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Tie-2

Tie-2

Los inhibidores de Tie-2 son compuestos que se dirigen al receptor Tie-2, una tirosina quinasa involucrada en la angiogénesis y la integridad vascular. La señalización de Tie-2 es crucial para el mantenimiento de los vasos sanguíneos, y su desregulación está asociada con el cáncer y las enfermedades vasculares. En CymitQuimica, ofrecemos inhibidores de Tie-2 para apoyar su investigación en angiogénesis, biología vascular y terapias contra el cáncer dirigidas.

Productos de "Tie-2"

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Hay 20 productos en esta categoría.
  • TIE2 Protein, Mouse, Recombinant (hFc)


    TIE2 Protein, Mouse, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag.
    Forma y color:Lyophilized Powder
    Peso molecular:107.7 kDa (predicted)

    Ref: TM-TMPY-01954

    1mg
    3.832,00€
    200µg
    608,00€
  • Anti-TIE2 Antibody-PE (1E654)


    Anti-TIE2 Antibody-PE (1E654) is a PE-conjugated Mouse antibody targeting TIE2. Anti-TIE2 Antibody-PE (1E654) can be used in FCM.
    Forma y color:Odour Liquid

    Ref: TM-TMAY-01087P

    25T
    87,00€
    100T
    264,00€
  • TIE2 Protein, Mouse, Recombinant (aa 770-1122, His & GST)


    TIE2 Protein, Mouse, Recombinant (aa 770-1122, His & GST) is expressed in Baculovirus insect cells with His and GST tag.
    Forma y color:Lyophilized Powder
    Peso molecular:68.2kDa (predicted); 68 kDa (reducing conditions)

    Ref: TM-TMPY-04575

    50µg
    410,00€
  • Anti-TIE2 Antibody (7A105)


    Anti-TIE2 Antibody (7A105) is a Mouse antibody targeting TIE2. Anti-TIE2 Antibody (7A105) can be used in ELISA.
    Forma y color:Odour Liquid

    Ref: TM-TMAY-01086

    100µl
    204,00€
  • Anti-TIE2 Antibody-APC (1E654)


    Anti-TIE2 Antibody-APC (1E654) is a APC-conjugated Mouse antibody targeting TIE2. Anti-TIE2 Antibody-APC (1E654) can be used in FCM.
    Forma y color:Odour Liquid

    Ref: TM-TMAY-01087A

    25T
    110,00€
    100T
    266,00€
  • Anti-TIE2 Antibody-FITC (9U826)


    Anti-TIE2 Antibody-FITC (9U826) is a FITC-conjugated Rabbit antibody targeting TIE2. Anti-TIE2 Antibody-FITC (9U826) can be used in FCM.
    Forma y color:Odour Liquid

    Ref: TM-TMAY-01088F

    25T
    95,00€
    100T
    181,00€
  • Anti-TIE2 Antibody-PE (9U826)


    Anti-TIE2 Antibody-PE (9U826) is a PE-conjugated Rabbit antibody targeting TIE2. Anti-TIE2 Antibody-PE (9U826) can be used in FCM.
    Forma y color:Odour Liquid

    Ref: TM-TMAY-01088P

    25T
    95,00€
    100T
    265,00€
  • Anti-TIE2 Antibody (9U826)


    Anti-TIE2 Antibody (9U826) is a Rabbit antibody targeting TIE2. Anti-TIE2 Antibody (9U826) can be used in ELISA(Cap),FCM,ICC/IF.
    Forma y color:Odour Liquid

    Ref: TM-TMAY-01088

    20µl
    98,00€
    100µl
    276,00€
  • TIE2 Protein, Human, Recombinant (hFc)


    TIE2 Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with C-Fc tag.
    Forma y color:Lyophilized Powder
    Peso molecular:120-150 KDa (reducing condition)

    Ref: TM-TMPJ-00642

    1mg
    1.316,00€
    10µg
    72,00€
    50µg
    189,00€
    500µg
    880,00€
  • Anti-TIE2 Antibody (1E654)


    Anti-TIE2 Antibody (1E654) is a Mouse antibody targeting TIE2. Anti-TIE2 Antibody (1E654) can be used in FCM.
    Forma y color:Odour Liquid

    Ref: TM-TMAY-01087

    100µl
    205,00€
  • Razuprotafib

    CAS:
    Razuprotafib (AKB-9778) inhibits HPTPß (IC50: 50 nM), activates Tie-2, and guards against acute kidney injury.
    Fórmula:C26H26N4O6S3
    Pureza:98.53%
    Forma y color:Solid
    Peso molecular:586.7

    Ref: TM-T16724

    1mg
    240,00€
    5mg
    393,00€
    10mg
    588,00€
    25mg
    998,00€
    50mg
    1.301,00€
    100mg
    1.700,00€
    1mL*10mM (DMSO)
    507,00€
  • Tie2 kinase inhibitor 1

    CAS:
    Tie2 kinase inhibitor 1 (Tie2 kinase inhibitor), an optimized compound of SB-203580, is selective to Tie2 with IC50 of 0.25 μM, which is 200-fold more effective
    Fórmula:C26H21N3O2S
    Pureza:99.51%
    Forma y color:Solid
    Peso molecular:439.53

    Ref: TM-T6335

    1mg
    66,00€
    5mg
    150,00€
    10mg
    225,00€
    25mg
    404,00€
    50mg
    610,00€
    100mg
    838,00€
    500mg
    1.691,00€
  • Pexmetinib

    CAS:
    Pexmetinib (ARRY-614) is an orally bioavailable dual p38 MAPK/Tie-2 inhibitor.Cost-effective and quality-assured.
    Fórmula:C31H33FN6O3
    Pureza:98.41% - 99.66%
    Forma y color:Solid
    Peso molecular:556.63

    Ref: TM-T6934

    1mg
    47,00€
    5mg
    97,00€
    10mg
    139,00€
    25mg
    271,00€
    50mg
    435,00€
    100mg
    567,00€
    200mg
    810,00€
    1mL*10mM (DMSO)
    118,00€
  • Anti-TIE2 Antibody-FITC (1E654)


    Anti-TIE2 Antibody-FITC (1E654) is a FITC-conjugated Mouse antibody targeting TIE2. Anti-TIE2 Antibody-FITC (1E654) can be used in FCM.
    Forma y color:Odour Liquid

    Ref: TM-TMAY-01087F

    25T
    95,00€
    100T
    180,00€
  • BAY-826

    CAS:
    BAY-826 is a novel, potent and selective TIE-2 inhibitor that inhibits TIE-2 phosphorylation and can be used to study tumors.
    Fórmula:C26H19F5N6OS
    Pureza:98%
    Forma y color:Solid
    Peso molecular:558.53

    Ref: TM-T38930

    1mg
    75,00€
  • TIE2 Protein, Mouse, Recombinant (His), Biotinylated


    TIE2 Protein, Mouse, Recombinant (His), Biotinylated is expressed in HEK293 mammalian cells with His tag.
    Forma y color:Lyophilized Powder
    Peso molecular:82.03 kDa (predicted); 88.1 kDa (reducing conditions)

    Ref: TM-TMPY-06974

    20µg
    410,00€
    100µg
    954,00€
  • TIE2 Protein, Human, Recombinant (aa 23-745, His)


    TIE2 Protein, Human, Recombinant (aa 23-745, His) is expressed in HEK293 mammalian cells with C-6xHis tag.
    Forma y color:Lyophilized Powder
    Peso molecular:100-120 KDa (reducing condition)

    Ref: TM-TMPJ-00643

    1mg
    1.316,00€
    10µg
    62,00€
    50µg
    170,00€
    500µg
    880,00€
  • CE-245677 mesylate

    CAS:
    CE-245677 mesylate is a selective Tie2 kinase inhibitor with oral activity and potential anti-tumor effects, useful in pain research.
    Fórmula:C25H26Cl2N6O6S
    Pureza:99.42%
    Forma y color:Solid
    Peso molecular:609.48

    Ref: TM-T68286

    1mg
    279,00€
    5mg
    685,00€
    10mg
    938,00€
    25mg
    1.444,00€
    50mg
    1.882,00€
    100mg
    2.375,00€
  • CE-245677

    CAS:
    CE-245677 is a potent reversible inhibitor of Tie2 and TrkA/B kinases. With a cellular IC50s of 4.7 and 1 nM.
    Fórmula:C24H22Cl2N6O3
    Pureza:98.99% - 99.23%
    Forma y color:Solid
    Peso molecular:513.38

    Ref: TM-T14921

    1mg
    62,00€
    2mg
    87,00€
    5mg
    119,00€
    10mg
    187,00€
    25mg
    313,00€
    50mg
    432,00€
    100mg
    638,00€
    1mL*10mM (DMSO)
    136,00€
  • Anti-TIE2 Antibody-APC (9U826)


    Anti-TIE2 Antibody-APC (9U826) is a APC-conjugated Rabbit antibody targeting TIE2. Anti-TIE2 Antibody-APC (9U826) can be used in FCM.
    Forma y color:Odour Liquid

    Ref: TM-TMAY-01088A

    25T
    110,00€
    100T
    264,00€