Receptor de cannabinoides
Los receptores cannabinoides son GPCR que median los efectos de los cannabinoides endógenos (endocannabinoides) y los fitocannabinoides, como los encontrados en el cannabis. Los dos tipos principales de receptores cannabinoides, CB1 y CB2, están involucrados en la regulación de una amplia gama de procesos fisiológicos, incluida la percepción del dolor, el apetito, el estado de ánimo y la función inmunitaria. Los moduladores de los receptores cannabinoides tienen potencial terapéutico en el tratamiento de afecciones como el dolor crónico, la epilepsia y la esclerosis múltiple. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores cannabinoides de alta calidad para apoyar su investigación en neurofarmacología, manejo del dolor e inmunología.
Productos de "Receptor de cannabinoides"
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CB1/2 agonist 3
CAS:CB1/2 agonist 3 is a competitive and potent CB1/CB2 agonist with high affinity for hCB1 and hCB2 and can be used to study neurological disorders.Fórmula:C25H41NO2Pureza:98.78%Forma y color:SolidPeso molecular:387.6β-Caryophyllene
CAS:β-Caryophyllene ((-)-(E)-Caryophyllene) acts as an CB2 receptor agonist.Fórmula:C15H24Pureza:95.43% - 99.11%Forma y color:Turpentine (Ntp 1992)Peso molecular:204.35Pregnenolone monosulfate sodium
CAS:Pregnenolone monosulfate sodium salt is an neurosteroid, enhances NMDA receptor,CREB phosphorylation, TRPM3 channels, and may inhibit GABA A receptors.Fórmula:C21H31NaO5SPureza:99.763%Forma y color:SolidPeso molecular:418.52Noladin ether
CAS:Noladin ether (2-AG ether) is a cannabinoid CB1 receptor agonist.Fórmula:C23H40O3Forma y color:SolidPeso molecular:364.56Otenabant
CAS:Otenabant (CP-945598) has been investigated for the treatment of Obesity.Fórmula:C25H25Cl2N7OPureza:100%Forma y color:SolidPeso molecular:510.42OMDM-6
CAS:OMDM-6 is a dual agonist of TRPV1(EC50 = 75 nM) and CB1 (Ki = 3.2 μM). OMDM-6 inhibits anandamide cellular uptake with a Ki of 7.0 μM.Fórmula:C28H42N2O3Pureza:99.49%Forma y color:SolidPeso molecular:454.64Ref: TM-T12307
1mg115,00€5mg255,00€10mg375,00€25mg562,00€50mg787,00€100mg1.074,00€200mg1.444,00€1mL*10mM (DMSO)283,00€CB1R antagonist 1
CAS:CB1R antagonist 1 is a potent CB1R antagonist that can be used to study diseases related to the nervous system.Fórmula:C18H23F3N2O3SPureza:99.65%Forma y color:SolidPeso molecular:404.45(±)-Ibipinabant
CAS:(±)-Ibipinabant ((±)-SLV319) has been used in trials studying the treatment of Obesity and Obesity and Type 2 Diabetes.Fórmula:C23H20Cl2N4O2SPureza:99.28% - 99.83%Forma y color:SolidPeso molecular:487.4Olorinab
CAS:Olorinab (APD 371) (APD 371) is a highly potent, selective and fully efficacious cannabinoid receptor type 2 (CB2) agonist. With an EC50 of 6.2 nM for hCB2.Fórmula:C18H23N5O3Pureza:97.13% - 97.67%Forma y color:SolidPeso molecular:357.41BAY 38-7271
CAS:BAY 38-7271: potent neuroprotective, selective CB1/CB2 agonist, Ki of 1.85 nM (CB1) & 5.96 nM (CB2).Fórmula:C20H21F3O5SPureza:98%Forma y color:SolidPeso molecular:430.44CB2R agonist 2
CB2R agonist 2 (cis-17-para) is a CB2R agonist [1].Pureza:98%Forma y color:Odour SolidCannabigerol
CAS:Cannabigerol is a high affinity α±2-adrenergic receptor agonist, moderate affinity 5-HT1A receptor antagonist, and low affinity CB1 receptor antagonist ; alsoFórmula:C21H32O2Pureza:99.23% - 99.92%Forma y color:SolidPeso molecular:316.48Ref: TM-TN1465
1mg145,00€2mg215,00€5mg314,00€10mg474,00€25mg808,00€50mg1.111,00€100mg1.501,00€1mL*10mM (DMSO)324,00€Dehydroabiethylamine
CAS:Dehydroabiethylamine (NSC-2955) boosts liver CYP2B, blocks PDKs & cholesterol transport, and has anti-tumor effects.Fórmula:C20H31NPureza:97.24%Forma y color:Pale Yellow Viscous Liquid /Technical Grade/ Viscous Colorless To Amber LiquidPeso molecular:285.47MDA77
CAS:MDA77 is a CB2 agonist with an EC50 value of 5.82 nM and exhibits no activity towards CB1.Fórmula:C21H23N3O3Forma y color:SolidPeso molecular:365.43TRPV1/CB2 agonist 1
TRPV1/CB2 agonist 1 (compound 41) is a dual agonist targeting hTRPV1 and CB2 receptors, with an EC50 value of 26.8 μM for hTRPV1. It is applicable in research related to the nervous system.Forma y color:Odour SolidO-1602
CAS:O-1602 is a novel GPR55 agonist, an atypical cannabinoid associated with the central nervous system and obesity, and is a candidate compound for the treatmentFórmula:C17H22O2Pureza:99.4%Forma y color:SolidPeso molecular:258.36CB1 inverse agonist 1
CAS:MRL-650 is an oral, selective CB1 agonist; IC50: CB1=7.5 nM, CB2=4100 nM; anorexigenic effects noted.Fórmula:C25H18Cl3N3O3Pureza:99.12%Forma y color:SolidPeso molecular:514.79Ref: TM-T10694
1mg77,00€5mg158,00€10mg225,00€25mg338,00€50mg472,00€100mg645,00€200mg869,00€1mL*10mM (DMSO)187,00€NESS 0327
CAS:NESS 0327 is a high selectivity antagonist of the cannabinoid CB1 receptor. NESS 0327 is more than 60,000-fold selective for the CB1 receptor.Fórmula:C24H23Cl3N4OPureza:99.74%Forma y color:SolidPeso molecular:489.82CB1 agonist 1
CAS:CB1 agonist 1 is a potent CB1 agonist with a pIC50 value of 5.7 for CB1 receptors.CB1 agonist 1 can be used to study brain disorders, pain, and inflammation.Fórmula:C24H24N2O5SPureza:98.56%Forma y color:SolidPeso molecular:452.52Tetrahydromagnolol
CAS:Tetrahydromagnolol can activate cannabinoid (CB) receptors.Fórmula:C18H22O2Pureza:100% - 99.82%Forma y color:SolidPeso molecular:270.37
