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Receptor de dopamina

Receptor de dopamina

Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.

Productos de "Receptor de dopamina"

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productos por página.Hay 309 productos en esta categoría.
  • NRA-0160

    CAS:
    NRA-0160 is a selective antagonist of dopamine D4 receptor(Ki of 0.48 nM)
    Fórmula:C24H23F2N3OS
    Pureza:98%
    Forma y color:Solid
    Peso molecular:439.52

    Ref: TM-T12252

    25mg
    1.444,00€
    50mg
    1.882,00€
    100mg
    2.375,00€
  • Tiaspirone hydrochloride

    CAS:
    Tiaspirone hydrochloride (BMY-13859 hydrochloride) exhibits antipsychotic activity and influences the electrophysiological activity of dopaminergic neurons.
    Fórmula:C24H33ClN4O2S
    Pureza:99.98%
    Forma y color:Soild
    Peso molecular:477.06

    Ref: TM-T24885L

    1mg
    185,00€
    5mg
    459,00€
    10mg
    657,00€
    25mg
    1.026,00€
    50mg
    1.415,00€
    1mL*10mM (DMSO)
    47,00€
  • 5-HT6/7 antagonist 1

    CAS:
    5-HT6/7 antagonist 1 is a dual 5-HT6/7/2A and D2 receptor antagonist for the study of dementia and Alzheimer's disease.
    Fórmula:C22H20FN3O3
    Pureza:98.55% - 98.78%
    Forma y color:Solid
    Peso molecular:393.41

    Ref: TM-T61807

    1mg
    665,00€
    5mg
    1.681,00€
  • Benperidol

    CAS:
    Benperidol (Anquil), a butanone derivative, has antipsychotic effects and blocks D2 receptors; useful in PET scans.
    Fórmula:C22H24FN3O2
    Pureza:97.39%
    Forma y color:Solid
    Peso molecular:381.44

    Ref: TM-T26360

    1mg
    116,00€
    5mg
    276,00€
    10mg
    410,00€
    25mg
    680,00€
    50mg
    938,00€
    100mg
    1.293,00€
    500mg
    2.593,00€
    1mL*10mM (DMSO)
    279,00€
  • Liafensine

    CAS:
    Liafensine(BMS-820836): Selective inhibitor for serotonin, norepinephrine, dopamine reuptake; targets major depression, CNS disorders.
    Fórmula:C24H22N4
    Pureza:99.46%
    Forma y color:Solid
    Peso molecular:366.46

    Ref: TM-T32737

    1mg
    368,00€
    5mg
    877,00€
    10mg
    1.198,00€
    25mg
    1.776,00€
    50mg
    2.395,00€
  • Asenapine

    CAS:
    Asenapine (Org 5222) is a 5-HT receptor, adrenergic receptor, and histamine receptor antagonist with antipsychotic properties for the treatment of schizophrenia
    Fórmula:C17H16ClNO
    Pureza:99.16%
    Forma y color:Coa
    Peso molecular:285.77

    Ref: TM-T21360

    1mg
    38,00€
    5mg
    79,00€
    10mg
    97,00€
    25mg
    165,00€
    50mg
    235,00€
    100mg
    346,00€
    1mL*10mM (DMSO)
    88,00€
  • SLV-310

    CAS:
    SLV-310 is a D2 receptor antagonist and 5-HT reuptake receptor inhibitor for the study of neurological disorders such as bipolar disorder and schizophrenia.
    Fórmula:C25H24FN3O2
    Pureza:98.91%
    Forma y color:Solid
    Peso molecular:417.48

    Ref: TM-T28809

    1mg
    279,00€
    5mg
    685,00€
    10mg
    938,00€
    25mg
    1.444,00€
    50mg
    1.882,00€
    100mg
    2.375,00€
  • D3R/MOR antagonist 1


    Compound 114 (D3R/MOR antagonist 1) exhibits dual antagonistic activity at dopamine D3 receptors (D3R) and mu-opioid receptors (MOR), with K i values of 46.5 nM
    Fórmula:C22H27Cl2N3O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:420.38

    Ref: TM-T78778

    5mg
    A consultar
    50mg
    A consultar
  • Metoclopramide hydrochloride

    CAS:
    Metoclopramide hydrochloride (Metoclopramide HCl) is a selective dopamine D2 receptor antagonist, used as an antiemetic.
    Fórmula:C14H22ClN3O2·HCl
    Pureza:99.99%
    Forma y color:White To Off-White Powder
    Peso molecular:336.26

    Ref: TM-T1069

    10mg
    39,00€
    25mg
    55,00€
    50mg
    78,00€
    100mg
    90,00€
    200mg
    144,00€
    500mg
    230,00€
    1mL*10mM (DMSO)
    47,00€
  • NMI 8739

    CAS:
    NMI 8739 (n-docosahexaenoyl dopamine) is an agonist of D2 autoreceptor.
    Fórmula:C30H41NO3
    Pureza:98.51%
    Forma y color:Solid
    Peso molecular:463.65

    Ref: TM-T11079

    1mg
    40,00€
    5mg
    85,00€
    10mg
    120,00€
    25mg
    207,00€
    50mg
    303,00€
    100mg
    449,00€
    200mg
    652,00€
    1mL*10mM (DMSO)
    90,00€
  • Itopride hydrochloride

    CAS:
    Itopride hydrochloride (Ganaton) is an AChE and D2DR inhibitor.
    Fórmula:C20H27ClN2O4
    Pureza:99.59%
    Forma y color:White Or Pale Brownish Crystal
    Peso molecular:394.9

    Ref: TM-T1552

    50mg
    35,00€
    100mg
    49,00€
    500mg
    81,00€
    1mL*10mM (DMSO)
    50,00€
  • Oxolinic acid

    CAS:
    Oxolinic acid (Nidantin) is a synthetic antimicrobial related to NALIDIXIC ACID and used in URINARY TRACT INFECTIONS.
    Fórmula:C13H11NO5
    Pureza:98.39% - 99.72%
    Forma y color:Crystals From Dimethylformamide White Crystalline Powder
    Peso molecular:261.23

    Ref: TM-T1233

    1g
    37,00€
    5g
    70,00€
    10g
    104,00€
  • Fluphenazine decanoate

    CAS:
    Fluphenazine decanoate is dopamine D2 receptor blocke,and is a long-acting phenothiazine neuroleptic that used to treat schizophrenia.
    Fórmula:C32H44F3N3O2S
    Pureza:100% - 98.14%
    Forma y color:Solid
    Peso molecular:591.77

    Ref: TM-T7943

    5mg
    43,00€
    10mg
    66,00€
    25mg
    90,00€
    50mg
    104,00€
    100mg
    170,00€
    200mg
    255,00€
    1mL*10mM (DMSO)
    51,00€
  • Benztropine mesylate

    CAS:
    Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON
    Fórmula:C21H25NO·CH4SO3
    Pureza:98.41% - 99.96%
    Forma y color:White Crystalline Powder; Odourless Or Almost Odourless
    Peso molecular:403.53

    Ref: TM-T1336

    500mg
    34,00€
  • Syrosingopine

    CAS:
    Syrosingopine is a dual inhibitor of MCT1 and MCT4, 60 times more potent against MCT4, preventing lactate and H+ efflux.Cost-effective and quality-assured.
    Fórmula:C35H42N2O11
    Pureza:99.25% - 99.78%
    Forma y color:Solid
    Peso molecular:666.71

    Ref: TM-TN2252

    1mg
    66,00€
    5mg
    142,00€
    10mg
    212,00€
    25mg
    361,00€
    50mg
    543,00€
    100mg
    750,00€
    1mL*10mM (DMSO)
    202,00€
  • GR 103691

    CAS:
    GR 103691 is a potent, selective dopamine D3 receptor antagonist (Ki: 0.4 nM).
    Fórmula:C30H35N3O3
    Pureza:98.94% - 99.29%
    Forma y color:Solid
    Peso molecular:485.62

    Ref: TM-T11463

    2mg
    46,00€
    5mg
    66,00€
    10mg
    99,00€
    25mg
    197,00€
    50mg
    311,00€
    100mg
    505,00€
    500mg
    1.121,00€
    1mL*10mM (DMSO)
    74,00€
  • PF-00217830

    CAS:
    PF-00217830: agonist at serotonin 1A & dopamine D2, antagonist at serotonin 2A, potential schizophrenia study drug.
    Fórmula:C26H30N4O2
    Pureza:98.30%
    Forma y color:Solid
    Peso molecular:430.54

    Ref: TM-T24613

    1mg
    94,00€
    5mg
    205,00€
    10mg
    303,00€
    25mg
    490,00€
    50mg
    710,00€
    100mg
    998,00€
    200mg
    1.349,00€
  • Aniracetam

    CAS:
    Aniracetam (Ro 13-5057)(Ro 13-5057), a nootropic and neuroprotective drug, selectively modulates the AMPA receptor and nAChR.
    Fórmula:C12H13NO3
    Pureza:99.88% - 99.89%
    Forma y color:White Crystalline Or Crystalline Powde
    Peso molecular:219.24

    Ref: TM-T0333

    1g
    52,00€
    1mL*10mM (DMSO)
    34,00€
  • Oxidopamine hydrobromide

    CAS:
    Oxidopamine hydrobromide (6-OHDA hydrobromide) is a neurotransmitter dopamine antagonist.
    Fórmula:C8H12BrNO3
    Pureza:98.1% - 99.88%
    Forma y color:Beige To Brown Fine Crystalline Powder
    Peso molecular:250.09

    Ref: TM-T12352L

    1g
    263,00€
    100mg
    62,00€
    200mg
    89,00€
    500mg
    168,00€
  • Flunarizine dihydrochloride

    CAS:
    Flunarizine dihydrochloride: a calcium blocker also targeting calmodulin and histamine H1, used for migraine, vertigo, vascular disease, and epilepsy aid.
    Fórmula:C26H28Cl2F2N2
    Pureza:99.53% - 99.89%
    Forma y color:White Crystalline Powder Odorless And Tasteless
    Peso molecular:477.42

    Ref: TM-T0806

    1g
    66,00€
    500mg
    48,00€
    1mL*10mM (DMSO)
    50,00€