Beta-bloqueante
Los betabloqueantes, también conocidos como agentes bloqueadores beta-adrenérgicos, son compuestos que bloquean la acción de la epinefrina (adrenalina) en los receptores beta, lo que reduce la frecuencia cardíaca y la presión arterial. A menudo se utilizan para tratar afecciones como la hipertensión, las arritmias y la insuficiencia cardíaca. En CymitQuimica, ofrecemos una variedad de betabloqueantes para fines de investigación en estudios cardiovasculares y clínicos.
Subcategorías de "Beta-bloqueante"
Productos de "Beta-bloqueante"
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Carvedilol EP Impurity B (Carvedilol USP Related Compound B) (Mixture of Diastereomers)
CAS:Fórmula:C39H39N3O6Forma y color:White To Off-White SolidPeso molecular:645.76Hydrochlorothiazide Dimer
CAS:Impurity Hydrochlorothiazide EP Impurity C Applications N-[[7-(Aminosulfonyl)-6-chloro-2,3-dihydro-1,1-dioxo-4H-1,2,4-benzothiadiazin-4-yl]methyl]-6-chloro-3,4-dihydro-1,1-dioxo-2H-1,2,4-benzothiadiazine-7-sulfonamide (Hydrochlorothiazide EP Impurity C) is an impurity in bulk Hydrochlorothiazide. Dimer Impurity C. References Daniels, S.L., et al.: J. Pharm. Sci., 70, 211 (1981), Fang, X., et al.: Pharm. Res., 14, 691 (1997),Fórmula:C15H16Cl2N6O8S4Forma y color:Off-WhitePeso molecular:607.495-Nitrosopyrimidine-2,4,6-triamine (Nitrosotriaminopyrimidine)
CAS:Producto controladoFórmula:C4H6N6OForma y color:NeatPeso molecular:154.13Carvedilol USP Related Compound D
CAS:Fórmula:C15H13NO2Forma y color:Pale Brown SolidPeso molecular:239.27Desfluoro Nebivolol (Mixture of Diastereomers)
CAS:Fórmula:C22H26FNO4Forma y color:White To Off-White SolidPeso molecular:387.45Nebivolol Impurity 15 HCl (Mixture of Diastereomers)
CAS:Fórmula:C29H31F2NO4·HClForma y color:White To Off-White SolidPeso molecular:495.57 36.462-[[2-[[(4RS)-4-(2-Chlorophenyl)-3-(ethoxycarbonyl)-5-(methoxycarbonyl)-6-methyl-1,4-dihydropyridin-2-yl]methoxy]ethyl]carbamoyl]benzoic Acid
CAS:Producto controladoFórmula:C28H29ClN2O8Forma y color:NeatPeso molecular:556.99Lovastatin-d9 (Mixture of Diastereomers)
CAS:Producto controladoApplications Lovastatin-d9, is the labeled analogue of Lovastatin (L472225), an antihypercholesterolemic agent. A fungal metabolite, which is a potent inhibitor of HMG-CoA reductase. References Bilheimer, D.W., et al.: Proc. Nat. Acad. Sci. USA, 80, 4124 (1983),Fórmula:C24H27D9O5Forma y color:NeatPeso molecular:413.6N,N'-Bis[2-(3,4-dimethoxyphenyl)ethyl]-N,N'-dimethylpropane-1,3-diamine Dihydrochloride
CAS:Producto controladoForma y color:Neat1-[4-(2-Methoxyethyl)phenoxy]-2,3-epoxypropane
CAS:Producto controladoFórmula:C12H16O3Forma y color:NeatPeso molecular:208.25Ezetimibe Tetrahydropyran Impurity
CAS:Impurity Ezetimibe Tetrahydropyran Impurity Applications Ezetimibe (E975000) tetrahydropyran impurity.Fórmula:C24H21F2NO3Forma y color:White To Off-WhitePeso molecular:409.43Ethyl Methyl 4-(2,3-Dichlorophenyl)-2,6-dimethylpyridine-3,5-dicarboxylate
CAS:Producto controladoFórmula:C18H17Cl2NO4Forma y color:NeatPeso molecular:382.24cis-7,10,13,16-Docosatetraenoic Acid Ethyl Ester-d5
CAS:Producto controladoApplications cis-7,10,13,16-Docosatetraenoic Acid Ethyl Ester-d5 is an isotopic analog of cis-7,10,13,16-Docosatetraenoic Acid Ethyl Ester. cis-7,10,13,16-Docosatetraenoic Acid Ethyl Ester is an ethyl analog of cis-7,10,13,16-Docosatetraenoic Acid (D494510). cis-7,10,13,16-Docosatetraenoic Acid has been identified as a protein kinase inhibitor, affecting serotonin levels in studies. References Mirnikjoo, B. et al.: J. Biol. Chem., 276, 10888 (2001);Fórmula:C24D5H35O2Forma y color:NeatPeso molecular:365.604p-Torasemide (1-(1-Methylethyl)-3-[[4-[(4-methylphenyl)amino]pyridin-3-yl]sulfonyl]urea)
CAS:Fórmula:C16H20N4O3SAlthiazide
CAS:Applications Diuretic and antihypertensive. References Twagirumukiza, M., et al.: Trop. Med. Int. Health, 15, 350 (2010), Gohil, V., et al.: Nat. Biotechnol., 28, 249 (2010), Peters, R., et al.: Anal. Bioanal. Chem., 396, 2583 (2010),Fórmula:C11H14ClN3O4S3Forma y color:NeatPeso molecular:383.895-[[4-[[2-(1-Methylethoxy)ethoxy]methyl]phenoxy]methyl]-3-(1-methylethyl)-2-oxazolidinone
CAS:Producto controladoForma y color:NeatCaptopril Methyl Ester
CAS:Producto controladoFórmula:C10H17NO3SForma y color:NeatPeso molecular:231.314’-Hydroxyphenyl Carvedilol
CAS:Producto controladoApplications A metabolite of Carvedilol (C184625). It is used in the treatment of hypertension. References Sponer, G., et al.: J. Cardiovasc. Pharmacol., 9, 317 (1987), Fujimaki, M., ET AL.: Xenobiotica, 20, 1025 (1990), Ruffolo, R., et al.: Eur. J. Clin. Pharmacol., 38, S82 (1990), Schaefer, W.H., et al.: Drug Metab. Dispos., 26, 10, 958 (1998),Fórmula:C24H26N2O5Forma y color:Off White SolidPeso molecular:422.47Fluocinolone Acetonide-21-aldehyde
CAS:Impurity Fluocinolone Acetonide EP Impurity D Stability Hygroscopic Applications Fluocinolone acetonide-21-aldehyde, is a derivative of Fluocinolone Acetonide (F455800), which is a Corticosteroid, used in dermatology to reduce skin inflammation and relieve itching. References Sammul, et al.: J. Assoc. Off. Agric. Chem., 47, 952 (1964), Emerson, M.V., et al.: BioDrugs, 21, 245 (2007),Fórmula:C24H28F2O6Forma y color:White To Light YellowPeso molecular:450.47Deiodo Amiodarone
CAS:Producto controladoImpurity Amiodarone EP Impurity C /Amiodarone USP Related Compound C Applications An intermediate of Amiodarone (A632950). Amiodarone EP Impurity C References Weir, S., et al.: J. Pharm. Sci., 74, 460 (1985), Ramanathan, R., et al.: Anal. Chem., 72, 1352 (2000),Fórmula:C25H30INO3Forma y color:NeatPeso molecular:519.415Esmolol hydrochloride
CAS:Esmolol is a cardioselective beta-blocker used in parenteral forms in the treatment of arrhythmias and severe hypertension.Fórmula:C16H25NO4·HClPureza:98.72% - 99.48%Forma y color:White SolidPeso molecular:331.15Bezafibrate 100 µg/mL in Acetonitrile
CAS:Producto controladoFórmula:C19H20ClNO4Forma y color:Single SolutionPeso molecular:361.82Carvedilol Impurity 12
CAS:Fórmula:C33H36N2O6Forma y color:White To Off-White SolidPeso molecular:556.66Hydroxyatenolol-d7
CAS:Producto controladoApplications Hydroxyatenolol-d7 is the isotope labelled analog of Hydroxyatenolol (H802480); a metabolite of Atenolol (A790075) which is a cardioselective β-adrenergic blocker, antihypertensive, antianginal, and antiarrhythmic (class II). References Escher, B., et al.: Environ. Sci. Technol., 40, 7402 (2006); Caplar, V., et al.: Anal. Profiles Drug Subs., 13, 1 (1984)Fórmula:C14H15D7N2O4Forma y color:NeatPeso molecular:289.38Simvastatin-d6
CAS:Producto controladoStability Hygroscopic Applications Deuterated Simvastatin, a competitive inhibitor of HMG-CoA reductase. A synthetic analog of Lovastatin. Antilipemic. References Hoffman, W.F., et al.: J. Med. Chem., 29, 849 (1986), Mol, M.J., et al.: Lancet, 2, 936 (1986),Fórmula:C25H32D6O5Forma y color:White To Off-WhitePeso molecular:424.6Nebivolol Impurity 21 (Mixture of Diastereomers)
CAS:Fórmula:C11H11FO2Forma y color:Colorless LiquidPeso molecular:194.21Desmethyl Ranolazine-d5
CAS:Producto controladoApplications A labelled metabolite of Ranolazine (R122500). References Chaitman, B.R., et al.: J. Am. Coll. Cardial., 43, 1375 (2004), McCormack, J.G., et al.: Gen. Pharmacol., 30, 639 (1998), Schofield, J.A.H., et al.: Expert Opin. Invest. Drugs, 11, 117 (2002),Fórmula:C23H26D5N3O4Forma y color:NeatPeso molecular:418.54Hexobendine Dihydrochloride
CAS:Producto controladoApplications Hexobendine is used as vasodilator (coronary). References Rdudolph, et al.: Arzneim.-Forsch., 20, 637 (1970), Kolassa, P., et al.: Biochem. Pharmacol., 20, 490 (1971), Zommer-Urbanska, S., et al.: Pharmazie, 40, 419 (1985),Fórmula:C30H44N2O10·2ClHForma y color:NeatPeso molecular:665.60Betamethasone 100 µg/mL in Acetonitrile
CAS:Fórmula:C22H29FO5Forma y color:Single SolutionPeso molecular:392.466-Methyl Pergolide
CAS:Producto controladoApplications 6-Methyl Pergolide is a potent antagonist of 5-HT2A and 5-HT2B receptors on porcine cardiac valves, it also activates brain dopaminergic receptors and lowers cranial DOPAC levels in rats (1,2). References (1) Fuller, R.W., et al.: Neuroendocrinol., 36, 285 (1983)(2) Goernemann, T., et al.: J. Pharmacol. Exp. Ther., 324, 1136 (2008)Fórmula:C17H22N2SForma y color:NeatPeso molecular:286.43N-Nitroso Nebivolol
CAS:Fórmula:C22H24F2N2O5Forma y color:White To Off-White SolidPeso molecular:434.445-(4-Fluorophenyl)-2,3-dihydro-3-(1-methylethyl)-2-oxo-N,4-diphenyl-1-[2-tetrahydro-4-hydroxy-6-oxo-2H-pyran-2-yl]ethyl]-1H-pyrrole-3-carboxamide
CAS:Producto controladoApplications 5-(4-Fluorophenyl)-2,3-dihydro-3-(1-methylethyl)-2-oxo-N,4-diphenyl-1-[2-tetrahydro-4-hydroxy-6-oxo-2H-pyran-2-yl]ethyl]-1H-pyrrole-3-carboxamide is a photodegradation product of Atorvastatin (A791750). References Cermola, F., et al.: Tetrahedron., 62, 7390 (2006);Fórmula:C33H33FN2O5Forma y color:NeatPeso molecular:556.62Metoprolol EP Impurity O-d7 HCl (Metoprolol USP Related Compound D-d7) (Mixture of Diastereomers)
CAS:Fórmula:C27H34D7NO6·HClPeso molecular:482.67 36.46Propranolol-d7 (Naphthalenyl-d7)
CAS:Fórmula:C16H14D7NO2Forma y color:White To Off-White SolidPeso molecular:266.39Atorvastatin-d5 Sodium Salt
CAS:Producto controladoStability Hygroscopic Applications A deuterated selective, competitive HMG-CoA reductase inhibitor. Atorvastatin is the only drug in its class specfically indicated for lowering both elevated LDL-cholesterol and triglycerides in patients with hypercholesterolemia. References Kearney, A.S., et al.: Pharm. Res., 10, 1461 (1993), Heinonen, T.M., et al.: Clin. Ther., 18, 853 (1996), Whitfield, L.R., et al.: Eur. J. Drug Metab. Pharmacokinet., 25, 97 (2000),Fórmula:C332H5H29FN2O5·NaPureza:>90%Forma y color:Off-White To Light BrownPeso molecular:585.651,1-Dimethyl-1-propanol-d6
CAS:Producto controladoFórmula:C5H6D6OForma y color:NeatPeso molecular:94.19Nebivolol Related Compound 3 HCl (Mixture of (RS,SR), (SR,SR) and (SR,RS) Isomers)
Fórmula:C22H25F2NO4·HClForma y color:White To Off-White SolidPeso molecular:405.45 36.46Amlodipine Mesilate
CAS:Producto controladoFórmula:C20H25ClN2O5Forma y color:NeatPeso molecular:408.88Atenolol
CAS:Producto controladoApplications Cardioselective β-adrenergic blocker. Antihypertensive, antianginal, antiarrhythmic (class II). References Caplar, V., et al.: Anal. Profiles Drug Subs., 13, 1 (1984),Fórmula:C14H22N2O3Forma y color:WhitePeso molecular:266.344-Hydroxy Atorvastatin Lactone-d5
CAS:Producto controladoApplications A labelled metabolite of Atorvastatin, a selective, competitive HMG-CoA reductase inhibitor. Atorvastatin is the only drug in its class specfically indicated for lowering both elevated LDL-cholesterol and triglycerides in patients with hypercholesterolemia.Fórmula:C332H5H28FN2O5Forma y color:NeatPeso molecular:561.65(2RS)-1-[4-(2-Butoxyethyl)phenoxy]-3-[(1-methylethyl)amino]propan-2-ol Hydrochloride
CAS:Forma y color:Neat(3R,5R)-6-Cyano-3,5-dihydroxy-hexanoic Acid tert-Butyl Ester
CAS:Producto controladoFórmula:C11H19NO4Forma y color:NeatPeso molecular:229.27rac-Diacetolol
CAS:Rac-Diacetolol is a racemic mixture of two isomers, (+) and (-), of acebutolol. Rac-Diacetolol is used to treat bowel disease, chronic oral inflammation and cardiac arrhythmias. It is also used as an experimental solubility probe in the study of the interactions between drugs and biological membranes. Rac-Diacetolol has been shown to have a low affinity for cytochrome P450 enzymes, which are responsible for metabolizing many drugs in the body. Rac-Diacetolol has been found to reduce plasma concentrations of PCSK9 antibody in patients with inflammatory bowel disease. The drug also has anti-inflammatory properties that may be due to its inhibition of prostaglandin synthesis.Fórmula:C16H24N2O4Pureza:Min. 95%Forma y color:PowderPeso molecular:308.37 g/molFosinopril USP Related Compound H
CAS:Producto controladoFórmula:C10H15O3PForma y color:NeatPeso molecular:214.20Olmesartan 100 µg/mL in Acetonitrile:Methanol
CAS:Producto controladoFórmula:C24H26N6O3Forma y color:Single SolutionPeso molecular:446.50Carvedilol N’-2-Hydroxy-3-[[2-(methoxyphenoxy)ethyl]amine
CAS:Producto controladoImpurity Carvedilol Impurity A; Carvedilol USP A Applications An impurity from the process of Carvedilol (C184625). Carvedilol impurity A. Carvedilol USP A.Fórmula:C36H43N3O7Forma y color:NeatPeso molecular:629.74O-Desmethylmetoprolol (1-(4-(2-hydroxyethyl)phenoxy)-3-(isopropylamino)propan-2-ol)
CAS:Amino-alcohols, other than those containing more than one kind of oxygen function, their ethers and esters, salts thereof, nesoiFórmula:C14H23NO3Forma y color:White Off-White SolidPeso molecular:253.16779Diazoxide
CAS:Producto controladoApplications Diazoxide reduces status epilepticus neuron damage in diabetes. A potassium channel opener References Baba, A., et al.: J. Neurosci., 23, 7737 (2003), Bancila, V., et al.: J. Neurochem., 90, 1243 (2004), Bancila, V., et al.: J. Biol. Chem., 280, 8793 (2005),Fórmula:C8H7ClN2O2SForma y color:NeatPeso molecular:230.677-Hydroxy Propranolol Glucuronide (Mixture of Diastereomers)
CAS:Fórmula:C22H29NO9Forma y color:White To Off-White SolidPeso molecular:451.48Carvedilol USP Related Compound E
CAS:Fórmula:C9H13NO2Forma y color:Yellowish-Brown LiquidPeso molecular:167.215-Oxorosuvastatin Methyl Ester
CAS:Producto controladoFórmula:C23H28FN3O6SForma y color:NeatPeso molecular:493.551-(3,4-Dihydroxyphenyl)-2-(methylamino)ethanone Hydrochloride (Adrenalone Hydrochloride)
CAS:Fórmula:C9H11NO3·ClH(2RS)-1-[Benzyl[2-(2-methoxyphenoxy)ethyl]amino]-3-(9H-carbazol-4-yloxy)propan-2-ol
CAS:Forma y color:Neat(2S)-2-[(3S,8aR)-3-(4-Aminobutyl)-1,4-dioxohexahydropyrrolo[1,2-a]pyrazin-2(1H)-yl]-4-phenylbutanoic Acid (R,S,S-Diketopiperazine)
CAS:Producto controladoFórmula:C21H29N3O4Forma y color:NeatPeso molecular:387.47Felodipine 100 µg/mL in Acetonitrile
CAS:Fórmula:C18H19Cl2NO4Forma y color:Single SolutionPeso molecular:384.25Dopamine-d4 Hydrochloride
CAS:Producto controladoApplications Labelled Dopamine. Endogenous catecholamine with α and β-adrenergic activity. Cardiotonic; antihypotensive. Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package References Carter, J.E., et al.: Anal. Profiles Drug Subs., 11, 257 (1982), Dasta, J.F., et al.: Pharmacotherapy, 6, 304 (1986),Fórmula:C8H4H7NO2·ClHForma y color:White To Light BrownPeso molecular:193.66Mexiletine-d6 Hydrochloride
CAS:Producto controladoStability Hygroscopic Applications Labelled Mexiletine (M340800). Antiarrhythmic (class IB). References Singh, E.M., et al.: Br. J. Pharmacol., 44, 1 (1972), Scott, K.N., et al.: Drug Metab. Dispos., 1, 506 (1973), Chew, C.Y.C., et al.: Drugs, 17, 161 (1979), Abounassif, M.A., et al.: Anal. Profiles Drug Subs., 20, 433 (1991),Fórmula:C11H12D6ClNOForma y color:White To Off-WhitePeso molecular:221.765'-Hydroxyphenyl Carvedilol-d5
CAS:Producto controladoApplications A Labelled metabolite of Carvedilol which is a multiple-action, neurohormonal antagonist that is used in the treatment of hypertension. References Schaefer, W.H., et al.: Drug Metab. Dispos., 26, 958 (1998).Fórmula:C24H21D5N2O5Forma y color:NeatPeso molecular:427.5Timolol EP Impurity F (Timolol USP Related Compound F)
CAS:Fórmula:C6H8ClN3OSForma y color:Pale Yellow To Off-White SolidPeso molecular:205.67(±)-Epinephrine hydrochloride
CAS:Producto controladoFórmula:C9H13NO3·ClHForma y color:NeatPeso molecular:219.67Betaxolol
CAS:Betaxolol (Kerlone) is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension and glaucoma.Fórmula:C18H29NO3Pureza:99.01%Forma y color:White Crystalline SolidPeso molecular:307.431-[4-(2-Methoxyethyl)phenoxy]propan-2-one
CAS:Producto controladoFórmula:C12H16O3Forma y color:NeatPeso molecular:208.25Dimethyl (4RS)-2-[(2-Aminoethoxy)methyl]-4-(2-chlorophenyl)-6-methyl-1,4-dihydropyridine-3,5-dicarboxylate
CAS:Producto controladoFórmula:C19H23ClN2O5Forma y color:NeatPeso molecular:394.854-(2,3-Epoxypropoxy)phenylacetamide
CAS:Impurity Atenolol EP Impurity C Applications 4-(2,3-Epoxypropoxy)phenylacetamide (Atenolol EP Impurity C) is an impurity of Atenolol, a cardioselective β-adrenergic blocker. References Caplar, V., et al.: Anal. Profiles Drug Subs., 13, 1 (1984)Fórmula:C11H13NO3Forma y color:NeatPeso molecular:207.23(3R,5R)-Rosuvastatin Sodium Salt
CAS:Impurity Rosuvastatin EP Impurity B Stability Hygroscopic Applications A diastereomer of Rosuvastatin (R700500) used for treatment, prevention and combination therapy of lipid-related disorders. Rosuvastatin EP Impurity BFórmula:C22H27FN3NaO6SForma y color:White To Light YellowPeso molecular:503.52(S)-Propranolol HCl
CAS:Fórmula:C16H21NO2·HClForma y color:White To Off-White SolidPeso molecular:259.35 36.46Metoprolol EP Impurity M DiHCl
CAS:Fórmula:C9H22N2O·2HClForma y color:White To Off-White SolidPeso molecular:174.29 2*36.46(S)-Propranolol Glucuronide
Fórmula:C22H29NO8Forma y color:White To Off-White SolidPeso molecular:435.48Bunitrolol
CAS:Applications Bunitrolol is a beta adrenoceptor antagonist that is used as an antihypertensive and antianginal agent. References Narimatsu, S., et al.: Chirality, 11, 1 (1999); Tsuchihashi, H., et al.: Jpn. J. Pharmacol., 45, 349 (1987)Fórmula:C14H20N2O2Forma y color:Colourless To Light YellowPeso molecular:248.32
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