NMDAR
Los inhibidores del receptor de N-Metil-D-Aspartato (NMDAR) son compuestos que bloquean la actividad de los NMDARs, un subtipo de receptores de glutamato que desempeñan un papel crítico en la plasticidad sináptica, el aprendizaje y la memoria. La sobreactivación de los NMDARs está implicada en la excitotoxicidad, que puede llevar a daño neuronal y está asociada con condiciones como el accidente cerebrovascular, el trauma craneoencefálico y enfermedades neurodegenerativas. Los inhibidores de NMDAR son herramientas esenciales para estudiar la excitotoxicidad y para desarrollar terapias neuroprotectoras. En CymitQuimica, ofrecemos una gama de inhibidores de NMDAR para apoyar su investigación en función sináptica, neuroprotección y trastornos cognitivos.
Productos de "NMDAR"
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AV-101
CAS:AV-101 (4-Cl-KYN) is a prodrug antagonist at the glycine site of the NMDA receptor with antidepressant activity that reduces dyskinesia.Fórmula:C10H11ClN2O3Pureza:97.84% - 98.27%Forma y color:SolidPeso molecular:242.66BZAD01
CAS:BZAD01 is a selective NMDA NR1A/2B receptor antagonist.Fórmula:C16H12F6N2OPureza:99.51% - 99.78%Forma y color:SolidPeso molecular:362.27Ref: TM-T25196
5mg50,00€10mg84,00€25mg150,00€50mg226,00€100mg375,00€200mg523,00€1mL*10mM (DMSO)71,00€Aptiganel
CAS:Aptiganel (CNS-1102) is a non-competitive NMDA antagonist, a peptide that may be used to study acute ischemic stroke.Fórmula:C20H21N3Pureza:98.19% - 98.90%Forma y color:SolidPeso molecular:303.4Delucemine Hydrochloride
CAS:Delucemine Hydrochloride (Delucemine) is a polyamine NMDA receptor antagonist used in the study of neurological disorders such as depression.Fórmula:C16H18ClF2NPureza:98.14% - 99.53%Forma y color:SolidPeso molecular:297.77Mephenesin
CAS:Mephenesin (Cresoxydiol) is a centrally acting muscle relaxant with a short duration of action.Fórmula:C10H14O3Pureza:99.49%Forma y color:SolidPeso molecular:182.22ZL006
CAS:ZL006 is an effective inhibitor of nNOS/PSD-95 interaction. ZL006 also inhibits NMDA receptor-mediated NO synthesis.Fórmula:C14H11Cl2NO4Pureza:98.29%Forma y color:SolidPeso molecular:328.15Ref: TM-T17293
5mg50,00€10mg66,00€25mg117,00€50mg180,00€100mg306,00€200mg444,00€1mL*10mM (DMSO)52,00€(-)-Dizocilpine maleate
CAS:(-)-Dizocilpine maleate ((-)-MK 801 (Maleate)) is a potent, selective and non-competitive NMDA receptor antagonist with Kd of 37.2 nM in rat brain membranes.Fórmula:C20H19NO4Pureza:99.89%Forma y color:White SolidPeso molecular:337.37RPR104632
CAS:RPR104632 is a novel and potent antagonist located at the NMDA glycine site with neuroprotective activity.Fórmula:C15H11BrCl2N2O4SPureza:99.06%Forma y color:SolidPeso molecular:466.13Alaproclate
CAS:Alaproclate is a non-competitive NMDA receptor antagonist and a new selective 5-HT uptake inhibitor for the study of depression and dementia.Fórmula:C13H18ClNO2Pureza:98.51% - 98.64%Forma y color:SolidPeso molecular:255.74Dizocilpine
CAS:MK-801 (Dizocilpine (MK-801)) is a potent N-methyl-D-aspartate (NMDA) receptor antagonist with Ki of 30.5 nM.Fórmula:C16H15NPureza:99.75% - 99.97%Forma y color:SolidPeso molecular:221.3MDL-29951
CAS:MDL-29951 is a novel glycine antagonist of NMDA receptor activation.Fórmula:C12H9Cl2NO4Pureza:99.07% - 99.49%Forma y color:SolidPeso molecular:302.11Ref: TM-T1897
1mg50,00€5mg104,00€10mg180,00€25mg325,00€50mg469,00€100mg645,00€200mg868,00€1mL*10mM (DMSO)108,00€Gacyclidine
CAS:Gacyclidine (OTO311), an NMDA receptor blocker, treats tinnitus and injuries in the brain and spinal cord.Fórmula:C16H25NSPureza:100% - 99%Forma y color:SolidPeso molecular:263.44BDBM50597431
CAS:BDBM50597431 is an NMDA receptor modulator that may have can be used to study Alzheimer's disease and Parkinson's syndrome.Fórmula:C27H43F3O2Pureza:98.64% - 99.28%Forma y color:SoildPeso molecular:456.62ALDH3A1-IN-1
CAS:ALDH3A1-IN-1 (Compound 18) is a potent inhibitor of ALDH3A1 with IC50 of 1.61 μM, outperforms DEAB in prostate cancer cells.Fórmula:C13H18N2O3Pureza:99.86%Forma y color:SolidPeso molecular:250.29Ro 25-6981
CAS:Ro 25-6981: potent, selective NMDA receptor blocker (NR2B), IC50: 0.009 μM (NR1C/NR2B), 52 μM (NR1C/NR2A), useful in Parkinson's research.Fórmula:C22H29NO2Pureza:99.44%Forma y color:SolidPeso molecular:339.47L-Cysteine S-sulfate
CAS:L-Cysteine S-sulfate (S-Sulfo-L-cysteine) is an effective N-methyl-d-aspartate (NMDA) glutamatergic receptors agonist.Fórmula:C3H7NO5S2Pureza:98.92% - 99.92%Forma y color:SolidPeso molecular:201.22PEAQX
CAS:PEAQX (NVP-AAM077) is an oral NMDA antagonist, inhibits 1A/2A receptors (IC50: 270 nM), less so 1A/2B (IC50: 29,600 nM).Fórmula:C17H17BrN3O5PPureza:100% - ≥98%Forma y color:SolidPeso molecular:454.21Ref: TM-T4171
1mg34,00€2mg46,00€5mg74,00€10mg125,00€25mg216,00€50mg338,00€100mg470,00€200mg680,00€1mL*10mM (DMSO)97,00€Co 101244 hydrochloride
CAS:Co 101244 hydrochloride (4-Piperidinol, 1-[2-(4-hydroxyphenoxy)ethyl]-4-[(4-Methylphenyl)Methyl]-,hydrochloride) is an NR2B-containing NMDA receptor antagonist.Fórmula:C21H28ClNO3Pureza:98.44%Forma y color:SolidPeso molecular:377.9MRZ 2-514
CAS:MRZ 2-514 (8-bromo-4,5-dihydroxypyridazino[4,5-b]quinolin-1-one) is a strychnine-insensitive modulatory site of the NMDA receptor (glycineB)antagonist with KiFórmula:C11H6BrN3O3Pureza:98.13%Forma y color:SolidPeso molecular:308.09Ref: TM-T12110
1mg96,00€5mg202,00€10mg329,00€25mg655,00€50mg1.103,00€100mg1.483,00€1mL*10mM (DMSO)224,00€Rapastinel
CAS:Rapastinel (TPPT-amide) (GLYX-13) is an N-methyl-D-aspartate receptor (NMDAR) modulator.Fórmula:C18H31N5O6Pureza:97.18%Forma y color:SolidPeso molecular:413.47SDZ 220-040 ammonium
SDZ 220-040 ammonium is a competitive glutamate ionotropic receptor NMDA antagonist used in the study of neurological disorders.Fórmula:C16H19Cl2N2O6PPureza:97.31%Forma y color:SolidPeso molecular:437.21TCN 201
CAS:TCN 201 is a selective antagonist of NMDA receptors containing the NR2A subunit.Fórmula:C21H17ClFN3O4SPureza:98.50%Forma y color:SolidPeso molecular:461.89TCN 213
CAS:TCN 213 is an antagonist of NMDA receptor that has a selective for NR1/NR2A over NR1/NR2BFórmula:C18H24N4OS2Pureza:99.68%Forma y color:SolidPeso molecular:376.54Neboglamine hydrochloride
CAS:Neboglamine (CR-2249, XY-2401) hydrochloride boosts NMDA receptor, aids schizophrenia research, and is orally active.Fórmula:C13H25ClN2O3Pureza:97.15% - 99.11%Forma y color:SolidPeso molecular:292.8DL-AP5
CAS:DL-AP5 is the racemic form of a selective N-methyl-D-aspartate (NMDA) receptor antagonist with anticonvulsant effects.Fórmula:C5H12NO5PPureza:99.33%Forma y color:White Fine Crystalline PowderPeso molecular:197.13NMDA-IN-1
CAS:NMDA-IN-1 is a potent and NR2B-selective antagonist of NMDA(NMDA Ki of 0.85 nM; NR2B Ca2+ influx IC50 is 9.7 nM).Fórmula:C20H23ClFN3OPureza:97.01%Forma y color:SolidPeso molecular:375.87Ref: TM-T12234
1mg71,00€5mg135,00€10mg226,00€25mg371,00€50mg520,00€100mg702,00€200mg944,00€1mL*10mM (DMSO)149,00€L-701252
CAS:L-701252, a potent glycine site NMDA receptor antagonist, exhibits an inhibition concentration (IC50) of 420 nM.Fórmula:C13H10ClNO3Pureza:98.53%Forma y color:White Crystalline SolidPeso molecular:263.68Felbamate
CAS:Felbamate (W-554) is an Anti-epileptic Agent.Fórmula:C11H14N2O4Pureza:100% - 99.44%Forma y color:White Powder SolidPeso molecular:238.24UBP551
CAS:UBP551 is a potent and selective NMDA receptors modulator.Fórmula:C11H8O4Pureza:98.69%Forma y color:SolidPeso molecular:204.18Ref: TM-T8351
5mg55,00€10mg82,00€25mg126,00€50mg182,00€100mg273,00€200mg409,00€500mg677,00€1mL*10mM (DMSO)64,00€R-(+)-EU-1180-453
CAS:R-(+)-EU-1180-453 is a novel GluN2C/D selective NMDAR-positive modulator for the study of neurological disorders.Fórmula:C22H21FN2O3Pureza:100%Forma y color:SolidPeso molecular:380.41CNS-5161 hydrochloride
CAS:CNS-5161 hydrochloride (CNS 5161A) is a new antagonist of NMDA ion-channel.Fórmula:C16H19Cl2N3S2Pureza:99.53%Forma y color:SolidPeso molecular:388.385,7-Dichlorokynurenic acid
CAS:5,7-Dichlorokynurenic acid (5,7-dichlorokynurenic acid sodium) is an NMDA receptor antagonist.Fórmula:C10H5Cl2NO3Pureza:99.56%Forma y color:SolidPeso molecular:258.06QNZ46
CAS:QNZ46 is a NR2C/NR2D-selective NMDA receptor non-competitive antagonist.Fórmula:C24H17N3O6Pureza:99.65%Forma y color:SolidPeso molecular:443.41UK-240455
CAS:UK-240455: Potent NMDA glycine antagonist with neuroprotection and motor function benefits in Parkinson's.Fórmula:C11H11Cl2N3O5SPureza:98.34% - 99.83%Forma y color:SolidPeso molecular:368.19Ref: TM-T13248
1mg333,00€5mg787,00€10mg1.074,00€25mg1.510,00€50mg1.882,00€100mg2.375,00€500mg4.655,00€1mL*10mM (DMSO)680,00€Radiprodil
CAS:Radiprodil (RGH-896) is an oral NMDA NR2B antagonist for potential DPNP neuropathic pain treatment.Fórmula:C21H20FN3O4Pureza:99.74%Forma y color:SolidPeso molecular:397.4Ref: TM-T5385
1mg48,00€2mg65,00€5mg96,00€10mg153,00€25mg240,00€50mg354,00€100mg532,00€1mL*10mM (DMSO)96,00€N20C hydrochloride
CAS:N20C hydrochloride (2-((3,3-diphenylpropyl)amino)acetamide hydrochloride) is a non-competitive NMDA receptor open-channel blocker.Fórmula:C17H21ClN2OPureza:98.58%Forma y color:SolidPeso molecular:304.81D-AP5
CAS:D-AP5 (D-APV) is a NMDA receptor antagonist.Fórmula:C5H12NO5PPureza:100% - 98.77%Forma y color:White Fine Crystalline PowderPeso molecular:197.13CGP 37849
CAS:CGP 37849: oral NMDA antagonist (Ki=35 nM), anticonvulsant, with antidepressant/anxiolytic effects.Fórmula:C6H12NO5PPureza:99.87%Forma y color:White SolidPeso molecular:209.14Ref: TM-T7720
1mg127,00€5mg283,00€10mg432,00€25mg697,00€50mg938,00€100mg1.293,00€1mL*10mM (DMSO)281,00€Gavestinel sodium
CAS:Gavestinel (GV 150526): potent, selective oral NMDA antagonist; binds glycine site, pKi 8.5; studied for acute ischemic stroke.Fórmula:C18H11Cl2N2NaO3Pureza:99.04%Forma y color:SolidPeso molecular:397.19Ro 8-4304
CAS:Ro 8-4304 Hydrochloride is an antagonist of NMDA receptor with IC50 of 0.4 μMFórmula:C21H23FN2O3Pureza:98%Forma y color:SolidPeso molecular:370.42Dizocilpine Maleate
CAS:Dizocilpine Maleate (MK 801) is a potent noncompetitive antagonist of the NMDA receptor with Kd of 37.2 nM in rat brain membranes.Fórmula:C20H19NO4Pureza:99% - 99.96%Forma y color:White SolidPeso molecular:337.38SDZ 220-040
CAS:SDZ 220-040 是一种选择性哺乳动物 NMDA 受体拮抗剂,可诱导根系生长的部分无重力模式 。Fórmula:C16H16Cl2NO6PPureza:99.33%Forma y color:SolidPeso molecular:420.18L-689560
CAS:L-689560, a radiolabeled ligand, studies NMDA receptors, is an antagonist at GluN1 glycine site.Fórmula:C17H15Cl2N3O3Pureza:98%Forma y color:SolidPeso molecular:380.23CIQ
CAS:CIQ is a subunit-selective potentiator of NMDA receptors containing the NR2C or NR2D subunit. EC50 value: 2.7 μM for NR2C and 2.8 μM for NR2D.Fórmula:C26H26ClNO5Pureza:99.50%Forma y color:SolidPeso molecular:467.94Dalzanemdor
CAS:Dalzanemdor (SAGE-718) is an NMDA receptor-positive modulator of metabolism that can be used to study Huntington's chorea, Alzheimer's disease, and cognitiveFórmula:C27H43F3O2Pureza:100% - 98.20%Forma y color:SolidPeso molecular:456.621-Aminocyclobutanecarboxylic acid
CAS:1-Aminocyclobutanecarboxylic acid (ACBC) is a NMDA receptor partial agonist. 1-Aminocyclobutanecarboxylic acid act at the glycine site, NR1[1].Fórmula:C5H9NO2Pureza:99.94%Forma y color:White To Tan Powder Crystals Crystalline Powder And/Or With ChunksPeso molecular:115.13Aptiganel hydrochloride
CAS:Aptiganel hydrochloride(Cerestat) is the salt form of Aptiganel.Aptiganel is a non-competitive NMDA antagonist with neuroprotective effects used in the treatment of stroke and focal cerebral ischemia.Fórmula:C20H22ClN3Pureza:99.89%Forma y color:SolidPeso molecular:339.86Ref: TM-T38068
1mg38,00€5mg80,00€10mg126,00€25mg267,00€50mg462,00€100mg700,00€200mg995,00€1mL*10mM (DMSO)88,00€Cycloleucine
CAS:Cycloleucine is an antagonist of NMDA receptor associated glycine receptor with a Ki of 600 μM.Fórmula:C6H11NO2Pureza:98.13%Forma y color:SolidPeso molecular:129.16Flupirtine maleate
CAS:Flupirtine maleate (Katadolon maleate), a centrally acting non-opioid analgesia, is the salt form of Flupirtine. Flupirtine is an NMDA receptor antagonist.Fórmula:C15H17FN4O2·C4H4O4Pureza:99.50% - 99.9%Forma y color:Off-White Crystalline PowderPeso molecular:420.39Flutriafol
CAS:Flutriafol is a pesticide, demethylation inhibitor, and NMDA receptor agonistFórmula:C16H13F2N3OPureza:98.75%Forma y color:SolidPeso molecular:301.29
