
Receptor de dopamina
Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.
Productos de "Receptor de dopamina"
Ordenar por
NRA-0160
CAS:NRA-0160 is a selective antagonist of dopamine D4 receptor(Ki of 0.48 nM)Fórmula:C24H23F2N3OSPureza:98%Forma y color:SolidPeso molecular:439.52Tiaspirone hydrochloride
CAS:Tiaspirone hydrochloride (BMY-13859 hydrochloride) exhibits antipsychotic activity and influences the electrophysiological activity of dopaminergic neurons.Fórmula:C24H33ClN4O2SPureza:99.98%Forma y color:SoildPeso molecular:477.065-HT6/7 antagonist 1
CAS:5-HT6/7 antagonist 1 is a dual 5-HT6/7/2A and D2 receptor antagonist for the study of dementia and Alzheimer's disease.Fórmula:C22H20FN3O3Pureza:98.55% - 98.78%Forma y color:SolidPeso molecular:393.41Benperidol
CAS:Benperidol (Anquil), a butanone derivative, has antipsychotic effects and blocks D2 receptors; useful in PET scans.Fórmula:C22H24FN3O2Pureza:97.39%Forma y color:SolidPeso molecular:381.44Ref: TM-T26360
1mg116,00€5mg276,00€10mg410,00€25mg680,00€50mg938,00€100mg1.293,00€500mg2.593,00€1mL*10mM (DMSO)279,00€Liafensine
CAS:Liafensine(BMS-820836): Selective inhibitor for serotonin, norepinephrine, dopamine reuptake; targets major depression, CNS disorders.Fórmula:C24H22N4Pureza:99.46%Forma y color:SolidPeso molecular:366.46Asenapine
CAS:Asenapine (Org 5222) is a 5-HT receptor, adrenergic receptor, and histamine receptor antagonist with antipsychotic properties for the treatment of schizophreniaFórmula:C17H16ClNOPureza:99.16%Forma y color:CoaPeso molecular:285.77SLV-310
CAS:SLV-310 is a D2 receptor antagonist and 5-HT reuptake receptor inhibitor for the study of neurological disorders such as bipolar disorder and schizophrenia.Fórmula:C25H24FN3O2Pureza:98.91%Forma y color:SolidPeso molecular:417.48D3R/MOR antagonist 1
Compound 114 (D3R/MOR antagonist 1) exhibits dual antagonistic activity at dopamine D3 receptors (D3R) and mu-opioid receptors (MOR), with K i values of 46.5 nMFórmula:C22H27Cl2N3OPureza:98%Forma y color:SolidPeso molecular:420.38Metoclopramide hydrochloride
CAS:Metoclopramide hydrochloride (Metoclopramide HCl) is a selective dopamine D2 receptor antagonist, used as an antiemetic.Fórmula:C14H22ClN3O2·HClPureza:99.99%Forma y color:White To Off-White PowderPeso molecular:336.26NMI 8739
CAS:NMI 8739 (n-docosahexaenoyl dopamine) is an agonist of D2 autoreceptor.Fórmula:C30H41NO3Pureza:98.51%Forma y color:SolidPeso molecular:463.65Ref: TM-T11079
1mg40,00€5mg85,00€10mg120,00€25mg207,00€50mg303,00€100mg449,00€200mg652,00€1mL*10mM (DMSO)90,00€Itopride hydrochloride
CAS:Itopride hydrochloride (Ganaton) is an AChE and D2DR inhibitor.Fórmula:C20H27ClN2O4Pureza:99.59%Forma y color:White Or Pale Brownish CrystalPeso molecular:394.9Oxolinic acid
CAS:Oxolinic acid (Nidantin) is a synthetic antimicrobial related to NALIDIXIC ACID and used in URINARY TRACT INFECTIONS.Fórmula:C13H11NO5Pureza:98.39% - 99.72%Forma y color:Crystals From Dimethylformamide White Crystalline PowderPeso molecular:261.23Fluphenazine decanoate
CAS:Fluphenazine decanoate is dopamine D2 receptor blocke,and is a long-acting phenothiazine neuroleptic that used to treat schizophrenia.Fórmula:C32H44F3N3O2SPureza:100% - 98.14%Forma y color:SolidPeso molecular:591.77Benztropine mesylate
CAS:Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSONFórmula:C21H25NO·CH4SO3Pureza:98.41% - 99.96%Forma y color:White Crystalline Powder; Odourless Or Almost OdourlessPeso molecular:403.53Syrosingopine
CAS:Syrosingopine is a dual inhibitor of MCT1 and MCT4, 60 times more potent against MCT4, preventing lactate and H+ efflux.Cost-effective and quality-assured.Fórmula:C35H42N2O11Pureza:99.25% - 99.78%Forma y color:SolidPeso molecular:666.71Ref: TM-TN2252
1mg66,00€5mg142,00€10mg212,00€25mg361,00€50mg543,00€100mg750,00€1mL*10mM (DMSO)202,00€GR 103691
CAS:GR 103691 is a potent, selective dopamine D3 receptor antagonist (Ki: 0.4 nM).Fórmula:C30H35N3O3Pureza:98.94% - 99.29%Forma y color:SolidPeso molecular:485.62Ref: TM-T11463
2mg46,00€5mg66,00€10mg99,00€25mg197,00€50mg311,00€100mg505,00€500mg1.121,00€1mL*10mM (DMSO)74,00€PF-00217830
CAS:PF-00217830: agonist at serotonin 1A & dopamine D2, antagonist at serotonin 2A, potential schizophrenia study drug.Fórmula:C26H30N4O2Pureza:98.30%Forma y color:SolidPeso molecular:430.54Aniracetam
CAS:Aniracetam (Ro 13-5057)(Ro 13-5057), a nootropic and neuroprotective drug, selectively modulates the AMPA receptor and nAChR.Fórmula:C12H13NO3Pureza:99.88% - 99.89%Forma y color:White Crystalline Or Crystalline PowdePeso molecular:219.24Oxidopamine hydrobromide
CAS:Oxidopamine hydrobromide (6-OHDA hydrobromide) is a neurotransmitter dopamine antagonist.Fórmula:C8H12BrNO3Pureza:98.1% - 99.88%Forma y color:Beige To Brown Fine Crystalline PowderPeso molecular:250.09Flunarizine dihydrochloride
CAS:Flunarizine dihydrochloride: a calcium blocker also targeting calmodulin and histamine H1, used for migraine, vertigo, vascular disease, and epilepsy aid.Fórmula:C26H28Cl2F2N2Pureza:99.53% - 99.89%Forma y color:White Crystalline Powder Odorless And TastelessPeso molecular:477.42