CymitQuimica logo
Receptor adrenérgico

Receptor adrenérgico

Los receptores adrenérgicos son GPCR que son activados por catecolaminas, como la adrenalina y la noradrenalina. Estos receptores se clasifican en subtipos alfa y beta, cada uno de los cuales juega un papel clave en la regulación de la frecuencia cardíaca, la presión arterial y la respuesta de lucha o huida. Los moduladores de los receptores adrenérgicos son esenciales en el tratamiento de enfermedades cardiovasculares, asma y trastornos de ansiedad. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores adrenérgicos de alta calidad para apoyar su investigación en endocrinología, farmacología cardiovascular y respuesta al estrés.

Subcategorías de "Receptor adrenérgico"

Productos de "Receptor adrenérgico"

Ordenar por

productos por página.Hay 310 productos en esta categoría.
  • L748337

    CAS:
    L748337 is a β3-adrenoceptor antagonist that inhibits β3-, β2-, and β1-adrenoceptors and inhibits the protective effects of CL316243.
    Fórmula:C26H31N3O5S
    Pureza:99.67% - 99.67%
    Forma y color:Solid
    Peso molecular:497.61

    Ref: TM-T22905

    1mg
    69,00€
  • Tetrahydrozoline

    CAS:
    Tetrahydrozoline (Tetryzoline) is an alpha-adrenergic agonist that causes vasoconstriction and is widely used in the study of nasal and conjunctival congestion.
    Fórmula:C13H16N2
    Pureza:97.85% - 99.77%
    Forma y color:Solid
    Peso molecular:200.28

    Ref: TM-T0397

    50mg
    39,00€
    100mg
    52,00€
    500mg
    127,00€
  • Sertindole

    CAS:
    Sertindole, atypical antipsychotic, targets D2, 5-HT1D, 5-HT2A, 5-HT2C receptors (Kds: 2.7, 20, 0.14, 6 nM).
    Fórmula:C24H26ClFN4O
    Pureza:99.74%
    Forma y color:Off-White To Pale Yellow Solid
    Peso molecular:440.94

    Ref: TM-T5858

    5mg
    49,00€
    10mg
    65,00€
    25mg
    143,00€
    50mg
    275,00€
    100mg
    375,00€
    1mL*10mM (DMSO)
    52,00€
  • ADRA1D receptor antagonist 1 HCl

    CAS:
    ADRA1D receptor antagonist 1 HCl is a selective α1D adrenergic receptor antagonist (Ki: 1.6 nM) with potential antiproliferative activity.
    Fórmula:C15H14Cl2N4O
    Pureza:98.13%
    Forma y color:Solid
    Peso molecular:337.2

    Ref: TM-T10250

    1mg
    190,00€
  • Medetomidine hydrochloride

    CAS:
    Medetomidine hydrochloride (MPV785) is a selective α2-adrenoceptor agonist, with Ki of 1.08 nM, exhibts 1620-fold selectivity over α1-adrenoceptor.
    Fórmula:C13H16N2·HCl
    Pureza:99.96%
    Forma y color:White Or Off White Crystalline Powder
    Peso molecular:236.74

    Ref: TM-T6579

    10mg
    35,00€
    25mg
    52,00€
    50mg
    88,00€
    100mg
    115,00€
    500mg
    243,00€
    1mL*10mM (DMSO)
    35,00€
  • Imiloxan

    CAS:
    Imiloxan (RS-21361) is an α2 adrenergic receptor antagonist used in the treatment of major depressive disorder.
    Fórmula:C14H16N2O2
    Pureza:100% - 98.89%
    Forma y color:Solid
    Peso molecular:244.29

    Ref: TM-T27599

    1mg
    393,00€
    5mg
    933,00€
    25mg
    1.872,00€
  • Tizanidine hydrochloride

    CAS:
    Tizanidine hydrochloride (Tizanidine HCl), an α2-adrenergic receptor agonist, inhibits neurotransmitter release from CNS noradrenergic neurons.
    Fórmula:C9H9Cl2N5S
    Pureza:99.96%
    Forma y color:Solid White
    Peso molecular:290.17

    Ref: TM-T0290

    10mg
    51,00€
    25mg
    64,00€
    50mg
    95,00€
    100mg
    105,00€
    200mg
    133,00€
    500mg
    212,00€
    1mL*10mM (DMSO)
    42,00€
  • SR59230A hydrochloride

    CAS:
    SR59230A hydrochloride (SR59230A HCl) is a beta3-adrenergic receptor antagonist that inhibits ultradian brown adipose tissue thermogenesis.
    Fórmula:C21H28ClNO2
    Pureza:99.49%
    Forma y color:Solid
    Peso molecular:361.91

    Ref: TM-T13016L

    1mg
    46,00€
    5mg
    89,00€
    10mg
    116,00€
    25mg
    183,00€
    50mg
    271,00€
    100mg
    401,00€
    1mL*10mM (DMSO)
    97,00€
  • Pipoxazole

    CAS:
    Pipoxazole, an adrenergic receptor antagonist, is used potentially for the treatment of depression.
    Fórmula:C14H20N4O
    Pureza:97.88% - 99.19%
    Forma y color:Solid
    Peso molecular:260.33

    Ref: TM-T28419

    1mg
    279,00€
    5mg
    683,00€
    10mg
    938,00€
    25mg
    1.415,00€
    50mg
    1.882,00€
    100mg
    2.612,00€
  • Bambuterol hydrochloride

    CAS:
    Bambuterol hydrochloride (KWD-2183 hydrochloride) , a long-acting beta-adrenoceptor agonist, is utilized for the treating of asthma.
    Fórmula:C18H30ClN3O5
    Pureza:99.53% - 99.61%
    Forma y color:White Solid
    Peso molecular:403.91

    Ref: TM-T1446

    10mg
    48,00€
    25mg
    69,00€
    50mg
    88,00€
    100mg
    97,00€
    200mg
    133,00€
    500mg
    212,00€
    1mL*10mM (DMSO)
    44,00€
  • Brexpiprazole

    CAS:
    Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.
    Fórmula:C25H27N3O2S
    Pureza:99.06% - 99.96%
    Forma y color:Solid
    Peso molecular:433.57

    Ref: TM-T2306

    5mg
    49,00€
    10mg
    66,00€
    25mg
    80,00€
    50mg
    93,00€
    100mg
    99,00€
    200mg
    147,00€
    500mg
    274,00€
  • Salmeterol

    CAS:
    Salmeterol (GR33343X) is a long-acting agonist of beta2-adrenergic receptor (beta 2AR) used for treatment ofasthma.
    Fórmula:C25H37NO4
    Pureza:99.2% - 99.9%
    Forma y color:Solid
    Peso molecular:415.57

    Ref: TM-T12829

    5mg
    55,00€
    10mg
    88,00€
    25mg
    154,00€
    50mg
    274,00€
    1mL*10mM (DMSO)
    77,00€
  • A 61603

    CAS:
    Cixutumumab (IMC-A12) is a humanized IgG monoclonal antibody targeting the IGF1R with anticancer activity.
    Fórmula:C14H20BrN3O3S
    Forma y color:Solid
    Peso molecular:390.3

    Ref: TM-T21927

    1mg
    A consultar
    5mg
    A consultar
    10mg
    A consultar
  • Brefonalol HCl


    Brefonalol HCl, ADRA blocker for neurological/cardiovascular issues, treats angina, arrhythmias, hypertension.
    Fórmula:C22H29ClN2O2
    Pureza:99.45%
    Forma y color:Solid
    Peso molecular:388.93

    Ref: TM-T30586L

    1mg
    185,00€
    5mg
    409,00€
    10mg
    605,00€
    25mg
    938,00€
    50mg
    1.293,00€
    100mg
    1.738,00€
    500mg
    3.496,00€
  • 5-Bromoimidazo[1,2-A]Pyrazine

    CAS:
    5-Bromoimidazo[1,2-a]pyrazine inhibits phosphodiesterase and beta-adrenergic receptors.5-Bromoimidazo[1,2-a]pyrazine shows antibronchospastic activity in vitro.
    Fórmula:C6H4BrN3
    Pureza:97.04%
    Forma y color:Solid
    Peso molecular:198.02

    Ref: TM-T77641

    1mg
    115,00€
    5mg
    245,00€
    10mg
    363,00€
    25mg
    562,00€
    50mg
    775,00€
    100mg
    1.035,00€
    200mg
    1.406,00€
  • Cyclazosin HCl

    CAS:
    Cyclazosin HCl is an α-adrenergic receptor antagonist that can be used to study non-arteritic ischemic optic neuropathy.
    Fórmula:C23H28ClN5O4
    Pureza:99.44%
    Forma y color:Solid
    Peso molecular:473.95

    Ref: TM-T70585

    1mg
    279,00€
    5mg
    685,00€
    10mg
    938,00€
    25mg
    1.444,00€
    50mg
    1.882,00€
  • Ancarolol

    CAS:
    Ancarolol is a blocking agent of beta-adrenergic.
    Fórmula:C18H24N2O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:332.39

    Ref: TM-T14287

    25mg
    1.444,00€
    50mg
    1.882,00€
    100mg
    2.375,00€
  • Bucumolol

    CAS:
    Bucumolol (Bucumarol) is a β-adrenergic blocking agent and a local anesthetic with antihypertensive activity and can be used to study myocardial infarction.
    Fórmula:C17H23NO4
    Pureza:99.70%
    Forma y color:Soild
    Peso molecular:305.37

    Ref: TM-T30606L

    1mg
    201,00€
    5mg
    497,00€
    10mg
    701,00€
    25mg
    1.094,00€
    50mg
    1.508,00€
    100mg
    1.931,00€
  • 1-(2-Pyridyl)piperazine

    CAS:
    1-(2-Pyridyl)piperazine (NSC-13778) is a selective α2-adrenoceptor antagonists.
    Fórmula:C9H13N3
    Pureza:98.92%
    Forma y color:Clear Colorless To Pale Yellow Liquid
    Peso molecular:163.22

    Ref: TM-T5105

    1g
    34,00€
    1mL*10mM (DMSO)
    34,00€
  • OPC-28326

    CAS:
    OPC-28326: an α2-adrenergic blocker; dilates blood vessels; inhibits α2A/B/C receptors with Ki 2040/285/55 nM.
    Fórmula:C26H35N3O2
    Pureza:98.56%
    Forma y color:Solid
    Peso molecular:421.58

    Ref: TM-T13804

    1mg
    187,00€
    5mg
    455,00€
    10mg
    620,00€
    25mg
    940,00€
    50mg
    1.264,00€
    100mg
    1.663,00€
    200mg
    2.252,00€
    1mL*10mM (DMSO)
    567,00€