Receptor de glucagón
Los receptores de glucagón son GPCR que median los efectos del glucagón, una hormona involucrada en la regulación de la homeostasis de la glucosa al promover la descomposición del glucógeno y la liberación de glucosa desde el hígado. Estos receptores son cruciales en la gestión de los niveles de azúcar en sangre y son de particular interés en el estudio de la diabetes y los trastornos metabólicos. Los antagonistas de los receptores de glucagón se están explorando como posibles tratamientos para la hiperglucemia en la diabetes tipo 2. En CymitQuimica, ofrecemos una variedad de moduladores de receptores de glucagón de alta calidad para apoyar su investigación en endocrinología, diabetes y regulación metabólica.
Productos de "Receptor de glucagón"
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Hay 39 productos en esta categoría.
(S, R)-LSN 3318839
CAS:(S,R)-LSN 3318839 enhances GLP-1R, shows strong blood sugar lowering in animals, works with sitagliptin.Fórmula:C26H23Cl2N3O2Pureza:99.57%Forma y color:SoildPeso molecular:480.39NNC 92-1687
CAS:NNC 92-1687 is a selective glucagon receptor antagonist that can be used to study type 2 diabetes.Fórmula:C15H12N2O3SPureza:100% - 99.72%Forma y color:SolidPeso molecular:300.33Avexitide
CAS:Avexitide (Exendin-3 (9-39) amide) (Exendin (9-39)) is a specific and competitive antagonist of glucagon-like peptide-1 (GLP-1) receptor.Fórmula:C149H234N40O47SPureza:98% - 99.65%Forma y color:SolidPeso molecular:3369.76Exendin-4 acetate
CAS:Exendin-4 acetate is a 39 amino acid peptide.Exendin-4 acetate is a long-acting GLP-1 receptor agonist(IC50 = 3.22 nM).Fórmula:C186H286N50O62SPureza:98.65%Forma y color:SolidPeso molecular:4247Lotiglipron
CAS:Lotiglipron (PF-07081532) is a GLP-1R agonist that lowers blood glucose and may be used in the study of type 2 diabetes mellitus (T2DM) and excess obesity.Fórmula:C31H31ClN4O5Pureza:98.3%Forma y color:SolidPeso molecular:575.05V-0219
CAS:V-0219 is a positive allosteric modulator of GLP-1 and can be used in studies about obesity-associated diabetes.Fórmula:C20H25F3N4O2Pureza:100%Forma y color:SoildPeso molecular:410.43Orforglipron
CAS:Orforglipron (LY3502970; GLP-1 receptor agonist 1) is an orally available glucagon-like peptide (GLP-1) receptor agonist for the study of obesity and type 1Fórmula:C48H48F2N10O5Pureza:99.15% - 99.61%Forma y color:SolidPeso molecular:882.96Ref: TM-T11408
1mg244,00€5mg597,00€10mg938,00€25mg1.882,00€50mg2.593,00€100mg3.505,00€1mL*10mM (DMSO)47,00€V-0219 hydrochloride
V-0219 hydrochloride: oral GLP-1R PAM for obesity-linked diabetes study.Fórmula:C20H26ClF3N4O2Pureza:100%Forma y color:SoildPeso molecular:446.89Ref: TM-T60047L
1mg59,00€5mg125,00€10mg205,00€25mg393,00€50mg585,00€100mg832,00€200mg1.121,00€1mL*10mM (DMSO)136,00€Semaglutide
CAS:Semaglutide is a glucagon-like peptide 1 receptor (GLP-1R) agonist(EC50 of 6.2 pM in a reporter assay using BHK cells expressing the human receptor).Fórmula:C187H291N45O59Pureza:96.92% - 99.78%Forma y color:SolidPeso molecular:4114Ref: TM-T19850
1mg126,00€5mg264,00€10mg378,00€25mg562,00€50mg780,00€100mg1.054,00€200mg1.419,00€500µg85,00€GLP-1 (9-36) amide
CAS:GLP-1 (9-36) amide is an antagonist at the human GLP-1 receptor.Fórmula:C140H214N36O43Pureza:97%Forma y color:SolidPeso molecular:3089.41LGD-6972
CAS:LGD-6972 is an antagonist of glucagon receptor.Fórmula:C43H46N2O5SPureza:98.8% - 99.33%Forma y color:SolidPeso molecular:702.9Ref: TM-T11845
1mg88,00€5mg187,00€10mg274,00€25mg472,00€50mg692,00€100mg938,00€1mL*10mM (DMSO)283,00€Shanzhiside methyl ester
CAS:Shanzhiside methylester soothes neuropathic pain by triggering spinal GLP-1 receptors, boosting microglial β-endorphin through p38 MAPK.Fórmula:C17H26O11Pureza:99.32%Forma y color:SolidPeso molecular:406.38GLP-1 receptor agonist 9
CAS:1H-Benzimidazole-6-carboxylic acid is a GLP-1 receptor agonist.Fórmula:C32H31ClFN3O5Pureza:98%Forma y color:SolidPeso molecular:592.06Tirzepatide
CAS:Tirzepatide (LY-3298176) is a dual agonist of GIP and GLP-1 receptors with neuroprotective activity and can be used to study diabetes and obesity.Fórmula:C225H348N48O68Pureza:99.52% - 99.99%Forma y color:SolidPeso molecular:4813.45Exendin-4
CAS:Exenatide: GLP-1 receptor agonist, 39-amino acid, longer half-life (2.4 hrs), IC50 of 3.22 nM.Fórmula:C184H282N50O60SPureza:97.71% - 99.72%Forma y color:SolidPeso molecular:4186.57PF-06882961 Tris
CAS:PF-06882961 Tris (UNII-2HJV78O0SS) is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.Fórmula:C35H41FN6O7Pureza:98.11% - 99.79%Forma y color:SolidPeso molecular:676.7GLP-1(7-37) acetate(106612-94-6 free base)
CAS:Glp-1(7-37) acetate is an intestinal insulin hormone that enhances glucose-induced insulin secretion.Fórmula:C151H228N40O47Pureza:98.89%Forma y color:SolidPeso molecular:3355.67PF-06291874
CAS:PF-06291874 (Glucagon receptor antagonists-4) (Glucagon receptor antagonists-4) is a highly effective and orally active antagonist of the glucagon receptor.Fórmula:C26H28F3N3O4Pureza:99.12%Forma y color:SolidPeso molecular:503.51GLP-1(7-36), amide
CAS:GLP-1 secretion by human enteroendocrine NCI-H716 cells is augmented in a dose-dependent manner by the addition of CPE.Cost-effective and quality-assured.Fórmula:C149H226N40O45Pureza:99.85%Forma y color:White PowderPeso molecular:3297.63Adomeglivant
CAS:Adomeglivant (LY2409021) is a potent and selective glucagon receptor antagonist. Which is used in clinical trial for type 2 diabetes mellitus.Fórmula:C32H36F3NO4Pureza:99.97%Forma y color:SolidPeso molecular:555.63Ref: TM-T14130
5mg116,00€10mg188,00€25mg323,00€50mg568,00€100mg949,00€200mg1.424,00€1mL*10mM (DMSO)137,00€PF-06882961
CAS:PF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.Fórmula:C31H30FN5O4Pureza:95.1% - 99.54%Forma y color:SolidPeso molecular:555.6GLP-1 receptor agonist 9 citrate
GLP-1 receptor agonist 9 citrate is an agonist of GLP-1.Fórmula:C38H39ClFN3O12Pureza:95%Forma y color:SolidPeso molecular:784.18GLP-1R modulator C5
CAS:GLP-1R modulator C5 is a GLP-1R modulator that enhances GLP-1 binding to GLP-1R via transmembrane sites and can be used in the study of type II diabetes.Fórmula:C24H21NO3Pureza:99.59%Forma y color:SolidPeso molecular:371.43BETP
CAS:BETP is an agonist of GLP-1 receptor (EC50s: 0.66 and 0.755 μM for human and rat GLP-1 receptor).Fórmula:C20H17F3N2O2SPureza:98.51%Forma y color:SolidPeso molecular:406.42Lixisenatide acetate (320367-13-3 free base)
CAS:Lixisenatide acetate is a receptor agonist similar to glucagon-like peptide-1 (glp-1) for the treatment of type 2 diabetes mellitus (T2DM).Fórmula:C215H347N61O65S·6C2H4O2Pureza:98% - 99.9%Forma y color:SolidPeso molecular:5218.88Secretin (33-59), rat
CAS:Secretin (33-59), rat (Secretin (rat)) is a classical hormone in the gastrointestinal system and a neuropeptide.Fórmula:C129H216N42O42Pureza:98.12%Forma y color:SolidPeso molecular:3027.35GRA Ex-25
CAS:GRA Ex-25 (GRA-Ex-25) is an inhibitor of glucagon receptor.Fórmula:C29H36F3N3O5Pureza:98.2% - 98.88%Forma y color:SolidPeso molecular:563.61Ref: TM-T3422
1mg63,00€2mg88,00€5mg139,00€10mg205,00€25mg419,00€50mg617,00€100mg879,00€1mL*10mM (DMSO)187,00€LSN3318839
CAS:LSN3318839 is a potent and orally available glucagon-like peptide-1 receptor (GLP-1R) modulator.LSN3318839 enhances GLP-1R G-protein-coupled signaling and canFórmula:C26H23Cl2N3O2Pureza:99.43%Forma y color:SolidPeso molecular:480.39Retatrutide
CAS:Retatrutide (LY3437943) is a triple agonist of GCGR, GIPR and GLP-1R that can be used to study obesity.Fórmula:C221H342N46O68Pureza:98.31%Forma y color:SolidPeso molecular:4732.09Glucagon (1-29), bovine, human, porcine hydrochloride
CAS:Glucagon (1-29), bovine, human, porcine hydrochloride is a peptide hormone, produced by pancreatic α-cells. Glucagon increases HNF4α phosphorylation.Fórmula:C153H225N43O49S·ClHPureza:95.65% - 98.03%Forma y color:SolidPeso molecular:3519.21GLP-1R agonist 3
CAS:GLP-1R agonist 3 is a GLP-1R agonist, an imidazole derivative.GLP-1R agonist 3 can be used to study diabetes and obesity.Fórmula:C31H28FN5O4Pureza:97.19%Forma y color:SolidPeso molecular:553.58GLP-1R modulator C16
CAS:GLP-1R modulator C16 is a variable modulator that significantly increases the binding affinity of GLP-4.Fórmula:C21H26ClFN2O3Pureza:99.6% - 99.6%Forma y color:SolidPeso molecular:408.89Liraglutide
CAS:Liraglutide (Liraglutida) is a synthetic analog of GLP-1, an agonist of the GLP-1 receptor. Liraglutide is an antidiabetic agent. Cost effective and quality assured.Fórmula:C172H265N43O51Pureza:99.04%Forma y color:SolidPeso molecular:3751.25NNC-0640
CAS:NNC-0640 is a negative allosteric modulator of Human Glucagon Receptor with an IC50 of 69.2 nM.Fórmula:C29H31N7O4SPureza:97.04%Forma y color:SolidPeso molecular:573.67Ref: TM-T7364
1mg48,00€2mg65,00€5mg96,00€10mg169,00€25mg298,00€50mg454,00€100mg655,00€1mL*10mM (DMSO)96,00€GLP-1R Antagonist 1
CAS:GLP-1R Antagonist 1 is an orally active, CNS penetrant and non-competitive glucagon-like peptide 1 receptor (GLP-1R) antagonist (IC50: 650 nM).Fórmula:C16H11ClF6N4O2Pureza:99.64%Forma y color:SolidPeso molecular:440.73Semaglutide TFA
Semaglutide TFA is a glucagon-like peptide-1 congener that induces weight loss, lowers blood glucose levels and reduces cardiovascular risk in diabetic patientsFórmula:C189H290F3N45O61Pureza:99.69%Forma y color:SolidPeso molecular:4225.6482L-168049
CAS:L-168049: Human glucagon receptor antagonist, IC50 - 3.7 nM human, 63 nM murine, 60 nM canine.Fórmula:C24H20BrClN2OPureza:100%Forma y color:SolidPeso molecular:467.79Ref: TM-T22893
1mg52,00€5mg111,00€10mg180,00€25mg378,00€50mg560,00€100mg800,00€500mg1.644,00€1mL*10mM (DMSO)123,00€GLP-1R Agonist DMB
CAS:GLP-1R Agonist DMB is an agonist of glucagon-like peptide 1 receptor (GLP-1R; KB = 26.3 nM for the recombinant human receptor).Fórmula:C13H15Cl2N3O2SPureza:99.52%Forma y color:SolidPeso molecular:348.25Anti-GCGR Antibody (7J909)
Anti-GCGR Antibody (7J909) is an antibody targeting GCGR. Anti-GCGR Antibody (7J909) can be used in ELISA.Forma y color:Odour Liquid
