
Receptor GNRH
Los receptores de la hormona liberadora de gonadotropinas (GnRH) son GPCR que se unen a la GnRH, una hormona responsable de regular la liberación de la hormona luteinizante (LH) y la hormona foliculoestimulante (FSH) de la glándula pituitaria. Estos receptores son cruciales para la función reproductiva y son el objetivo de terapias para condiciones como el cáncer de próstata, la endometriosis y la infertilidad. Los agonistas y antagonistas de los receptores de GnRH también se utilizan en tecnologías de reproducción asistida. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de GnRH de alta calidad para apoyar su investigación en salud reproductiva, endocrinología y terapia hormonal.
Productos de "Receptor GNRH"
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Hay 14 productos en esta categoría.
Relugolix
CAS:Relugolix (RVT-601) is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, withFórmula:C29H27F2N7O5SPureza:98.64% - 99.67%Forma y color:SolidPeso molecular:623.63Ref: TM-T3630
1mg37,00€5mg79,00€10mg116,00€25mg198,00€50mg329,00€100mg512,00€500mg1.093,00€1mL*10mM (DMSO)96,00€Goserelin acetate
CAS:Goserelin acetate (Fertilan) is a synthetic long-acting agonist of gonadotropin-releasing hormone, used in treatments of cancer.Fórmula:C61H88N18O16Pureza:100% - 99.86%Forma y color:White Crystalline PowderPeso molecular:1329.46Alarelin Acetate
CAS:Alarelin Acetate is a synthetic GnRH agonist which can directly inhibit proliferation and DNA synthesis of rat GSMC through GnRH receptors.Fórmula:C56H78N16O12Pureza:100% - 99.81%Forma y color:White PowderPeso molecular:1167.34Ref: TM-T1494
5mg58,00€10mg95,00€25mg115,00€50mg156,00€100mg180,00€500mg452,00€1mL*10mM (DMSO)120,00€GnRH-R antagonist 1
CAS:Compound 21a: Oral GnRH-R antagonist, IC50=0.57 nM, potent against prostate cancer/prevents LH surges.Fórmula:C31H28F5N7O6SPureza:98%Forma y color:SolidPeso molecular:721.65Abarelix
CAS:Abarelix (PPI 149) is a potent gonadotrophin-releasing hormone (GnRH) antagonist, which is used for prostate cancer treatment.Fórmula:C72H95ClN14O14Pureza:100%Forma y color:SolidPeso molecular:1416.06GnRH antagonist 2
CAS:GnRH antagonist 2 is a GnRH receptor antagonist, useful for studying endocrine diseases.Fórmula:C28H27F2N9O5Pureza:98.08%Forma y color:SolidPeso molecular:607.57Elagolix sodium
CAS:Elagolix sodium (NBI-56418 sodium) is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM, respectively).Fórmula:C32H29F5N3NaO5Pureza:99.71%Forma y color:SolidPeso molecular:653.57Fertirelin
CAS:Fertirelin, or fertirelin acetate, sold under the brand name Ovalyse, is a gonadotropin-releasing hormone agonist (GnRH agonist).Fórmula:C55H76N16O12Pureza:100%Forma y color:SolidPeso molecular:1153.29Ref: TM-TP1288
1mg47,00€2mg63,00€5mg96,00€10mg135,00€50mg177,00€100mg264,00€200mg393,00€1mL*10mM (DMSO)170,00€Linzagolix
CAS:Linzagolix is a small-molecule, non-peptide, orally active gonadotropin-releasing hormone antagonist (GnRH antagonist) which is under development by KisseiFórmula:C22H15F3N2O7SPureza:99.68%Forma y color:SolidPeso molecular:508.42Cetrorelix Acetate
CAS:Cetrorelix Acetate is gonadotropin-releasing hormone (GnRH) receptor antagonist with an IC50 of 1.21 nM.Fórmula:C70H92ClN17O14·xC2H4O2Pureza:97.96%Forma y color:SolidPeso molecular:1491.11Linzagolix choline
CAS:Linzagolix choline is a GnRH antagonist. It can be used to study pain associated with uterine fibroids and endometriosis.Fórmula:C27H28F3N3O8SPureza:99.64%Forma y color:SolidPeso molecular:611.59(R)-Elagolix
CAS:(R)-Elagolix (NBI-56418) is an orally active, highly selective, short-term potent antagonist of the non-peptide gonadotropin-releasing hormone receptor.Fórmula:C32H30F5N3O5Pureza:97.63%Forma y color:SolidPeso molecular:631.59Ref: TM-T11174
1mg38,00€2mg49,00€5mg79,00€10mg111,00€25mg188,00€50mg329,00€100mg487,00€200mg695,00€1mL*10mM (DMSO)96,00€Cetrorelix diacetate
CAS:Cetrorelix diacetate (NS-75A) is is a gonadotropin-releasing hormone antagonist.Fórmula:C74H100ClN17O18Pureza:98.38%Forma y color:SolidPeso molecular:1551.17Ref: TM-T5520L
1mg52,00€5mg90,00€10mg150,00€25mg291,00€50mg437,00€100mg642,00€500mg1.359,00€1mL*10mM (DMSO)251,00€Opigolix
CAS:Opigolix is a Gonadotropin-releasing hormone receptor antagonist.Fórmula:C25H19F3N4O5SPureza:98.07% - 99.54%Forma y color:SolidPeso molecular:544.5