Forma y color:SolidPeso molecular:455.47DGAT-1 inhibitor 2
CAS:DGAT-1 inhibitor 2: effective against obesity, targets enzyme in triglyceride synthesis for diabetes treatment.Fórmula:C24H28N4O3Pureza:98.27%Forma y color:SolidPeso molecular:420.5Ref: TM-T11016
1mg65,00€5mg140,00€10mg216,00€25mg399,00€50mg612,00€100mg842,00€1mL*10mM (DMSO)156,00€Eliglustat
CAS:Eliglustat (Genz 99067) is an oral inhibitor of glucosylceramide synthase which is used in the therapy of type 1 Gaucher disease.Fórmula:C23H36N2O4Pureza:99% - 99.51%Forma y color:SolidPeso molecular:404.54Ref: TM-T3663
1mg57,00€2mg74,00€5mg95,00€10mg124,00€25mg183,00€50mg240,00€100mg444,00€500mg998,00€1mL*10mM (DMSO)93,00€CBHcy
CAS:CBHcy, a dual substrate analog, is a specific BHMT inhibitor that may induce cysteinemia.Fórmula:C9H17NO4SPureza:100% - 100%Forma y color:SolidPeso molecular:235.3α-2,3-sialyltransferase-IN-1
CAS:α-2,3-sialyltransferase-IN-1 is a noncompetitive inhibitor of α-2,3-sialyltransferase(IC50 of 6 μM).Fórmula:C28H45NO6Pureza:98% - 98%Forma y color:SolidPeso molecular:491.66FSG67
CAS:FSG67 is an inhibitor of glycerol 3-phosphate acyltransferase (IC 50 =24 μM) [1].Fórmula:C16H25NO4SForma y color:SolidPeso molecular:327.44ABT-046
CAS:ABT-046 is an orally active, selective, and highly efficient Diacylglycerol Acyltransferase 1 (DGAT-1) inhibitor that can be used in metabolic disease research.Fórmula:C20H22N4O2Pureza:98.13%Forma y color:SolidPeso molecular:350.41GGTI-2418
CAS:GGTI-2418 is a GGTase I inhibitor with potential antitumor activity and inhibits the growth of human breast tumors.Fórmula:C23H31N5O4Pureza:99.18%Forma y color:SolidPeso molecular:441.523,5-Dinitrocatechol
CAS:OR-486 is an inhibitor of catechol-O-methyl-transferase(COMT) and can be used to prepare the molybdenum (VI)- 3,5-Dinitrocatechol complex.Fórmula:C6H4N2O6Pureza:99.88%Forma y color:SolidPeso molecular:200.11Sinbaglustat
CAS:Sinbaglustat (OGT2378), an oral N-alkyl iminosugar, inhibits GCS/GBA2 and treats lysosomal storage and neurodegenerative disorders.Fórmula:C11H23NO4Pureza:99.93%Forma y color:SolidPeso molecular:233.3Ref: TM-T40542
1mg93,00€5mg226,00€10mg339,00€25mg540,00€50mg735,00€100mg979,00€200mg1.320,00€1mL*10mM (DMSO)205,00€BMS-214662
CAS:BMS-214662 is a selective farnesyl transferase inhibitor with anti-tumor activity, used in research on pancreatic cancer, head and neck cancer, and lung cancer.Fórmula:C25H23N5O2S2Pureza:99.58% - 99.58%Forma y color:SolidPeso molecular:489.61AZD3988
CAS:AZD3988 is an orally active and highly potent inhibitor of diacylglycerol acyltransferase-1 (DGAT-1) for the study of diabetes and obesity.Fórmula:C23H22F2N4O4Pureza:99.19% - 99.82%Forma y color:SolidPeso molecular:456.44Tipifarnib (S enantiomer)
CAS:Tipifarnib S enantiomer ((S)-(-)-R-115777) is the S-enantiomer of Tipifarnib. Tipifarnib is a potent and specific farnesyltransferase inhibitor (IC50: 0.6 nM).Fórmula:C27H22Cl2N4OPureza:99.05%Forma y color:SolidPeso molecular:489.4Ref: TM-T17102
1mg51,00€5mg107,00€10mg172,00€25mg300,00€50mg432,00€100mg610,00€200mg822,00€1mL*10mM (DMSO)115,00€Ibiglustat (L-Malic acid)
CAS:Ibiglustat (L-Malic acid) (Ibiglustat L-Malic acid) is a selective, brain-penetrant, and allosteric inhibitor of glucosylceramide synthase.Fórmula:C24H30FN3O7SPureza:99.79%Forma y color:SolidPeso molecular:523.57Ref: TM-T11599
1mg60,00€2mg88,00€5mg153,00€10mg217,00€25mg368,00€50mg547,00€100mg782,00€1mL*10mM (DMSO)170,00€GGTI-2133
CAS:GGTI-2133: potent GGTase I inhibitor, IC50=38 nM; blocks inflammatory cell invasion in mice asthma.Fórmula:C27H28N4O3Pureza:99.80%Forma y color:SolidPeso molecular:456.54GPAT-IN-1
CAS:GPAT-IN-1 is a glycerol 3-phosphate acyltransferase (GPAT) inhibitor, which can be used to study obesity and diabetes.Fórmula:C21H26ClNO4SPureza:99.61% - 99.61%Forma y color:SolidPeso molecular:423.95P-3FAX-Neu5Ac
CAS:P-3FAX-Neu5Ac is a sialic acid analog and a sialyltransferase inhibitor.Fórmula:C22H30FNO14Pureza:97.08%Forma y color:SolidPeso molecular:551.47Nitecapone
CAS:Nitecapone is a reversible inhibitor of S-COMT (IC50 values of 300 nM in rat liver)Fórmula:C12H11NO6Pureza:98.39%Forma y color:SolidPeso molecular:265.22CP-609754
CAS:CP-609754 shows selective inhibition of farnesyltransferase.Fórmula:C29H22ClN3O2Pureza:98.8% - 99.04%Forma y color:SolidPeso molecular:479.96Ref: TM-T38050
1mg55,00€5mg116,00€10mg187,00€25mg319,00€50mg449,00€100mg638,00€200mg840,00€1mL*10mM (DMSO)134,00€GSK2973980A
CAS:GSK2973980A is a selective Acyl-CoA:diacylglycerol acyltransferase 1 (DGAT1) inhibitor (IC50: 3 nM).Fórmula:C25H19F5N4O4Pureza:98%Forma y color:SolidPeso molecular:534.43LB42708
CAS:LB42708 is an orally active farnesyltransferase (FTase) inhibitor (IC50: 0.8/1.2/2.0 nM toward H/N/K-ras).Fórmula:C30H27BrN4O2Pureza:97.83%Forma y color:SolidPeso molecular:555.47Ref: TM-T2678
1mg49,00€2mg64,00€5mg96,00€10mg145,00€25mg278,00€50mg414,00€100mg580,00€1mL*10mM (DMSO)133,00€Lucerastat
CAS:Lucerastat(NBDGJ) is an orally available inhibitor of GCS for Fabry disease by reducing harmful substrates.. GCS is a key enzyme in sphingolipid synthesiss.Fórmula:C10H21NO4Pureza:98%Forma y color:SolidPeso molecular:219.28Risedronic Acid
CAS:Risedronic Acid (Risedronate), a pyridinyl biphosphonate, can inhibit osteoclast-mediated bone resorption.Fórmula:C7H11NO7P2Pureza:99.77% - 99.85%Forma y color:White Crystalline PowderPeso molecular:283.11Lapaquistat acetate
CAS:Lapaquistat acetate (TAK-475) is a squalene synthase inhibitor that reduces the cytotoxicity induced by statins in human skeletal muscle cells.Fórmula:C33H41ClN2O9Pureza:100% - 99.74%Forma y color:SolidPeso molecular:645.14Entacapone acid
CAS:Entacapone acid (AG 1290) is a selective and reversible inhibitor of catechol-O-methyltransferase(COMT).Fórmula:C10H6N2O6Pureza:99.76%Forma y color:SolidPeso molecular:250.16GGsTop
CAS:GGsTop (Nahlsgen) is a GGT inhibitor with anti-aging activity.Fórmula:C13H18NO7PPureza:98.96%Forma y color:SolidPeso molecular:331.26OU749
CAS:OU749 is a γ-glutamyl transferase (GGT) inhibitor with an intrinsic Ki of 17.6 μM.Fórmula:C16H15N3O3S2Pureza:99.7%Forma y color:SolidPeso molecular:361.44Ref: TM-T22128
2mg49,00€5mg88,00€10mg127,00€25mg208,00€50mg309,00€100mg460,00€500mg1.008,00€1mL*10mM (DMSO)70,00€JNJ-DGAT2-A
CAS:JNJ-DGAT2-A, a specific inhibitor of DGAT2(IC50 = 0.14 μM), can be used in studies about the synthesis of triglycerides.Fórmula:C24H16BrFN4O2SPureza:98.2%Forma y color:SolidPeso molecular:523.38Tipifarnib
CAS:Tipifarnib (IND 58359), a quinolinone, inhibits farnesyl transferase, blocks Ras activation, arrests cell growth, and curbs angiogenesis.Fórmula:C27H22Cl2N4OPureza:97.1% - 99.22%Forma y color:Off-White To Pale Beige SolidPeso molecular:489.4FGTI-2734
CAS:FGTI-2734, a dual FT/GGT-1 inhibitor (IC50: 250/520 nM), blocks KRAS membrane binding and curbs KRAS-driven pancreatic cancer.Fórmula:C26H31FN6O2SPureza:99.36%Forma y color:SolidPeso molecular:510.63Ref: TM-T11282
1mg51,00€5mg119,00€10mg188,00€25mg393,00€50mg587,00€100mg835,00€1mL*10mM (DMSO)136,00€Minodronic acid monohydrate
CAS:Minodronic acid monohydrate 是一种法尼基二磷酸合成酶抑制剂,可作为骨吸收抑制剂。Fórmula:C9H14N2O8P2Pureza:≥95%Forma y color:SolidPeso molecular:340.16Entacapone
CAS:Entacapone (OR-611) is a selective and reversible inhibitor of catechol-O-methyltransferase (COMT).Fórmula:C14H15N3O5Pureza:100% - 99.79%Forma y color:Yellow Crystalline SolidPeso molecular:305.29Ref: TM-T2216
5mg35,00€10mg51,00€25mg80,00€50mg96,00€100mg144,00€200mg207,00€500mg350,00€1mL*10mM (DMSO)49,00€Ibiglustat
CAS:Ibiglustat (GZ402671) inhibits Glucosylceramide synthase, may treat Fabry disease by preventing GL-3 synthesis.Fórmula:C20H24FN3O2SPureza:97.97% - 99.14%Forma y color:SolidPeso molecular:389.49Ref: TM-T4473
1mg39,00€5mg97,00€10mg168,00€25mg298,00€50mg430,00€100mg605,00€200mg815,00€1mL*10mM (DMSO)90,00€Miglustat hydrochloride
CAS:Miglustat hydrochloride (N-Butyldeoxynojirimycin hydrochloride) is an inhibitor of glucosylceramide synthase and can be used for studies about Type I GaucherFórmula:C10H22ClNO4Pureza:99.61%Forma y color:SolidPeso molecular:255.74Ref: TM-TQ0155
1mg40,00€2mg52,00€5mg88,00€10mg140,00€25mg273,00€50mg472,00€100mg687,00€1mL*10mM (DMSO)87,00€Ervogastat
CAS:Ervogastat (PF-06865571) is a potent and well-tolerated diacylglycerol acyltransferase 2 inhibitor.Fórmula:C21H21N5O4Pureza:99.97%Forma y color:SolidPeso molecular:407.42Ref: TM-T9186
1mg130,00€5mg306,00€10mg512,00€25mg825,00€50mg1.121,00€100mg1.510,00€1mL*10mM (DMSO)319,00€DGAT1-IN-1
CAS:DGAT1-IN-1 is a potent inhibitor of diacylglycerol O- acyltransferase type 1(DGAT1, IC50 of < 10 nM).Fórmula:C30H28F3N3O4Pureza:99.15%Forma y color:SolidPeso molecular:551.56Ref: TM-T15109
1mg62,00€2mg87,00€5mg119,00€10mg187,00€25mg359,00€50mg540,00€100mg778,00€1mL*10mM (DMSO)145,00€L-739750 2HCl
L-739750 2HCl is a potent inhibitor of peptidomimetic farnesyltransferase, a novel pseudopeptide mimetic with potential anticancer activity.Fórmula:C23H41Cl2N3O6S2Pureza:98.69% - 99.34%Forma y color:SoildPeso molecular:590.62FDW028
CAS:FDW028 is a FUT8 inhibitor with antitumor activity that works by promoting B7-H3 lysosomal degradation through defucosylation and CMA pathways.Fórmula:C22H24N6OPureza:98.73% - 99.55%Forma y color:SoildPeso molecular:388.47Ref: TM-T77809
1mg70,00€5mg150,00€10mg235,00€25mg408,00€50mg562,00€100mg800,00€200mg1.074,00€1mL*10mM (DMSO)166,00€OSMI-1
CAS:OSMI-1: cell-permeable OGT inhibitor, blocks O-GlcNAcylation (IC50: 2.7 μM), no effect on other cell glycans.Fórmula:C28H25N3O6S2Pureza:96.79% - 99.83%Forma y color:SolidPeso molecular:563.64Ref: TM-T16409
1mg40,00€2mg52,00€5mg85,00€10mg124,00€25mg197,00€50mg350,00€100mg522,00€1mL*10mM (DMSO)96,00€
