Receptor de cannabinoides
Los receptores cannabinoides son GPCR que median los efectos de los cannabinoides endógenos (endocannabinoides) y los fitocannabinoides, como los encontrados en el cannabis. Los dos tipos principales de receptores cannabinoides, CB1 y CB2, están involucrados en la regulación de una amplia gama de procesos fisiológicos, incluida la percepción del dolor, el apetito, el estado de ánimo y la función inmunitaria. Los moduladores de los receptores cannabinoides tienen potencial terapéutico en el tratamiento de afecciones como el dolor crónico, la epilepsia y la esclerosis múltiple. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores cannabinoides de alta calidad para apoyar su investigación en neurofarmacología, manejo del dolor e inmunología.
Productos de "Receptor de cannabinoides"
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LY2828360
CAS:LY2828360: CB2 agonist, Ki=40.3 nM; biases CB2 over CB1 with EC50s of 20.1 nM and >100 μM.Fórmula:C22H27ClN6OPureza:98.45% - 99.51%Forma y color:SolidPeso molecular:426.94FDU-PB-22
CAS:FDU-PB-22, a novel synthetic cannabinoid, undergoes rapid metabolism in human liver microsomes (HLM) with a half-life of 12.4 minutes.Fórmula:C26H18FNO2Forma y color:SolidPeso molecular:395.43CB1 antagonist 1
CAS:CB1 antagonist 1 is a CB1 receptor antagonist, used in the research of obesity and metabolic syndrome, neuroinflammatory disorders, cognitive disorders, andFórmula:C26H22Cl2N4Pureza:98%Forma y color:SolidPeso molecular:461.39APP-FUBINACA
CAS:APP-FUBINACA is a cannabinoid receptor agonist, classified as a phenylalanine amide-based indazole-3-carboxamide derivative. It exhibits neurostimulatory effects.Fórmula:C24H21FN4O2Forma y color:SolidPeso molecular:416.45MJ 15
CAS:MJ 15 is a CB1 receptor antagonist with specificity for the study of obesity-induced diseases.Fórmula:C23H17Cl3N4OPureza:99.63%Forma y color:SolidPeso molecular:471.77Afubiata
CAS:ADB-FUBIATA is a synthetic cannabinoid studied for its metabolic profile, along with AFUBIATA, CH-FUBIATA, and CH-PIATA. This in vitro analysis by Watanabe S, et al., examines these compounds, as published in "Arch Toxicol," 2023 Dec;97(12):3085-3094.Fórmula:C27H29FN2OForma y color:SolidPeso molecular:416.53AM281
CAS:AM 281, a cannabinoid antagonist, reduces neurologic dysfunction and mortality rate after cecal ligation and puncture in rats.Fórmula:C21H19Cl2IN4O2Pureza:100% - 99.2%Forma y color:White To Off-White SolidPeso molecular:557.21Ref: TM-T2264
1mg85,00€5mg172,00€10mg274,00€25mg552,00€50mg792,00€100mg1.093,00€500mg2.175,00€1mL*10mM (DMSO)245,00€PSB-SB-487
CAS:PSB-SB-487 is antagonist of GPR55.Fórmula:C26H32O4Pureza:98.53%Forma y color:SolidPeso molecular:408.53Ref: TM-T8975
1mg38,00€5mg85,00€10mg126,00€25mg245,00€50mg364,00€100mg507,00€200mg697,00€1mL*10mM (DMSO)93,00€MDA7
CAS:MDA7 is a selective agonist of the cannabinoid receptor 2 (CB2), demonstrating an EC50 of 128 nM in human CB2 receptors and 67.4 nM in rat CB2 receptors. The compound exhibits good affinity for CB2 receptors, with Ki values of 422 nM for humans and 238 nM for rats. In rat models, MDA7 shows analgesic activity.Fórmula:C22H25NO2Forma y color:SolidPeso molecular:335.439Drinabant
CAS:Drinabant (AVE-1625) is an orally active CB1 receptor antagonist.Fórmula:C23H20Cl2F2N2O2SPureza:99.8%Forma y color:SolidPeso molecular:497.38Ref: TM-T21861
1mg87,00€2mg116,00€5mg170,00€10mg259,00€25mg425,00€50mg598,00€100mg810,00€500mg1.624,00€AM6545
CAS:AM6545 is a CB1 receptor antagonist used in the study of obesity and diabetes.Fórmula:C26H23Cl2N5O3SPureza:97.03%Forma y color:SolidPeso molecular:556.46PSNCBAM-1
CAS:PSNCBAM-1 (PSNCBAM 1) is a CB1 receptor negative allosteric modulator (EC50 = 0.1 μM) with hypophagic effects in vivo.Fórmula:C22H21ClN4OPureza:98.18%Forma y color:SolidPeso molecular:392.88L-α-lysophosphatidylinositol sodium
CAS:L-α-lysophosphatidylinositol sodium is an endogenous ligand of GPR55 and an endocannabinoid neurotransmitter.Fórmula:C25H48NaO12PForma y color:SolidPeso molecular:594.6Falcarinol
CAS:Falcarinol, also known as Panaxynol, is a naturally occurring compound that acts as an orally active inhibitor of Hsp90.Fórmula:C17H24OPureza:98%Forma y color:SolidPeso molecular:244.37AM1241
CAS:AM-1241 is a selective cannabinoid CB2 receptor agonist with Ki of 3.4 nM, exhibits 82-fold selectivity over CB1 receptor.Fórmula:C22H22IN3O3Pureza:98.82% - 99.10%Forma y color:SolidPeso molecular:503.33Ref: TM-T6755
2mg38,00€5mg51,00€10mg88,00€25mg172,00€50mg290,00€100mg523,00€500mg1.130,00€1mL*10mM (DMSO)93,00€GW 405833
CAS:GW 405833 (L-768242) is an agonist of cannabinoid-2 (CB(2)) receptor-selectiveFórmula:C23H24Cl2N2O3Pureza:99.82% - 99.93%Forma y color:SolidPeso molecular:447.35Linoleoyl Ethanolamide
CAS:Linoleoyl Ethanolamide is an endocannabinoid agent.Fórmula:C20H37NO2Pureza:99.97%Forma y color:SolidPeso molecular:323.51Ref: TM-T8425
1mg35,00€5mg67,00€10mg90,00€25mg164,00€50mg239,00€100mg348,00€200mg522,00€1mL*10mM (DMSO)85,00€Anandamide
CAS:Anandamide ((5Z,8Z,11Z,14Z)-N-(2-Hydroxyethyl)icosa-5,8,11,14-tetraenamide), an immune modulator, acts via not only cannabinoid receptors (CB1 and CB2) but alsoFórmula:C22H37NO2Pureza:98.76% - 99.22%Forma y color:Light Yellow OilPeso molecular:347.53Ref: TM-T14046
1mg35,00€2mg49,00€5mg74,00€10mg131,00€25mg246,00€50mg366,00€100mg538,00€200mg752,00€1mL*10mM (DMSO)81,00€exo-Tetrahydrocannabivarin
CAS:exo-Tetrahydrocannabivarin (Compound 12) is an analog of Δ9,11-THC. It weakly binds to cannabinoid receptors (CB) with an IC50 of 1.4 μM. In mice, exo-Tetrahydrocannabivarin exhibits activity related to both motor function and analgesia.Fórmula:C19H26O2Forma y color:SolidPeso molecular:286.41Arvanil
CAS:Arvanil (N-Vanillylarachidonamide) is a synthetic capsaicin-amphetamine hybrid that acts as a ligand for VR1 and CB1, offering neuroprotective effects.Fórmula:C28H41NO3Pureza:99.49%Forma y color:SolidPeso molecular:439.63
