Receptores acoplados de proteína G y receptores 7-TM
Los receptores acoplados a proteínas G (GPCR) y los receptores de 7 dominios transmembrana (7-TM) son una gran familia de proteínas de membrana que desempeñan un papel clave en la comunicación celular y la transducción de señales. Estos receptores están involucrados en una amplia gama de procesos fisiológicos, incluyendo la percepción sensorial, la respuesta inmunitaria y la regulación hormonal. Los GPCR son objetivos principales en el descubrimiento de fármacos, lo que los convierte en esenciales para la investigación en farmacología y medicina. En CymitQuimica, ofrecemos una amplia selección de reactivos y compuestos de alta calidad relacionados con los GPCR y los receptores 7-TM para apoyar su investigación y esfuerzos en el desarrollo de medicamentos.
Productos de "Receptores acoplados de proteína G y receptores 7-TM"
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ML-335
CAS:ML-335, a μ-δ targeted agonist and MOR/DOR ligand, may lead to isomer-biased drugs with pain-relief properties.Fórmula:C25H32N2O3Pureza:98.52%Forma y color:SolidPeso molecular:408.53Ref: TM-T23002
2mg40,00€5mg62,00€10mg87,00€25mg170,00€50mg264,00€100mg380,00€200mg540,00€1mL*10mM (DMSO)35,00€Fananserin
CAS:Fananserin: Oral 5-HT2A antagonist (Ki=0.37 nM, rat), blocks human D4 receptor (Ki=2.93 nM).Fórmula:C23H24FN3O2SPureza:99.78%Forma y color:SolidPeso molecular:425.52Ref: TM-T15270
2mg42,00€5mg56,00€10mg81,00€25mg116,00€50mg170,00€100mg250,00€200mg369,00€1mL*10mM (DMSO)62,00€(S)-FTY720-phosphonate
CAS:FTY720 (S)-Phosphate, an S1P receptor 1 (S1PR1) agonist, is utilized in studying acute inflammatory diseases, including acute lung injury.Fórmula:C20H36NO4PPureza:98%Forma y color:SolidPeso molecular:385.48Pimavanserin tartrate
CAS:Pimavanserin tartrate is a potent 5-HT 2A receptor inverse agonist used to treat Parkinson's disease-related psychosis.Cost-effective and quality-assured.Fórmula:C50H68F2N6O4·C4H6O6Pureza:100% - 99.98%Forma y color:SolidPeso molecular:1005.2Amosulalol
CAS:Amosulalol is a combined alpha and beta adrenoceptor antagonist.Fórmula:C18H24N2O5SPureza:98.91%Forma y color:SolidPeso molecular:380.46Ref: TM-T30027
1mg185,00€2mg279,00€5mg425,00€10mg625,00€25mg938,00€50mg1.311,00€100mg1.795,00€1mL*10mM (DMSO)454,00€Adenosine amine congener
CAS:Adenosine amine congener (ADAC) (ADAC) is an agonist of selective A1 adenosine receptor,.Fórmula:C28H32N8O6Pureza:97.86%Forma y color:SolidPeso molecular:576.6Efloxate
CAS:Efloxate (Angorlisin), a vasodilator, is utilized in the treatment of chronic coronary insufficiency.Fórmula:C19H16O5Pureza:100%Forma y color:SolidPeso molecular:324.33Ziprasidone
CAS:Ziprasidone (Geodon) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.Fórmula:C21H21ClN4OSPureza:100% - 99.53%Forma y color:Tan SolidPeso molecular:412.94CYM50358
CAS:N-(4-(aminomethyl)-2,6-dimethylphenyl)-5 is a potent, selective antagonist of the sphingosine-1-phosphate receptor 4 (S1P4).Fórmula:C20H18Cl2N2O2Pureza:98.05% - 99.76%Forma y color:SolidPeso molecular:389.28Gastrin/CCK antagonist 1
CAS:Gastrin/CCK antagonist 1 is a potent gastrin/CCK antagonist for the study of metabolic system-related diseases.Fórmula:C28H32FN5O4Pureza:98.33%Forma y color:SolidPeso molecular:521.58Pranlukast
CAS:Cysteinyl leukotriene receptor antagonistFórmula:C27H23N5O4Pureza:Min. 95%Peso molecular:481.5 g/molIodophenpropit dihydrobromide
CAS:Iodophenpropit dihydrobromide: selective histamine H3 antagonist, reversible binding, high affinity (KD: 0.32 nM).Fórmula:C15H20BrIN4SPureza:98%Forma y color:SolidPeso molecular:495.22ATI-2341
CAS:ATI-2341, pepducin targeting the CXCR4, is an allosteric agonist activating the Gi to promote inhibition of cAMP production and induce calcium mobilization.Fórmula:C104H178N26O25S2Forma y color:SolidPeso molecular:2256.82Maropitant
CAS:Maropitant is a selective neurokinin (NK1) receptor antagonist.Fórmula:C32H40N2OPureza:97.35% - 99.75%Forma y color:SolidPeso molecular:468.67BMS-986224
CAS:BMS-986224 is an orally active, potent and selective APJ receptor agonist.BMS-986224 is a candidate compound for the treatment of heart failure.Fórmula:C24H23ClN4O6Pureza:98.61% - 98.82%Forma y color:SolidPeso molecular:498.92human GALP (3-32)
Human GALP (3-32) (Galanin-like peptide (3-32)) serves as a high-affinity agonist for galanin receptors GalR1 (IC50 = 33 nM) and GalR2 (IC50 = 15 nM), asFórmula:C137H213N43O38SPureza:98%Forma y color:SolidPeso molecular:3102.49(Rac)-Rotigotine hydrochloride
CAS:(Rac)-Rotigotine hydrochloride is a racemate of Rotigotine. Rotigotine is a full agonist of dopamine receptor, a partial the 5-HT1A receptor agonist.Fórmula:C19H26ClNOSForma y color:SolidPeso molecular:351.93GM-60186
GM-60186, a potent inhibitor of the 5-HT receptor 2B (HTR2B) with an IC50 of 257 nM, effectively suppresses the proliferation and migration of colorectal cancer cells.Fórmula:C30H33FN2O4Forma y color:SolidPeso molecular:504.59Docosahexaenoic acid ethyl ester
CAS:Docosahexaenoic acid ethyl ester (Ethyl docosahexaenoate) enhances 6-hydroxydopamine-induced neuronal damage by inducing lipid peroxidation in the mouse striatum, and can be used to study oxidative diseases of the retina or neurons.Fórmula:C24H36O2Forma y color:SolidPeso molecular:356.54ONO-8130
CAS:ONO-8130 is an orally available antagonist of EP1 receptor.Fórmula:C25H28N2O5S2Pureza:97.82%Forma y color:SolidPeso molecular:500.63
